AP2011005745A0 - Modulators of toll-like receptors. - Google Patents

Modulators of toll-like receptors.

Info

Publication number
AP2011005745A0
AP2011005745A0 AP2011000745A AP2011000745A AP2011005745A0 AP 2011005745 A0 AP2011005745 A0 AP 2011005745A0 AP 2011000745 A AP2011000745 A AP 2011000745A AP 2011000745 A AP2011000745 A AP 2011000745A AP 2011005745 A0 AP2011005745 A0 AP 2011005745A0
Authority
AP
ARIPO
Prior art keywords
toll
modulators
receptors
Prior art date
Application number
AP2011000745A
Other languages
English (en)
Inventor
Manoj C Desai
Ryan Mc Fadden
Randall L Halcomb
Original Assignee
Gilead Sciences Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41621203&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AP2011005745(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gilead Sciences Inc filed Critical Gilead Sciences Inc
Publication of AP2011005745A0 publication Critical patent/AP2011005745A0/xx

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
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    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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    • A61K31/7076—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines containing purines, e.g. adenosine, adenylic acid
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    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
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    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D475/00—Heterocyclic compounds containing pteridine ring systems
    • C07D475/06—Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D475/00—Heterocyclic compounds containing pteridine ring systems
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    • C07D475/06—Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4
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    • C07D487/04—Ortho-condensed systems
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    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
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  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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AP2011000745A 2008-12-09 2009-12-07 Modulators of toll-like receptors. AP2011005745A0 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US12106108P 2008-12-09 2008-12-09
US17040409P 2009-04-17 2009-04-17
US22438609P 2009-07-09 2009-07-09
US22737809P 2009-07-21 2009-07-21
US24263509P 2009-09-15 2009-09-15

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AP2011005745A0 true AP2011005745A0 (en) 2011-06-30

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AP2011000745A AP2011005745A0 (en) 2008-12-09 2009-12-07 Modulators of toll-like receptors.

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US (8) US8367670B2 (xx)
EP (3) EP2818469B1 (xx)
JP (3) JP5600116B2 (xx)
KR (2) KR101787309B1 (xx)
CN (2) CN103497192B (xx)
AP (1) AP2011005745A0 (xx)
AR (1) AR074506A1 (xx)
AU (1) AU2009333559B2 (xx)
BR (1) BRPI0923305B1 (xx)
CA (1) CA2745295C (xx)
CL (1) CL2011001392A1 (xx)
CO (1) CO6362010A2 (xx)
CY (1) CY1115176T1 (xx)
DK (1) DK2364314T3 (xx)
EA (3) EA026557B1 (xx)
EC (2) ECSP11011189A (xx)
ES (2) ES2467108T3 (xx)
HK (2) HK1161880A1 (xx)
HR (1) HRP20140539T1 (xx)
IL (2) IL213101A (xx)
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PE (1) PE20120106A1 (xx)
PL (1) PL2364314T3 (xx)
PT (2) PT2364314E (xx)
RS (1) RS53347B (xx)
SG (1) SG172060A1 (xx)
SI (1) SI2364314T1 (xx)
SM (1) SMT201400083B (xx)
TW (5) TWI480268B (xx)
UY (1) UY32306A (xx)
WO (1) WO2010077613A1 (xx)
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Families Citing this family (236)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PE20120106A1 (es) 2008-12-09 2012-02-20 Gilead Sciences Inc Moduladores de receptores tipo toll
DK2459216T3 (da) 2009-09-02 2013-12-09 Novartis Ag Immunogene sammensætninger omfattende tlr-aktivitetsmodulatorer
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US8629142B2 (en) 2014-01-14
ECSP11011310A (es) 2011-10-31
US9127006B2 (en) 2015-09-08
JP5945567B2 (ja) 2016-07-05
CA2745295A1 (en) 2010-07-08
US11110091B2 (en) 2021-09-07
CN103497192A (zh) 2014-01-08
CN102272134B (zh) 2013-10-16
US20180085370A1 (en) 2018-03-29
EP2818469B1 (en) 2017-02-15
EA021377B9 (ru) 2015-09-30
ES2467108T3 (es) 2014-06-11
BRPI0923305B1 (pt) 2019-01-22
US20170065592A1 (en) 2017-03-09
ES2623794T3 (es) 2017-07-12

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