LT3030227T - Prailginto atpalaidavimo jak1 inhibitoriaus dozavimo formos - Google Patents

Prailginto atpalaidavimo jak1 inhibitoriaus dozavimo formos

Info

Publication number
LT3030227T
LT3030227T LTEP14753182.6T LT14753182T LT3030227T LT 3030227 T LT3030227 T LT 3030227T LT 14753182 T LT14753182 T LT 14753182T LT 3030227 T LT3030227 T LT 3030227T
Authority
LT
Lithuania
Prior art keywords
dosage forms
sustained release
release dosage
jak1 inhibitor
jak1
Prior art date
Application number
LTEP14753182.6T
Other languages
English (en)
Inventor
Krishnaswamy Yeleswaram
Bhavnish Parikh
Dilip P. MODI
Trupti SHETH
Original Assignee
Incyte Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Incyte Corporation filed Critical Incyte Corporation
Publication of LT3030227T publication Critical patent/LT3030227T/lt

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2009—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
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    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
    • A—HUMAN NECESSITIES
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    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
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    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
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    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
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    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/14—Drugs for disorders of the endocrine system of the thyroid hormones, e.g. T3, T4
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    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
    • A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Neurology (AREA)
  • Dermatology (AREA)
  • Hematology (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Endocrinology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Inorganic Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychiatry (AREA)
  • Emergency Medicine (AREA)
  • Transplantation (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Cardiology (AREA)
  • Oncology (AREA)
LTEP14753182.6T 2013-08-07 2014-08-06 Prailginto atpalaidavimo jak1 inhibitoriaus dozavimo formos LT3030227T (lt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361863325P 2013-08-07 2013-08-07
US201361913066P 2013-12-06 2013-12-06
PCT/US2014/049940 WO2015021153A1 (en) 2013-08-07 2014-08-06 Sustained release dosage forms for a jak1 inhibitor

Publications (1)

Publication Number Publication Date
LT3030227T true LT3030227T (lt) 2020-06-10

Family

ID=51383933

Family Applications (1)

Application Number Title Priority Date Filing Date
LTEP14753182.6T LT3030227T (lt) 2013-08-07 2014-08-06 Prailginto atpalaidavimo jak1 inhibitoriaus dozavimo formos

Country Status (30)

Country Link
US (4) US9655854B2 (lt)
EP (2) EP3721873A1 (lt)
JP (5) JP6334700B2 (lt)
KR (3) KR20220103810A (lt)
CN (3) CN116036089A (lt)
AU (3) AU2014305989B2 (lt)
BR (1) BR122020001831A8 (lt)
CA (2) CA2920108C (lt)
CL (1) CL2016000292A1 (lt)
CR (3) CR20230316A (lt)
CY (1) CY1123314T1 (lt)
DK (1) DK3030227T3 (lt)
EA (1) EA201690357A1 (lt)
ES (1) ES2792549T3 (lt)
HR (1) HRP20200955T1 (lt)
HU (1) HUE049345T2 (lt)
IL (2) IL277554B2 (lt)
LT (1) LT3030227T (lt)
MX (2) MX2016001639A (lt)
MY (1) MY195091A (lt)
PE (2) PE20160223A1 (lt)
PH (3) PH12016500243B1 (lt)
PL (1) PL3030227T3 (lt)
PT (1) PT3030227T (lt)
RS (1) RS60469B1 (lt)
SG (3) SG11201600815WA (lt)
SI (1) SI3030227T1 (lt)
TW (3) TWI789516B (lt)
UA (1) UA120499C2 (lt)
WO (1) WO2015021153A1 (lt)

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DK3030227T3 (da) 2020-04-20
TW202320789A (zh) 2023-06-01
EP3030227B1 (en) 2020-04-08
CA2920108A1 (en) 2015-02-12
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JP2020079317A (ja) 2020-05-28
US10561616B2 (en) 2020-02-18
PT3030227T (pt) 2020-06-25
CR20160102A (es) 2016-07-28
MX2019013381A (es) 2020-02-20
AU2014305989A1 (en) 2016-03-10
US20220016036A1 (en) 2022-01-20
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WO2015021153A1 (en) 2015-02-12
PH12019502074A1 (en) 2020-02-24
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AU2019257368B2 (en) 2021-02-25
CA3155500A1 (en) 2015-02-12
CN105579032A (zh) 2016-05-11
CN114010611A (zh) 2022-02-08
KR102419714B1 (ko) 2022-07-13
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MX2016001639A (es) 2016-10-07
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PH12019502072A1 (en) 2020-07-13
AU2014305989B2 (en) 2019-11-28
HRP20200955T1 (hr) 2020-10-02
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NZ717230A (en) 2021-05-28
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