CY1123314T1 - Μορφες δοσολογιας παρατεταμενης απελευθερωσης για αναστολεα jak1 - Google Patents

Μορφες δοσολογιας παρατεταμενης απελευθερωσης για αναστολεα jak1

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Publication number
CY1123314T1
CY1123314T1 CY20201100572T CY201100572T CY1123314T1 CY 1123314 T1 CY1123314 T1 CY 1123314T1 CY 20201100572 T CY20201100572 T CY 20201100572T CY 201100572 T CY201100572 T CY 201100572T CY 1123314 T1 CY1123314 T1 CY 1123314T1
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CY
Cyprus
Prior art keywords
dosage forms
release dosage
extended release
jak1 inhibitor
jak1
Prior art date
Application number
CY20201100572T
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English (en)
Inventor
Krishnaswamy Yeleswaram
Bhavnish Parikh
Dilip P. MODI
Trupti SHETH
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Incyte Corporation
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Publication date
Application filed by Incyte Corporation filed Critical Incyte Corporation
Publication of CY1123314T1 publication Critical patent/CY1123314T1/el

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    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
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    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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Abstract

Η εφεύρεση αυτή αφορά σε μορφές δοσολογίας παρατεταμένης απελευθέρωσης που περιλαμβάνουν {1 -{1 -[3-φθορο-2-(τριφθορομεθυλ)ισονικοτινοϋλ]πιπεριδιν-4-υλ}-3-[4-(7Η-πυρρολο[2,3-d]πυριμιδιν-4-υλ)- 1Η-πυραζολ-1-υλ]αζετιδιν-3-υλ}ακετονιτρίλιο, ή φαρμακευτικώς αποδεκτό άλας αυτού, και δόσεις και μεθόδους που σχετίζονται με αυτό.
CY20201100572T 2013-08-07 2020-06-23 Μορφες δοσολογιας παρατεταμενης απελευθερωσης για αναστολεα jak1 CY1123314T1 (el)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361863325P 2013-08-07 2013-08-07
US201361913066P 2013-12-06 2013-12-06
PCT/US2014/049940 WO2015021153A1 (en) 2013-08-07 2014-08-06 Sustained release dosage forms for a jak1 inhibitor

Publications (1)

Publication Number Publication Date
CY1123314T1 true CY1123314T1 (el) 2021-12-31

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Country Status (30)

Country Link
US (4) US9655854B2 (el)
EP (2) EP3721873A1 (el)
JP (5) JP6334700B2 (el)
KR (3) KR20220103810A (el)
CN (3) CN105579032A (el)
AU (3) AU2014305989B2 (el)
BR (1) BR122020001831A8 (el)
CA (2) CA2920108C (el)
CL (1) CL2016000292A1 (el)
CR (3) CR20190343A (el)
CY (1) CY1123314T1 (el)
DK (1) DK3030227T3 (el)
EA (1) EA201690357A1 (el)
ES (1) ES2792549T3 (el)
HR (1) HRP20200955T1 (el)
HU (1) HUE049345T2 (el)
IL (2) IL277554B2 (el)
LT (1) LT3030227T (el)
MX (2) MX2016001639A (el)
MY (1) MY195091A (el)
PE (2) PE20220579A1 (el)
PH (3) PH12016500243B1 (el)
PL (1) PL3030227T3 (el)
PT (1) PT3030227T (el)
RS (1) RS60469B1 (el)
SG (3) SG10201801069QA (el)
SI (1) SI3030227T1 (el)
TW (3) TWI730935B (el)
UA (1) UA120499C2 (el)
WO (1) WO2015021153A1 (el)

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