US2985589A
(en)
|
1957-05-22 |
1961-05-23 |
Universal Oil Prod Co |
Continuous sorption process employing fixed bed of sorbent and moving inlets and outlets
|
US3632836A
(en)
|
1968-10-25 |
1972-01-04 |
Dow Chemical Co |
Solid curable polyepoxides modified with hydrolyzed liquid polyepoxides
|
US3832460A
(en)
|
1971-03-19 |
1974-08-27 |
C Kosti |
Anesthetic-vasoconstrictor-antihistamine composition for the treatment of hypertrophied oral tissue
|
US4140755A
(en)
|
1976-02-13 |
1979-02-20 |
Hoffmann-La Roche Inc. |
Sustained release tablet formulations
|
DE3036390A1
(de)
|
1980-09-26 |
1982-05-13 |
Troponwerke GmbH & Co KG, 5000 Köln |
Neue pyrrolo-pyrimidine, verfahren zu ihrer herstellung und ihre verwendung bei der herstellung von biologischen wirkstoffen
|
DE3220113A1
(de)
|
1982-05-28 |
1983-12-01 |
Basf Ag, 6700 Ludwigshafen |
Difluormethoxiphenylthiophosphorsaeureester
|
US4402832A
(en)
|
1982-08-12 |
1983-09-06 |
Uop Inc. |
High efficiency continuous separation process
|
US4404335A
(en)
|
1982-08-16 |
1983-09-13 |
The Dow Chemical Company |
Hydrolyzing epoxy resins in absence of solvent and in presence of oxalic acid and a phosphonium compound
|
US4548990A
(en)
|
1983-08-15 |
1985-10-22 |
Ciba-Geigy Corporation |
Crosslinked, porous polymers for controlled drug delivery
|
US4498991A
(en)
|
1984-06-18 |
1985-02-12 |
Uop Inc. |
Serial flow continuous separation process
|
NL8403224A
(nl)
|
1984-10-24 |
1986-05-16 |
Oce Andeno Bv |
Dioxafosforinanen, de bereiding ervan en de toepassing voor het splitsen van optisch actieve verbindingen.
|
CA1306260C
(en)
|
1985-10-18 |
1992-08-11 |
Shionogi & Co., Ltd. |
Condensed imidazopyridine derivatives
|
CA2067221C
(en)
|
1989-10-11 |
1997-04-15 |
Yasuji Sakuma |
Fused pyrimidine derivative, process for preparation of same and pharmaceutical preparation comprising same as active ingredient
|
US5403593A
(en)
|
1991-03-04 |
1995-04-04 |
Sandoz Ltd. |
Melt granulated compositions for preparing sustained release dosage forms
|
IT1258781B
(it)
|
1992-01-16 |
1996-02-29 |
Zambon Spa |
Composizione farmaceutica oftalmica contenente n-acetilcisteina e polivinilalcol
|
US5521184A
(en)
|
1992-04-03 |
1996-05-28 |
Ciba-Geigy Corporation |
Pyrimidine derivatives and processes for the preparation thereof
|
FR2695126B1
(fr)
|
1992-08-27 |
1994-11-10 |
Sanofi Elf |
Dérivés d'acide thiényl ou pyrrolyl carboxyliques, leur préparation et médicaments les contenant.
|
AU671491B2
(en)
|
1992-12-18 |
1996-08-29 |
F. Hoffmann-La Roche Ag |
N-oxycarbonyl substituted 5'-deoxy-5-fluorcytidines
|
JPH0710876A
(ja)
|
1993-06-24 |
1995-01-13 |
Teijin Ltd |
4位に環状アミノ基を有するピロロ[2,3―d]ピリミジン
|
USH1439H
(en)
|
1993-10-18 |
1995-05-02 |
The Dow Chemical Company |
Method to increase the level of α-glycol in liquid epoxy resin
|
EP0727217A3
(en)
|
1995-02-10 |
1997-01-15 |
Suntory Ltd |
Pharmaceutical and cosmetic compositions containing God-type ellagitannin as an active ingredient
|
IL117580A0
(en)
|
1995-03-29 |
1996-07-23 |
Merck & Co Inc |
Inhibitors of farnesyl-protein transferase and pharmaceutical compositions containing them
|
US5856326A
(en)
|
1995-03-29 |
1999-01-05 |
Merck & Co., Inc. |
Inhibitors of farnesyl-protein transferase
|
BR9609613A
(pt)
|
1995-07-05 |
1999-05-25 |
Du Pont |
Composto composição fungicida e método de controle de doenças de plantas
|
DE69619114T2
(de)
|
1995-07-06 |
2002-10-02 |
Novartis Ag, Basel |
Pyrolopyrimidine und verfahren zu ihrer herstellung
|
US5630943A
(en)
|
1995-11-30 |
1997-05-20 |
Merck Patent Gesellschaft Mit Beschrankter Haftung |
Discontinuous countercurrent chromatographic process and apparatus
|
GB9604361D0
(en)
|
1996-02-29 |
1996-05-01 |
Pharmacia Spa |
4-Substituted pyrrolopyrimidine compounds as tyrosine kinase inhibitors
|
CA2250232A1
(en)
|
1996-04-03 |
1997-10-09 |
Allen I. Oliff |
A method of treating cancer
|
AU2802297A
(en)
|
1996-04-18 |
1997-11-07 |
Merck & Co., Inc. |
A method of treating cancer
|
US5795909A
(en)
|
1996-05-22 |
1998-08-18 |
Neuromedica, Inc. |
DHA-pharmaceutical agent conjugates of taxanes
|
JP2000508335A
(ja)
|
1996-05-30 |
2000-07-04 |
メルク エンド カンパニー インコーポレーテッド |
癌の治療方法
|
US6624138B1
(en)
|
2001-09-27 |
2003-09-23 |
Gp Medical |
Drug-loaded biological material chemically treated with genipin
|
WO1998044797A1
(en)
|
1997-04-07 |
1998-10-15 |
Merck & Co., Inc. |
A method of treating cancer
|
US6063284A
(en)
|
1997-05-15 |
2000-05-16 |
Em Industries, Inc. |
Single column closed-loop recycling with periodic intra-profile injection
|
US6060038A
(en)
|
1997-05-15 |
2000-05-09 |
Merck & Co., Inc. |
Radiolabeled farnesyl-protein transferase inhibitors
|
CA2295620A1
(en)
|
1997-08-11 |
1999-02-18 |
Boehringer Ingelheim Pharmaceuticals, Inc. |
5,6-heteroaryl-dipyrido¬2,3-b:3',2'-f|azepines and their use in the prevention or treatment of hiv infection
|
US7153845B2
(en)
|
1998-08-25 |
2006-12-26 |
Columbia Laboratories, Inc. |
Bioadhesive progressive hydration tablets
|
US6075056A
(en)
|
1997-10-03 |
2000-06-13 |
Penederm, Inc. |
Antifungal/steroid topical compositions
|
US6025366A
(en)
|
1998-04-02 |
2000-02-15 |
Merck & Co., Inc. |
Antagonists of gonadotropin releasing hormone
|
US6232320B1
(en)
|
1998-06-04 |
2001-05-15 |
Abbott Laboratories |
Cell adhesion-inhibiting antiinflammatory compounds
|
CN1332743A
(zh)
|
1998-06-04 |
2002-01-23 |
艾博特公司 |
抑制细胞粘附抗炎化合物
|
PA8474101A1
(es)
|
1998-06-19 |
2000-09-29 |
Pfizer Prod Inc |
Compuestos de pirrolo [2,3-d] pirimidina
|
ID26698A
(id)
|
1998-06-19 |
2001-02-01 |
Pfizer Prod Inc |
SENYAWA-SENYAWA PIROLO [2,3-d] PIRIMIDINA
|
JP4516690B2
(ja)
|
1998-08-11 |
2010-08-04 |
ノバルティス アーゲー |
血管形成阻害活性を有するイソキノリン誘導体
|
JP2000119271A
(ja)
|
1998-08-12 |
2000-04-25 |
Hokuriku Seiyaku Co Ltd |
1h―イミダゾピリジン誘導体
|
JP5026635B2
(ja)
|
1998-09-10 |
2012-09-12 |
ニュコメデ ダンマルク アンパーツセルスカブ |
医薬物質の迅速放出医薬組成物
|
US6413419B1
(en)
|
1998-10-29 |
2002-07-02 |
Institut Francais Du Petrole |
Process and device for separation with variable-length chromatographic
|
FR2785196B1
(fr)
|
1998-10-29 |
2000-12-15 |
Inst Francais Du Petrole |
Procede et dispositif de separation avec des zones chromatographiques a longueur variable
|
US6375839B1
(en)
|
1998-10-29 |
2002-04-23 |
Institut Francais Du Petrole |
Process and device for separation with variable-length chromatographic zones
|
US6133031A
(en)
|
1999-08-19 |
2000-10-17 |
Isis Pharmaceuticals Inc. |
Antisense inhibition of focal adhesion kinase expression
|
EP1165084A4
(en)
|
1999-03-03 |
2002-05-15 |
Merck & Co Inc |
PRENYL PROTEIN TRANSFERASES INHIBITORS
|
GB9905075D0
(en)
|
1999-03-06 |
1999-04-28 |
Zeneca Ltd |
Chemical compounds
|
US6217895B1
(en)
|
1999-03-22 |
2001-04-17 |
Control Delivery Systems |
Method for treating and/or preventing retinal diseases with sustained release corticosteroids
|
US6239113B1
(en)
|
1999-03-31 |
2001-05-29 |
Insite Vision, Incorporated |
Topical treatment or prevention of ocular infections
|
AU3565999A
(en)
|
1999-04-16 |
2000-11-02 |
Coelacanth Chemical Corporation |
Synthesis of azetidine derivatives
|
US6921763B2
(en)
|
1999-09-17 |
2005-07-26 |
Abbott Laboratories |
Pyrazolopyrimidines as therapeutic agents
|
ATE275141T1
(de)
|
1999-10-13 |
2004-09-15 |
Banyu Pharma Co Ltd |
Substituierte imidazolin-derivate
|
US7235258B1
(en)
|
1999-10-19 |
2007-06-26 |
Nps Pharmaceuticals, Inc. |
Sustained-release formulations for treating CNS-mediated disorders
|
DE60007552T2
(de)
|
1999-12-10 |
2004-09-23 |
Pfizer Products Inc., Groton |
PYRROLO[2,3-d]PYRIMIDIN-VERBINDUNGEN ALS PROTEIN KINASEN HEMMER
|
OA12514A
(en)
|
1999-12-24 |
2006-05-29 |
Aventis Pharma Ltd |
Azaindoles.
|
GB0004890D0
(en)
|
2000-03-01 |
2000-04-19 |
Astrazeneca Uk Ltd |
Chemical compounds
|
US7235551B2
(en)
|
2000-03-02 |
2007-06-26 |
Smithkline Beecham Corporation |
1,5-disubstituted-3,4-dihydro-1h-pyrimido[4,5-d]pyrimidin-2-one compounds and their use in treating csbp/p38 kinase mediated diseases
|
DE60100866T2
(de)
|
2000-04-07 |
2004-07-29 |
Laboratoire Medidom S.A. |
Cyklosporin, Hyaluronsäure und Polysorbate enthaltenes Augenarzneimittel
|
AU4878601A
(en)
|
2000-04-20 |
2001-11-07 |
Mitsubishi Corporation |
Aromatic amide compounds
|
ES2527754T3
(es)
|
2000-04-25 |
2015-01-29 |
Icos Corporation |
Inhibidores de la isoforma delta de la fosfatidilinositol 3-quinasa humana
|
US7498304B2
(en)
|
2000-06-16 |
2009-03-03 |
Curis, Inc. |
Angiogenesis-modulating compositions and uses
|
US20030022819A1
(en)
|
2000-06-16 |
2003-01-30 |
Ling Leona E. |
Angiogenesis-modulating compositions and uses
|
US6335342B1
(en)
|
2000-06-19 |
2002-01-01 |
Pharmacia & Upjohn S.P.A. |
Azaindole derivatives, process for their preparation, and their use as antitumor agents
|
AU2001274598A1
(en)
|
2000-06-23 |
2002-01-02 |
Mitsubishi Pharma Corporation |
Antitumor effect potentiators
|
DE60137734D1
(de)
|
2000-06-26 |
2009-04-02 |
Pfizer Prod Inc |
PyrroloÄ2,3-DÜpyrimidin Verbindungen als Immunosuppressive Wirkstoffe
|
EP1294358B1
(en)
|
2000-06-28 |
2004-08-18 |
Smithkline Beecham Plc |
Wet milling process
|
WO2002016370A1
(fr)
|
2000-08-22 |
2002-02-28 |
Hokuriku Seiyaku Co., Ltd. |
Derives de 1h-imidazopyridine
|
AU2002228783A1
(en)
|
2000-12-05 |
2002-06-18 |
Vertex Pharmaceuticals Incorporated |
Inhibitors of c-jun n-terminal kinases (jnk) and other protein kinases
|
GB0100622D0
(en)
|
2001-01-10 |
2001-02-21 |
Vernalis Res Ltd |
Chemical compounds V111
|
US20040077654A1
(en)
|
2001-01-15 |
2004-04-22 |
Bouillot Anne Marie Jeanne |
Aryl piperidine and piperazine derivatives as inducers of ldl-receptor expression
|
JP2004528295A
(ja)
|
2001-01-30 |
2004-09-16 |
サイトピア ピーティワイ リミテッド |
キナーゼ阻害方法
|
CA2446864C
(en)
|
2001-05-16 |
2011-02-15 |
Vertex Pharmaceuticals Incorporated |
Inhibitors of src and other protein kinases
|
US7301023B2
(en)
|
2001-05-31 |
2007-11-27 |
Pfizer Inc. |
Chiral salt resolution
|
GB0115109D0
(en)
|
2001-06-21 |
2001-08-15 |
Aventis Pharma Ltd |
Chemical compounds
|
GB0115393D0
(en)
|
2001-06-23 |
2001-08-15 |
Aventis Pharma Ltd |
Chemical compounds
|
WO2003011285A1
(en)
|
2001-08-01 |
2003-02-13 |
Merck & Co., Inc. |
BENZIMIDAZO[4,5-f]ISOQUINOLINONE DERIVATIVES
|
AU2002337142B2
(en)
|
2001-09-19 |
2007-10-11 |
Aventis Pharma S.A. |
Indolizines as kinase protein inhibitors
|
US6429231B1
(en)
|
2001-09-24 |
2002-08-06 |
Bradley Pharmaceuticals, Inc. |
Compositions containing antimicrobials and urea for the treatment of dermatological disorders and methods for their use
|
DK1441737T3
(da)
|
2001-10-30 |
2006-11-13 |
Novartis Ag |
Staurosporin-derivater som inhibitorer af FLT3-receptor-tyrosinkinase-aktivitet
|
JP2003155285A
(ja)
|
2001-11-19 |
2003-05-27 |
Toray Ind Inc |
環状含窒素誘導体
|
US6949668B2
(en)
|
2001-11-30 |
2005-09-27 |
Teijin Limited |
Process for producing 5-(3-cyanophenyl)-3-formylbenzoic acid compound
|
GT200200234A
(es)
|
2001-12-06 |
2003-06-27 |
|
Compuestos cristalinos novedosos
|
US6995144B2
(en)
|
2002-03-14 |
2006-02-07 |
Eisai Co., Ltd. |
Nitrogen containing heterocyclic compounds and medicines containing the same
|
AU2003237807B2
(en)
|
2002-04-15 |
2008-10-23 |
Rb Health (Us) Llc |
Sustained release of guaifenesin combination drugs
|
TW200403058A
(en)
|
2002-04-19 |
2004-03-01 |
Bristol Myers Squibb Co |
Heterocyclo inhibitors of potassium channel function
|
US7304061B2
(en)
|
2002-04-26 |
2007-12-04 |
Vertex Pharmaceuticals Incorporated |
Heterocyclic inhibitors of ERK2 and uses thereof
|
ATE381332T1
(de)
|
2002-05-02 |
2008-01-15 |
Merck & Co Inc |
Tyrosinkinase-hemmer
|
EP1503731A1
(en)
|
2002-05-07 |
2005-02-09 |
Control Delivery Systems, Inc. |
Processes for forming a drug delivery device
|
CN100558715C
(zh)
|
2002-05-23 |
2009-11-11 |
西托匹亚有限公司 |
蛋白激酶抑制剂
|
TW200406374A
(en)
|
2002-05-29 |
2004-05-01 |
Novartis Ag |
Diaryl urea derivatives useful for the treatment of protein kinase dependent diseases
|
US7385018B2
(en)
|
2002-06-26 |
2008-06-10 |
Idemitsu Kosan Co., Ltd. |
Hydrogenated copolymer, process for producing the same, and hot-melt adhesive composition containing the same
|
GB0215676D0
(en)
|
2002-07-05 |
2002-08-14 |
Novartis Ag |
Organic compounds
|
GB0215844D0
(en)
|
2002-07-09 |
2002-08-14 |
Novartis Ag |
Organic compounds
|
EP1541563A4
(en)
|
2002-07-10 |
2007-11-07 |
Ono Pharmaceutical Co |
ANTAGONIST OF CCR4 AND CORRESPONDING MEDICINAL USE
|
BR0314603A
(pt)
|
2002-09-20 |
2005-07-26 |
Alcon Inc |
Uso de inibidores da sìntese de citoquina para o tratamento de distúrbios de olhos secos
|
US20040204404A1
(en)
|
2002-09-30 |
2004-10-14 |
Robert Zelle |
Human N-type calcium channel blockers
|
ES2289349T3
(es)
|
2002-11-04 |
2008-02-01 |
Vertex Pharmaceuticals Incorporated |
Derivados de heteroaril-pirimidina como inhibidores de jak.
|
US8034831B2
(en)
|
2002-11-06 |
2011-10-11 |
Celgene Corporation |
Methods for the treatment and management of myeloproliferative diseases using 4-(amino)-2-(2,6-Dioxo(3-piperidyl)-isoindoline-1,3-dione in combination with other therapies
|
CL2003002353A1
(es)
|
2002-11-15 |
2005-02-04 |
Vertex Pharma |
Compuestos derivados de diaminotriazoles, inhibidores d ela proteina quinasa; composicion farmaceutica; procedimiento de preparacion; y su uso del compuesto en el tratamiento de enfermedades de desordenes alergicos, proliferacion, autoinmunes, condic
|
US20040099204A1
(en)
|
2002-11-25 |
2004-05-27 |
Nestor John J. |
Sheet, page, line, position marker
|
AU2003276591A1
(en)
|
2002-11-26 |
2004-06-18 |
Pfizer Products Inc. |
Method of treatment of transplant rejection
|
UA80767C2
(en)
|
2002-12-20 |
2007-10-25 |
Pfizer Prod Inc |
Pyrimidine derivatives for the treatment of abnormal cell growth
|
UY28126A1
(es)
|
2002-12-24 |
2004-06-30 |
Alcon Inc |
Uso de glucocorticoides selectivos para la superficie ocular en el tratamiento de la sequedad ocular
|
US7135493B2
(en)
|
2003-01-13 |
2006-11-14 |
Astellas Pharma Inc. |
HDAC inhibitor
|
US7444183B2
(en)
|
2003-02-03 |
2008-10-28 |
Enteromedics, Inc. |
Intraluminal electrode apparatus and method
|
AU2004212421B2
(en)
|
2003-02-07 |
2009-08-20 |
Vertex Pharmaceuticals Incorporated |
Heteroaryl substituted pyrolls useful as inhibitors of protein kinases
|
GB0305929D0
(en)
|
2003-03-14 |
2003-04-23 |
Novartis Ag |
Organic compounds
|
US7547794B2
(en)
|
2003-04-03 |
2009-06-16 |
Vertex Pharmaceuticals Incorporated |
Compositions useful as inhibitors of protein kinases
|
SE0301373D0
(sv)
|
2003-05-09 |
2003-05-09 |
Astrazeneca Ab |
Novel compounds
|
SE0301372D0
(sv)
|
2003-05-09 |
2003-05-09 |
Astrazeneca Ab |
Novel compounds
|
FR2857454B1
(fr)
|
2003-07-08 |
2006-08-11 |
Aventis Pasteur |
Dosage des acides techoiques des bacteries gram+
|
US20050043346A1
(en)
|
2003-08-08 |
2005-02-24 |
Pharmacia Italia S.P.A. |
Pyridylpyrrole derivatives active as kinase inhibitors
|
WO2005020921A2
(en)
|
2003-08-29 |
2005-03-10 |
Exelixis, Inc. |
C-kit modulators and methods of use
|
EP1678147B1
(en)
|
2003-09-15 |
2012-08-08 |
Lead Discovery Center GmbH |
Pharmaceutically active 4,6-disubstituted aminopyrimidine derivatives as modulators of protein kinases
|
AR045944A1
(es)
|
2003-09-24 |
2005-11-16 |
Novartis Ag |
Derivados de isoquinolina 1.4-disustituidas
|
DK1679074T3
(da)
|
2003-10-24 |
2011-03-21 |
Santen Pharmaceutical Co Ltd |
Terapeutisk middel til keratoconjunktive forstyrrelser
|
US7387793B2
(en)
|
2003-11-14 |
2008-06-17 |
Eurand, Inc. |
Modified release dosage forms of skeletal muscle relaxants
|
MY141220A
(en)
|
2003-11-17 |
2010-03-31 |
Astrazeneca Ab |
Pyrazole derivatives as inhibitors of receptor tyrosine kinases
|
BRPI0416909A
(pt)
|
2003-11-25 |
2007-01-16 |
Pfizer Prod Inc |
método de tratamento de aterosclerose
|
CN1893952A
(zh)
|
2003-12-17 |
2007-01-10 |
辉瑞产品公司 |
用于治疗移植排斥的吡咯并[2,3-d]嘧啶化合物
|
CA2550189A1
(en)
|
2003-12-19 |
2005-07-21 |
Schering Corporation |
Thiadiazoles as cxc- and cc- chemokine receptor ligands
|
CA2550361C
(en)
|
2003-12-19 |
2014-04-29 |
Prabha Ibrahim |
Compounds and methods for development of ret modulators
|
CA2548374C
(en)
|
2003-12-23 |
2014-05-27 |
Astex Therapeutics Limited |
Pyrazole derivatives as protein kinase modulators
|
US20050187389A1
(en)
|
2004-01-13 |
2005-08-25 |
Ambit Biosciences Corporation |
Pyrrolopyrimidine derivatives and analogs and their use in the treatment and prevention of diseases
|
WO2005089502A2
(en)
|
2004-03-18 |
2005-09-29 |
The Brigham And Women's Hospital, Inc. |
Methods for the treatment of synucleinopathies
|
DK2332940T3
(da)
|
2004-03-30 |
2013-02-11 |
Vertex Pharma |
Azaindoler, der kan anvendes som inhibitorer af JAK og andre proteinkinaser
|
JP5213229B2
(ja)
|
2004-04-23 |
2013-06-19 |
エグゼリクシス, インコーポレイテッド |
キナーゼ調節因子および使用方法
|
US20060106020A1
(en)
|
2004-04-28 |
2006-05-18 |
Rodgers James D |
Tetracyclic inhibitors of Janus kinases
|
US7558717B2
(en)
|
2004-04-28 |
2009-07-07 |
Vertex Pharmaceuticals Incorporated |
Crystal structure of human JAK3 kinase domain complex and binding pockets thereof
|
MXPA06012663A
(es)
|
2004-05-03 |
2007-01-16 |
Novartis Ag |
Combinaciones que comprenden un agonista del receptor s1p y un inhibidor de quinasa jak3.
|
US20060074102A1
(en)
|
2004-05-14 |
2006-04-06 |
Kevin Cusack |
Kinase inhibitors as therapeutic agents
|
PE20060426A1
(es)
|
2004-06-02 |
2006-06-28 |
Schering Corp |
DERIVADOS DE ACIDO TARTARICO COMO INHIBIDORES DE MMPs, ADAMs, TACE Y TNF-alfa
|
MXPA06014247A
(es)
|
2004-06-10 |
2007-03-12 |
Irm Llc |
Compuestos y composiciones como inhibidores de la proteina quinasa.
|
EP1760071A4
(en)
|
2004-06-23 |
2008-03-05 |
Ono Pharmaceutical Co |
COMPOUND WITH S1P RECEPTOR BINDING ABILITY AND USE THEREOF
|
CA2572058A1
(en)
|
2004-06-30 |
2006-01-12 |
Vertex Pharmaceuticals Incorporated |
Azaindoles useful as inhibitors of protein kinases
|
US7138423B2
(en)
|
2004-07-20 |
2006-11-21 |
Bristol-Myers Squibb Company |
Arylpyrrolidine derivatives as NK-1 /SSRI antagonists
|
FR2873691B1
(fr)
|
2004-07-29 |
2006-10-06 |
Sanofi Synthelabo |
Derives d'amino-piperidine, leur preparation et leur application en therapeutique
|
WO2006013114A1
(en)
|
2004-08-06 |
2006-02-09 |
Develogen Aktiengesellschaft |
Use of a timp-2 secreted protein product for preventing and treating pancreatic diseases and/or obesity and/or metabolic syndrome
|
WO2006022459A1
(en)
|
2004-08-23 |
2006-03-02 |
Mogam Biotechnology Institute |
Primer and probe for detection of sars coronavirus, kit comprising the primer and/or the probe, and detection method thereof
|
US20070054916A1
(en)
|
2004-10-01 |
2007-03-08 |
Amgen Inc. |
Aryl nitrogen-containing bicyclic compounds and methods of use
|
SI1802625T1
(sl)
|
2004-10-13 |
2008-10-31 |
Hoffmann La Roche |
Disubstituirani pirazolobenzodiazepini, koristni kot inhibitorji za cdk2 in angiogenezo ter za zdravljenje prsnega raka, raka kolona, pljuäśnega rakain raka prostate
|
MY179032A
(en)
|
2004-10-25 |
2020-10-26 |
Cancer Research Tech Ltd |
Ortho-condensed pyridine and pyrimidine derivatives (e.g.purines) as protein kinase inhibitors
|
UY29177A1
(es)
|
2004-10-25 |
2006-05-31 |
Astex Therapeutics Ltd |
Derivados sustituidos de purina, purinona y deazapurina, composiciones que los contienen métodos para su preparación y sus usos
|
AU2005304784B2
(en)
|
2004-11-04 |
2011-03-24 |
Vertex Pharmaceuticals Incorporated |
Pyrazolo[1,5-a]pyrimidines useful as inhibitors of protein kinases
|
RU2007123675A
(ru)
|
2004-11-24 |
2008-12-27 |
Новартис АГ (CH) |
Комбинации ингибиторов jak
|
US7517870B2
(en)
|
2004-12-03 |
2009-04-14 |
Fondazione Telethon |
Use of compounds that interfere with the hedgehog signaling pathway for the manufacture of a medicament for preventing, inhibiting, and/or reversing ocular diseases related with ocular neovascularization
|
WO2006065916A1
(en)
|
2004-12-14 |
2006-06-22 |
Alcon, Inc. |
Method of treating dry eye disorders using 13(s)-hode and its analogs
|
AR054416A1
(es)
|
2004-12-22 |
2007-06-27 |
Incyte Corp |
Pirrolo [2,3-b]piridin-4-il-aminas y pirrolo [2,3-b]pirimidin-4-il-aminas como inhibidores de las quinasas janus. composiciones farmaceuticas.
|
WO2006067445A2
(en)
|
2004-12-22 |
2006-06-29 |
Astrazeneca Ab |
Csf-1r kinase inhibitors
|
CA2595574A1
(en)
|
2005-01-20 |
2006-07-27 |
Pfizer Limited. |
Chemical compounds
|
ES2320487T3
(es)
|
2005-02-03 |
2009-05-22 |
Vertex Pharmaceuticals, Inc. |
Pirrolopirimidinas utiles como inhibidores de proteina quinasas.
|
WO2007044050A2
(en)
|
2005-02-04 |
2007-04-19 |
Bristol-Myers Squibb Company |
1h-imidazo[4,5-d]thieno[3,2-b]pyridine based tricyclic compounds and pharmaceutical compositions comprising same
|
BRPI0608513A2
(pt)
|
2005-03-15 |
2010-01-05 |
Irm Llc |
compostos e composições como inibidores da proteìna quinase
|
MX2007012393A
(es)
|
2005-04-05 |
2008-02-22 |
Pharmacopeia Inc |
Derivados de purina e imidazopiridina para la inmunosupresion.
|
GB0510139D0
(en)
|
2005-05-18 |
2005-06-22 |
Addex Pharmaceuticals Sa |
Novel compounds B1
|
CA2609126A1
(en)
|
2005-05-20 |
2006-11-30 |
Vertex Pharmaceuticals Incorporated |
Pyrrolopyridines useful as inhibitors of protein kinase
|
GB0510390D0
(en)
|
2005-05-20 |
2005-06-29 |
Novartis Ag |
Organic compounds
|
CN105348203B
(zh)
|
2005-06-08 |
2018-09-18 |
里格尔药品股份有限公司 |
抑制jak途径的组合物和方法
|
WO2006136823A1
(en)
|
2005-06-21 |
2006-12-28 |
Astex Therapeutics Limited |
Heterocyclic containing amines as kinase b inhibitors
|
EP1893612B1
(en)
|
2005-06-22 |
2011-08-03 |
Plexxikon, Inc. |
Pyrrolo [2, 3-b]pyridine derivatives as protein kinase inhibitors
|
CN102127078A
(zh)
|
2005-07-14 |
2011-07-20 |
安斯泰来制药株式会社 |
Janus激酶3的杂环类抑制剂
|
FR2889662B1
(fr)
|
2005-08-11 |
2011-01-14 |
Galderma Res & Dev |
Emulsion de type huile-dans-eau pour application topique en dermatologie
|
US20070049591A1
(en)
|
2005-08-25 |
2007-03-01 |
Kalypsys, Inc. |
Inhibitors of MAPK/Erk Kinase
|
CA2621261C
(en)
|
2005-09-22 |
2014-05-20 |
Incyte Corporation |
Azepine inhibitors of janus kinases
|
AU2006297351A1
(en)
|
2005-09-30 |
2007-04-12 |
Vertex Pharmaceuticals Incorporated |
Deazapurines useful as inhibitors of janus kinases
|
WO2007044894A2
(en)
|
2005-10-11 |
2007-04-19 |
Chembridge Research Laboratories, Inc. |
Cell-free protein expression systems and methods of use thereof
|
CA2623202C
(en)
|
2005-10-14 |
2014-09-16 |
Sumitomo Chemical Company, Limited |
Hydrazide compound and pesticidal use of the same
|
BRPI0618011A2
(pt)
|
2005-10-28 |
2011-08-16 |
Astrazeneca Ab |
composto ou um sal farmaceuticamente aceitável do mesmo, processo para a preparação do mesmo, composição farmacêutica, uso de um composto ou um sal farmaceuticamente aceitável do mesmo, e, métodos para produzir um efeito anti-proliferativo e um efeito pró-apoptósico em um animal de sangue quente, para tratar doença e para produzir um efeito inibidor de jak em um animal de sangue quente
|
NZ567851A
(en)
|
2005-11-01 |
2011-09-30 |
Targegen Inc |
Bi-aryl meta-pyrimidine inhibitors of kinases
|
WO2007062459A1
(en)
|
2005-11-29 |
2007-06-07 |
Cytopia Research Pty Ltd |
Selective kinase inhibitors based on pyridine scaffold
|
US20130137681A1
(en)
|
2005-12-13 |
2013-05-30 |
Incyte Corporation |
HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS
|
SI2348023T1
(sl)
|
2005-12-13 |
2015-10-30 |
Incyte Corporation |
S heteroarilom substituirani pirolo (2,3-b)piridini in pirolo (2,3-b)pirimidini kot zaviralci janus kinaze
|
EP1968568A4
(en)
|
2005-12-22 |
2011-04-13 |
Glaxosmithkline Llc |
HEMMER OF NUTS ACTIVITY
|
PT1962830E
(pt)
|
2005-12-23 |
2013-05-29 |
Glaxosmithkline Llc |
Inibidores azaindólicos de cinases aurora
|
JP4643455B2
(ja)
|
2006-01-12 |
2011-03-02 |
株式会社ユニバーサルエンターテインメント |
遊技システム
|
TW201412738A
(zh)
|
2006-01-17 |
2014-04-01 |
Vertex Pharma |
適合作為傑納斯激酶(janus kinase)抑制劑之氮雜吲哚
|
US20070208053A1
(en)
|
2006-01-19 |
2007-09-06 |
Arnold Lee D |
Fused heterobicyclic kinase inhibitors
|
EP1981887A2
(en)
|
2006-02-01 |
2008-10-22 |
SmithKline Beecham Corporation |
Pyrrolo[2,3,b]pyridine derivatives useful as raf kinase inhibitors
|
US7745477B2
(en)
|
2006-02-07 |
2010-06-29 |
Hoffman-La Roche Inc. |
Heteroaryl and benzyl amide compounds
|
PL1842534T3
(pl)
|
2006-02-24 |
2012-05-31 |
Teva Pharma |
Tabletki bursztynianu metoprololu o przedłużonym uwalnianiu oraz sposoby ich wytwarzania
|
CA2644368A1
(en)
|
2006-03-10 |
2007-09-20 |
Ono Pharmaceutical Co., Ltd. |
Nitrogenated heterocyclic derivative, and pharmaceutical agent comprising the derivative as active ingredient
|
BRPI0709866B8
(pt)
|
2006-04-03 |
2021-05-25 |
Astellas Pharma Inc |
compostos héteros e composição farmacêutica compreendendo ditos compostos
|
EP2001884A1
(en)
|
2006-04-05 |
2008-12-17 |
Vertex Pharmaceuticals, Inc. |
Deazapurines useful as inhibitors of janus kinases
|
US20090124636A1
(en)
|
2006-04-12 |
2009-05-14 |
Pfizer Inc. |
Chemical compounds
|
WO2007129195A2
(en)
|
2006-05-04 |
2007-11-15 |
Pfizer Products Inc. |
4-pyrimidine-5-amino-pyrazole compounds
|
US20080051427A1
(en)
|
2006-05-18 |
2008-02-28 |
Fritz Schuckler |
Pharmaceutical Compositions and Methods of Using Same
|
US7691811B2
(en)
|
2006-05-25 |
2010-04-06 |
Bodor Nicholas S |
Transporter-enhanced corticosteroid activity and methods and compositions for treating dry eye
|
JO3235B1
(ar)
|
2006-05-26 |
2018-03-08 |
Astex Therapeutics Ltd |
مركبات بيررولوبيريميدين و استعمالاتها
|
NZ573174A
(en)
|
2006-06-01 |
2012-01-12 |
Msd Consumer Care Inc |
Sustained release pharmaceutical dosage form containing phenylephrine
|
EP2044061A2
(en)
|
2006-07-20 |
2009-04-08 |
Mehmet Kahraman |
Benzothiophene inhibitors of rho kinase
|
WO2008013622A2
(en)
|
2006-07-27 |
2008-01-31 |
E. I. Du Pont De Nemours And Company |
Fungicidal azocyclic amides
|
US8492378B2
(en)
|
2006-08-03 |
2013-07-23 |
Takeda Pharmaceutical Company Limited |
GSK-3β inhibitor
|
CA2660560A1
(en)
|
2006-08-16 |
2008-02-21 |
Boehringer Ingelheim International Gmbh |
Pyrazine compounds, their use and methods of preparation
|
JP2010502675A
(ja)
|
2006-09-08 |
2010-01-28 |
ノバルティス アクチエンゲゼルシャフト |
リンパ球相互作用が介在する疾患または障害を処置するために有用なn−ビアリール(ヘテロ)アリールスルホンアミド誘導体
|
WO2008035376A2
(en)
|
2006-09-19 |
2008-03-27 |
Council Of Scientific & Industrial Research |
A novel bio-erodible insert for ophthalmic applications and a process for the preparation thereof
|
CL2007002867A1
(es)
|
2006-10-04 |
2008-06-27 |
Pharmacopeia Inc |
Compuestos derivados de 2-(bencimidazolil)purina, inhibidores de janus quinasa 3; composicion farmaceutica que los contiene; y su uso para tratar enfermedades autoinmune, inflamatorias, cardiovasculares, rechazo de implante, entre otras.
|
CL2007002866A1
(es)
|
2006-10-04 |
2008-07-04 |
Pharmacopeia Inc |
Compuestos derivados de 6-sustituidos-2-(bencimidazolil) purina y purinona; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto en el tratamiento de enfermedades autoinmunes, enfermedad inflamatoria, enfermedad mediada por m
|
US20120225057A1
(en)
*
|
2006-10-11 |
2012-09-06 |
Deciphera Pharmaceuticals, Llc |
Methods and compositions for the treatment of myeloproliferative diseases and other proliferative diseases
|
WO2008058126A2
(en)
|
2006-11-06 |
2008-05-15 |
Supergen, Inc. |
Imidazo[1,2-b]pyridazine and pyrazolo[1,5-a]pyrimidine derivatives and their use as protein kinase inhibitors
|
US20080119496A1
(en)
|
2006-11-16 |
2008-05-22 |
Pharmacopeia Drug Discovery, Inc. |
7-Substituted Purine Derivatives for Immunosuppression
|
ME01507B
(me)
|
2006-11-22 |
2014-04-20 |
Incyte Holdings Corp |
Imidazotriazini i imidazopirimidini kao inhibitori kinaze
|
WO2008067119A2
(en)
|
2006-11-27 |
2008-06-05 |
Smithkline Beecham Corporation |
Novel compounds
|
CA2672616A1
(en)
|
2006-12-15 |
2008-06-26 |
Abbott Laboratories |
Novel oxadiazole compounds
|
WO2008079291A2
(en)
|
2006-12-20 |
2008-07-03 |
Amgen Inc. |
Substituted heterocycles and methods of use
|
ES2387471T3
(es)
|
2006-12-20 |
2012-09-24 |
Amgen Inc. |
Compuestos heterocíclicos y su uso en el tratamiento de la inflamación, la angiogénesis y el cáncer
|
MX2009005644A
(es)
|
2006-12-22 |
2009-06-08 |
Sigma Tau Ind Farmaceuti |
Gel util para el suministro de farmacos oftalmicos.
|
JP5492565B2
(ja)
|
2006-12-22 |
2014-05-14 |
インサイト・コーポレイション |
Janusキナーゼ阻害剤としての置換複素環
|
KR20080062876A
(ko)
|
2006-12-29 |
2008-07-03 |
주식회사 대웅제약 |
신규한 항진균성 트리아졸 유도체
|
WO2008082839A2
(en)
|
2006-12-29 |
2008-07-10 |
Abbott Laboratories |
Pim kinase inhibitors as cancer chemotherapeutics
|
WO2008082840A1
(en)
|
2006-12-29 |
2008-07-10 |
Abbott Laboratories |
Pim kinase inhibitors as cancer chemotherapeutics
|
US8822497B2
(en)
|
2007-03-01 |
2014-09-02 |
Novartis Ag |
PIM kinase inhibitors and methods of their use
|
ES2420113T3
(es)
|
2007-04-03 |
2013-08-22 |
Array Biopharma, Inc. |
Compuestos de imidazo[1,2-a]piridina como inhibidores de receptores tirosina quinasa
|
US8188178B2
(en)
|
2007-05-07 |
2012-05-29 |
3M Innovative Properties Company |
Cold shrinkable article including an epichlorohydrin composition
|
GB0709031D0
(en)
|
2007-05-10 |
2007-06-20 |
Sareum Ltd |
Pharmaceutical compounds
|
WO2008145681A2
(en)
|
2007-05-31 |
2008-12-04 |
Boehringer Ingelheim International Gmbh |
Ccr2 receptor antagonists and uses thereof
|
GB0710528D0
(en)
|
2007-06-01 |
2007-07-11 |
Glaxo Group Ltd |
Novel compounds
|
CL2008001709A1
(es)
|
2007-06-13 |
2008-11-03 |
Incyte Corp |
Compuestos derivados de pirrolo [2,3-b]pirimidina, moduladores de quinasas jak; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como cancer, psoriasis, artritis reumatoide, entre otras.
|
CU24179B1
(es)
|
2007-06-13 |
2016-04-25 |
Incyte Corp |
SALES DE ÁCIDO MALEICO Y DE ÁCIDO SULFÚRICO DE (R)-3-(4-(7H-PIRROLO[2,3-d]PIRIMIDIN-4-IL)-1H-PIRAZOL-1-IL)-3-CICLOPENTILPROPANITRILO
|
CA2691914C
(en)
|
2007-07-11 |
2012-06-26 |
Pfizer Inc. |
Pharmaceutical compositions and methods of treating dry eye disorders
|
WO2009016460A2
(en)
|
2007-08-01 |
2009-02-05 |
Pfizer Inc. |
Pyrazole compounds and their use as raf inhibitors
|
WO2009049028A1
(en)
|
2007-10-09 |
2009-04-16 |
Targegen Inc. |
Pyrrolopyrimidine compounds and their use as janus kinase modulators
|
EP2217235A4
(en)
|
2007-11-15 |
2011-01-12 |
Musc Found For Res Dev |
PROTEIN INHIBITORS PIM KINASES, COMPOSITIONS AND METHODS FOR TREATING CANCER
|
BRPI0820544A2
(pt)
|
2007-11-16 |
2015-06-16 |
Incyte Corp |
4-pirazolil-n-arilpirimidin-2-aminas e pirazolil-n-heteroarilpirimidin-2-aminas como inibidores de janus cinase
|
GB0723815D0
(en)
|
2007-12-05 |
2008-01-16 |
Glaxo Group Ltd |
Compounds
|
CN101977923B
(zh)
|
2008-01-18 |
2014-10-08 |
捷克有机化学和生物化学研究院 |
抑制细胞生长的7-脱氮嘌呤核苷
|
CA2714181C
(en)
|
2008-02-04 |
2013-12-24 |
Mercury Therapeutics, Inc. |
Ampk modulators
|
AR070531A1
(es)
|
2008-03-03 |
2010-04-14 |
Novartis Ag |
Inhibidores de cinasa pim y metodos para su uso
|
BRPI0909040B8
(pt)
|
2008-03-11 |
2021-05-25 |
Incyte Holdings Corp |
derivados de azetidina e ciclobutano, seus usos, e composição
|
AU2009227013B2
(en)
|
2008-03-21 |
2013-01-10 |
Novartis Ag |
Novel heterocyclic compounds and uses therof
|
WO2009155156A1
(en)
|
2008-06-18 |
2009-12-23 |
Merck & Co., Inc. |
Inhibitors of janus kinases
|
CA2726836C
(en)
|
2008-06-26 |
2019-06-18 |
Anterios, Inc. |
Use of nanoemulsions in the manufacture of a medicament for treating skin disorders
|
TWI461423B
(zh)
|
2008-07-02 |
2014-11-21 |
Astrazeneca Ab |
用於治療Pim激酶相關病狀及疾病之噻唑啶二酮化合物
|
FR2933409B1
(fr)
|
2008-07-03 |
2010-08-27 |
Centre Nat Rech Scient |
NOUVEAUX PYRROLO °2,3-a! CARBAZOLES ET LEUR UTILISATION COMME INHIBITEURS DES KINASES PIM
|
WO2010022081A1
(en)
|
2008-08-19 |
2010-02-25 |
Array Biopharma Inc. |
Triazolopyridine compounds as pim kinase inhibitors
|
TWI496779B
(zh)
|
2008-08-19 |
2015-08-21 |
Array Biopharma Inc |
作為pim激酶抑制劑之三唑吡啶化合物
|
SI2384326T1
(sl)
|
2008-08-20 |
2014-06-30 |
Zoetis Llc |
Pirolo(2,3-d)pirimidinske spojine
|
BRPI0918846A2
(pt)
|
2008-09-02 |
2019-09-24 |
Novartis Ag |
inibidores de cinase heterocíclica
|
US8329732B2
(en)
|
2008-09-02 |
2012-12-11 |
Novartis Ag |
Kinase inhibitors and methods of their use
|
KR20110058866A
(ko)
|
2008-09-02 |
2011-06-01 |
노파르티스 아게 |
비시클릭 키나제 억제제
|
CL2009001884A1
(es)
*
|
2008-10-02 |
2010-05-14 |
Incyte Holdings Corp |
Uso de 3-ciclopentil-3-[4-(7h-pirrolo[2,3-d]pirimidin-4-il)-1h-pirazol-1-il)propanonitrilo, inhibidor de janus quinasa, y uso de una composición que lo comprende para el tratamiento del ojo seco.
|
EP2350054A4
(en)
|
2008-10-17 |
2012-03-28 |
Merck Canada Inc |
AZETIDINE DERIVATIVES AS INHIBITORS OF THE STEAROYL COENZYME A DELTA 9 DESATURASE
|
JOP20190230A1
(ar)
|
2009-01-15 |
2017-06-16 |
Incyte Corp |
طرق لاصلاح مثبطات انزيم jak و المركبات الوسيطة المتعلقة به
|
EP2210890A1
(en)
|
2009-01-19 |
2010-07-28 |
Almirall, S.A. |
Oxadiazole derivatives as S1P1 receptor agonists
|
US8263601B2
(en)
|
2009-02-27 |
2012-09-11 |
Concert Pharmaceuticals, Inc. |
Deuterium substituted xanthine derivatives
|
HUE046493T2
(hu)
|
2009-05-22 |
2020-03-30 |
Incyte Holdings Corp |
3-[4-(7H-Pirrolo[2,3-d]pirimidin-4-il)-lH-pirazol-l-il]oktán- vagy heptán-nitril JAK inhibitorokként
|
US8716303B2
(en)
|
2009-05-22 |
2014-05-06 |
Incyte Corporation |
N-(hetero)aryl-pyrrolidine derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines and pyrrol-3-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors
|
UA110324C2
(en)
*
|
2009-07-02 |
2015-12-25 |
Genentech Inc |
Jak inhibitory compounds based on pyrazolo pyrimidine
|
EP2451813B1
(en)
|
2009-07-08 |
2014-10-01 |
Leo Pharma A/S |
Heterocyclic compounds as jak receptor and protein tyrosine kinase inhibitors
|
US20120157500A1
(en)
|
2009-08-24 |
2012-06-21 |
Weikang Tao |
Jak inhibition blocks rna interference associated toxicities
|
TW201111385A
(en)
|
2009-08-27 |
2011-04-01 |
Biocryst Pharm Inc |
Heterocyclic compounds as janus kinase inhibitors
|
TW201113285A
(en)
|
2009-09-01 |
2011-04-16 |
Incyte Corp |
Heterocyclic derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors
|
SG10201405568UA
(en)
|
2009-09-08 |
2014-11-27 |
Hoffmann La Roche |
4-substituted pyridin-3-yl-carboxamide compounds and methods of use
|
EP2305660A1
(en)
|
2009-09-25 |
2011-04-06 |
Almirall, S.A. |
New thiadiazole derivatives
|
PT2486041E
(pt)
|
2009-10-09 |
2013-11-14 |
Incyte Corp |
Derivados hidroxilo, ceto e glucuronido de 3-(4-(7h-pirrolo[2,3-d]pirimidin-4-il)-1h-pirazol-1-il)-3-ciclopentil-propanonitrilo
|
EP2491039A1
(en)
*
|
2009-10-20 |
2012-08-29 |
Cellzome Limited |
Heterocyclyl pyrazolopyrimidine analogues as jak inhibitors
|
US8671402B2
(en)
*
|
2009-11-09 |
2014-03-11 |
Bank Of America Corporation |
Network-enhanced control of software updates received via removable computer-readable medium
|
EP2332917B1
(en)
|
2009-11-11 |
2012-08-01 |
Sygnis Bioscience GmbH & Co. KG |
Compounds for PIM kinase inhibition and for treating malignancy
|
WO2011066378A2
(en)
|
2009-11-24 |
2011-06-03 |
Alder Biopharmaceuticals, Inc. |
Antagonists of il-6 to prevent or treat thrombosis
|
US20130129675A1
(en)
|
2009-12-04 |
2013-05-23 |
Board Of Regents, The University Of Texas System |
Interferon therapies in combination with blockade of stat3 activation
|
ES2461967T3
(es)
*
|
2009-12-18 |
2014-05-21 |
Pfizer Inc. |
Compuestos de pirrolo[2,3-d]pirimidina
|
US8461328B2
(en)
|
2010-01-12 |
2013-06-11 |
Genentech, Inc. |
Tricyclic heterocyclic compounds, compositions and methods of use thereof
|
SA111320200B1
(ar)
*
|
2010-02-17 |
2014-02-16 |
ديبيوفارم اس ايه |
مركبات ثنائية الحلقة واستخداماتها كمثبطات c-src/jak مزدوجة
|
JP5858434B2
(ja)
*
|
2010-02-18 |
2016-02-10 |
インサイト・ホールディングス・コーポレイションIncyte Holdings Corporation |
Janusキナーゼ阻害薬としてのシクロブタンおよびメチルシクロブタン誘導体
|
DK3050882T3
(en)
*
|
2010-03-10 |
2018-03-19 |
Incyte Holdings Corp |
PIPERIDIN-4-YL-AZETIDINE DERIVATIVES AS JAK1 INHIBITORS
|
UA109131C2
(ru)
|
2010-04-14 |
2015-07-27 |
Еррей Біофарма Інк. |
5,7-ЗАМЕЩЕННЫЕ ИМИДАЗО[1,2-c]ПИРИМИДИНЫ КАК ИНГИБИТОРЫ JAK-КИНАЗ
|
EP2390252A1
(en)
|
2010-05-19 |
2011-11-30 |
Almirall, S.A. |
New pyrazole derivatives
|
ME02445B
(me)
|
2010-05-21 |
2016-09-20 |
Incyte Holdings Corp |
Topikalna formulacija za inhibiciju jak-a
|
US8637529B2
(en)
|
2010-06-11 |
2014-01-28 |
AbbYie Inc. |
Pyrazolo[3,4-d]pyrimidine compounds
|
US9351943B2
(en)
|
2010-07-01 |
2016-05-31 |
Matthew T. McLeay |
Anti-fibroblastic fluorochemical emulsion therapies
|
WO2012045010A1
(en)
|
2010-09-30 |
2012-04-05 |
Portola Pharmaceuticals, Inc. |
Combinations of 4-(3-(2h-1,2,3-triazo-2-yl) phenylamino)-2-((1r,2s)-2-aminocyclohexylamino) pyrimidine-5-carboxamide and fludarabine
|
UA113156C2
(xx)
|
2010-11-19 |
2016-12-26 |
|
Циклобутилзаміщені похідні піролопіридину й піролопіримідину як інгібітори jak
|
JP5917544B2
(ja)
|
2010-11-19 |
2016-05-18 |
インサイト・ホールディングス・コーポレイションIncyte Holdings Corporation |
Jak阻害剤としての複素環置換ピロロピリジンおよびピロロピリミジン
|
CN104473933A
(zh)
|
2010-12-03 |
2015-04-01 |
Ym生物科学澳大利亚私人有限公司 |
Jak-2 介导的病症的治疗
|
JP5936628B2
(ja)
|
2011-02-18 |
2016-06-22 |
ノバルティス・ファルマ・アクチェンゲゼルシャフトNovartis Pharma AG |
mTOR/JAK阻害剤併用療法
|
CN102247368B
(zh)
|
2011-05-19 |
2013-05-29 |
安徽永生堂药业有限责任公司 |
一种复方阿伐斯汀缓释片及其制备方法
|
CN102218042A
(zh)
|
2011-05-26 |
2011-10-19 |
青岛黄海制药有限责任公司 |
富马酸喹硫平组合物的缓释片剂及其制备方法
|
US8691807B2
(en)
|
2011-06-20 |
2014-04-08 |
Incyte Corporation |
Azetidinyl phenyl, pyridyl or pyrazinyl carboxamide derivatives as JAK inhibitors
|
WO2013007765A1
(en)
|
2011-07-13 |
2013-01-17 |
F. Hoffmann-La Roche Ag |
Fused tricyclic compounds for use as inhibitors of janus kinases
|
WO2013007768A1
(en)
|
2011-07-13 |
2013-01-17 |
F. Hoffmann-La Roche Ag |
Tricyclic heterocyclic compounds, compositions and methods of use thereof as jak inhibitors
|
WO2013023119A1
(en)
|
2011-08-10 |
2013-02-14 |
Novartis Pharma Ag |
JAK P13K/mTOR COMBINATION THERAPY
|
TW201313721A
(zh)
|
2011-08-18 |
2013-04-01 |
Incyte Corp |
作為jak抑制劑之環己基氮雜環丁烷衍生物
|
UA111854C2
(uk)
*
|
2011-09-07 |
2016-06-24 |
Інсайт Холдінгс Корпорейшн |
Способи і проміжні сполуки для отримання інгібіторів jak
|
TW201406761A
(zh)
|
2012-05-18 |
2014-02-16 |
Incyte Corp |
做爲jak抑制劑之哌啶基環丁基取代之吡咯并吡啶及吡咯并嘧啶衍生物
|
US10155987B2
(en)
|
2012-06-12 |
2018-12-18 |
Dana-Farber Cancer Institute, Inc. |
Methods of predicting resistance to JAK inhibitor therapy
|
CA2876306C
(en)
|
2012-06-15 |
2024-02-20 |
Concert Pharmaceuticals, Inc. |
Deuterated derivatives of ruxolitinib
|
US20150246043A1
(en)
|
2012-07-27 |
2015-09-03 |
Ratiopharm Gmbh |
Oral dosage forms for modified release comprising ruxolitinib
|
CN102772384A
(zh)
|
2012-08-07 |
2012-11-14 |
四川百利药业有限责任公司 |
一种盐酸米诺环素缓释片及其制备方法
|
WO2014036016A1
(en)
*
|
2012-08-31 |
2014-03-06 |
Principia Biopharma Inc. |
Benzimidazole derivatives as itk inhibitors
|
SG10201703533VA
(en)
|
2012-11-01 |
2017-06-29 |
Incyte Corp |
Tricyclic fused thiophene derivatives as jak inhibitors
|
PE20151157A1
(es)
|
2012-11-15 |
2015-08-19 |
Incyte Corp |
Formas de dosificacion de ruxolitinib de liberacion sostenida
|
PE20151902A1
(es)
|
2013-03-06 |
2015-12-26 |
Incyte Corp |
Proceso e intermedios para hacer un inhibidor de jak
|
EP4275756A3
(en)
|
2013-05-17 |
2024-02-07 |
Incyte Holdings Corporation |
Bipyrazole derivatives as jak inhibitors
|
RS60469B1
(sr)
|
2013-08-07 |
2020-07-31 |
Incyte Corp |
Dozni oblici sa produženim oslobađanjem za jak1 inhibitor
|
MX2016002165A
(es)
*
|
2013-08-20 |
2017-01-05 |
Incyte Corp |
Beneficio de supervivencia en pacientes con tumores solidos con niveles elevados de proteina c reactiva.
|
SI3110409T1
(sl)
|
2014-02-28 |
2018-11-30 |
Incyte Corporation |
Inhibitorji JAK1 za zdravljenje mielodisplastičnih sindromov
|
MA54622A
(fr)
|
2014-04-08 |
2021-11-03 |
Incyte Corp |
Traitement d'affections malignes par lymphocytes b par un inhibiteur jak et pi3k combiné
|
SG11201609016VA
(en)
|
2014-04-30 |
2016-11-29 |
Incyte Corp |
Processes of preparing a jak1 inhibitor and new forms thereto
|
ES2946179T3
(es)
|
2014-05-28 |
2023-07-13 |
Onco Tracker Inc |
Efectos antineoplásicos de inhibidores de JAK2 en combinación con derivados de talidomida y glucocorticoides
|
US9498467B2
(en)
|
2014-05-30 |
2016-11-22 |
Incyte Corporation |
Treatment of chronic neutrophilic leukemia (CNL) and atypical chronic myeloid leukemia (aCML) by inhibitors of JAK1
|
US10766900B2
(en)
|
2017-12-29 |
2020-09-08 |
Formosa Laboratories, Inc. |
Baricitinib intermediate, method for forming Baricitinib intermediate, and method for preparing Baricitinib or pharmaceutically acceptable salt thereof
|
KR20210124345A
(ko)
|
2019-02-06 |
2021-10-14 |
콘서트 파마슈티컬즈, 인크. |
거울상 이성질체 풍부한 jak 억제제를 제조하는 방법
|