SE0301373D0 - Novel compounds - Google Patents

Novel compounds

Info

Publication number
SE0301373D0
SE0301373D0 SE0301373A SE0301373A SE0301373D0 SE 0301373 D0 SE0301373 D0 SE 0301373D0 SE 0301373 A SE0301373 A SE 0301373A SE 0301373 A SE0301373 A SE 0301373A SE 0301373 D0 SE0301373 D0 SE 0301373D0
Authority
SE
Sweden
Prior art keywords
novel compounds
imidazo
formula
methods
pharmaceutical compositions
Prior art date
Application number
SE0301373A
Other languages
English (en)
Inventor
Martin Hemmerling
Thomas Klingstedt
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Priority to SE0301373A priority Critical patent/SE0301373D0/sv
Publication of SE0301373D0 publication Critical patent/SE0301373D0/sv
Priority to EP04731525A priority patent/EP1625126B1/en
Priority to BRPI0410081-6A priority patent/BRPI0410081A/pt
Priority to CNA200480012617XA priority patent/CN1784402A/zh
Priority to CA002524624A priority patent/CA2524624A1/en
Priority to SI200430618T priority patent/SI1625126T1/sl
Priority to PT04731525T priority patent/PT1625126E/pt
Priority to PL04731525T priority patent/PL1625126T3/pl
Priority to AT04731525T priority patent/ATE384061T1/de
Priority to US10/556,228 priority patent/US20060287355A1/en
Priority to PCT/SE2004/000694 priority patent/WO2004099204A1/en
Priority to DE602004011330T priority patent/DE602004011330T2/de
Priority to AU2004236144A priority patent/AU2004236144B2/en
Priority to ES04731525T priority patent/ES2298754T3/es
Priority to EP07119970A priority patent/EP1887007A3/en
Priority to DK04731525T priority patent/DK1625126T3/da
Priority to MXPA05012025A priority patent/MXPA05012025A/es
Priority to JP2006508045A priority patent/JP2006525997A/ja
Priority to CY20081100279T priority patent/CY1107301T1/el

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
SE0301373A 2003-05-09 2003-05-09 Novel compounds SE0301373D0 (sv)

Priority Applications (19)

Application Number Priority Date Filing Date Title
SE0301373A SE0301373D0 (sv) 2003-05-09 2003-05-09 Novel compounds
JP2006508045A JP2006525997A (ja) 2003-05-09 2004-05-06 Ｊａｋ３キナーゼ阻害剤としてのイミダゾ及びチアゾロピリジン
AT04731525T ATE384061T1 (de) 2003-05-09 2004-05-06 Imidazo- und thiazolopyridine als jak3-kinase- inhibitoren
PCT/SE2004/000694 WO2004099204A1 (en) 2003-05-09 2004-05-06 Imidazo and thiazolopyridines as jak3 kinase inhibitors
CNA200480012617XA CN1784402A (zh) 2003-05-09 2004-05-06 用作jak3激酶抑制剂的咪唑并和噻唑并吡啶化合物
CA002524624A CA2524624A1 (en) 2003-05-09 2004-05-06 Imidazo and thiazolopyridines as jak3 kinase inhibitors
SI200430618T SI1625126T1 (sl) 2003-05-09 2004-05-06 Imidazo- in tiazolopiridini kot inhibitorji JAK3-kinaze
PT04731525T PT1625126E (pt) 2003-05-09 2004-05-06 Imidazo- e tiazolopiridinas como inibidores de cinase jak3
PL04731525T PL1625126T3 (pl) 2003-05-09 2004-05-06 Imidazo- i tiazolopirydyny jako inhibitory kinazy JAK3
EP04731525A EP1625126B1 (en) 2003-05-09 2004-05-06 Imidazo and thiazolopyridines as jak3 kinase inhibitors
US10/556,228 US20060287355A1 (en) 2003-05-09 2004-05-06 Imidazo and thiazolopyridines as jak3 kinase inhibitors
BRPI0410081-6A BRPI0410081A (pt) 2003-05-09 2004-05-06 composto, composição farmacêutica, método de tratamento de uma doença ou condição mediada por jak3, e, processo para a preparação de um composto
DE602004011330T DE602004011330T2 (de) 2003-05-09 2004-05-06 Imidazo- und thiazolopyridine als jak3-kinase-inhibitoren
AU2004236144A AU2004236144B2 (en) 2003-05-09 2004-05-06 Imidazo and thiazolopyridines as JAK3 kinase inhibitors
ES04731525T ES2298754T3 (es) 2003-05-09 2004-05-06 Imidazo- y tiazolopiridinas como inhibidores de jak3 quinasa.
EP07119970A EP1887007A3 (en) 2003-05-09 2004-05-06 Imidazo- and Thiazolopyridine as JAK3 Kinase Inhibitors
DK04731525T DK1625126T3 (da) 2003-05-09 2004-05-06 Imidazo- og thiazolopyridiner som JAK3-kinaseinhibitorer
MXPA05012025A MXPA05012025A (es) 2003-05-09 2004-05-06 Imidazo y tiazolopiridinas como inhibidores de cinasa jak3.
CY20081100279T CY1107301T1 (el) 2003-05-09 2008-03-12 Ιμιδαζο και θειαζολοπυριδινες ως αναστολεις κινασης jak3

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE0301373A SE0301373D0 (sv) 2003-05-09 2003-05-09 Novel compounds

Publications (1)

Publication Number Publication Date
SE0301373D0 true SE0301373D0 (sv) 2003-05-09

Family

ID=20291271

Family Applications (1)

Application Number Title Priority Date Filing Date
SE0301373A SE0301373D0 (sv) 2003-05-09 2003-05-09 Novel compounds

Country Status (17)

Country Link
US (1) US20060287355A1 (sv)
EP (2) EP1625126B1 (sv)
JP (1) JP2006525997A (sv)
CN (1) CN1784402A (sv)
AT (1) ATE384061T1 (sv)
AU (1) AU2004236144B2 (sv)
BR (1) BRPI0410081A (sv)
CA (1) CA2524624A1 (sv)
CY (1) CY1107301T1 (sv)
DE (1) DE602004011330T2 (sv)
DK (1) DK1625126T3 (sv)
ES (1) ES2298754T3 (sv)
MX (1) MXPA05012025A (sv)
PL (1) PL1625126T3 (sv)
PT (1) PT1625126E (sv)
SE (1) SE0301373D0 (sv)
WO (1) WO2004099204A1 (sv)

Families Citing this family (65)

* Cited by examiner, † Cited by third party
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