EA200801608A1 - Производные бензимидазолонкарбоновой кислоты - Google Patents
Производные бензимидазолонкарбоновой кислотыInfo
- Publication number
- EA200801608A1 EA200801608A1 EA200801608A EA200801608A EA200801608A1 EA 200801608 A1 EA200801608 A1 EA 200801608A1 EA 200801608 A EA200801608 A EA 200801608A EA 200801608 A EA200801608 A EA 200801608A EA 200801608 A1 EA200801608 A1 EA 200801608A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- benzimidazolonic
- derivatives
- carbonic acid
- carbonic
- compounds
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/10—Laxatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/26—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
Abstract
Настоящее изобретение относится к соединениям формулы (XI), где каждый из R
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2004177488A JP4129445B2 (ja) | 2004-06-15 | 2004-06-15 | ベンズイミダゾロンカルボン酸誘導体 |
US60704804P | 2004-09-02 | 2004-09-02 | |
US60700804P | 2004-09-02 | 2004-09-02 | |
US60703504P | 2004-09-02 | 2004-09-02 |
Publications (1)
Publication Number | Publication Date |
---|---|
EA200801608A1 true EA200801608A1 (ru) | 2008-10-30 |
Family
ID=35414645
Family Applications (3)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200801608A EA200801608A1 (ru) | 2004-06-15 | 2005-06-01 | Производные бензимидазолонкарбоновой кислоты |
EA200602122A EA010891B9 (ru) | 2004-06-15 | 2005-06-01 | Производные бензимидазолонкарбоновой кислоты |
EA200801607A EA200801607A1 (ru) | 2004-06-15 | 2005-06-01 | Производные бензимидазолонкарбоновой кислоты |
Family Applications After (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200602122A EA010891B9 (ru) | 2004-06-15 | 2005-06-01 | Производные бензимидазолонкарбоновой кислоты |
EA200801607A EA200801607A1 (ru) | 2004-06-15 | 2005-06-01 | Производные бензимидазолонкарбоновой кислоты |
Country Status (24)
Country | Link |
---|---|
US (3) | US7705020B2 (ru) |
EP (1) | EP1758891A2 (ru) |
KR (1) | KR100875558B1 (ru) |
AR (1) | AR049353A1 (ru) |
AU (1) | AU2005254800B2 (ru) |
BR (1) | BRPI0512046A (ru) |
CA (1) | CA2569654C (ru) |
CR (1) | CR8756A (ru) |
EA (3) | EA200801608A1 (ru) |
EC (1) | ECSP067079A (ru) |
GE (1) | GEP20094638B (ru) |
GT (1) | GT200500156A (ru) |
HK (1) | HK1104031A1 (ru) |
IL (1) | IL179612A (ru) |
MA (1) | MA28667B1 (ru) |
MX (1) | MXPA06014486A (ru) |
NL (1) | NL1029250C2 (ru) |
NO (1) | NO20065160L (ru) |
PA (1) | PA8636901A1 (ru) |
PE (1) | PE20060298A1 (ru) |
SV (1) | SV2008002145A (ru) |
TW (1) | TWI298635B (ru) |
UY (1) | UY28961A1 (ru) |
WO (1) | WO2005123718A2 (ru) |
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WO1998003167A1 (en) | 1996-07-24 | 1998-01-29 | Warner-Lambert Company | Isobutylgaba and its derivatives for the treatment of pain |
BRPI0414105B8 (pt) * | 2003-09-03 | 2021-05-25 | Askat Inc | compostos de benzimidazolona com atividade agonista do receptor 5-ht4 |
WO2005123718A2 (en) * | 2004-06-15 | 2005-12-29 | Pfizer Japan Inc. | Benzimidazolone carboxylic acid derivatives |
US7396933B2 (en) * | 2004-11-05 | 2008-07-08 | Theravance, Inc. | Quinolinone-carboxamide compounds |
JP5086091B2 (ja) * | 2004-11-05 | 2012-11-28 | セラヴァンス, インコーポレーテッド | 5−ht4受容体アゴニスト化合物 |
CN101080406A (zh) * | 2004-12-22 | 2007-11-28 | 施万制药 | 吲唑-甲酰胺化合物 |
EP1856110B1 (en) | 2005-02-22 | 2011-06-22 | Pfizer Inc. | Oxyindole derivatives as 5ht4 receptor agonists |
CN101163701A (zh) * | 2005-03-02 | 2008-04-16 | 施万制药 | 作为5-ht4受体激动剂的喹啉酮化合物 |
JP2008533121A (ja) * | 2005-03-15 | 2008-08-21 | ファイザー株式会社 | Cb2受容体リガンドとしてのベンズイミダゾロン誘導体 |
AU2006262101A1 (en) * | 2005-06-23 | 2007-01-04 | Merck & Co., Inc. | 3-fluoro-piperidine T-type calcium channel antagonists |
US8501773B2 (en) * | 2005-06-29 | 2013-08-06 | Merck Sharp & Dohme Corp. | 4-fluoro-piperidine T-type calcium channel antagonists |
GB0525068D0 (en) | 2005-12-08 | 2006-01-18 | Novartis Ag | Organic compounds |
KR20140147142A (ko) * | 2006-01-24 | 2014-12-29 | 가부시키가이샤 아루떼꾸 우에노 | 바이-사이클릭 화합물을 함유하는 약학적 조성물 및 바이-사이클릭 화합물의 안정화 방법 |
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CA2716367C (en) | 2008-02-20 | 2015-05-26 | The Curators Of The University Of Missouri | Composition comprising a combination of omeprazole and lansoprazole, and a buffering agent, and methods of using same |
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US8835444B2 (en) | 2010-02-02 | 2014-09-16 | Novartis Ag | Cyclohexyl amide derivatives as CRF receptor antagonists |
US8980922B2 (en) | 2010-02-12 | 2015-03-17 | Raqualia Pharma Inc. | 5-HT4 receptor agonists for the treatment of dementia |
UY34094A (es) | 2011-05-27 | 2013-01-03 | Novartis Ag | Derivados de la piperidina 3-espirocíclica como agonistas de receptores de la ghrelina |
PE20142443A1 (es) | 2012-05-03 | 2015-01-28 | Novartis Ag | Sal de l-malato de derivados de 2,7-diaza-espiro[4,5]dec-7-ilo y formas cristalinas de los mismos como agonistas del receptor de grelina |
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- 2005-06-01 WO PCT/IB2005/001825 patent/WO2005123718A2/en active Application Filing
- 2005-06-01 CA CA2569654A patent/CA2569654C/en not_active Expired - Fee Related
- 2005-06-01 GE GEAP20059755A patent/GEP20094638B/en unknown
- 2005-06-01 EA EA200801608A patent/EA200801608A1/ru unknown
- 2005-06-01 MX MXPA06014486A patent/MXPA06014486A/es active IP Right Grant
- 2005-06-01 BR BRPI0512046-2A patent/BRPI0512046A/pt not_active IP Right Cessation
- 2005-06-01 KR KR1020067026378A patent/KR100875558B1/ko not_active IP Right Cessation
- 2005-06-01 EA EA200602122A patent/EA010891B9/ru not_active IP Right Cessation
- 2005-06-01 EA EA200801607A patent/EA200801607A1/ru unknown
- 2005-06-01 EP EP05750293A patent/EP1758891A2/en not_active Withdrawn
- 2005-06-01 AU AU2005254800A patent/AU2005254800B2/en not_active Ceased
- 2005-06-13 PE PE2005000671A patent/PE20060298A1/es not_active Application Discontinuation
- 2005-06-14 NL NL1029250A patent/NL1029250C2/nl not_active IP Right Cessation
- 2005-06-14 UY UY28961A patent/UY28961A1/es not_active Application Discontinuation
- 2005-06-14 US US11/153,775 patent/US7705020B2/en not_active Expired - Fee Related
- 2005-06-14 US US11/153,757 patent/US7595329B2/en not_active Expired - Fee Related
- 2005-06-14 AR ARP050102433A patent/AR049353A1/es not_active Application Discontinuation
- 2005-06-14 TW TW094119692A patent/TWI298635B/zh not_active IP Right Cessation
- 2005-06-15 GT GT200500156A patent/GT200500156A/es unknown
- 2005-06-15 SV SV2005002145A patent/SV2008002145A/es unknown
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2006
- 2006-11-09 NO NO20065160A patent/NO20065160L/no not_active Application Discontinuation
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- 2006-12-13 EC EC2006007079A patent/ECSP067079A/es unknown
- 2006-12-15 MA MA29536A patent/MA28667B1/fr unknown
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2007
- 2007-07-27 HK HK07108217.3A patent/HK1104031A1/xx not_active IP Right Cessation
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2008
- 2008-01-09 US US11/971,265 patent/US20080108660A1/en not_active Abandoned
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