UA101493C2 - Производные азетидина и циклобутана как ингибиторы jak - Google Patents

Производные азетидина и циклобутана как ингибиторы jak

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Publication number
UA101493C2
UA101493C2 UAA201010917A UAA201010917A UA101493C2 UA 101493 C2 UA101493 C2 UA 101493C2 UA A201010917 A UAA201010917 A UA A201010917A UA A201010917 A UAA201010917 A UA A201010917A UA 101493 C2 UA101493 C2 UA 101493C2
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UA
Ukraine
Prior art keywords
azetidine
jak inhibitors
cyclobutane derivatives
jak
cyclobutane
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UAA201010917A
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English (en)
Ukrainian (uk)
Inventor
Джеймс Д. Роджерс
Стейси Шепард
Юнь-Лун Ли
Цзячен Чжоу
Пинли Лю
Дейвид Мелони
Майкл Ся
Original Assignee
Инсайт Корпорейшн
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Application filed by Инсайт Корпорейшн filed Critical Инсайт Корпорейшн
Publication of UA101493C2 publication Critical patent/UA101493C2/ru

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  • Health & Medical Sciences (AREA)
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Abstract

Изобретение касается производных азетидина и циклобутана, а также композиций, содержащих эти соединения, их применения и способов получения, которые являются ингибиторами JAK, полезными при лечении обусловленных JAK заболеваний, в том числе, например, воспалительных и аутоимунных расстройств, а также рака.
UAA201010917A 2008-03-11 2009-03-10 Производные азетидина и циклобутана как ингибиторы jak UA101493C2 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US3566208P 2008-03-11 2008-03-11
US14498209P 2009-01-15 2009-01-15
PCT/US2009/036635 WO2009114512A1 (en) 2008-03-11 2009-03-10 Azetidine and cyclobutane derivatives as jak inhibitors

Publications (1)

Publication Number Publication Date
UA101493C2 true UA101493C2 (ru) 2013-04-10

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ID=40591836

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Application Number Title Priority Date Filing Date
UAA201010917A UA101493C2 (ru) 2008-03-11 2009-03-10 Производные азетидина и циклобутана как ингибиторы jak

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EP (1) EP2288610B8 (ru)
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KR (2) KR20120108042A (ru)
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AR (1) AR070828A1 (ru)
AU (1) AU2009223640B2 (ru)
BR (1) BRPI0909040B8 (ru)
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