GT199900216A - Polimorfos de acido 2-(3-ciano-4-isobutiloxifenil)-4-metil-5-tiazol carboxilico y metodo de produccion de los mismos. - Google Patents

Polimorfos de acido 2-(3-ciano-4-isobutiloxifenil)-4-metil-5-tiazol carboxilico y metodo de produccion de los mismos.

Info

Publication number
GT199900216A
GT199900216A GT199900216A GT199900216A GT199900216A GT 199900216 A GT199900216 A GT 199900216A GT 199900216 A GT199900216 A GT 199900216A GT 199900216 A GT199900216 A GT 199900216A GT 199900216 A GT199900216 A GT 199900216A
Authority
GT
Guatemala
Prior art keywords
polymorphes
acid
isobutiloxifenil
tiazol
ciano
Prior art date
Application number
GT199900216A
Other languages
English (en)
Inventor
Matsumoto Koichi
Watanabe Kenzo
Hiramatsu Toshiyuki
Kitamura Mitsutaka
Original Assignee
Teijin Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=15953825&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=GT199900216(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Teijin Ltd filed Critical Teijin Ltd
Publication of GT199900216A publication Critical patent/GT199900216A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Physical Education & Sports Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

LA PRESENTE INVENCION PROVEE UNA TECNICA PARA PRODUCIR SELECTIVAMENTE UN POLIMORFO DESEADO DE ACIDO 2(CIANO4ISOBUTILOXIFENIL)4METIL5TIAZOL CARBOXILICO (VER FÒRMULA I). ESTA PROVEE TAMBIEN UN METODO PARA PRODUCIR VARIOS POLIMORFOS, QUE COMPRENDE CRISTALIZAR BAJO LAS CONDICIONES DEFINIDAS POR UNA TEMPERATURA ESPECIFICA Y UNA COMPOSICION DE UN SOLVENTE MIXTO DE METANOL Y AGUA, Y LOS POLIMORFOS OBTENIDOS POR EL MEODO.
GT199900216A 1998-06-19 1999-12-16 Polimorfos de acido 2-(3-ciano-4-isobutiloxifenil)-4-metil-5-tiazol carboxilico y metodo de produccion de los mismos. GT199900216A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP17307998 1998-06-19

Publications (1)

Publication Number Publication Date
GT199900216A true GT199900216A (es) 2001-06-08

Family

ID=15953825

Family Applications (1)

Application Number Title Priority Date Filing Date
GT199900216A GT199900216A (es) 1998-06-19 1999-12-16 Polimorfos de acido 2-(3-ciano-4-isobutiloxifenil)-4-metil-5-tiazol carboxilico y metodo de produccion de los mismos.

Country Status (39)

Country Link
US (1) US6225474B1 (es)
EP (4) EP1956014B1 (es)
JP (1) JP3547707B2 (es)
KR (1) KR100511183B1 (es)
CN (3) CN102659712A (es)
AT (2) ATE449765T1 (es)
AU (1) AU748026B2 (es)
BE (1) BE2010C024I2 (es)
BG (1) BG64734B1 (es)
BR (1) BR9906539A (es)
CA (2) CA2301863C (es)
CY (3) CY1109720T1 (es)
CZ (1) CZ298170B6 (es)
DE (2) DE122010000013I1 (es)
DK (3) DK1956014T3 (es)
ES (3) ES2718467T3 (es)
FR (1) FR10C0022I2 (es)
GT (1) GT199900216A (es)
HK (2) HK1029788A1 (es)
HR (2) HRP20000092C1 (es)
HU (2) HU229405B1 (es)
ID (1) ID25775A (es)
IL (1) IL134594A (es)
IN (1) IN191537B (es)
IS (4) IS9020A (es)
LT (1) LT1956014T (es)
LU (1) LU91682I2 (es)
NO (1) NO321308B1 (es)
NZ (1) NZ503326A (es)
PL (1) PL200710B1 (es)
PT (3) PT1956015E (es)
RU (1) RU2198169C3 (es)
SI (3) SI1020454T2 (es)
SK (2) SK287946B6 (es)
TR (1) TR200000458T1 (es)
TW (1) TWI248439B (es)
UA (1) UA57611C2 (es)
WO (1) WO1999065885A1 (es)
ZA (1) ZA200000737B (es)

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Also Published As

Publication number Publication date
IL134594A0 (en) 2001-04-30
HK1029788A1 (en) 2001-04-12
RU2198169C3 (ru) 2017-07-20
AU4289299A (en) 2000-01-05
PL200710B1 (pl) 2009-01-30
PT1956014T (pt) 2019-04-24
ES2336287T5 (es) 2013-04-02
EP2404910A3 (en) 2014-10-29
HK1118293A1 (es) 2009-02-06
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