LT1956014T - 2-(3-ciano-4-izobutiloksifenil)-4-metil-5-tiazolkarboksirūgšties polimorfai ir jų gamybos būdas - Google Patents

2-(3-ciano-4-izobutiloksifenil)-4-metil-5-tiazolkarboksirūgšties polimorfai ir jų gamybos būdas

Info

Publication number
LT1956014T
LT1956014T LTEP08005933.0T LT08005933T LT1956014T LT 1956014 T LT1956014 T LT 1956014T LT 08005933 T LT08005933 T LT 08005933T LT 1956014 T LT1956014 T LT 1956014T
Authority
LT
Lithuania
Prior art keywords
polymorphs
producing
isobutyloxyphenyl
cyano
methyl
Prior art date
Application number
LTEP08005933.0T
Other languages
English (en)
Inventor
Kolchi Matsumoto
Kenzo Watanabe
Toshiyuki Hiramatsu
Mitsutaka Kitamura
Original Assignee
Teijin Pharma Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=15953825&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=LT1956014(T) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Teijin Pharma Limited filed Critical Teijin Pharma Limited
Publication of LT1956014T publication Critical patent/LT1956014T/lt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/56Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/06Antigout agents, e.g. antihyperuricemic or uricosuric agents
LTEP08005933.0T 1998-06-19 1999-06-18 2-(3-ciano-4-izobutiloksifenil)-4-metil-5-tiazolkarboksirūgšties polimorfai ir jų gamybos būdas LT1956014T (lt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP17307998 1998-06-19

Publications (1)

Publication Number Publication Date
LT1956014T true LT1956014T (lt) 2019-03-25

Family

ID=15953825

Family Applications (1)

Application Number Title Priority Date Filing Date
LTEP08005933.0T LT1956014T (lt) 1998-06-19 1999-06-18 2-(3-ciano-4-izobutiloksifenil)-4-metil-5-tiazolkarboksirūgšties polimorfai ir jų gamybos būdas

Country Status (39)

Country Link
US (1) US6225474B1 (lt)
EP (4) EP1956015B2 (lt)
JP (1) JP3547707B2 (lt)
KR (1) KR100511183B1 (lt)
CN (3) CN102659712A (lt)
AT (2) ATE522512T2 (lt)
AU (1) AU748026B2 (lt)
BE (1) BE2010C024I2 (lt)
BG (1) BG64734B1 (lt)
BR (1) BR9906539A (lt)
CA (2) CA2566652C (lt)
CY (3) CY1109720T1 (lt)
CZ (1) CZ298170B6 (lt)
DE (2) DE122010000013I1 (lt)
DK (3) DK1956015T4 (lt)
ES (3) ES2718467T3 (lt)
FR (1) FR10C0022I2 (lt)
GT (1) GT199900216A (lt)
HK (2) HK1029788A1 (lt)
HR (2) HRP20000092C1 (lt)
HU (2) HU229405B1 (lt)
ID (1) ID25775A (lt)
IL (1) IL134594A (lt)
IN (1) IN191537B (lt)
IS (4) IS9020A (lt)
LT (1) LT1956014T (lt)
LU (1) LU91682I2 (lt)
NO (1) NO321308B1 (lt)
NZ (1) NZ503326A (lt)
PL (1) PL200710B1 (lt)
PT (3) PT1956015E (lt)
RU (1) RU2198169C3 (lt)
SI (3) SI1020454T2 (lt)
SK (2) SK287928B6 (lt)
TR (1) TR200000458T1 (lt)
TW (1) TWI248439B (lt)
UA (1) UA57611C2 (lt)
WO (1) WO1999065885A1 (lt)
ZA (1) ZA200000737B (lt)

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CN107540630A (zh) * 2016-06-29 2018-01-05 康普药业股份有限公司 一种非布司他化合物及制备方法
GR1009119B (el) 2016-06-30 2017-09-18 "Φαρματεν Α.Β.Ε.Ε." Φαρμακευτικο σκευασμα περιεχον ενα μη πουρινικο επιλεκτικο αναστολεα της οξειδασης της ξανθινης και μεθοδος παρασκευης αυτου
KR20180013563A (ko) * 2016-07-29 2018-02-07 한미정밀화학주식회사 고순도 결정형 페북소스타트의 개선된 제조 방법
CN106565627B (zh) * 2016-10-10 2020-01-10 扬子江药业集团有限公司 一种非布司他药用晶型的制备方法
GR1009659B (el) 2018-09-07 2019-11-28 Φαρματεν Α.Β.Ε.Ε. Φαρμακευτικο σκευασμα που περιλαμβανει ενα συμπλοκο αλατος της φεβουξοστατης με οξειδιο του μαγνησιου και μεθοδος για την παρασκευη αυτου
WO2020067275A1 (ja) * 2018-09-28 2020-04-02 株式会社カネカ 安定性に優れた還元型補酵素q10結晶の製造方法
CN112390766B (zh) * 2019-08-13 2022-09-06 浙江天宇药业股份有限公司 一种非布司他a晶型的制备方法
CN111004191A (zh) * 2019-10-24 2020-04-14 武汉光谷亚太医药研究院有限公司 一种大粒径非布司他a晶的制备方法
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CY2010006I2 (el) 2012-01-25
SI1956015T1 (sl) 2011-10-28
EP1956015A3 (en) 2008-09-17
HUP0004325A2 (hu) 2001-10-28
PT1020454E (pt) 2009-12-21
BE2010C024I2 (en) 2018-08-24
HRP20000092A2 (en) 2000-08-31
EP1956014A3 (en) 2008-08-20
IS3002B (is) 2018-09-15
IL134594A (en) 2004-12-15
WO1999065885A1 (en) 1999-12-23
CZ298170B6 (cs) 2007-07-11
CN102020617B (zh) 2019-04-23
IS2886B (is) 2014-07-15
ES2336287T3 (es) 2010-04-09
US6225474B1 (en) 2001-05-01
DK1020454T3 (da) 2010-01-04
EP1956014B1 (en) 2019-01-16
SI1956014T1 (sl) 2019-02-28
CZ2000582A3 (cs) 2000-07-12
CA2301863A1 (en) 1999-12-23
AU748026B2 (en) 2002-05-30
CN1275126A (zh) 2000-11-29
ATE449765T1 (de) 2009-12-15
BG64734B1 (bg) 2006-01-31
EP1020454B2 (en) 2013-01-23
SI1956015T2 (sl) 2018-12-31
SK287928B6 (sk) 2012-04-03
SI1020454T2 (sl) 2013-03-29
IN191537B (lt) 2003-12-06
KR100511183B1 (ko) 2005-08-30
CA2566652A1 (en) 1999-12-23
JP3547707B2 (ja) 2004-07-28
DK1020454T4 (da) 2013-11-25
GT199900216A (es) 2001-06-08
CY1109720T1 (el) 2012-01-25
EP2404910A3 (en) 2014-10-29
ES2336287T5 (es) 2013-04-02
CN102659712A (zh) 2012-09-12
ES2371786T3 (es) 2012-01-10
HRP20120217A2 (hr) 2012-05-31
RU2198169C3 (ru) 2017-07-20
NO20000789D0 (no) 2000-02-17
ATE522512T2 (de) 2011-09-15
AU4289299A (en) 2000-01-05
ZA200000737B (en) 2000-09-08
HRP20120217B1 (hr) 2019-04-05
PT1956014T (pt) 2019-04-24
HU229405B1 (en) 2013-12-30
NO20000789L (no) 2000-02-17
ES2371786T5 (es) 2019-04-22
HK1029788A1 (en) 2001-04-12
CN102020617A (zh) 2011-04-20
EP1956015A2 (en) 2008-08-13
EP1956015B1 (en) 2011-08-31
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