NO322470B1 - Cyklisk protein-tyrosin-kinase-inhibitor, anvendelse av slike for fremstilling av farmasøytiske preparater for behandling av lidelser og farmasøytiske preparater inneholdende slike. - Google Patents

Cyklisk protein-tyrosin-kinase-inhibitor, anvendelse av slike for fremstilling av farmasøytiske preparater for behandling av lidelser og farmasøytiske preparater inneholdende slike. Download PDF

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Publication number
NO322470B1
NO322470B1 NO20014970A NO20014970A NO322470B1 NO 322470 B1 NO322470 B1 NO 322470B1 NO 20014970 A NO20014970 A NO 20014970A NO 20014970 A NO20014970 A NO 20014970A NO 322470 B1 NO322470 B1 NO 322470B1
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Norway
Prior art keywords
amino
thiazolecarboxamide
chloro
methylphenyl
methyl
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Application number
NO20014970A
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English (en)
Norwegian (no)
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NO20014970L (no
NO20014970D0 (no
Inventor
Jagabandhu Das
Joel C Barrish
John Wityak
Ramesh Padmanabha
Ping Chen
Derek J Norris
Arthur M Doweyko
Original Assignee
Bristol Myers Squibb Co
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Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of NO20014970D0 publication Critical patent/NO20014970D0/no
Publication of NO20014970L publication Critical patent/NO20014970L/no
Publication of NO322470B1 publication Critical patent/NO322470B1/no

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    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
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    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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    • C07D491/10—Spiro-condensed systems
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NO20014970A 1999-04-15 2001-10-12 Cyklisk protein-tyrosin-kinase-inhibitor, anvendelse av slike for fremstilling av farmasøytiske preparater for behandling av lidelser og farmasøytiske preparater inneholdende slike. NO322470B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US12951099P 1999-04-15 1999-04-15
PCT/US2000/009753 WO2000062778A1 (en) 1999-04-15 2000-04-12 Cyclic protein tyrosine kinase inhibitors

Publications (3)

Publication Number Publication Date
NO20014970D0 NO20014970D0 (no) 2001-10-12
NO20014970L NO20014970L (no) 2001-12-10
NO322470B1 true NO322470B1 (no) 2006-10-09

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ID=22440334

Family Applications (3)

Application Number Title Priority Date Filing Date
NO20014970A NO322470B1 (no) 1999-04-15 2001-10-12 Cyklisk protein-tyrosin-kinase-inhibitor, anvendelse av slike for fremstilling av farmasøytiske preparater for behandling av lidelser og farmasøytiske preparater inneholdende slike.
NO2007005C NO2007005I1 (no) 1999-04-15 2007-03-27 N-(2-klor-6-metylfenyl)-2-[[6-[4-(2-hydroksyetyl)-1-piperazinyl]-2-metyl-4-pyrimidinyl]amino]5-tiazolkarboksamid
NO2019016C NO2019016I1 (no) 1999-04-15 2019-04-05 dasatinib

Family Applications After (2)

Application Number Title Priority Date Filing Date
NO2007005C NO2007005I1 (no) 1999-04-15 2007-03-27 N-(2-klor-6-metylfenyl)-2-[[6-[4-(2-hydroksyetyl)-1-piperazinyl]-2-metyl-4-pyrimidinyl]amino]5-tiazolkarboksamid
NO2019016C NO2019016I1 (no) 1999-04-15 2019-04-05 dasatinib

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