JP2005525291A5 - - Google Patents
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- JP2005525291A5 JP2005525291A5 JP2003520733A JP2003520733A JP2005525291A5 JP 2005525291 A5 JP2005525291 A5 JP 2005525291A5 JP 2003520733 A JP2003520733 A JP 2003520733A JP 2003520733 A JP2003520733 A JP 2003520733A JP 2005525291 A5 JP2005525291 A5 JP 2005525291A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- solvate
- salt
- compound
- formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE0102764A SE0102764D0 (sv) | 2001-08-17 | 2001-08-17 | Compounds |
| PCT/GB2002/003745 WO2003015774A1 (en) | 2001-08-17 | 2002-08-15 | Compounds effecting glucokinase |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2005168987A Division JP4441446B2 (ja) | 2001-08-17 | 2005-06-09 | グルコキナーゼ化合物 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2005525291A JP2005525291A (ja) | 2005-08-25 |
| JP2005525291A5 true JP2005525291A5 (enExample) | 2006-01-05 |
| JP3987829B2 JP3987829B2 (ja) | 2007-10-10 |
Family
ID=20285065
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003520733A Expired - Fee Related JP3987829B2 (ja) | 2001-08-17 | 2002-08-15 | グルコキナーゼ化合物 |
| JP2005168987A Expired - Fee Related JP4441446B2 (ja) | 2001-08-17 | 2005-06-09 | グルコキナーゼ化合物 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2005168987A Expired - Fee Related JP4441446B2 (ja) | 2001-08-17 | 2005-06-09 | グルコキナーゼ化合物 |
Country Status (31)
| Country | Link |
|---|---|
| US (3) | US7390908B2 (enExample) |
| EP (12) | EP1661567B1 (enExample) |
| JP (2) | JP3987829B2 (enExample) |
| KR (1) | KR100920439B1 (enExample) |
| CN (4) | CN101584691A (enExample) |
| AR (1) | AR037898A1 (enExample) |
| AT (11) | ATE359781T1 (enExample) |
| AU (1) | AU2002321462B2 (enExample) |
| BR (1) | BR0212008A (enExample) |
| CA (1) | CA2457410C (enExample) |
| CO (1) | CO5560563A2 (enExample) |
| CY (5) | CY1105746T1 (enExample) |
| DE (11) | DE60227119D1 (enExample) |
| DK (5) | DK1568367T5 (enExample) |
| ES (10) | ES2309862T3 (enExample) |
| HU (1) | HUP0401213A3 (enExample) |
| IL (2) | IL160219A0 (enExample) |
| IS (1) | IS7150A (enExample) |
| MX (1) | MXPA04001500A (enExample) |
| MY (1) | MY146279A (enExample) |
| NO (1) | NO20040686L (enExample) |
| NZ (1) | NZ531193A (enExample) |
| PL (1) | PL368970A1 (enExample) |
| PT (5) | PT1669068E (enExample) |
| RU (1) | RU2329043C9 (enExample) |
| SE (1) | SE0102764D0 (enExample) |
| SI (5) | SI1661569T1 (enExample) |
| TW (1) | TWI333855B (enExample) |
| UA (1) | UA83182C2 (enExample) |
| WO (1) | WO2003015774A1 (enExample) |
| ZA (1) | ZA200401015B (enExample) |
Families Citing this family (147)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE0102299D0 (sv) | 2001-06-26 | 2001-06-26 | Astrazeneca Ab | Compounds |
| SE0102300D0 (sv) * | 2001-06-26 | 2001-06-26 | Astrazeneca Ab | Compounds |
| SE0102764D0 (sv) * | 2001-08-17 | 2001-08-17 | Astrazeneca Ab | Compounds |
| JP2004123732A (ja) * | 2002-09-10 | 2004-04-22 | Takeda Chem Ind Ltd | 5員複素環化合物 |
| WO2004024705A1 (ja) * | 2002-09-10 | 2004-03-25 | Takeda Pharmaceutical Company Limited | 5員複素環化合物 |
| PL375021A1 (en) | 2002-10-03 | 2005-11-14 | Novartis Ag | Substituted (thiazol-2-yl) -amide or sulfonamide as glycokinase activators useful in the treatment of type 2 diabetes |
| GB0226930D0 (en) | 2002-11-19 | 2002-12-24 | Astrazeneca Ab | Chemical compounds |
| GB0226931D0 (en) | 2002-11-19 | 2002-12-24 | Astrazeneca Ab | Chemical compounds |
| PL378117A1 (pl) | 2003-02-11 | 2006-03-06 | Prosidion Limited | Tricyklopodstawione związki amidowe |
| BRPI0407283A (pt) | 2003-02-13 | 2006-01-31 | Banyu Pharma Co Ltd | Composto, composição farmacêutica, e, agente ativador de glucoquinase, agentes terapêuticos e/ou agentes preventivos para diabetes melito e obesidade |
| WO2004076420A1 (ja) | 2003-02-26 | 2004-09-10 | Banyu Pharmaceutical Co., Ltd. | ヘテロアリールカルバモイルベンゼン誘導体 |
| JP2006525361A (ja) * | 2003-05-02 | 2006-11-09 | エラン ファーマシューティカルズ,インコーポレイテッド | ブラジキニンb1受容体アンタゴニストとしての選択された置換ピラゾール誘導体および関連化合物 |
| ATE410161T1 (de) * | 2003-05-02 | 2008-10-15 | Elan Pharm Inc | 4-bromo-5-(2-chloro-benzoylamino)-1h-pyrazol-3- carbonsäureamid-derivate und verwandte verbindungen als bradykinin b1 rezeptor antagonisten zur behandlung von entzündlichen erkrankungen |
| BRPI0411699A (pt) * | 2003-06-20 | 2006-08-29 | Hoffmannn La Roche Ag F | compostos para uso como substáncia terapeuticamente ativa; método para o tratamento e/ou profilaxia de doenças que estão associadas à modulação de receptores cb1 e uso destes compostos |
| ES2222822B1 (es) * | 2003-07-28 | 2005-12-16 | Laboratorios Farmaceuticos Rovi, S.A. | Diamidas de aminoacidos en posicion no alfa utiles como adyuvantes para la administracion de agentes biologicos activos. |
| WO2005046683A1 (en) | 2003-10-07 | 2005-05-26 | Renovis, Inc. | Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same |
| GB0325402D0 (en) * | 2003-10-31 | 2003-12-03 | Astrazeneca Ab | Compounds |
| GB0328178D0 (en) * | 2003-12-05 | 2004-01-07 | Astrazeneca Ab | Compounds |
| JP2007523905A (ja) * | 2004-02-18 | 2007-08-23 | アストラゼネカ アクチボラグ | 化合物 |
| EP2048137A1 (en) * | 2004-02-18 | 2009-04-15 | AstraZeneca AB | Benzamide derivatives and their use as glucokinase activating agents. |
| US7781451B2 (en) | 2004-04-02 | 2010-08-24 | Novartis Ag | Thiazolopyridine derivatives, pharmaceut ical conditions containing them and methods of treating glucokinase mediated conditions |
| US20080125403A1 (en) | 2004-04-02 | 2008-05-29 | Merck & Co., Inc. | Method of Treating Men with Metabolic and Anthropometric Disorders |
| PT1735322E (pt) | 2004-04-02 | 2012-01-12 | Novartis Ag | Derivados de sulfonamido-tiazolopiridina como activadores de glucoquinase úteis para o tratamento de diabetes de tipo 2 |
| TW200600086A (en) * | 2004-06-05 | 2006-01-01 | Astrazeneca Ab | Chemical compound |
| RU2403246C2 (ru) * | 2004-06-05 | 2010-11-10 | Астразенека Аб | Гетероарилбензамидные производные для применения в качестве активаторов глюкокиназы (glk) в лечении диабета |
| KR100739367B1 (ko) * | 2004-07-14 | 2007-07-16 | 크리스탈지노믹스(주) | 설파마이드 유도체 및 이를 함유하는 지방대사 촉진용약학적 조성물 |
| GB0423044D0 (en) * | 2004-10-16 | 2004-11-17 | Astrazeneca Ab | Compounds |
| BRPI0516595A (pt) | 2004-10-16 | 2008-09-23 | Astrazeneca Ab | processo para fabricar um composto, e, composto |
| GB0423043D0 (en) * | 2004-10-16 | 2004-11-17 | Astrazeneca Ab | Compounds |
| US7576099B2 (en) | 2005-02-28 | 2009-08-18 | Renovis, Inc. | Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same |
| BRPI0609464A2 (pt) * | 2005-05-23 | 2010-04-13 | Japan Tobacco Inc | composto de pirazol e agente terapêutico para diabetes compreendendo o mesmo |
| EP1891069A1 (en) * | 2005-05-24 | 2008-02-27 | AstraZeneca AB | 2-phenyl substituted imidazol [4,5b]pyridine/ pyrazine and purine derivatives as glucokinase modulators |
| TW200714597A (en) * | 2005-05-27 | 2007-04-16 | Astrazeneca Ab | Chemical compounds |
| GB0510852D0 (en) * | 2005-05-27 | 2005-07-06 | Astrazeneca Ab | Chemical compounds |
| EP2027113A1 (en) * | 2005-07-09 | 2009-02-25 | AstraZeneca AB | Heteroaryl benzamide derivatives for use as glk activators in the treatment of diabetes |
| US20110053910A1 (en) * | 2005-07-09 | 2011-03-03 | Mckerrecher Darren | 2 -heterocyclyloxybenzoyl amino heterocyclyl compounds as modulators of glucokinase for the treatment of type 2 diabetes |
| KR20110084339A (ko) | 2005-07-09 | 2011-07-21 | 아스트라제네카 아베 | 당뇨병 치료에 있어 glk 활성화제로서 사용하기 위한 헤테로아릴 벤즈아미드 유도체 |
| GB0514173D0 (en) * | 2005-07-09 | 2005-08-17 | Astrazeneca Ab | Chemical compounds |
| RU2415141C2 (ru) * | 2005-07-09 | 2011-03-27 | Астразенека Аб | Производные гетероарилбензамида для применения в качестве активаторов glk в лечении диабета |
| ES2426345T3 (es) | 2005-07-20 | 2013-10-22 | Eli Lilly And Company | Compuesto unidos en posición 1-amino |
| US9202182B2 (en) * | 2005-08-11 | 2015-12-01 | International Business Machines Corporation | Method and system for analyzing business architecture |
| JP2007063225A (ja) | 2005-09-01 | 2007-03-15 | Takeda Chem Ind Ltd | イミダゾピリジン化合物 |
| NZ566877A (en) | 2005-09-29 | 2010-05-28 | Sanofi Aventis | Phenyl-1,2,4-oxadiazolone derivatives, processes for their preparation and their use as pharmaceuticals |
| GT200600429A (es) | 2005-09-30 | 2007-04-30 | Compuestos organicos | |
| GT200600428A (es) | 2005-09-30 | 2007-05-21 | Compuestos organicos | |
| CN101312940B (zh) | 2005-11-17 | 2012-11-14 | 伊莱利利公司 | 胰高血糖素受体拮抗剂、制备和治疗用途 |
| TW200738621A (en) | 2005-11-28 | 2007-10-16 | Astrazeneca Ab | Chemical process |
| EP2001875A2 (en) | 2006-03-08 | 2008-12-17 | Takeda San Diego, Inc. | Glucokinase activators |
| EP2010520B1 (en) * | 2006-04-20 | 2012-09-12 | Pfizer Products Inc. | Heterobicyclic amides for the prevention and treatment of glucokinase-mediated diseases |
| EP2019824A2 (en) | 2006-04-28 | 2009-02-04 | Transtech Pharma, Inc. | Benzamide glucokinase activators |
| CA2669708A1 (en) * | 2006-04-28 | 2007-11-08 | Transtech Pharma, Inc. | Benzamide glucokinase activators |
| PE20080251A1 (es) | 2006-05-04 | 2008-04-25 | Boehringer Ingelheim Int | Usos de inhibidores de dpp iv |
| UA93548C2 (uk) | 2006-05-05 | 2011-02-25 | Айерем Елелсі | Сполуки та композиції як модулятори хеджхогівського сигнального шляху |
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| US7888504B2 (en) * | 2006-07-06 | 2011-02-15 | Bristol-Myers Squibb Company | Glucokinase activators and methods of using same |
| US7910747B2 (en) | 2006-07-06 | 2011-03-22 | Bristol-Myers Squibb Company | Phosphonate and phosphinate pyrazolylamide glucokinase activators |
| JP2009544648A (ja) | 2006-07-24 | 2009-12-17 | エフ.ホフマン−ラ ロシュ アーゲー | グルコキナーゼ活性化剤としてのピラゾール類 |
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