HK1172341A1 - Novel crystalline heteroaromatic fluoroglycoside hydrates, pharmaceuticals comprising these compounds and their use - Google Patents

Novel crystalline heteroaromatic fluoroglycoside hydrates, pharmaceuticals comprising these compounds and their use

Info

Publication number
HK1172341A1
HK1172341A1 HK12113296.0A HK12113296A HK1172341A1 HK 1172341 A1 HK1172341 A1 HK 1172341A1 HK 12113296 A HK12113296 A HK 12113296A HK 1172341 A1 HK1172341 A1 HK 1172341A1
Authority
HK
Hong Kong
Prior art keywords
hydrates
pharmaceuticals
compounds
novel crystalline
fluoroglycoside
Prior art date
Application number
HK12113296.0A
Other languages
English (en)
Inventor
David Rigal
Franceska Fischer
Bernd Becker
Martin Feth
Norbert Nagel
Bruno Baumgartner
Martin Broeckelmann
Original Assignee
Sanofi Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Sa filed Critical Sanofi Sa
Publication of HK1172341A1 publication Critical patent/HK1172341A1/xx

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/02—Heterocyclic radicals containing only nitrogen as ring hetero atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Diabetes (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
HK12113296.0A 2009-08-26 2012-12-24 Novel crystalline heteroaromatic fluoroglycoside hydrates, pharmaceuticals comprising these compounds and their use HK1172341A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP09290650 2009-08-26
PCT/EP2010/062461 WO2011023754A1 (fr) 2009-08-26 2010-08-26 Nouveaux hydrates de fluoroglycoside hétéroaromatiques cristallins, substances pharmaceutiques comprenant ces composés et leur utilisation

Publications (1)

Publication Number Publication Date
HK1172341A1 true HK1172341A1 (en) 2013-04-19

Family

ID=41426365

Family Applications (1)

Application Number Title Priority Date Filing Date
HK12113296.0A HK1172341A1 (en) 2009-08-26 2012-12-24 Novel crystalline heteroaromatic fluoroglycoside hydrates, pharmaceuticals comprising these compounds and their use

Country Status (17)

Country Link
US (1) US8785608B2 (fr)
EP (1) EP2470552B1 (fr)
JP (1) JP2013503135A (fr)
KR (1) KR20120060207A (fr)
CN (1) CN102482312A (fr)
AU (1) AU2010288523A1 (fr)
BR (1) BR112012003973A2 (fr)
CA (1) CA2771278A1 (fr)
DK (1) DK2470552T3 (fr)
ES (1) ES2443016T3 (fr)
HK (1) HK1172341A1 (fr)
IL (1) IL218225A0 (fr)
MX (1) MX2012001729A (fr)
PT (1) PT2470552E (fr)
RU (1) RU2012111354A (fr)
SG (1) SG178880A1 (fr)
WO (1) WO2011023754A1 (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR101721831B1 (ko) * 2014-11-06 2017-03-31 주식회사 종근당 로베글리타존을 함유하는 경구 투여용 약제학적 조성물
JP2023509800A (ja) * 2020-01-10 2023-03-09 コンシナンス セラピューティクス， インコーポレイテッド 薬物の治療的組み合わせ及びそれらの使用方法

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WO2011023754A1 (fr) 2011-03-03
IL218225A0 (en) 2012-04-30
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BR112012003973A2 (pt) 2015-09-08
KR20120060207A (ko) 2012-06-11
ES2443016T3 (es) 2014-02-17
CA2771278A1 (fr) 2011-03-03
AU2010288523A1 (en) 2012-03-15
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PT2470552E (pt) 2014-01-30

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