AU2001292670A1 - Pyrazole compounds useful as protein kinase inhibitors - Google Patents

Pyrazole compounds useful as protein kinase inhibitors

Info

Publication number
AU2001292670A1
AU2001292670A1 AU2001292670A AU9267001A AU2001292670A1 AU 2001292670 A1 AU2001292670 A1 AU 2001292670A1 AU 2001292670 A AU2001292670 A AU 2001292670A AU 9267001 A AU9267001 A AU 9267001A AU 2001292670 A1 AU2001292670 A1 AU 2001292670A1
Authority
AU
Australia
Prior art keywords
ring
optionally substituted
aliphatic
halo
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2001292670A
Other languages
English (en)
Inventor
David Bebbington
Jean-Damien Charrier
Robert Davies
Julian M.C. Golec
Ronald Knegtel
Pan Li
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Vertex Pharmaceuticals Inc
Original Assignee
Vertex Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27398347&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AU2001292670(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Vertex Pharmaceuticals Inc filed Critical Vertex Pharmaceuticals Inc
Publication of AU2001292670A1 publication Critical patent/AU2001292670A1/en
Abandoned legal-status Critical Current

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    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
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    • C07—ORGANIC CHEMISTRY
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    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
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    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
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    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Endocrinology (AREA)
  • Rheumatology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Neurosurgery (AREA)
  • Pulmonology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychiatry (AREA)
  • Emergency Medicine (AREA)
  • Oncology (AREA)
  • Hospice & Palliative Care (AREA)
  • Dermatology (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Pain & Pain Management (AREA)
  • Transplantation (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
AU2001292670A 2000-09-15 2001-09-14 Pyrazole compounds useful as protein kinase inhibitors Abandoned AU2001292670A1 (en)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US23279500P 2000-09-15 2000-09-15
US60232795 2000-09-15
US25788700P 2000-12-21 2000-12-21
US60257887 2000-12-21
US28694901P 2001-04-27 2001-04-27
US60286949 2001-04-27
PCT/US2001/028793 WO2002022605A1 (en) 2000-09-15 2001-09-14 Pyrazole compounds useful as protein kinase inhibitors

Publications (1)

Publication Number Publication Date
AU2001292670A1 true AU2001292670A1 (en) 2002-03-26

Family

ID=27398347

Family Applications (9)

Application Number Title Priority Date Filing Date
AU2001292670A Abandoned AU2001292670A1 (en) 2000-09-15 2001-09-14 Pyrazole compounds useful as protein kinase inhibitors
AU2001294558A Abandoned AU2001294558A1 (en) 2000-09-15 2001-09-14 Pyrazole compounds useful as protein kinase inhibitors
AU2001290912A Abandoned AU2001290912A1 (en) 2000-09-15 2001-09-14 Pyrazole compounds useful as protein kinase inhibitors
AU2001290944A Abandoned AU2001290944A1 (en) 2000-09-15 2001-09-14 Pyrazole compounds useful as protein kinase inhibitors
AU2001296875A Abandoned AU2001296875A1 (en) 2000-09-15 2001-09-14 Triazole compounds useful as protein kinase inhibitors
AU2001296871A Abandoned AU2001296871A1 (en) 2000-09-15 2001-09-14 Pyrazole compounds useful as protein kinase inhibitors
AU2001290914A Abandoned AU2001290914A1 (en) 2000-09-15 2001-09-14 Pyrazole compounds useful as protein kinase inhibitors
AU2001291013A Abandoned AU2001291013A1 (en) 2000-09-15 2001-09-14 Pyrazole compounds useful as protein kinase inhibitors
AU2008252044A Abandoned AU2008252044A1 (en) 2000-09-15 2008-12-03 Compounds Useful as Protein Kinase Inhibitors

Family Applications After (8)

Application Number Title Priority Date Filing Date
AU2001294558A Abandoned AU2001294558A1 (en) 2000-09-15 2001-09-14 Pyrazole compounds useful as protein kinase inhibitors
AU2001290912A Abandoned AU2001290912A1 (en) 2000-09-15 2001-09-14 Pyrazole compounds useful as protein kinase inhibitors
AU2001290944A Abandoned AU2001290944A1 (en) 2000-09-15 2001-09-14 Pyrazole compounds useful as protein kinase inhibitors
AU2001296875A Abandoned AU2001296875A1 (en) 2000-09-15 2001-09-14 Triazole compounds useful as protein kinase inhibitors
AU2001296871A Abandoned AU2001296871A1 (en) 2000-09-15 2001-09-14 Pyrazole compounds useful as protein kinase inhibitors
AU2001290914A Abandoned AU2001290914A1 (en) 2000-09-15 2001-09-14 Pyrazole compounds useful as protein kinase inhibitors
AU2001291013A Abandoned AU2001291013A1 (en) 2000-09-15 2001-09-14 Pyrazole compounds useful as protein kinase inhibitors
AU2008252044A Abandoned AU2008252044A1 (en) 2000-09-15 2008-12-03 Compounds Useful as Protein Kinase Inhibitors

Country Status (23)

Country Link
US (7) US7098330B2 (enrdf_load_stackoverflow)
EP (8) EP1318814B1 (enrdf_load_stackoverflow)
JP (9) JP4105949B2 (enrdf_load_stackoverflow)
KR (4) KR20030032035A (enrdf_load_stackoverflow)
CN (3) CN1469875A (enrdf_load_stackoverflow)
AP (1) AP2003002762A0 (enrdf_load_stackoverflow)
AT (8) ATE346064T1 (enrdf_load_stackoverflow)
AU (9) AU2001292670A1 (enrdf_load_stackoverflow)
BR (1) BR0114088A (enrdf_load_stackoverflow)
CA (8) CA2422377C (enrdf_load_stackoverflow)
DE (8) DE60128709T2 (enrdf_load_stackoverflow)
DK (1) DK1318997T3 (enrdf_load_stackoverflow)
ES (3) ES2242771T5 (enrdf_load_stackoverflow)
HU (4) HUP0302172A2 (enrdf_load_stackoverflow)
IL (6) IL154817A0 (enrdf_load_stackoverflow)
MX (8) MXPA03002291A (enrdf_load_stackoverflow)
NO (4) NO20031190L (enrdf_load_stackoverflow)
NZ (4) NZ525014A (enrdf_load_stackoverflow)
PE (1) PE20020451A1 (enrdf_load_stackoverflow)
PL (1) PL361676A1 (enrdf_load_stackoverflow)
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