SK283763B6 - Deriváty chinazolínu a etylestery 4,5-bis(2-metoxyetoxy)- benzoovej kyseliny ako medziprodukty na ich prípravu - Google Patents

Deriváty chinazolínu a etylestery 4,5-bis(2-metoxyetoxy)- benzoovej kyseliny ako medziprodukty na ich prípravu Download PDF

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Publication number
SK283763B6
SK283763B6 SK56-2003A SK562003A SK283763B6 SK 283763 B6 SK283763 B6 SK 283763B6 SK 562003 A SK562003 A SK 562003A SK 283763 B6 SK283763 B6 SK 283763B6
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SK
Slovakia
Prior art keywords
bis
methoxyethoxy
group
carbon atoms
alkyl
Prior art date
Application number
SK56-2003A
Other languages
English (en)
Slovak (sk)
Inventor
Caughren Schnur Rodney
Daniel Arnold Lee
Original Assignee
Pfizer Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23636708&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SK283763(B6) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Inc. filed Critical Pfizer Inc.
Publication of SK283763B6 publication Critical patent/SK283763B6/sk

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94Nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
SK56-2003A 1995-03-30 1996-03-25 Deriváty chinazolínu a etylestery 4,5-bis(2-metoxyetoxy)- benzoovej kyseliny ako medziprodukty na ich prípravu SK283763B6 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US41330095A 1995-03-30 1995-03-30
PCT/IB1995/000436 WO1996030347A1 (en) 1995-03-30 1995-06-06 Quinazoline derivatives

Publications (1)

Publication Number Publication Date
SK283763B6 true SK283763B6 (sk) 2004-01-08

Family

ID=23636708

Family Applications (2)

Application Number Title Priority Date Filing Date
SK56-2003A SK283763B6 (sk) 1995-03-30 1996-03-25 Deriváty chinazolínu a etylestery 4,5-bis(2-metoxyetoxy)- benzoovej kyseliny ako medziprodukty na ich prípravu
SK387-96A SK283762B6 (sk) 1995-03-30 1996-03-25 4-(Substituovaný fenylamino)chinazolínové deriváty, spôsob a medziprodukty na ich výrobu, ich použitie a farmaceutické prostriedky na ich báze

Family Applications After (1)

Application Number Title Priority Date Filing Date
SK387-96A SK283762B6 (sk) 1995-03-30 1996-03-25 4-(Substituovaný fenylamino)chinazolínové deriváty, spôsob a medziprodukty na ich výrobu, ich použitie a farmaceutické prostriedky na ich báze

Country Status (44)

Country Link
EP (5) EP2163546B1 (xx)
JP (1) JP3088018B2 (xx)
KR (1) KR100232335B1 (xx)
CN (1) CN1066142C (xx)
AP (1) AP735A (xx)
AR (1) AR002723A1 (xx)
AT (2) ATE205483T1 (xx)
AU (2) AU703638B2 (xx)
BR (1) BR9601200B1 (xx)
CA (1) CA2216796C (xx)
CO (1) CO4410333A1 (xx)
CZ (2) CZ295145B6 (xx)
DE (3) DE69536015D1 (xx)
DK (1) DK0817775T3 (xx)
EG (1) EG24229A (xx)
ES (2) ES2161290T3 (xx)
FI (1) FI120646B (xx)
FR (1) FR06C0010I2 (xx)
GR (1) GR3037070T3 (xx)
HK (1) HK1038740A1 (xx)
HR (1) HRP960147B1 (xx)
HU (2) HU229120B1 (xx)
IL (7) IL189037A (xx)
LU (1) LU91209I2 (xx)
MA (1) MA23831A1 (xx)
MX (1) MX9707453A (xx)
MY (1) MY117896A (xx)
NL (1) NL300214I2 (xx)
NO (2) NO308740B1 (xx)
NZ (1) NZ286263A (xx)
OA (1) OA10277A (xx)
PE (1) PE43897A1 (xx)
PL (1) PL186843B1 (xx)
PT (1) PT817775E (xx)
RU (2) RU2694252C3 (xx)
SA (1) SA96160707B1 (xx)
SG (1) SG43262A1 (xx)
SI (1) SI9600102A (xx)
SK (2) SK283763B6 (xx)
TR (1) TR199600265A1 (xx)
TW (1) TW454000B (xx)
UA (1) UA44254C2 (xx)
WO (1) WO1996030347A1 (xx)
ZA (1) ZA962522B (xx)

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