KR102179751B1 - 이중 glp1/글루카곤 작용제로서의 엑센딘-4 유도체 - Google Patents

이중 glp1/글루카곤 작용제로서의 엑센딘-4 유도체 Download PDF

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KR102179751B1
KR102179751B1 KR1020157010088A KR20157010088A KR102179751B1 KR 102179751 B1 KR102179751 B1 KR 102179751B1 KR 1020157010088 A KR1020157010088 A KR 1020157010088A KR 20157010088 A KR20157010088 A KR 20157010088A KR 102179751 B1 KR102179751 B1 KR 102179751B1
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carboxy
butyryl
ethoxy
amino acid
acid residue
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토르스텐 하아크
미하엘 바그너
베른트 헨켈
지그프리트 스텐겔린
안드레아스 에페르스
마르틴 보싸르트
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    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/605—Glucagons
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
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  • Proteomics, Peptides & Aminoacids (AREA)
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  • Diabetes (AREA)
  • Epidemiology (AREA)
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  • Urology & Nephrology (AREA)
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KR1020157010088A 2012-10-09 2013-10-08 이중 glp1/글루카곤 작용제로서의 엑센딘-4 유도체 Active KR102179751B1 (ko)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
EP12306232 2012-10-09
EP12306232.5 2012-10-09
EP13305222.5 2013-02-27
EP13305222 2013-02-27
PCT/EP2013/070882 WO2014056872A1 (en) 2012-10-09 2013-10-08 Exendin-4 derivatives as dual glp1/glucagon agonists

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Publication Number Publication Date
KR20150064093A KR20150064093A (ko) 2015-06-10
KR102179751B1 true KR102179751B1 (ko) 2020-11-17

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US (3) US9365632B2 (https=)
EP (1) EP2906595B1 (https=)
JP (1) JP6373270B2 (https=)
KR (1) KR102179751B1 (https=)
CN (1) CN104837864B (https=)
AR (1) AR092925A1 (https=)
AU (1) AU2013328802B2 (https=)
BR (1) BR112015007685A2 (https=)
CA (1) CA2887272C (https=)
CL (2) CL2015000811A1 (https=)
CR (1) CR20150200A (https=)
CY (1) CY1119987T1 (https=)
DK (1) DK2906595T3 (https=)
DO (1) DOP2015000073A (https=)
EA (1) EA030023B1 (https=)
ES (1) ES2647418T3 (https=)
GT (1) GT201500081A (https=)
HR (1) HRP20171726T1 (https=)
HU (1) HUE037150T2 (https=)
IL (1) IL237641B (https=)
LT (1) LT2906595T (https=)
MX (1) MX359533B (https=)
MY (1) MY168749A (https=)
NO (1) NO2906595T3 (https=)
NZ (1) NZ706898A (https=)
PE (1) PE20150900A1 (https=)
PH (1) PH12015500688A1 (https=)
PL (1) PL2906595T3 (https=)
PT (1) PT2906595T (https=)
RS (1) RS56515B1 (https=)
SG (1) SG11201501770WA (https=)
SI (1) SI2906595T1 (https=)
TN (1) TN2015000101A1 (https=)
TW (1) TWI613213B (https=)
UA (1) UA116217C2 (https=)
UY (1) UY35072A (https=)
WO (1) WO2014056872A1 (https=)
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