BR0314996A - Composição, composição farmaceuticamente aceitável, método para produzir a composição, métodos para estabilizar a exendina-4 (1-39) ou uma sua variante, derivado ou análogo contra a degradação, antes, durante ou após o uso pretendido, para tratar doenças, para tratar de estados de doenças associados com nìveis elevados de glicose do sangue, para a regulação dos nìveis de glicose do sangue, para a regulação do esvaziamento gástrico, para estimular a liberação de insulina em um mamìfero para reduzir o nìvel de glicose do sangue em um mamìfero, para reduzir o nìvel de lipìdeos plasmáticos em um mamìfero, para reduzir a mortalidade e a morbidez após o infarto miocárdico em um mamìfero, para estimular a liberação de insulina em um mamìfero, e para produzir uma exendina (1-39) estabilizada, e, exendina (1-39) estabilizada - Google Patents
Composição, composição farmaceuticamente aceitável, método para produzir a composição, métodos para estabilizar a exendina-4 (1-39) ou uma sua variante, derivado ou análogo contra a degradação, antes, durante ou após o uso pretendido, para tratar doenças, para tratar de estados de doenças associados com nìveis elevados de glicose do sangue, para a regulação dos nìveis de glicose do sangue, para a regulação do esvaziamento gástrico, para estimular a liberação de insulina em um mamìfero para reduzir o nìvel de glicose do sangue em um mamìfero, para reduzir o nìvel de lipìdeos plasmáticos em um mamìfero, para reduzir a mortalidade e a morbidez após o infarto miocárdico em um mamìfero, para estimular a liberação de insulina em um mamìfero, e para produzir uma exendina (1-39) estabilizada, e, exendina (1-39) estabilizadaInfo
- Publication number
- BR0314996A BR0314996A BR0314996-0A BR0314996A BR0314996A BR 0314996 A BR0314996 A BR 0314996A BR 0314996 A BR0314996 A BR 0314996A BR 0314996 A BR0314996 A BR 0314996A
- Authority
- BR
- Brazil
- Prior art keywords
- mammal
- exendin
- blood glucose
- composition
- reduce
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/46—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/57563—Vasoactive intestinal peptide [VIP]; Related peptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/46—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
- C07K14/47—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Abstract
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US41562602P | 2002-10-02 | 2002-10-02 | |
PCT/DK2003/000651 WO2004035623A2 (en) | 2002-10-02 | 2003-10-02 | Stabilized exendin-4 compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
BR0314996A true BR0314996A (pt) | 2005-08-09 |
Family
ID=32107880
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0314996-0A BR0314996A (pt) | 2002-10-02 | 2003-10-02 | Composição, composição farmaceuticamente aceitável, método para produzir a composição, métodos para estabilizar a exendina-4 (1-39) ou uma sua variante, derivado ou análogo contra a degradação, antes, durante ou após o uso pretendido, para tratar doenças, para tratar de estados de doenças associados com nìveis elevados de glicose do sangue, para a regulação dos nìveis de glicose do sangue, para a regulação do esvaziamento gástrico, para estimular a liberação de insulina em um mamìfero para reduzir o nìvel de glicose do sangue em um mamìfero, para reduzir o nìvel de lipìdeos plasmáticos em um mamìfero, para reduzir a mortalidade e a morbidez após o infarto miocárdico em um mamìfero, para estimular a liberação de insulina em um mamìfero, e para produzir uma exendina (1-39) estabilizada, e, exendina (1-39) estabilizada |
Country Status (13)
Country | Link |
---|---|
US (2) | US7544657B2 (pt) |
EP (1) | EP1546200A2 (pt) |
JP (1) | JP2006517908A (pt) |
KR (1) | KR20050083713A (pt) |
AU (2) | AU2003268621B2 (pt) |
BR (1) | BR0314996A (pt) |
CA (1) | CA2500295A1 (pt) |
MX (1) | MXPA05003335A (pt) |
NO (1) | NO20051585L (pt) |
PL (1) | PL377591A1 (pt) |
RU (1) | RU2376314C2 (pt) |
WO (1) | WO2004035623A2 (pt) |
ZA (1) | ZA200502571B (pt) |
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-
2003
- 2003-10-02 WO PCT/DK2003/000651 patent/WO2004035623A2/en active Application Filing
- 2003-10-02 CA CA002500295A patent/CA2500295A1/en not_active Abandoned
- 2003-10-02 RU RU2005113291/04A patent/RU2376314C2/ru not_active IP Right Cessation
- 2003-10-02 AU AU2003268621A patent/AU2003268621B2/en not_active Ceased
- 2003-10-02 MX MXPA05003335A patent/MXPA05003335A/es active IP Right Grant
- 2003-10-02 JP JP2004543971A patent/JP2006517908A/ja not_active Ceased
- 2003-10-02 US US10/529,858 patent/US7544657B2/en not_active Expired - Fee Related
- 2003-10-02 PL PL377591A patent/PL377591A1/pl not_active Application Discontinuation
- 2003-10-02 BR BR0314996-0A patent/BR0314996A/pt not_active IP Right Cessation
- 2003-10-02 EP EP03747852A patent/EP1546200A2/en not_active Withdrawn
- 2003-10-02 KR KR1020057005716A patent/KR20050083713A/ko not_active Application Discontinuation
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2005
- 2005-03-29 NO NO20051585A patent/NO20051585L/no not_active Application Discontinuation
- 2005-03-30 ZA ZA200502571A patent/ZA200502571B/en unknown
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2009
- 2009-04-15 AU AU2009201477A patent/AU2009201477A1/en not_active Abandoned
- 2009-05-04 US US12/435,295 patent/US20090208565A1/en not_active Abandoned
Also Published As
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WO2004035623A3 (en) | 2004-06-03 |
PL377591A1 (pl) | 2006-02-06 |
NO20051585L (no) | 2005-06-20 |
AU2003268621B2 (en) | 2009-01-15 |
AU2003268621A1 (en) | 2004-05-04 |
RU2005113291A (ru) | 2006-01-20 |
US20090208565A1 (en) | 2009-08-20 |
ZA200502571B (en) | 2006-02-22 |
MXPA05003335A (es) | 2005-07-05 |
AU2009201477A1 (en) | 2009-05-07 |
CA2500295A1 (en) | 2004-04-29 |
RU2376314C2 (ru) | 2009-12-20 |
US7544657B2 (en) | 2009-06-09 |
US20060194719A1 (en) | 2006-08-31 |
EP1546200A2 (en) | 2005-06-29 |
JP2006517908A (ja) | 2006-08-03 |
WO2004035623A2 (en) | 2004-04-29 |
KR20050083713A (ko) | 2005-08-26 |
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