JP2013519675A - アリールメトキシイソインドリン誘導体、それを含む組成物、及びその使用方法 - Google Patents

アリールメトキシイソインドリン誘導体、それを含む組成物、及びその使用方法 Download PDF

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JP2013519675A
JP2013519675A JP2012552978A JP2012552978A JP2013519675A JP 2013519675 A JP2013519675 A JP 2013519675A JP 2012552978 A JP2012552978 A JP 2012552978A JP 2012552978 A JP2012552978 A JP 2012552978A JP 2013519675 A JP2013519675 A JP 2013519675A
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JP2013519675A5 (enExample
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マン ホン−ワフ
ダブリュー．ムルレル ゲオルゲ
ルチェルマン アレクアンデル
エム．クハリル エハブ
スヘン−チュ チェン ロゲル
ズハング ウエイホング
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Celgene Corp
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Celgene Corp
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    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4412—Non condensed pyridines; Hydrogenated derivatives thereof having oxo groups directly attached to the heterocyclic ring
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  • Chemical & Material Sciences (AREA)
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  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Oncology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Vascular Medicine (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Epidemiology (AREA)
  • Molecular Biology (AREA)
  • Anesthesiology (AREA)
  • Ophthalmology & Optometry (AREA)
  • AIDS & HIV (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
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JP2012552978A 2010-02-11 2011-02-10 アリールメトキシイソインドリン誘導体、それを含む組成物、及びその使用方法 Withdrawn JP2013519675A (ja)

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US30361810P 2010-02-11 2010-02-11
US61/303,618 2010-02-11
PCT/US2011/024269 WO2011100380A1 (en) 2010-02-11 2011-02-10 Arylmethoxy isoindoline derivatives and compositions comprising and methods of using the same

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JP2016004951A Division JP6215976B2 (ja) 2010-02-11 2016-01-14 アリールメトキシイソインドリン誘導体、それを含む組成物、及びその使用方法

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JP2013519675A true JP2013519675A (ja) 2013-05-30
JP2013519675A5 JP2013519675A5 (enExample) 2014-03-27

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JP2012552978A Withdrawn JP2013519675A (ja) 2010-02-11 2011-02-10 アリールメトキシイソインドリン誘導体、それを含む組成物、及びその使用方法
JP2016004951A Active JP6215976B2 (ja) 2010-02-11 2016-01-14 アリールメトキシイソインドリン誘導体、それを含む組成物、及びその使用方法
JP2016080097A Withdrawn JP2016172746A (ja) 2010-02-11 2016-04-13 アリールメトキシイソインドリン誘導体、それを含む組成物、及びその使用方法
JP2016171451A Active JP6270944B2 (ja) 2010-02-11 2016-09-02 アリールメトキシイソインドリン誘導体、それを含む組成物、及びその使用方法
JP2017125219A Pending JP2017200944A (ja) 2010-02-11 2017-06-27 アリールメトキシイソインドリン誘導体、それを含む組成物、及びその使用方法

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JP2016004951A Active JP6215976B2 (ja) 2010-02-11 2016-01-14 アリールメトキシイソインドリン誘導体、それを含む組成物、及びその使用方法
JP2016080097A Withdrawn JP2016172746A (ja) 2010-02-11 2016-04-13 アリールメトキシイソインドリン誘導体、それを含む組成物、及びその使用方法
JP2016171451A Active JP6270944B2 (ja) 2010-02-11 2016-09-02 アリールメトキシイソインドリン誘導体、それを含む組成物、及びその使用方法
JP2017125219A Pending JP2017200944A (ja) 2010-02-11 2017-06-27 アリールメトキシイソインドリン誘導体、それを含む組成物、及びその使用方法

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Cited By (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2015524478A (ja) * 2012-08-09 2015-08-24 セルジーン コーポレイション ３−（４−（（４−（モルホリノメチル）ベンジル）オキシ）−１−オキソイソインドリン−２−イル）ピペリジン−２，６−ジオンを使用する癌の治療方法
JP2016532657A (ja) * 2013-10-08 2016-10-20 セルジーン コーポレイション （ｓ）−３−（４−（（４−（モルホリノメチル）ベンジル）オキシ）−１−オキソイソインドリン−２−イル）ピペリジン−２，６−ジオンの製剤
JP2017501400A (ja) * 2013-12-06 2017-01-12 セルジーン コーポレイション びまん性大細胞型ｂ細胞リンパ腫、多発性骨髄腫、及び骨髄癌の治療の薬効を決定するための方法
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