JP2013512923A5 - - Google Patents

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JP2013512923A5
JP2013512923A5 JP2012542215A JP2012542215A JP2013512923A5 JP 2013512923 A5 JP2013512923 A5 JP 2013512923A5 JP 2012542215 A JP2012542215 A JP 2012542215A JP 2012542215 A JP2012542215 A JP 2012542215A JP 2013512923 A5 JP2013512923 A5 JP 2013512923A5
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JP5852005B2 (ja
JP2013512923A (ja
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JP2012542215A 2009-12-03 2010-12-03 高コレステロール血症、アテローム性動脈硬化症、冠動脈性心疾患、胆石、肥満症、および他の心血管疾患の処置のために有用なグアニル酸シクラーゼのアゴニスト Active JP5852005B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US12/630,654 US8969514B2 (en) 2007-06-04 2009-12-03 Agonists of guanylate cyclase useful for the treatment of hypercholesterolemia, atherosclerosis, coronary heart disease, gallstone, obesity and other cardiovascular diseases
US12/630,654 2009-12-03
PCT/US2010/058848 WO2011069038A2 (en) 2009-12-03 2010-12-03 Agonists of guanylate cyclase useful for the treatment of hypercholesterolemia, atherosclerosis, coronary heart disease, gallstone, obesity and other cardiovascular diseases

Related Child Applications (1)

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JP2015126368A Division JP5942023B2 (ja) 2009-12-03 2015-06-24 高コレステロール血症、アテローム性動脈硬化症、冠動脈性心疾患、胆石、肥満症、および他の心血管疾患の処置のために有用なグアニル酸シクラーゼのアゴニスト

Publications (3)

Publication Number Publication Date
JP2013512923A JP2013512923A (ja) 2013-04-18
JP2013512923A5 true JP2013512923A5 (OSRAM) 2014-01-30
JP5852005B2 JP5852005B2 (ja) 2016-02-03

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Family Applications (6)

Application Number Title Priority Date Filing Date
JP2012542215A Active JP5852005B2 (ja) 2009-12-03 2010-12-03 高コレステロール血症、アテローム性動脈硬化症、冠動脈性心疾患、胆石、肥満症、および他の心血管疾患の処置のために有用なグアニル酸シクラーゼのアゴニスト
JP2015126368A Active JP5942023B2 (ja) 2009-12-03 2015-06-24 高コレステロール血症、アテローム性動脈硬化症、冠動脈性心疾患、胆石、肥満症、および他の心血管疾患の処置のために有用なグアニル酸シクラーゼのアゴニスト
JP2016102368A Expired - Fee Related JP6106313B2 (ja) 2009-12-03 2016-05-23 高コレステロール血症、アテローム性動脈硬化症、冠動脈性心疾患、胆石、肥満症、および他の心血管疾患の処置のために有用なグアニル酸シクラーゼのアゴニスト
JP2017040593A Active JP6251432B2 (ja) 2009-12-03 2017-03-03 高コレステロール血症、アテローム性動脈硬化症、冠動脈性心疾患、胆石、肥満症、および他の心血管疾患の処置のために有用なグアニル酸シクラーゼのアゴニスト
JP2017226132A Withdrawn JP2018065834A (ja) 2009-12-03 2017-11-24 高コレステロール血症、アテローム性動脈硬化症、冠動脈性心疾患、胆石、肥満症、および他の心血管疾患の処置のために有用なグアニル酸シクラーゼのアゴニスト
JP2019191828A Withdrawn JP2020023551A (ja) 2009-12-03 2019-10-21 高コレステロール血症、アテローム性動脈硬化症、冠動脈性心疾患、胆石、肥満症、および他の心血管疾患の処置のために有用なグアニル酸シクラーゼのアゴニスト

Family Applications After (5)

Application Number Title Priority Date Filing Date
JP2015126368A Active JP5942023B2 (ja) 2009-12-03 2015-06-24 高コレステロール血症、アテローム性動脈硬化症、冠動脈性心疾患、胆石、肥満症、および他の心血管疾患の処置のために有用なグアニル酸シクラーゼのアゴニスト
JP2016102368A Expired - Fee Related JP6106313B2 (ja) 2009-12-03 2016-05-23 高コレステロール血症、アテローム性動脈硬化症、冠動脈性心疾患、胆石、肥満症、および他の心血管疾患の処置のために有用なグアニル酸シクラーゼのアゴニスト
JP2017040593A Active JP6251432B2 (ja) 2009-12-03 2017-03-03 高コレステロール血症、アテローム性動脈硬化症、冠動脈性心疾患、胆石、肥満症、および他の心血管疾患の処置のために有用なグアニル酸シクラーゼのアゴニスト
JP2017226132A Withdrawn JP2018065834A (ja) 2009-12-03 2017-11-24 高コレステロール血症、アテローム性動脈硬化症、冠動脈性心疾患、胆石、肥満症、および他の心血管疾患の処置のために有用なグアニル酸シクラーゼのアゴニスト
JP2019191828A Withdrawn JP2020023551A (ja) 2009-12-03 2019-10-21 高コレステロール血症、アテローム性動脈硬化症、冠動脈性心疾患、胆石、肥満症、および他の心血管疾患の処置のために有用なグアニル酸シクラーゼのアゴニスト

Country Status (11)

Country Link
US (3) US8969514B2 (OSRAM)
EP (3) EP2506865B1 (OSRAM)
JP (6) JP5852005B2 (OSRAM)
CN (2) CN105963676B (OSRAM)
AU (2) AU2010325900B2 (OSRAM)
CA (2) CA3068416A1 (OSRAM)
ES (1) ES2540326T3 (OSRAM)
HK (1) HK1215387A1 (OSRAM)
IL (2) IL220090B (OSRAM)
MX (2) MX2012006263A (OSRAM)
WO (1) WO2011069038A2 (OSRAM)

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WO2012037380A2 (en) 2010-09-15 2012-03-22 Synergy Pharmaceuticals Inc. Formulations of guanylate cyclase c agonists and methods of use
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US9486494B2 (en) 2013-03-15 2016-11-08 Synergy Pharmaceuticals, Inc. Compositions useful for the treatment of gastrointestinal disorders
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US20160184387A1 (en) 2013-08-09 2016-06-30 Dominique Charmot Compounds and methods for inhibiting phosphate transport
US20160220630A1 (en) * 2013-10-10 2016-08-04 Synergy Pharmaceuticals, Inc. Agonists of guanylate cyclase useful for the treatment of opioid induced dysfunctions
CN103694320B (zh) * 2013-12-11 2015-11-11 深圳翰宇药业股份有限公司 一种普利卡那肽的制备方法
SG11201702496XA (en) 2014-11-14 2017-04-27 Gemphire Therapeutics Inc PROCESSES AND INTERMEDIATES FOR PREPARING α,ω-DICARBOXYLIC ACID-TERMINATED DIALKANE ETHERS
JP2018536710A (ja) * 2015-11-06 2018-12-13 ジェンファイア・セラピューティクス・インコーポレイテッドＧｅｍｐｈｉｒｅ Ｔｈｅｒａｐｅｕｔｉｃｓ Ｉｎｃ． 混合型脂質異常症の治療
EP3402804A1 (en) 2016-01-11 2018-11-21 Synergy Pharmaceuticals Inc. Formulations and methods for treating ulcerative colitis
JP2020516622A (ja) 2017-04-18 2020-06-11 ジェムフィアー セラピューティクス インコーポレイテッド ゲムカベン、薬学的に許容されるその塩、その組成物、およびその使用方法
WO2020087031A1 (en) 2018-10-26 2020-04-30 The Research Foundation For The State University Of New York Combination serotonin specific reuptake inhibitor and serotonin 1a receptor partial agonist for reducing l-dopa-induced dyskinesia
EP3972599B1 (en) 2019-05-21 2025-10-22 Ardelyx, Inc. Combination for lowering serum phosphate in a patient
AR119267A1 (es) 2019-06-12 2021-12-09 Novartis Ag Anticuerpos de receptor de péptido natriurético 1 y métodos de uso
CN113481153A (zh) * 2021-07-25 2021-10-08 南通美韦德生命科学有限公司 一种脂肪间充质干细胞的分离培养方法

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