HRP20000092C1 - Polymorphic modifications of 2-(3-cyano-4-isobutyloxyphenyl)-4-methyl-5-thiazole-carboxylic acid and processes for the preparation thereof - Google Patents

Polymorphic modifications of 2-(3-cyano-4-isobutyloxyphenyl)-4-methyl-5-thiazole-carboxylic acid and processes for the preparation thereof

Info

Publication number
HRP20000092C1
HRP20000092C1 HR20000092A HRP20000092A HRP20000092C1 HR P20000092 C1 HRP20000092 C1 HR P20000092C1 HR 20000092 A HR20000092 A HR 20000092A HR P20000092 A HRP20000092 A HR P20000092A HR P20000092 C1 HRP20000092 C1 HR P20000092C1
Authority
HR
Croatia
Prior art keywords
isobutyloxyphenyl
cyano
methyl
thiazole
processes
Prior art date
Application number
HR20000092A
Other languages
English (en)
Croatian (hr)
Inventor
Matsumoto Koichi
Watanabe Kenzo
Hiramatsu Toshiyuki
Kitamura Mitsutaka
Original Assignee
Teijin Pharma Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=15953825&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HRP20000092(C1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Teijin Pharma Limited filed Critical Teijin Pharma Limited
Publication of HRP20000092A2 publication Critical patent/HRP20000092A2/hr
Publication of HRPK20000092B1 publication Critical patent/HRPK20000092B1/xx
Publication of HRP20000092C1 publication Critical patent/HRP20000092C1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
HR20000092A 1998-06-19 2000-02-18 Polymorphic modifications of 2-(3-cyano-4-isobutyloxyphenyl)-4-methyl-5-thiazole-carboxylic acid and processes for the preparation thereof HRP20000092C1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP17307998 1998-06-19
PCT/JP1999/003258 WO1999065885A1 (en) 1998-06-19 1999-06-18 Polymorphic modifications of 2-(3-cyano-4-isobutyloxyphenyl)-4-methyl-5-thiazole-carboxylic acid and processes for the preparation thereof

Publications (3)

Publication Number Publication Date
HRP20000092A2 HRP20000092A2 (en) 2000-08-31
HRPK20000092B1 HRPK20000092B1 (en) 2001-10-31
HRP20000092C1 true HRP20000092C1 (en) 2012-04-30

Family

ID=15953825

Family Applications (2)

Application Number Title Priority Date Filing Date
HR20000092A HRP20000092C1 (en) 1998-06-19 2000-02-18 Polymorphic modifications of 2-(3-cyano-4-isobutyloxyphenyl)-4-methyl-5-thiazole-carboxylic acid and processes for the preparation thereof
HRP20120217AA HRP20120217B1 (hr) 1998-06-19 2012-03-07 Polimorfne modifikacije 2-(3-cijano-4-izobutiloksifenil)-4-metil-5-tiazol-karboksilne kiseline i postupak njihova dobivanja

Family Applications After (1)

Application Number Title Priority Date Filing Date
HRP20120217AA HRP20120217B1 (hr) 1998-06-19 2012-03-07 Polimorfne modifikacije 2-(3-cijano-4-izobutiloksifenil)-4-metil-5-tiazol-karboksilne kiseline i postupak njihova dobivanja

Country Status (39)

Country Link
US (1) US6225474B1 (hu)
EP (4) EP1020454B2 (hu)
JP (1) JP3547707B2 (hu)
KR (1) KR100511183B1 (hu)
CN (3) CN102659712A (hu)
AT (2) ATE522512T2 (hu)
AU (1) AU748026B2 (hu)
BE (1) BE2010C024I2 (hu)
BG (1) BG64734B1 (hu)
BR (1) BR9906539A (hu)
CA (2) CA2301863C (hu)
CY (3) CY1109720T1 (hu)
CZ (1) CZ298170B6 (hu)
DE (2) DE69941672D1 (hu)
DK (3) DK1956015T4 (hu)
ES (3) ES2718467T3 (hu)
FR (1) FR10C0022I2 (hu)
GT (1) GT199900216A (hu)
HK (2) HK1029788A1 (hu)
HR (2) HRP20000092C1 (hu)
HU (2) HU229405B1 (hu)
ID (1) ID25775A (hu)
IL (1) IL134594A (hu)
IN (1) IN191537B (hu)
IS (4) IS9020A (hu)
LT (1) LT1956014T (hu)
LU (1) LU91682I2 (hu)
NO (1) NO321308B1 (hu)
NZ (1) NZ503326A (hu)
PL (1) PL200710B1 (hu)
PT (3) PT1956015E (hu)
RU (1) RU2198169C3 (hu)
SI (3) SI1956014T1 (hu)
SK (2) SK287928B6 (hu)
TR (1) TR200000458T1 (hu)
TW (1) TWI248439B (hu)
UA (1) UA57611C2 (hu)
WO (1) WO1999065885A1 (hu)
ZA (1) ZA200000737B (hu)

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GR1009119B (el) 2016-06-30 2017-09-18 "Φαρματεν Α.Β.Ε.Ε." Φαρμακευτικο σκευασμα περιεχον ενα μη πουρινικο επιλεκτικο αναστολεα της οξειδασης της ξανθινης και μεθοδος παρασκευης αυτου
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CN106565627B (zh) * 2016-10-10 2020-01-10 扬子江药业集团有限公司 一种非布司他药用晶型的制备方法
GR1009659B (el) 2018-09-07 2019-11-28 Φαρματεν Α.Β.Ε.Ε. Φαρμακευτικο σκευασμα που περιλαμβανει ενα συμπλοκο αλατος της φεβουξοστατης με οξειδιο του μαγνησιου και μεθοδος για την παρασκευη αυτου
CN113166017B (zh) * 2018-09-28 2024-03-29 株式会社钟化 稳定性优异的还原型辅酶q10结晶的制造方法
CN112390766B (zh) * 2019-08-13 2022-09-06 浙江天宇药业股份有限公司 一种非布司他a晶型的制备方法
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Publication number Publication date
IS5377A (is) 2000-02-17
NO20000789L (no) 2000-02-17
IS2886B (is) 2014-07-15
ES2336287T5 (es) 2013-04-02
CA2301863C (en) 2009-01-27
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