EA006973B1 - Производные замещенных алкиламинов и их применение - Google Patents

Производные замещенных алкиламинов и их применение Download PDF

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Publication number
EA006973B1
EA006973B1 EA200300788A EA200300788A EA006973B1 EA 006973 B1 EA006973 B1 EA 006973B1 EA 200300788 A EA200300788 A EA 200300788A EA 200300788 A EA200300788 A EA 200300788A EA 006973 B1 EA006973 B1 EA 006973B1
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EA
Eurasian Patent Office
Prior art keywords
amino
ylmethyl
nicotinamide
substituted
alkyl
Prior art date
Application number
EA200300788A
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English (en)
Russian (ru)
Other versions
EA200300788A1 (ru
Inventor
Гуокинг Чен
Джеффри Адамс
Джин Бемис
Шон Букер
Гуолин Каи
Майкл Крогэн
Люсиан Дипьетро
Селиа Домингэз
Дэниел Елбаум
Джули Гермэйн
Стефани Гюнс-Мейер
Майкл Хэндли
Ки Хуанг
Джозеф Л. Ким
Тае-Сеонг КИМ
Александр Киселев
Ксиаоху Оуянг
Винод Ф. Пэтел
Леон М. Смит
Маркиан Стек
Эндрю Тэскер
Нинг Кси
Шимин Ксу
Честер Ченгуанг Юан
Original Assignee
Амген Инк.
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Publication date
Application filed by Амген Инк. filed Critical Амген Инк.
Publication of EA200300788A1 publication Critical patent/EA200300788A1/ru
Publication of EA006973B1 publication Critical patent/EA006973B1/ru

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    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
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