JP2005508905A5 - - Google Patents

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JP2005508905A5
JP2005508905A5 JP2003528544A JP2003528544A JP2005508905A5 JP 2005508905 A5 JP2005508905 A5 JP 2005508905A5 JP 2003528544 A JP2003528544 A JP 2003528544A JP 2003528544 A JP2003528544 A JP 2003528544A JP 2005508905 A5 JP2005508905 A5 JP 2005508905A5
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pharmaceutically acceptable
compound
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formula
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JP2005508905A (ja
JP3795044B2 (ja
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Priority claimed from PCT/US2002/029017 external-priority patent/WO2003024448A2/en
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Claims (6)

  1. 式Ｃｙ３−ＮＨ−ＣＨ２−（ｐ−フェニル）−ＣＯ−ＮＨ−（ｏ−アニリニル）の化合物であって、Ｃｙ３が、Ｃ３〜Ｃ７−複素環で置換されたピリミジルである化合物、又はその薬剤として許容される塩。
  2. Ｃ３〜Ｃ７−複素環が、メトキシピリジン又は置換されていないピリジンである請求項１記載の化合物。
  3. Ｃ３〜Ｃ７−複素環がモルホリノである請求項１記載の化合物。
  4. 式
    Figure 2005508905

    を有する化合物、又はその薬剤として許容される塩。
  5. 式
    Figure 2005508905

    を有する化合物、又はその薬剤として許容される塩。
  6. 薬剤として許容される担体、賦形剤又は希釈剤と一緒に、請求項１〜５のいずれか一項に記載の化合物を少なくとも１つ含む組成物。
JP2003528544A 2001-09-14 2002-09-12 ヒストンデアセチラーゼの阻害剤 Expired - Fee Related JP3795044B2 (ja)

Applications Claiming Priority (3)

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US32240201P 2001-09-14 2001-09-14
US39172802P 2002-06-26 2002-06-26
PCT/US2002/029017 WO2003024448A2 (en) 2001-09-14 2002-09-12 Inhibitors of histone deacetylase

Related Child Applications (1)

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JP2005080310A Division JP2005255683A (ja) 2001-09-14 2005-03-18 ヒストンデアセチラーゼの阻害剤

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JP2005508905A JP2005508905A (ja) 2005-04-07
JP2005508905A5 true JP2005508905A5 (ja) 2005-12-22
JP3795044B2 JP3795044B2 (ja) 2006-07-12

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JP2003528544A Expired - Fee Related JP3795044B2 (ja) 2001-09-14 2002-09-12 ヒストンデアセチラーゼの阻害剤
JP2005080310A Pending JP2005255683A (ja) 2001-09-14 2005-03-18 ヒストンデアセチラーゼの阻害剤
JP2010013418A Abandoned JP2010168382A (ja) 2001-09-14 2010-01-25 ヒストンデアセチラーゼの阻害剤

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JP2005080310A Pending JP2005255683A (ja) 2001-09-14 2005-03-18 ヒストンデアセチラーゼの阻害剤
JP2010013418A Abandoned JP2010168382A (ja) 2001-09-14 2010-01-25 ヒストンデアセチラーゼの阻害剤

Country Status (10)

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US (1) US7595343B2 (ja)
EP (1) EP1429765A2 (ja)
JP (3) JP3795044B2 (ja)
KR (2) KR20100107509A (ja)
CN (2) CN101851173A (ja)
AU (1) AU2002327627B2 (ja)
BR (1) BR0212510A (ja)
CA (1) CA2465978C (ja)
MX (1) MXPA04002397A (ja)
WO (1) WO2003024448A2 (ja)

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