CN1953417B
(zh)
*
|
1996-09-04 |
2010-12-29 |
英特托拉斯技术公司 |
一种从用户站点向外部站点发布使用数据的方法
|
US6184226B1
(en)
*
|
1998-08-28 |
2001-02-06 |
Scios Inc. |
Quinazoline derivatives as inhibitors of P-38 α
|
US6982260B1
(en)
|
1999-11-22 |
2006-01-03 |
Warner-Lambert Company |
Quinazolines and their use for inhibiting cyclin-dependent kinase enzymes
|
SK288019B6
(sk)
|
1999-12-24 |
2012-11-05 |
Aventis Pharma Limited |
Azaindoles derivatives, their use and pharmaceutical composition containing thereof
|
US6660731B2
(en)
*
|
2000-09-15 |
2003-12-09 |
Vertex Pharmaceuticals Incorporated |
Pyrazole compounds useful as protein kinase inhibitors
|
US6638926B2
(en)
*
|
2000-09-15 |
2003-10-28 |
Vertex Pharmaceuticals Incorporated |
Pyrazole compounds useful as protein kinase inhibitors
|
US7473691B2
(en)
*
|
2000-09-15 |
2009-01-06 |
Vertex Pharmaceuticals Incorporated |
Pyrazole compounds useful as protein kinase inhibitors
|
EP1347972A1
(en)
*
|
2000-12-19 |
2003-10-01 |
Smithkline Beecham Plc |
Pyrazolo 3,4-c]pyridines as gsk-3 inhibitors
|
CN100436452C
(zh)
*
|
2000-12-21 |
2008-11-26 |
沃泰克斯药物股份有限公司 |
可用作蛋白激酶抑制剂的吡唑化合物
|
MXPA03005696A
(es)
*
|
2000-12-21 |
2003-10-06 |
Glaxo Group Ltd |
Pirimidinaminas como moduladores de angiogenesis.
|
WO2002079163A1
(en)
*
|
2001-03-30 |
2002-10-10 |
Smithkline Beecham Corporation |
Aminopyridine derivatives as estrogen receptor modulators
|
JP4316893B2
(ja)
|
2001-05-16 |
2009-08-19 |
バーテックス ファーマシューティカルズ インコーポレイテッド |
Srcおよび他のプロテインキナーゼのインヒビター
|
GB0115109D0
(en)
|
2001-06-21 |
2001-08-15 |
Aventis Pharma Ltd |
Chemical compounds
|
US6939874B2
(en)
|
2001-08-22 |
2005-09-06 |
Amgen Inc. |
Substituted pyrimidinyl derivatives and methods of use
|
US7115617B2
(en)
|
2001-08-22 |
2006-10-03 |
Amgen Inc. |
Amino-substituted pyrimidinyl derivatives and methods of use
|
US20030176437A1
(en)
|
2001-08-31 |
2003-09-18 |
D.M. Watterson |
Anti-inflammatory and protein kinase inhibitor compositions and related methods for downregulation of detrimental cellular responses and inhibition of cell death
|
WO2003030909A1
(en)
*
|
2001-09-25 |
2003-04-17 |
Bayer Pharmaceuticals Corporation |
2- and 4-aminopyrimidines n-substtituded by a bicyclic ring for use as kinase inhibitors in the treatment of cancer
|
JP4542338B2
(ja)
|
2001-09-26 |
2010-09-15 |
ファイザー イタリア ソシエタ ア レスポンサビリタ リミタータ |
キナーゼ阻害因子として活性なアミノインダゾール誘導体、それらの製造方法及びそれらを含有する医薬組成物
|
TWI330183B
(US07585860-20090908-C00112.png)
*
|
2001-10-22 |
2010-09-11 |
Eisai R&D Man Co Ltd |
|
SE0104140D0
(sv)
*
|
2001-12-07 |
2001-12-07 |
Astrazeneca Ab |
Novel Compounds
|
EP2198867A1
(en)
|
2001-12-07 |
2010-06-23 |
Vertex Pharmaceuticals, Inc. |
Pyrimidine-based compounds useful as GSK-3 inhibitors
|
US20030187026A1
(en)
|
2001-12-13 |
2003-10-02 |
Qun Li |
Kinase inhibitors
|
AU2002357164A1
(en)
|
2001-12-17 |
2003-06-30 |
Smithkline Beecham Corporation |
Pyrazolopyridazine derivatives
|
US20030158195A1
(en)
|
2001-12-21 |
2003-08-21 |
Cywin Charles L. |
1,6 naphthyridines useful as inhibitors of SYK kinase
|
WO2003055866A1
(en)
*
|
2001-12-21 |
2003-07-10 |
Bayer Pharmaceuticals Corporation |
Quinazoline and quinoline derivative compounds as inhibitors of prolylpeptidase, inducers of apoptosis and cancer treatment agents
|
EP1471910A2
(en)
*
|
2002-01-17 |
2004-11-03 |
Neurogen Corporation |
Substituted quinazolin-4-ylamine analogues as modulators of capsaicin receptors
|
TWI329105B
(en)
|
2002-02-01 |
2010-08-21 |
Rigel Pharmaceuticals Inc |
2,4-pyrimidinediamine compounds and their uses
|
US20040034037A1
(en)
*
|
2002-02-06 |
2004-02-19 |
Harbeson Scott L. |
Heteroaryl compounds useful as inhibitors of GSK-3
|
ATE466580T1
(de)
|
2002-03-15 |
2010-05-15 |
Vertex Pharma |
Azolylaminoazine als proteinkinasehemmer
|
AU2003225800A1
(en)
|
2002-03-15 |
2003-09-29 |
Hayley Binch |
Azolylaminoazine as inhibitors of protein kinases
|
EP1485380B1
(en)
*
|
2002-03-15 |
2010-05-19 |
Vertex Pharmaceuticals Incorporated |
Azolylaminoazines as inhibitors of protein kinases
|
CA2479520A1
(en)
*
|
2002-04-05 |
2003-10-16 |
Birgit Jung |
P38 kinase inhibitors for treating mucus hypersecretion_
|
ES2340475T3
(es)
|
2002-05-01 |
2010-06-04 |
Vertex Pharmaceuticals Incorporated |
Estructura cristalizada de proteina aurora-2 y sus bolsillos de union.
|
ATE493987T1
(de)
*
|
2002-05-22 |
2011-01-15 |
Amgen Inc |
Aminopyrimidin-derivate zur verwendung als vanilloid-rezeptor-liganden zur behandlung von schmerzen
|
AU2003242252A1
(en)
|
2002-06-07 |
2003-12-22 |
Kyowa Hakko Kogyo Co., Ltd. |
Bicyclic pyrimidine derivatives
|
AU2003251721A1
(en)
|
2002-06-14 |
2003-12-31 |
Laboratoires Serono Sa |
Azole methylidene cyanide derivatives and their use as protein kinase modulators
|
MY141867A
(en)
*
|
2002-06-20 |
2010-07-16 |
Vertex Pharma |
Substituted pyrimidines useful as protein kinase inhibitors
|
AU2003249369A1
(en)
|
2002-06-21 |
2004-01-06 |
Cellular Genomics, Inc. |
Certain amino-substituted monocycles as kinase modulators
|
DE60320560T2
(de)
*
|
2002-07-17 |
2008-12-11 |
Pfizer Italia S.R.L. |
Heterobicyclische pyrazolderivate als kinaseinhibitoren
|
CA2494367A1
(en)
*
|
2002-07-25 |
2004-02-05 |
Scios Inc. |
Methods for improvement of lung function using tgf-.beta. inhibitors
|
CN1678321A
(zh)
|
2002-07-29 |
2005-10-05 |
里格尔药品股份有限公司 |
用2,4-嘧啶二胺化合物治疗或者预防自体免疫性疾病的方法
|
SI1532145T1
(sl)
*
|
2002-08-02 |
2007-02-28 |
Vertex Pharma |
Pirazolni sestavki, koristni kot inhibitorji GSK-3
|
CN101037438A
(zh)
*
|
2002-08-02 |
2007-09-19 |
沃泰克斯药物股份有限公司 |
用作gsk-3的抑制剂的吡唑组合物
|
DE60325865D1
(de)
*
|
2002-08-13 |
2009-03-05 |
Merck Sharp & Dohme |
Phenylpyridazin derivative als liganden für gaba-rezeptoren
|
BR0313397A
(pt)
|
2002-08-14 |
2005-06-28 |
Vertex Pharmaceuticals Incorpo |
Inibidores de proteina cinase e usos destes
|
KR101166745B1
(ko)
|
2002-09-05 |
2012-07-23 |
아방티 파르마 소시에테 아노님 |
의약으로서의 신규한 아미노인다졸 유도체 및 이를 함유하는 약제학적 조성물
|
FR2844267B1
(fr)
*
|
2002-09-05 |
2008-02-15 |
Aventis Pharma Sa |
Nouveaux derives d'aminoindazoles a titre de medicaments et compositions pharmaceutiques les renfermant
|
UA80295C2
(en)
|
2002-09-06 |
2007-09-10 |
Biogen Inc |
Pyrazolopyridines and using the same
|
CN1694708A
(zh)
*
|
2002-09-10 |
2005-11-09 |
西奥斯股份有限公司 |
TGFβ的抑制剂
|
CA2506772A1
(en)
|
2002-11-01 |
2004-05-21 |
Vertex Pharmaceuticals Incorporated |
Compositions useful as inhibitors of jak and other protein kinases
|
CA2507406A1
(en)
|
2002-11-05 |
2004-05-21 |
Vertex Pharmaceuticals Incorporated |
Compounds useful as inhibitors of jak and other protein kinases
|
WO2004048365A1
(en)
*
|
2002-11-21 |
2004-06-10 |
Chiron Corporation |
2,4,6-trisubstituted pyrimidines as phosphotidylinositol (pi) 3-kinase inhibitors and their use in the treatment of cancer
|
SI2316831T1
(sl)
*
|
2002-11-21 |
2013-07-31 |
Novartis Ag |
2-(morfolin-4-il)pirimidini kot inhibitorji fosfotidilinozitol (PI) 3-kinaze in njihova uporaba pri zdravljenju raka
|
US7759336B2
(en)
*
|
2002-12-10 |
2010-07-20 |
Ono Pharmaceutical Co., Ltd. |
Nitrogen-containing heterocyclic compounds and medicinal use thereof
|
FR2848554A1
(fr)
*
|
2002-12-12 |
2004-06-18 |
Aventis Pharma Sa |
Nouveaux derives d'aminoindazoles a titre de medicaments et compositions pharmaceutiques les renfermant
|
PL376789A1
(pl)
|
2002-12-12 |
2006-01-09 |
Aventis Pharma S.A. |
Pochodne aminoindazoli i ich zastosowanie jako inhibitorów kinazy
|
BR0317168A
(pt)
|
2002-12-13 |
2005-11-01 |
Neurogen Corp |
Composto ou uma forma farmaceuticamente aceitável do mesmo, composição farmacêutica, métodos de reduzir condutância de cálcio de um receptor de capsaicina celular, e de inibir ligação de ligante vanilóide a um receptor de capsaicina, métodos de tratar uma condição responsiva à modulação de receptor de capsaicina, dor, coceira, tosse ou soluços, incontinência urinária, de promover perda de peso em paciente, e de determinar a presença ou ausência de receptor de capsaicina em uma amostra, preparação farmacêutica embalada, e, uso de um composto
|
WO2004072029A2
(en)
*
|
2003-02-06 |
2004-08-26 |
Vertex Pharmaceuticals Incorporated |
Pyrazolopyridazines useful as inhibitors of protein kinases
|
US7157455B2
(en)
*
|
2003-02-10 |
2007-01-02 |
Hoffmann-La Roche Inc. |
4-Aminopyrimidine-5-one derivatives
|
JP2006521398A
(ja)
*
|
2003-03-28 |
2006-09-21 |
サイオス・インコーポレーテツド |
TGFβの二−環式ピリミジン阻害剤
|
AU2004230928B2
(en)
*
|
2003-04-09 |
2010-12-02 |
Exelixis, Inc. |
Tie-2 modulators and methods of use
|
WO2004096130A2
(en)
*
|
2003-04-24 |
2004-11-11 |
Merck & Co., Inc. |
Inhibitors of akt activity
|
WO2004096808A1
(en)
*
|
2003-04-28 |
2004-11-11 |
De Novo Pharmaceuticals Limited |
Triazine compounds and their use
|
CA2528834A1
(en)
*
|
2003-06-13 |
2005-02-10 |
Arena Pharmaceuticals, Inc. |
5-substituted 2h-pyrazole-3-carboxylic acid derivatives as agonists for the nicotinic acid receptor rup25 for the treatment of dyslipidemia and related diseases
|
MXPA05013922A
(es)
*
|
2003-06-20 |
2006-02-24 |
Coley Pharm Group Inc |
Antagonistas de receptor tipo toll de molecula pequena.
|
TW200510373A
(en)
|
2003-07-14 |
2005-03-16 |
Neurogen Corp |
Substituted quinolin-4-ylamine analogues
|
US7329664B2
(en)
|
2003-07-16 |
2008-02-12 |
Neurogen Corporation |
Substituted (7-pyridyl-4-phenylamino-quinazolin-2-yl)-methanol analogues
|
PL2256106T3
(pl)
|
2003-07-22 |
2015-08-31 |
Astex Therapeutics Ltd |
Związki 3,4-pochodne 1h-pirazolu i ich zastosowanie jako kinazy zależne od cyklin (cdk) i modulatory kinazy syntazy glikogenu-3 (gsk-3)
|
US7122542B2
(en)
|
2003-07-30 |
2006-10-17 |
Rigel Pharmaceuticals, Inc. |
Methods of treating or preventing autoimmune diseases with 2,4-pyrimidinediamine compounds
|
EP1663994B1
(en)
*
|
2003-08-05 |
2012-03-07 |
Vertex Pharmaceuticals Incorporated |
Tetrahydroquinazoline compounds as inhibitors of voltage-gated ion channels
|
JP4889489B2
(ja)
*
|
2003-08-06 |
2012-03-07 |
バーテックス ファーマシューティカルズ インコーポレイテッド |
プロテインキナーゼのインヒビターとして有用なアミノトリアゾール化合物
|
EP1668013B1
(en)
*
|
2003-09-23 |
2012-02-22 |
Vertex Pharmaceuticals Incorporated |
Pyrazolopyrrole derivatives as protein kinase inhibitors
|
GB0323137D0
(en)
|
2003-10-03 |
2003-11-05 |
Chang Lisa C W |
2,4,6- Trisubstituted pyrimidines and their different uses
|
KR20060123164A
(ko)
|
2003-10-17 |
2006-12-01 |
아스트라제네카 아베 |
암 치료에 사용하기 위한 4-(피라졸-3-일아미노)피리미딘유도체
|
WO2005047268A2
(en)
*
|
2003-11-10 |
2005-05-26 |
X-Ceptor Therapeutics, Inc. |
Substituted pyrimidine compositions and methods of use
|
US7338951B2
(en)
|
2003-11-10 |
2008-03-04 |
Synta Pharmaceuticals Corp. |
Pyridine compounds
|
CN102127056B
(zh)
*
|
2003-12-03 |
2013-08-21 |
Ym生物科学澳大利亚私人有限公司 |
微管蛋白抑制剂
|
CN1902193B
(zh)
*
|
2003-12-04 |
2011-07-13 |
沃泰克斯药物股份有限公司 |
可用作蛋白激酶抑制剂的喹喔啉
|
EP1709045A1
(en)
*
|
2003-12-09 |
2006-10-11 |
Vertex Pharmaceuticals Incorporated |
Naphthyridine derivatives and their use as modulators of muscarinic receptors
|
EP1694686A1
(en)
*
|
2003-12-19 |
2006-08-30 |
Takeda San Diego, Inc. |
Kinase inhibitors
|
TW200530235A
(en)
|
2003-12-24 |
2005-09-16 |
Renovis Inc |
Bicycloheteroarylamine compounds as ion channel ligands and uses thereof
|
KR20070026390A
(ko)
|
2004-01-23 |
2007-03-08 |
암젠 인코포레이션 |
화합물 및 사용방법
|
WO2005073224A2
(en)
|
2004-01-23 |
2005-08-11 |
Amgen Inc |
Quinoline quinazoline pyridine and pyrimidine counds and their use in the treatment of inflammation angiogenesis and cancer
|
CA2556239A1
(en)
|
2004-02-11 |
2005-08-25 |
Amgen Inc. |
Vanilloid receptor ligands and their use in treatments
|
EP1742936A2
(en)
|
2004-04-13 |
2007-01-17 |
Icagen, Inc. |
Polycyclic pyridines as potassium ion channel modulators
|
EP1763524A1
(en)
*
|
2004-04-23 |
2007-03-21 |
Takeda San Diego, Inc. |
Indole derivatives and use thereof as kinase inhibitors
|
US7793137B2
(en)
|
2004-10-07 |
2010-09-07 |
Cisco Technology, Inc. |
Redundant power and data in a wired data telecommunincations network
|
PT1905773E
(pt)
|
2004-05-14 |
2012-10-25 |
Millennium Pharm Inc |
Compostos e métodos para inibir a progressão mitótica por inibição da quinase aurora
|
EP1604988A1
(en)
*
|
2004-05-18 |
2005-12-14 |
Sanofi-Aventis Deutschland GmbH |
Pyridazinone derivatives, methods for producing them and their use as pharmaceuticals
|
EP1598348A1
(en)
*
|
2004-05-18 |
2005-11-23 |
Aventis Pharma Deutschland GmbH |
Novel pyridazinone derivatives as inhibitors of CDK2
|
DE102004028862A1
(de)
*
|
2004-06-15 |
2005-12-29 |
Merck Patent Gmbh |
3-Aminoindazole
|
GB0415364D0
(en)
*
|
2004-07-09 |
2004-08-11 |
Astrazeneca Ab |
Pyrimidine derivatives
|
US20080261821A1
(en)
*
|
2004-07-21 |
2008-10-23 |
The Regents Of Te University Of California |
Mechanism-Based Crosslinkers
|
JP2008510734A
(ja)
*
|
2004-08-18 |
2008-04-10 |
タケダ サン ディエゴ インコーポレイテッド |
キナーゼ阻害剤
|
WO2006018256A2
(en)
|
2004-08-19 |
2006-02-23 |
Dsm Ip Assets B.V. |
Process for the rectification of mixtures of high-boiling air-and/or temperature-sensitive useful products
|
GB0419416D0
(en)
|
2004-09-01 |
2004-10-06 |
Inst Of Ex Botany Ascr |
4-Arylazo-3,5-Diamino-Pyrazole compounds and use thereof
|
US7335672B2
(en)
|
2004-09-13 |
2008-02-26 |
Amgen Inc. |
Vanilloid receptor ligands and their use in treatments
|
CA2581454A1
(en)
*
|
2004-09-23 |
2006-03-30 |
Reddy Us Therapeutics, Inc. |
Novel pyrimidine compounds, process for their preparation and compositions containing them
|
AR050948A1
(es)
|
2004-09-24 |
2006-12-06 |
Hoffmann La Roche |
Derivados de ftalazinona; su obtencion y su utilizacion en la fabricacion de medicamentos para el tratamiento del cancer.
|
US7285569B2
(en)
|
2004-09-24 |
2007-10-23 |
Hoff Hoffmann-La Roche Inc. |
Tricycles, their manufacture and use as pharmaceutical agents
|
TW200626157A
(en)
|
2004-09-30 |
2006-08-01 |
Tibotec Pharm Ltd |
HCV inhibiting bi-cyclic pyrimidines
|
TW200621251A
(en)
|
2004-10-12 |
2006-07-01 |
Neurogen Corp |
Substituted biaryl quinolin-4-ylamine analogues
|
US7713973B2
(en)
|
2004-10-15 |
2010-05-11 |
Takeda Pharmaceutical Company Limited |
Kinase inhibitors
|
TW200621257A
(en)
*
|
2004-10-20 |
2006-07-01 |
Astellas Pharma Inc |
Pyrimidine derivative fused with nonaromatic ring
|
WO2006050389A2
(en)
|
2004-11-02 |
2006-05-11 |
Northwestern University |
Pyridazine compounds, compositions and methods
|
CA2589102C
(en)
|
2004-11-02 |
2013-08-13 |
Northwestern University |
Pyridazine compounds and methods for using the compounds to treat inflammatory diseases
|
JP2008520713A
(ja)
|
2004-11-17 |
2008-06-19 |
ミイカナ セラピューティクス インコーポレイテッド |
キナーゼ阻害剤
|
DK1814878T3
(da)
|
2004-11-24 |
2012-05-07 |
Rigel Pharmaceuticals Inc |
Spiro-2, 4-pyrimidindiamin-forbindelser og anvendelser deraf
|
US7652009B2
(en)
|
2004-11-30 |
2010-01-26 |
Amgem Inc. |
Substituted heterocycles and methods of use
|
US20060128710A1
(en)
*
|
2004-12-09 |
2006-06-15 |
Chih-Hung Lee |
Antagonists to the vanilloid receptor subtype 1 (VR1) and uses thereof
|
CA2588220A1
(en)
*
|
2004-12-23 |
2006-06-29 |
Pfizer Products Inc. |
Heteroaromatic derivatives useful as anticancer agents
|
JP5208516B2
(ja)
*
|
2004-12-30 |
2013-06-12 |
エグゼリクシス, インコーポレイテッド |
キナーゼモジュレーターとしてのピリミジン誘導体および使用方法
|
DK1856135T3
(da)
|
2005-01-19 |
2010-04-12 |
Rigel Pharmaceuticals Inc |
Prodrugs af 2,4-pyrimidindiamin-forbindelser og deres anvendelser
|
US8404718B2
(en)
|
2005-01-21 |
2013-03-26 |
Astex Therapeutics Limited |
Combinations of pyrazole kinase inhibitors
|
AR054425A1
(es)
|
2005-01-21 |
2007-06-27 |
Astex Therapeutics Ltd |
Sales de adicion de piperidin 4-il- amida de acido 4-(2,6-dicloro-benzoilamino) 1h-pirazol-3-carboxilico.
|
JP4804480B2
(ja)
*
|
2005-01-26 |
2011-11-02 |
シェーリング コーポレイション |
癌の処置のためのプロテインキナーゼインヒビターとしての、3−(インダゾール−5−イル)−(1,2,4)トリアジン誘導体、および関連する化合物
|
SI2383268T1
(sl)
|
2005-02-04 |
2016-02-29 |
Astrazeneca Ab |
Derivati pirazolilaminopiridina uporabni kot kinazni inhibitorji
|
US20060178388A1
(en)
|
2005-02-04 |
2006-08-10 |
Wrobleski Stephen T |
Phenyl-substituted pyrimidine compounds useful as kinase inhibitors
|
PT1853588E
(pt)
|
2005-02-16 |
2008-08-25 |
Astrazeneca Ab |
Compostos químicos
|
US20080161278A1
(en)
*
|
2005-03-23 |
2008-07-03 |
Astrazeneca Ab |
2-Azetidinyl-4-(1H-Pyrazol-3-Ylamino) Pyrimidines as Inhibitors of Insulin-Like Growth Factor-1 Receptor Activity
|
US7402596B2
(en)
|
2005-03-24 |
2008-07-22 |
Renovis, Inc. |
Bicycloheteroaryl compounds as P2X7 modulators and uses thereof
|
ATE517897T1
(de)
|
2005-03-25 |
2011-08-15 |
Tibotec Pharm Ltd |
Heterobicyclische inhibitoren von hvc
|
DK1869032T3
(da)
*
|
2005-04-05 |
2008-11-10 |
Astrazeneca Ab |
Pyrimidindervater til anvendelse som anticancermidler
|
GB0507347D0
(en)
*
|
2005-04-12 |
2005-05-18 |
Astrazeneca Ab |
Chemical compounds
|
US7462639B2
(en)
|
2005-04-14 |
2008-12-09 |
Hoffmann-La Roche Inc. |
Aminopyrazole derivatives
|
JO2787B1
(en)
|
2005-04-27 |
2014-03-15 |
امجين إنك, |
Alternative amide derivatives and methods of use
|
WO2006118231A1
(ja)
|
2005-04-28 |
2006-11-09 |
Mitsubishi Tanabe Pharma Corporation |
シアノピリジン誘導体及びその医薬としての用途
|
EP1885454A2
(en)
|
2005-05-04 |
2008-02-13 |
DeveloGen Aktiengesellschaft |
Use of gsk-3 inhibitors for preventing and treating pancreatic autoimmune disorders
|
ES2552804T3
(es)
*
|
2005-05-04 |
2015-12-02 |
Evotec Ag |
Compuestos heterocíclicos condensados, y sus composiciones y usos
|
US20080194606A1
(en)
*
|
2005-05-05 |
2008-08-14 |
Astrazeneca |
Pyrazolyl-Amino-Substituted Pyrimidines and Their Use in the Treatment of Cancer
|
AR056347A1
(es)
|
2005-05-12 |
2007-10-03 |
Tibotec Pharm Ltd |
Uso de compuestos de pteridina para fabricar medicamentos y composiciones farmaceuticas
|
CA2608009A1
(en)
|
2005-05-16 |
2006-11-23 |
Astrazeneca Ab |
Pyrazolylaminopyrimidine derivatives useful as tyrosine kinase inhibitors
|
CA2612788A1
(en)
|
2005-06-24 |
2006-12-28 |
Steven Cesar Alfons De Jonghe |
Pyrido(3,2-d)pyrimidines and pharmaceutical compositions useful for treating hepatitis c
|
ES2270715B1
(es)
|
2005-07-29 |
2008-04-01 |
Laboratorios Almirall S.A. |
Nuevos derivados de pirazina.
|
CA2619517A1
(en)
*
|
2005-08-18 |
2007-02-22 |
Michael Mortimore |
Pyrazine kinase inhibitors
|
WO2007023382A2
(en)
*
|
2005-08-25 |
2007-03-01 |
Pfizer Inc. |
Pyrimidine amino pyrazole compounds, potent kinase inhibitors
|
EP2258359A3
(en)
|
2005-08-26 |
2011-04-06 |
Braincells, Inc. |
Neurogenesis by muscarinic receptor modulation with sabcomelin
|
EP2275095A3
(en)
|
2005-08-26 |
2011-08-17 |
Braincells, Inc. |
Neurogenesis by muscarinic receptor modulation
|
EP1934219A1
(en)
|
2005-09-16 |
2008-06-25 |
Ranbaxy Laboratories Limited |
Substituted pyrazolo [3,4-b] pyridines as phosphodiesterase inhibitors
|
KR20140025610A
(ko)
*
|
2005-09-30 |
2014-03-04 |
미카나 테라퓨틱스, 인크. |
치환된 피라졸 화합물
|
CN101316587B
(zh)
*
|
2005-09-30 |
2013-04-03 |
迈卡纳治疗股份有限公司 |
取代的吡唑化合物
|
ES2274712B1
(es)
|
2005-10-06 |
2008-03-01 |
Laboratorios Almirall S.A. |
Nuevos derivados imidazopiridina.
|
US8119655B2
(en)
*
|
2005-10-07 |
2012-02-21 |
Takeda Pharmaceutical Company Limited |
Kinase inhibitors
|
GB0520657D0
(en)
*
|
2005-10-11 |
2005-11-16 |
Ludwig Inst Cancer Res |
Pharmaceutical compounds
|
EP2377530A3
(en)
|
2005-10-21 |
2012-06-20 |
Braincells, Inc. |
Modulation of neurogenesis by PDE inhibition
|
ES2391783T3
(es)
|
2005-10-28 |
2012-11-29 |
Astrazeneca Ab |
Derivados de 4-(3-aminopirazol)pirimidina para su uso como agentes inhibidores de las tirosina cinasas en el tratamiento del cáncer
|
EP2314289A1
(en)
|
2005-10-31 |
2011-04-27 |
Braincells, Inc. |
Gaba receptor mediated modulation of neurogenesis
|
AU2006311830B2
(en)
*
|
2005-11-03 |
2013-03-14 |
Vertex Pharmaceuticals Incorporated |
Aminopyrimidines useful as kinase inhibitors
|
EP2404919B1
(en)
|
2005-11-08 |
2013-08-21 |
Vertex Pharmaceuticals Incorporated |
Heterocyclic compound useful as a modulator of ATP-binding cassette transporters.
|
US7713987B2
(en)
|
2005-12-06 |
2010-05-11 |
Rigel Pharmaceuticals, Inc. |
Pyrimidine-2,4-diamines and their uses
|
US8546404B2
(en)
|
2005-12-13 |
2013-10-01 |
Merck Sharp & Dohme |
Compounds that are ERK inhibitors
|
US7572809B2
(en)
|
2005-12-19 |
2009-08-11 |
Hoffmann-La Roche Inc. |
Isoquinoline aminopyrazole derivatives
|
CA2633584A1
(en)
*
|
2005-12-20 |
2007-07-05 |
Takeda Pharmaceutical Company Limited |
Glucokinase activators
|
WO2007084557A2
(en)
|
2006-01-17 |
2007-07-26 |
Vertex Pharmaceuticals Incorporated |
Azaindoles useful as inhibitors of janus kinases
|
JO2660B1
(en)
|
2006-01-20 |
2012-06-17 |
نوفارتيس ايه جي |
Pi-3 inhibitors and methods of use
|
EP1984331B1
(en)
|
2006-02-16 |
2010-10-20 |
Schering Corporation |
Pyrrolidine derivatives as erk inhibitors
|
US20100216734A1
(en)
*
|
2006-03-08 |
2010-08-26 |
Braincells, Inc. |
Modulation of neurogenesis by nootropic agents
|
AU2007223036A1
(en)
*
|
2006-03-08 |
2007-09-13 |
Braincells, Inc. |
Modulation of neurogenesis by nootropic agents
|
PE20080145A1
(es)
*
|
2006-03-21 |
2008-02-11 |
Janssen Pharmaceutica Nv |
Tetrahidro-pirimidoazepinas como moduladores de trpv1
|
AU2007235237B2
(en)
*
|
2006-04-11 |
2011-08-18 |
Vertex Pharmaceuticals Incorporated |
Thiazoles, imidazoles, and pyrazoles useful as inhibitors of protein kinases
|
CA2650711A1
(en)
|
2006-04-28 |
2007-11-08 |
Northwestern University |
Compositions and treatments using pyridazine compounds and cholinesterase inhibitors
|
WO2007134077A2
(en)
*
|
2006-05-09 |
2007-11-22 |
Braincells, Inc. |
5 ht receptor mediated neurogenesis
|
CA2651813A1
(en)
|
2006-05-09 |
2007-11-22 |
Braincells, Inc. |
Neurogenesis by modulating angiotensin
|
US20100009983A1
(en)
*
|
2006-05-09 |
2010-01-14 |
Braincells, Inc. |
5 ht receptor mediated neurogenesis
|
PT2248812E
(pt)
|
2006-06-27 |
2014-03-12 |
Takeda Pharmaceutical |
Compostos cíclicos fundidos como moduladores do receptor gpr40
|
JP2009541480A
(ja)
*
|
2006-06-30 |
2009-11-26 |
アストラゼネカ アクチボラグ |
癌の治療において有用なピリミジン誘導体
|
WO2008005538A2
(en)
*
|
2006-07-05 |
2008-01-10 |
Exelixis, Inc. |
Methods of using igf1r and abl kinase modulators
|
EP2049500B1
(en)
|
2006-07-06 |
2011-09-07 |
Array Biopharma, Inc. |
Cyclopenta [d] pyrimidines as akt protein kinase inhibitors
|
US8063050B2
(en)
|
2006-07-06 |
2011-11-22 |
Array Biopharma Inc. |
Hydroxylated and methoxylated pyrimidyl cyclopentanes as AKT protein kinase inhibitors
|
UA95641C2
(en)
*
|
2006-07-06 |
2011-08-25 |
Эррей Биофарма Инк. |
Hydroxylated cyclopenta [d] pyrimidines as akt protein kinase inhibitors
|
US8338435B2
(en)
|
2006-07-20 |
2012-12-25 |
Gilead Sciences, Inc. |
Substituted pyrido(3,2-D) pyrimidines and pharmaceutical compositions for treating viral infections
|
AU2007292848A1
(en)
*
|
2006-09-08 |
2008-03-13 |
Braincells, Inc. |
Combinations containing a 4-acylaminopyridine derivative
|
AU2007299920A1
(en)
*
|
2006-09-19 |
2008-03-27 |
Braincells, Inc. |
PPAR Mediated Modulation of Neurogenesis
|
US20100184806A1
(en)
|
2006-09-19 |
2010-07-22 |
Braincells, Inc. |
Modulation of neurogenesis by ppar agents
|
EP2223925A1
(en)
*
|
2006-10-09 |
2010-09-01 |
Takeda Pharmaceutical Company Limited |
Kinase inhibitors
|
US20100120717A1
(en)
|
2006-10-09 |
2010-05-13 |
Brown Jason W |
Kinase inhibitors
|
US8642598B2
(en)
|
2006-10-21 |
2014-02-04 |
Abbvie Inc. |
Heterocyclic compounds and their use as glycogen synthase kinase 3 inhibitors
|
AU2007317435A1
(en)
*
|
2006-11-02 |
2008-05-15 |
Vertex Pharmaceuticals Incorporated |
Aminopyridines and aminopyrimidines useful as inhibitors of protein kinases
|
WO2008077086A1
(en)
*
|
2006-12-19 |
2008-06-26 |
Vertex Pharmaceuticals Incorporated |
Aminopyrimidines useful as inhibitors of protein kinases
|
WO2008077650A1
(en)
|
2006-12-26 |
2008-07-03 |
Gilead Sciences, Inc. |
Pyrido(3,2-d)pyrimidines useful for treating viral infections
|
US8143394B2
(en)
|
2006-12-26 |
2012-03-27 |
Gilead Sciences, Inc. |
Pyrido(3,2-d)pyrimidines useful for treating viral infections
|
TW200840584A
(en)
|
2006-12-26 |
2008-10-16 |
Gilead Sciences Inc |
Pyrido(3,2-d)pyrimidines useful for treating viral infections
|
AU2008213808B2
(en)
|
2007-02-06 |
2011-11-10 |
Novartis Ag |
PI 3-kinase inhibitors and methods of their use
|
EP2121633A2
(en)
*
|
2007-02-12 |
2009-11-25 |
Merck & Co., Inc. |
Piperazine derivatives for treatment of ad and related conditions
|
EP2120573A4
(en)
*
|
2007-02-12 |
2011-05-25 |
Merck Sharp & Dohme |
DERIVATIVES OF PIPERIDINE
|
JPWO2008111441A1
(ja)
|
2007-03-05 |
2010-06-24 |
協和発酵キリン株式会社 |
医薬組成物
|
JP5520057B2
(ja)
*
|
2007-03-09 |
2014-06-11 |
バーテックス ファーマシューティカルズ インコーポレイテッド |
蛋白キナーゼの阻害剤として有用なアミノピリミジン
|
JP5393489B2
(ja)
*
|
2007-03-09 |
2014-01-22 |
バーテックス ファーマシューティカルズ インコーポレイテッド |
蛋白キナーゼの阻害剤として有用なアミノピリミジン
|
NZ579483A
(en)
*
|
2007-03-09 |
2012-07-27 |
Vertex Pharma |
Aminopyridines useful as inhibitors of protein kinases
|
MX2009011059A
(es)
|
2007-04-13 |
2009-11-26 |
Vertex Pharma |
Aminopirimidinas utiles como inhibidores de cinasas.
|
JP2010524911A
(ja)
*
|
2007-04-18 |
2010-07-22 |
アストラゼネカ アクチボラグ |
5−アミノピラゾール−3−イル−3H−イミダゾ[4,5−b]ピリジン誘導体と癌の治療のためのその使用
|
WO2008137621A1
(en)
*
|
2007-05-02 |
2008-11-13 |
Vertex Pharmaceuticals Incorporated |
Aminopyrimidines useful as kinase inhibitors
|
MX2009011811A
(es)
*
|
2007-05-02 |
2010-01-14 |
Vertex Pharma |
Aminopirimidinas utiles como inhibidores de cinasa.
|
CA2685876A1
(en)
|
2007-05-02 |
2008-11-13 |
Vertex Pharmaceuticals Incorporated |
Thiazoles and pyrazoles useful as kinase inhibitors
|
JP2010526048A
(ja)
*
|
2007-05-04 |
2010-07-29 |
アストラゼネカ アクチボラグ |
アミノ−チアゾリル−ピリミジン誘導体、および癌の治療のための該誘導体の使用
|
UA99459C2
(en)
*
|
2007-05-04 |
2012-08-27 |
Астразенека Аб |
9-(pyrazol-3-yl)- 9h-purine-2-amine and 3-(pyraz0l-3-yl)-3h-imidazo[4,5-b]pyridin-5-amine derivatives and their use for the treatment of cancer
|
US8969386B2
(en)
|
2007-05-09 |
2015-03-03 |
Vertex Pharmaceuticals Incorporated |
Modulators of CFTR
|
EP2164842A2
(en)
*
|
2007-05-24 |
2010-03-24 |
Vertex Pharmaceuticals Incorporated |
Thiazoles and pyrazoles useful as kinase inhibitors
|
JP2010529193A
(ja)
*
|
2007-06-11 |
2010-08-26 |
ミイカナ セラピューティクス インコーポレイテッド |
置換ピラゾール化合物
|
US8242150B2
(en)
*
|
2007-06-13 |
2012-08-14 |
Merck Sharp & Dohme Corp. |
Triazole derivatives for treating alzheimer'S disease and related conditions
|
US7956190B2
(en)
|
2007-06-25 |
2011-06-07 |
Hoffmann-La Roche Inc. |
Benzimidazole amido derivatives as kinase inhibitors
|
RU2486181C2
(ru)
|
2007-07-05 |
2013-06-27 |
Эррэй Биофарма Инк. |
Пиримидилциклопентаны как ингибиторы акт-протеинкиназ
|
SI2173723T1
(sl)
*
|
2007-07-05 |
2011-12-30 |
Array Biopharma Inc |
Pirimidil ciklopentani kot inhibitorji AKT-protein-kinaze
|
US9409886B2
(en)
|
2007-07-05 |
2016-08-09 |
Array Biopharma Inc. |
Pyrimidyl cyclopentanes as AKT protein kinase inhibitors
|
US8846683B2
(en)
|
2007-07-05 |
2014-09-30 |
Array Biopharma, Inc. |
Pyrimidyl cyclopentanes as Akt protein kinase inhibitors
|
WO2009015254A1
(en)
|
2007-07-25 |
2009-01-29 |
Bristol-Myers Squibb Company |
Triazine kinase inhibitors
|
CA2694499A1
(en)
*
|
2007-07-31 |
2009-02-05 |
Vertex Pharmaceuticals Incorporated |
Process for preparing 5-fluoro-1h-pyrazolo [3, 4-b] pyridin-3-amine and derivatives thereof
|
TW200906818A
(en)
*
|
2007-07-31 |
2009-02-16 |
Astrazeneca Ab |
Chemical compounds
|
US8404856B2
(en)
|
2007-11-20 |
2013-03-26 |
Merck Sharp & Dohme Corp. |
Non-nucleoside reverse transcriptase inhibitors
|
MX364936B
(es)
*
|
2007-12-07 |
2019-05-15 |
Vertex Pharma |
Procesos para producir acidos cicloalquilcarboxamido-piridin benzoicos.
|
PL2225230T3
(pl)
|
2007-12-07 |
2017-08-31 |
Vertex Pharmaceuticals Incorporated |
Stałe postacie kwasu 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioksol-5-ilo)cyklopropanokarboksyamido)-3-metylopirydyn-2-ylo)benzoesowego
|
JP2011032169A
(ja)
*
|
2007-12-11 |
2011-02-17 |
Genecare Research Institute Co Ltd |
4−アミノピリミジン誘導体および該化合物を含有する医薬組成物
|
EP2224929B1
(en)
|
2007-12-17 |
2016-05-04 |
Janssen Pharmaceutica, N.V. |
Imidazolo-, oxazolo-, and thiazolopyrimidine modulators of trpv1
|
EP2240483B8
(en)
|
2008-01-09 |
2013-04-03 |
Array Biopharma, Inc. |
Pyrimidyl cyclopentanes as akt protein kinase inhibitors
|
US8329709B2
(en)
*
|
2008-01-09 |
2012-12-11 |
Genentech, Inc. |
5H-cyclopenta[D]pyrimidines as AKT protein kinase inhibitors
|
US8716483B2
(en)
|
2008-02-21 |
2014-05-06 |
Merck Sharp & Dohme Corp. |
Compounds that are ERK inhibitors
|
ES2647531T3
(es)
|
2008-02-28 |
2017-12-22 |
Vertex Pharmaceuticals Incorporated |
Derivados de heteroarilo como moduladores de CFTR
|
EP2262498A2
(en)
*
|
2008-03-10 |
2010-12-22 |
Vertex Pharmceuticals Incorporated |
Pyrimidines and pyridines useful as inhibitors of protein kinases
|
CL2009000904A1
(es)
*
|
2008-04-21 |
2010-04-30 |
Shionogi & Co |
Compuestos derivados de ciclohexil sulfonamidas que tienen actividad antagonista en el receptor npy y5, composicion farmaceutica y formulacion farmaceutica que los comprende.
|
US8158656B2
(en)
*
|
2008-05-16 |
2012-04-17 |
Shenzhen Chipscreen Biosciences Ltd. |
2-indolinone derivatives as multi-target protein kinase inhibitors and histone deacetylase inhibitors
|
MX2010012703A
(es)
|
2008-05-21 |
2010-12-21 |
Ariad Pharma Inc |
Derivados fosforosos como inhibidores de cinasa.
|
UY31885A
(es)
*
|
2008-06-11 |
2010-01-29 |
Astrazeneca Ab |
Derivados de las 1, 3, 5-triazina-2, 4-diaminas-6-sustituidas-n-sustituidas y sales farmacéuticamente aceptables de los mismos, composiciones y aplicaciones.
|
PE20110061A1
(es)
|
2008-06-12 |
2011-01-31 |
Janssen Pharmaceutica Nv |
Derivados de diamino-piridina, pirimidina y piridazina como moduladores del receptor h4 de histamina
|
AU2009267161B2
(en)
*
|
2008-07-03 |
2014-11-06 |
Merck Patent Gmbh |
Naphthyridininones as Aurora kinase inhibitors
|
US8536187B2
(en)
|
2008-07-03 |
2013-09-17 |
Gilead Sciences, Inc. |
2,4,6-trisubstituted pyrido(3,2-d)pyrimidines useful for treating viral infections
|
AR073354A1
(es)
*
|
2008-07-31 |
2010-11-03 |
Genentech Inc |
Compuestos de pirimidina, composiciones farmaceuticas y su uso en el tratamiento del cancer.
|
WO2010019392A1
(en)
*
|
2008-08-13 |
2010-02-18 |
Merck Sharp & Dohme Corp. |
Purine derivatives for treatment of alzheimer's disease
|
WO2010027921A1
(en)
*
|
2008-09-03 |
2010-03-11 |
Vertex Pharmaceuticals Incorporated |
Co-crystals and pharmaceutical formulations comprising the same
|
WO2010031056A2
(en)
|
2008-09-15 |
2010-03-18 |
The Regents Of The University Of California |
Methods and compositions for modulating ire1, src, and abl activity
|
RU2011116928A
(ru)
*
|
2008-09-30 |
2012-11-20 |
Астразенека Аб (Se) |
Гетероциклические ингибиторы jак киназы
|
CA2744343A1
(en)
*
|
2008-11-19 |
2010-05-27 |
Renovis, Inc. |
6, 7 -dihydro- 5h- pyrrolo [3, 4-d] pyrimidin-4-yl] -quinolin-3 -ylamine compounds useful as faah modulators and uses thereof
|
KR101048448B1
(ko)
|
2008-11-21 |
2011-07-11 |
한국화학연구원 |
신규 피라졸로[4,3-b]피리딘 유도체 또는 이의 약학적으로허용가능한 염, 이의 제조방법 및 이를 유효성분으로 함유하는 약학적 조성물
|
EP3006031A1
(en)
|
2009-02-05 |
2016-04-13 |
Takeda Pharmaceutical Company Limited |
Pyridazinone compounds
|
US20100216805A1
(en)
|
2009-02-25 |
2010-08-26 |
Braincells, Inc. |
Modulation of neurogenesis using d-cycloserine combinations
|
TWI476192B
(zh)
*
|
2009-02-27 |
2015-03-11 |
Ambit Biosciences Corp |
Jak激酶調節化合物及其使用方法
|
EP2406236A4
(en)
*
|
2009-03-09 |
2013-07-24 |
Surface Logix Inc |
INHIBITORS OF RHO KINASE
|
WO2010111050A1
(en)
*
|
2009-03-23 |
2010-09-30 |
Banyu Pharmaceutical Co., Ltd. |
Novel aminopyridine derivatives having aurora a selective inhibitory action
|
US8263632B2
(en)
*
|
2009-03-24 |
2012-09-11 |
Vertex Pharmaceuticals Incoporated |
Aminopyridine derivatives having Aurora A selective inhibitory action
|
CA2755953A1
(en)
*
|
2009-03-24 |
2010-09-30 |
Vertex Pharmaceuticals Incorporated |
Novel aminopyridine derivatives having aurora a selective inhibitory action
|
US8211901B2
(en)
|
2009-05-22 |
2012-07-03 |
Shenzhen Chipscreen Biosciences Ltd. |
Naphthamide derivatives as multi-target protein kinase inhibitors and histone deacetylase inhibitors
|
CN101906076B
(zh)
|
2009-06-04 |
2013-03-13 |
深圳微芯生物科技有限责任公司 |
作为蛋白激酶抑制剂和组蛋白去乙酰化酶抑制剂的萘酰胺衍生物、其制备方法及应用
|
CN105175409A
(zh)
*
|
2009-06-08 |
2015-12-23 |
南特生物科学公司 |
三嗪衍生物及其治疗应用
|
JP5785940B2
(ja)
*
|
2009-06-09 |
2015-09-30 |
アブラクシス バイオサイエンス, エルエルシー |
トリアジン誘導体類及びそれらの治療応用
|
CA2765050A1
(en)
*
|
2009-06-09 |
2010-12-16 |
California Capital Equity, Llc |
Ureidophenyl substituted triazine derivatives and their therapeutical applications
|
CN102480961A
(zh)
*
|
2009-06-24 |
2012-05-30 |
健泰科生物技术公司 |
与含氧杂环稠合的嘧啶化合物、组合物和使用方法
|
US8637525B2
(en)
|
2009-07-31 |
2014-01-28 |
Bristol-Myers Squibb Company |
Compounds for the reduction of beta-amyloid production
|
TWI468402B
(zh)
*
|
2009-07-31 |
2015-01-11 |
必治妥美雅史谷比公司 |
降低β-類澱粉生成之化合物
|
US20110053916A1
(en)
|
2009-08-14 |
2011-03-03 |
Vertex Pharmaceuticals Incorporated |
Pyrimidine compounds as tuberculosis inhibitors
|
CN102020657A
(zh)
*
|
2009-09-11 |
2011-04-20 |
上海艾力斯医药科技有限公司 |
稠合杂芳基衍生物、制备方法及其应用
|
MX2012005463A
(es)
|
2009-11-12 |
2012-09-12 |
Hoffmann La Roche |
Compuestos de purina n/9 sustituida, composiciones y metodos de uso.
|
JP5572715B2
(ja)
*
|
2009-11-12 |
2014-08-13 |
エフ・ホフマン−ラ・ロシュ・アクチェンゲゼルシャフト |
N−7置換プリン及びピラゾロピリミジン化合物、組成物及び使用方法
|
EP2533639A4
(en)
*
|
2010-02-11 |
2013-08-21 |
Univ Vanderbilt |
COMPOUNDS OF PYRAZOLOPYRIDINE, PYRAZOLOPYRAZINE, PYRAZOLOPYRIMIDINE, PYRAZOLOTHIOPHENE AND PYRAZOLOTHIAZOLE AS ALLOSTERIC POTENTIALIZERS OF METABOTROPIC GLUTAMATE RECEPTOR SUBTYPE 4 (MGLUR4), COMPOUNDS AND METHODS FOR TREATING NEUROLOGICAL DYSFUNCTIONS
|
NZ602838A
(en)
|
2010-04-07 |
2015-06-26 |
Vertex Pharma |
Pharmaceutical compositions of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl) cyclopropanecarboxamido)-3-methylpyridin-2-yl)benzoic acid and administration thereof
|
AU2011254550B2
(en)
|
2010-05-21 |
2013-11-07 |
Noviga Research Ab |
Novel pyrimidine derivatives
|
JP5713367B2
(ja)
|
2010-06-04 |
2015-05-07 |
エフ.ホフマン−ラ ロシュ アーゲーF. Hoffmann−La Roche Aktiengesellschaft |
Lrrk2モジュレーターとしてのアミノピリミジン誘導体
|
US20110319409A1
(en)
*
|
2010-06-23 |
2011-12-29 |
Cox Christopher D |
7-aza-quinazoline pde10 inhibitors
|
CN103298805A
(zh)
|
2010-09-01 |
2013-09-11 |
埃姆比特生物科学公司 |
喹唑啉化合物及其使用方法
|
CA2810954A1
(en)
|
2010-09-27 |
2012-04-05 |
Abbott Gmbh & Co. Kg |
Heterocyclic compounds and their use as glycogen synthase kinase-3 inhibitors
|
WO2012059932A1
(en)
|
2010-11-01 |
2012-05-10 |
Aurigene Discovery Technologies Limited |
2, 4 -diaminopyrimidine derivatives as protein kinase inhibitors
|
WO2012060847A1
(en)
|
2010-11-07 |
2012-05-10 |
Targegen, Inc. |
Compositions and methods for treating myelofibrosis
|
CA3017869C
(en)
|
2010-11-10 |
2021-07-27 |
Genentech, Inc. |
Pyrazole aminopyrimidine derivatives as lrrk2 modulators
|
ES2650744T3
(es)
|
2010-12-14 |
2018-01-22 |
Electrophoretics Limited |
Inhibidores de la caseína quinasa 1 delta (CK1delta)
|
CN103270026A
(zh)
|
2010-12-21 |
2013-08-28 |
诺瓦提斯公司 |
作为vps34抑制剂的联-杂芳基化合物
|
US9090592B2
(en)
|
2010-12-30 |
2015-07-28 |
AbbVie Deutschland GmbH & Co. KG |
Heterocyclic compounds and their use as glycogen synthase kinase-3 inhibitors
|
WO2012101654A2
(en)
*
|
2011-01-25 |
2012-08-02 |
Sphaera Pharma Pvt. Ltd |
Novel triazine compounds
|
JP5886411B2
(ja)
|
2011-03-24 |
2016-03-16 |
ノビガ・リサーチ・エービーNoviga Research AB |
新規のピリミジン誘導体
|
MX2013011333A
(es)
|
2011-04-01 |
2014-04-16 |
Genentech Inc |
Combinaciones de compuestos inhibidores de akt y mek, y metodos de uso.
|
ES2620644T3
(es)
|
2011-04-01 |
2017-06-29 |
Genentech, Inc. |
Combinaciones de compuestos inhibidores de AKT y agentes quimioterapéuticos, y métodos de uso
|
RU2477723C2
(ru)
|
2011-06-16 |
2013-03-20 |
Общество С Ограниченной Ответственностью "Фьюжн Фарма" |
Ингибиторы протеинкиназ (варианты), их применение для лечения онкологических заболеваний и фармацевтическая композиция на их основе
|
CN103930422A
(zh)
|
2011-07-19 |
2014-07-16 |
无限药品股份有限公司 |
杂环化合物及其用途
|
US8846656B2
(en)
|
2011-07-22 |
2014-09-30 |
Novartis Ag |
Tetrahydropyrido-pyridine and tetrahydropyrido-pyrimidine compounds and use thereof as C5a receptor modulators
|
RU2014109897A
(ru)
|
2011-08-25 |
2015-09-27 |
Ф.Хоффманн-Ля Рош Аг |
Ингибиторы серин/треонин киназы рак1
|
IN2014CN02646A
(US07585860-20090908-C00112.png)
|
2011-09-14 |
2015-08-07 |
Samumed Llc |
|
CA2847540C
(en)
|
2011-09-22 |
2016-05-17 |
Pfizer Inc. |
Pyrrolopyrimidine and purine derivatives
|
MX342326B
(es)
|
2011-09-27 |
2016-09-26 |
Novartis Ag |
3-pirimidin-4-il-oxazolidin-2-onas como inhibidoras de idh mutante.
|
US8815877B2
(en)
|
2011-12-22 |
2014-08-26 |
Genentech, Inc. |
Serine/threonine kinase inhibitors
|
UY34632A
(es)
|
2012-02-24 |
2013-05-31 |
Novartis Ag |
Compuestos de oxazolidin- 2- ona y usos de los mismos
|
RU2014141674A
(ru)
*
|
2012-03-16 |
2016-05-10 |
Аксикин Фармасьютикалз, Инк. |
3,5-диаминопиразоловые ингибиторы киназы
|
AU2013237226A1
(en)
*
|
2012-03-19 |
2014-10-09 |
Emory University |
Quinazoline compounds and their use in therapy
|
US20130303519A1
(en)
|
2012-03-20 |
2013-11-14 |
Millennium Pharmaceuticals, Inc. |
Methods of treating cancer using aurora kinase inhibitors
|
PH12017500997A1
(en)
|
2012-04-04 |
2018-02-19 |
Samumed Llc |
Indazole inhibitors of the wnt signal pathway and therapeutic uses thereof
|
RS61664B1
(sr)
|
2012-04-24 |
2021-04-29 |
Vertex Pharma |
Inhibitori dna-pk
|
CN106279202A
(zh)
*
|
2012-05-03 |
2017-01-04 |
霍夫曼-拉罗奇有限公司 |
作为lrrk2调节剂用于治疗帕金森病的吡唑氨基嘧啶衍生物
|
CN106220615A
(zh)
*
|
2012-05-03 |
2016-12-14 |
霍夫曼-拉罗奇有限公司 |
作为lrrk2调节剂的吡唑氨基嘧啶衍生物
|
SG10201610869TA
(en)
|
2012-06-26 |
2017-02-27 |
Del Mar Pharmaceuticals |
Methods for treating tyrosine-kinase-inhibitor-resistant malignancies in patients with genetic polymorphisms or ahi1 dysregulations or mutations employing dianhydrogalactitol, diacetyldianhydrogalacti
|
CA2886495C
(en)
*
|
2012-09-28 |
2023-09-19 |
Ignyta, Inc. |
Azaquinazoline inhibitors of atypical protein kinase c
|
JO3470B1
(ar)
|
2012-10-08 |
2020-07-05 |
Merck Sharp & Dohme |
مشتقات 5- فينوكسي-3h-بيريميدين-4-أون واستخدامها كمثبطات ناسخ عكسي ل hiv
|
ES2644758T3
(es)
|
2012-10-16 |
2017-11-30 |
Tolero Pharmaceuticals, Inc. |
Moduladores de PKM2 y métodos para su uso
|
US9296733B2
(en)
|
2012-11-12 |
2016-03-29 |
Novartis Ag |
Oxazolidin-2-one-pyrimidine derivative and use thereof for the treatment of conditions, diseases and disorders dependent upon PI3 kinases
|
KR20150087850A
(ko)
*
|
2012-11-20 |
2015-07-30 |
제넨테크, 인크. |
Egfr 돌연변이체를 함유하는 t790m의 억제제로서의 아미노피리미딘 화합물
|
KR102275676B1
(ko)
|
2012-11-21 |
2021-07-12 |
피티씨 테라퓨틱스, 인크. |
치환된 리버스 피리미딘 bmi-1 저해제
|
CN103012428A
(zh)
|
2013-01-08 |
2013-04-03 |
中国药科大学 |
4-(五元杂环并嘧啶/吡啶取代)氨基-1H-3-吡唑甲酰胺类CDK/Aurora双重抑制剂及其用途
|
MX370487B
(es)
|
2013-01-08 |
2019-12-16 |
Samumed Llc |
Inhibidores de 3-(benzo-imidazol-2-il)-indazol de la senda de señalización de wnt y usos terapéuticos de los mismos.
|
TWI644899B
(zh)
|
2013-02-04 |
2018-12-21 |
健生藥品公司 |
Flap調節劑
|
EP3495359A1
(en)
*
|
2013-02-04 |
2019-06-12 |
Janssen Pharmaceutica NV |
Flap modulators
|
EP2769722A1
(en)
*
|
2013-02-22 |
2014-08-27 |
Ruprecht-Karls-Universität Heidelberg |
Compounds for use in inhibiting HIV capsid assembly
|
JO3377B1
(ar)
*
|
2013-03-11 |
2019-03-13 |
Takeda Pharmaceuticals Co |
مشتقات بيريدينيل وبيريدينيل مندمج
|
RS58374B1
(sr)
|
2013-03-12 |
2019-03-29 |
Vertex Pharma |
Inhibitori dnk-pk
|
MX355945B
(es)
|
2013-03-14 |
2018-05-07 |
Novartis Ag |
3-pirimidin-4-il-oxazolidin-2-onas como inhibidoras de idh mutante.
|
CN105209042B
(zh)
|
2013-03-22 |
2019-03-08 |
米伦纽姆医药公司 |
催化性mtorc 1/2抑制剂与选择性极光a激酶抑制剂的组合
|
WO2015013581A1
(en)
|
2013-07-26 |
2015-01-29 |
Update Pharma Inc. |
Combinatorial methods to improve the therapeutic benefit of bisantrene
|
KR102232595B1
(ko)
|
2013-08-30 |
2021-03-26 |
피티씨 테라퓨틱스, 인크. |
치환된 피리미딘 bmi-1 저해제
|
WO2015028848A1
(en)
*
|
2013-09-02 |
2015-03-05 |
Piramal Enterprises Limited |
Bicyclic heterocyclic compounds as multi-kinase inhibitors
|
LT3052096T
(lt)
|
2013-10-03 |
2018-04-10 |
Kura Oncology, Inc. |
Erk inhibitoriai ir jų panaudojimo būdai
|
EP3055301B1
(en)
*
|
2013-10-07 |
2019-11-20 |
Kadmon Corporation, LLC |
(2-(5-isoindolin-2-yl)pyrimidin-4-yl)-amine derivatives as rho kinase inhibitors for treating autoimmune diseases
|
EP3057953B1
(en)
|
2013-10-17 |
2018-08-15 |
Vertex Pharmaceuticals Incorporated |
Co-crystals of (s)-n-methyl-8-(1-((2'-methyl-[4,5'-bipyrimidin]-6-yl)amino)propan-2-yl)quinoline-4-carboxamide and deuterated derivatives thereof as dna-pk inhibitors
|
MX2016006118A
(es)
|
2013-11-12 |
2016-07-21 |
Vertex Pharma |
Proceso para preparar composiciones farmaceuticas para el tratamiento de enfermedades mediadas por regulador de la conductancia transmembrana de la fibrosis quistica (cftr).
|
US10584115B2
(en)
|
2013-11-21 |
2020-03-10 |
Ptc Therapeutics, Inc. |
Substituted pyridine and pyrazine BMI-1 inhibitors
|
US9975878B2
(en)
|
2013-11-21 |
2018-05-22 |
Ptc Therapeutics, Inc. |
Substituted triazine BMI-1 inhibitors
|
UA115388C2
(uk)
|
2013-11-21 |
2017-10-25 |
Пфайзер Інк. |
2,6-заміщені пуринові похідні та їх застосування в лікуванні проліферативних захворювань
|
CN104672250B
(zh)
*
|
2013-11-29 |
2017-11-07 |
广东东阳光药业有限公司 |
取代的杂芳基化合物及其组合物和用途
|
ES2813875T3
(es)
|
2014-01-01 |
2021-03-25 |
Medivation Tech Llc |
Compuestos y procedimientos de uso
|
WO2015112739A1
(en)
*
|
2014-01-22 |
2015-07-30 |
The United States Of America, As Represented By The Secretary, Department Of Health And Human Services |
Compounds and method for treating parp1-deficient cancers
|
CN104926795B
(zh)
*
|
2014-03-17 |
2017-11-10 |
广东东阳光药业有限公司 |
取代的杂芳基化合物及其组合物和用途
|
TWI675836B
(zh)
*
|
2014-03-25 |
2019-11-01 |
美商伊格尼塔公司 |
非典型蛋白質激酶c之氮雜喹唑啉抑制劑
|
WO2015155738A2
(en)
|
2014-04-09 |
2015-10-15 |
Christopher Rudd |
Use of gsk-3 inhibitors or activators which modulate pd-1 or t-bet expression to modulate t cell immunity
|
CN105367555B
(zh)
*
|
2014-08-07 |
2019-06-25 |
广东东阳光药业有限公司 |
取代的杂芳基化合物及其组合物和用途
|
WO2016040180A1
(en)
|
2014-09-08 |
2016-03-17 |
Samumed, Llc |
3-(1h-benzo[d]imidazol-2-yl)-1h-pyrazolo[3,4-c]pyridine and therapeutic uses thereof
|
WO2016040181A1
(en)
|
2014-09-08 |
2016-03-17 |
Samumed, Llc |
3-(1h-imidazo[4,5-c]pyridin-2-yl)-1h-pyrazolo[3,4-c]pyridine and therapeutic uses thereof
|
WO2016040190A1
(en)
|
2014-09-08 |
2016-03-17 |
Samumed, Llc |
3-(3h-imidazo[4,5-b]pyridin-2-yl)-1h-pyrazolo[3,4-b]pyridine and therapeutic uses thereof
|
WO2016040185A1
(en)
|
2014-09-08 |
2016-03-17 |
Samumed, Llc |
2-(1h-indazol-3-yl)-3h-imidazo[4,5-b]pyridine and therapeutic uses thereof
|
WO2016040184A1
(en)
|
2014-09-08 |
2016-03-17 |
Samumed, Llc |
3-(3h-imidazo[4,5-b]pyridin-2-yl)-1h-pyrazolo[3,4-c]pyridine and therapeutic uses thereof
|
WO2016040193A1
(en)
|
2014-09-08 |
2016-03-17 |
Samumed, Llc |
3-(1h-imidazo[4,5-c]pyridin-2-yl)-1h-pyrazolo[3,4-b]pyridine and therapeutic uses thereof
|
US10302602B2
(en)
|
2014-11-18 |
2019-05-28 |
Vertex Pharmaceuticals Incorporated |
Process of conducting high throughput testing high performance liquid chromatography
|
TWI704151B
(zh)
*
|
2014-12-22 |
2020-09-11 |
美商美國禮來大藥廠 |
Erk抑制劑
|
ES2700200T3
(es)
*
|
2014-12-22 |
2019-02-14 |
Lilly Co Eli |
Inhibidores de ERK
|
US10227343B2
(en)
|
2015-01-30 |
2019-03-12 |
Vanderbilt University |
Isoquiniline and napthalene-substituted compounds as mGluR4 allosteric potentiators, compositions, and methods of treating neurological dysfunction
|
EP3070084A1
(en)
*
|
2015-03-18 |
2016-09-21 |
Rottapharm Biotech S.r.l. |
New fyn kinase inhibitors
|
AU2016247858B2
(en)
|
2015-04-17 |
2020-10-15 |
Ludwig Institute For Cancer Research Ltd. |
PLK4 inhibitors
|
WO2016197009A1
(en)
|
2015-06-05 |
2016-12-08 |
Vertex Pharmaceuticals Incorporated |
Triazoles for the treatment of demyelinating diseases
|
WO2017023987A1
(en)
|
2015-08-03 |
2017-02-09 |
Samumed, Llc. |
3-(1h-pyrrolo[3,2-c]pyridin-2-yl)-1h-pyrazolo[3,4-b]pyridines and therapeutic uses thereof
|
US10166218B2
(en)
|
2015-08-03 |
2019-01-01 |
Samumed, Llc |
3-(1H-indol-2-yl)-1H-pyrazolo[3,4-C]pyridines and therapeutic uses thereof
|
US10195185B2
(en)
|
2015-08-03 |
2019-02-05 |
Samumed, Llc |
3-(1H-imidazo[4,5-C]pyridin-2-yl)-1H-pyrazolo[4,3-B]pyridines and therapeutic uses thereof
|
US10519169B2
(en)
|
2015-08-03 |
2019-12-31 |
Samumed, Llc |
3-(1H-pyrrolo[2,3-C]pyridin-2-yl)-1 H-pyrazolo[4,3-B]pyridines and therapeutic uses thereof
|
US10604512B2
(en)
|
2015-08-03 |
2020-03-31 |
Samumed, Llc |
3-(1H-indol-2-yl)-1H-indazoles and therapeutic uses thereof
|
US10392383B2
(en)
|
2015-08-03 |
2019-08-27 |
Samumed, Llc |
3-(1H-benzo[d]imidazol-2-yl)-1H-pyrazolo[4,3-b]pyridines and therapeutic uses thereof
|
WO2017024004A1
(en)
|
2015-08-03 |
2017-02-09 |
Samumed, Llc. |
3-(1h-pyrrolo[2,3-b]pyridin-2-yl)-1h-pyrazolo[4,3-b]pyridines and therapeutic uses thereof
|
WO2017023984A1
(en)
|
2015-08-03 |
2017-02-09 |
Samumed, Llc. |
3-(1h-pyrrolo[3,2-c]pyridin-2-yl)-1h-pyrazolo[3,4-c]pyridines and therapeutic uses thereof
|
WO2017024015A1
(en)
*
|
2015-08-03 |
2017-02-09 |
Samumed, Llc. |
3-(3h-imidazo[4,5-b]pyridin-2-yl)-1h-pyrazolo[4,3-b]pyridines and therapeutic uses thereof
|
WO2017024003A1
(en)
|
2015-08-03 |
2017-02-09 |
Samumed, Llc |
3-(1h-pyrrolo[3,2-c]pyridin-2-yl)-1h-pyrazolo[4,3-b]pyridines and therapeutic uses thereof
|
WO2017023996A1
(en)
|
2015-08-03 |
2017-02-09 |
Samumed, Llc. |
3-(1h-pyrrolo[2,3-b]pyridin-2-yl)-1h-pyrazolo[3,4-b]pyridines and therapeutic uses thereof
|
WO2017024021A1
(en)
|
2015-08-03 |
2017-02-09 |
Samumed, Llc |
3-(1h-pyrrolo[2,3-b]pyridin-2-yl)-1h-indazoles and therapeutic uses thereof
|
US10188634B2
(en)
|
2015-08-03 |
2019-01-29 |
Samumed, Llc |
3-(3H-imidazo[4,5-C]pyridin-2-yl)-1 H-pyrazolo[4,3-B]pyridines and therapeutic uses thereof
|
US10383861B2
(en)
|
2015-08-03 |
2019-08-20 |
Sammumed, LLC |
3-(1H-pyrrolo[2,3-C]pyridin-2-yl)-1H-pyrazolo[3,4-C]pyridines and therapeutic uses thereof
|
WO2017023993A1
(en)
|
2015-08-03 |
2017-02-09 |
Samumed, Llc. |
3-(1h-indol-2-yl)-1h-pyrazolo[4,3-b]pyridines and therapeutic uses thereof
|
US10285982B2
(en)
|
2015-08-03 |
2019-05-14 |
Samumed, Llc |
3-(1H-pyrrolo[2,3-B]pyridin-2-yl)-1H-pyrazolo[3,4-C]pyridines and therapeutic uses thereof
|
US10463651B2
(en)
|
2015-08-03 |
2019-11-05 |
Samumed, Llc |
3-(1H-pyrrolo[3,2-C]pyridin-2-YL)-1H-indazoles and therapeutic uses thereof
|
WO2017079759A1
(en)
|
2015-11-06 |
2017-05-11 |
Samumed, Llc |
2-(1h-indazol-3-yl)-3h-imidazo[4,5-c]pyridines and their anti-inflammatory uses thereof
|
GB201604647D0
(en)
*
|
2016-03-18 |
2016-05-04 |
Mission Therapeutics Ltd |
Novel compounds
|
HRP20221446T1
(hr)
|
2016-06-01 |
2023-01-06 |
Biosplice Therapeutics, Inc. |
Postupci za pripremu n-(5-(3-(7-(3-fluorofenil)-3h-imidazo[4,5-c]piridin-2-il)-1h-indazol-5-il)piridin-3-il)-3-metilbutanamida
|
TW201815418A
(zh)
|
2016-09-27 |
2018-05-01 |
Vertex Pharma |
使用dna破壞劑及dna-pk抑制劑之組合治療癌症的方法
|
BR112019008061A2
(pt)
|
2016-10-21 |
2019-09-17 |
Samumed Llc |
métodos de uso de indazol-3-carboxamidas e seu uso como inibidores da via de sinalização de wnt/b-catenina
|
WO2018085171A1
(en)
|
2016-11-01 |
2018-05-11 |
Merck Sharp & Dohme Corp. |
Substituted bicyclic heteroaryl allosteric modulators of nicotinic acetylcholine receptors
|
JP2019533702A
(ja)
|
2016-11-07 |
2019-11-21 |
サミュメッド リミテッド ライアビリティ カンパニー |
単回用量の調整済み注射用製剤
|
IT201700047189A1
(it)
*
|
2017-05-02 |
2018-11-02 |
Fondazione St Italiano Tecnologia |
Composti e composizioni per il trattamento di cancro, disordini della retina e cardiomiopatie
|
AR112027A1
(es)
|
2017-06-15 |
2019-09-11 |
Biocryst Pharm Inc |
Inhibidores de alk 2 quinasa que contienen imidazol
|
CA3063616A1
(en)
|
2017-06-30 |
2019-12-06 |
Beijing Tide Pharmaceutical Co., Ltd. |
Rho-associated protein kinase inhibitor, pharmaceutical composition comprising same, and preparation method and use thereof
|
WO2019000682A1
(zh)
*
|
2017-06-30 |
2019-01-03 |
北京泰德制药股份有限公司 |
Rho相关蛋白激酶抑制剂、包含其的药物组合物及其制备方法和用途
|
JP7039802B2
(ja)
|
2017-06-30 |
2022-03-23 |
ベイジン タイド ファーマシューティカル カンパニー リミテッド |
Rho-関連プロテインキナーゼ阻害剤、rho-関連プロテインキナーゼ阻害剤を含む医薬組成物、当該医薬組成物の調製方法及び使用
|
CN109384774B
(zh)
*
|
2017-08-11 |
2023-02-17 |
中国科学院上海药物研究所 |
一类多取代的吡嗪/三嗪酰胺类化合物及其制备方法和应用
|
CA3074034A1
(en)
|
2017-10-27 |
2019-05-02 |
Theravance Biopharma R&D Ip, Llc |
Pyrimidine compound as jak kinase inhibitor
|
GB201801226D0
(en)
|
2018-01-25 |
2018-03-14 |
Redx Pharma Plc |
Modulators of Rho-associated protein kinase
|
US12030857B2
(en)
*
|
2018-06-25 |
2024-07-09 |
Kadmon Corporation, Llc |
Glucose uptake inhibitors
|
EP3836932A2
(en)
|
2018-08-17 |
2021-06-23 |
PTC Therapeutics, Inc. |
Method for treating pancreatic cancer
|
WO2020045941A1
(ko)
*
|
2018-08-27 |
2020-03-05 |
주식회사 대웅제약 |
신규한 헤테로사이클릭아민 유도체 및 이를 포함하는 약학 조성물
|
KR102328682B1
(ko)
*
|
2018-08-27 |
2021-11-18 |
주식회사 대웅제약 |
신규한 헤테로사이클릭아민 유도체 및 이를 포함하는 약학 조성물
|
US11066404B2
(en)
|
2018-10-11 |
2021-07-20 |
Incyte Corporation |
Dihydropyrido[2,3-d]pyrimidinone compounds as CDK2 inhibitors
|
PL3902803T3
(pl)
*
|
2018-12-27 |
2023-05-22 |
Les Laboratoires Servier |
Aza-heterobicykliczne inhibitory mat2a i sposoby zastosowania do leczenia nowotworu
|
WO2020142748A1
(en)
|
2019-01-03 |
2020-07-09 |
University Of Pittsburgh - Of The Commonwealth System Of Higher Education |
Methods and materials for increasing transcription factor eb polypeptide levels
|
US20220133740A1
(en)
|
2019-02-08 |
2022-05-05 |
Frequency Therapeutics, Inc. |
Valproic acid compounds and wnt agonists for treating ear disorders
|
WO2020168197A1
(en)
|
2019-02-15 |
2020-08-20 |
Incyte Corporation |
Pyrrolo[2,3-d]pyrimidinone compounds as cdk2 inhibitors
|
TW202100520A
(zh)
|
2019-03-05 |
2021-01-01 |
美商英塞特公司 |
作為cdk2 抑制劑之吡唑基嘧啶基胺化合物
|
EP3941463A1
(en)
|
2019-03-22 |
2022-01-26 |
Sumitomo Dainippon Pharma Oncology, Inc. |
Compositions comprising pkm2 modulators and methods of treatment using the same
|
CA3134405A1
(en)
|
2019-03-28 |
2020-10-01 |
Jiangsu Hengrui Medicine Co., Ltd. |
Thienoheterocyclic derivative, preparation method therefor and medical use thereof
|
KR20210146956A
(ko)
|
2019-03-29 |
2021-12-06 |
지앙수 헨그루이 메디슨 컴퍼니 리미티드 |
피롤로헤테로고리형 유도체, 이의 제조 방법, 및 의약에서 이의 응용
|
US11919904B2
(en)
|
2019-03-29 |
2024-03-05 |
Incyte Corporation |
Sulfonylamide compounds as CDK2 inhibitors
|
CN109826608A
(zh)
*
|
2019-04-08 |
2019-05-31 |
中国科学院地质与地球物理研究所 |
一种分段压裂装置
|
TW202106681A
(zh)
|
2019-04-24 |
2021-02-16 |
美商施萬生物製藥研發Ip有限責任公司 |
用於治療皮膚疾病之嘧啶jak抑制劑
|
PL3958969T3
(pl)
|
2019-04-24 |
2024-05-20 |
Theravance Biopharma R&D Ip, Llc |
Estrowe i węglanowe związki pirymidynowe jako inhibitory kinaz
|
US11440914B2
(en)
|
2019-05-01 |
2022-09-13 |
Incyte Corporation |
Tricyclic amine compounds as CDK2 inhibitors
|
WO2020223558A1
(en)
|
2019-05-01 |
2020-11-05 |
Incyte Corporation |
Tricyclic amine compounds as cdk2 inhibitors
|
CN113825757B
(zh)
|
2019-05-24 |
2023-10-20 |
江苏恒瑞医药股份有限公司 |
取代的稠合双环类衍生物、其制备方法及其在医药上的应用
|
WO2020243519A1
(en)
*
|
2019-05-29 |
2020-12-03 |
Ifm Due, Inc. |
Compounds and compositions for treating conditions associated with sting activity
|
EP4013750A1
(en)
|
2019-08-14 |
2022-06-22 |
Incyte Corporation |
Imidazolyl pyrimidinylamine compounds as cdk2 inhibitors
|
US20220289692A1
(en)
*
|
2019-09-06 |
2022-09-15 |
Inflazome Limited |
Nlrp3 inhibitors
|
KR20220079597A
(ko)
*
|
2019-10-02 |
2022-06-13 |
톨레모 테라퓨틱스 아게 |
헤테로사이클릭 유도체, 약학 조성물 및 암의 치료 또는 개선에서 그들의 용도
|
WO2021072232A1
(en)
|
2019-10-11 |
2021-04-15 |
Incyte Corporation |
Bicyclic amines as cdk2 inhibitors
|
AU2021226411A1
(en)
*
|
2020-02-26 |
2022-09-22 |
Jaguahr Therapeutics Pte Ltd |
Pyridopyrimidine derivatives useful in modulation of AhR signalling
|
MX2022011826A
(es)
*
|
2020-03-27 |
2022-10-18 |
Dong A St Co Ltd |
Derivados de aminopirimidina y su uso como moduladores del receptor de hidrocarburos de arilo.
|
KR20230051500A
(ko)
|
2020-07-15 |
2023-04-18 |
키에시 파르마슈티시 엣스. 피. 에이. |
Alk5 억제제로서 피리다진일 아미노 유도체
|
WO2022032484A1
(zh)
*
|
2020-08-11 |
2022-02-17 |
北京诺诚健华医药科技有限公司 |
哒嗪-3-甲酰胺类化合物、其制备方法及其在医药学上的应用
|
CN114149410A
(zh)
*
|
2020-09-07 |
2022-03-08 |
四川科伦博泰生物医药股份有限公司 |
吡啶并环类化合物及其制备方法和用途
|
WO2022068860A1
(zh)
|
2020-09-29 |
2022-04-07 |
江苏恒瑞医药股份有限公司 |
一种吡咯并杂环类衍生物的晶型及其制备方法
|
WO2022107919A1
(ko)
*
|
2020-11-19 |
2022-05-27 |
주식회사 보로노이 |
N을 포함하는 헤테로아릴 유도체 및 이를 유효성분으로 포함하는 단백질 키나아제 관련 질환의 예방 또는 치료용 약학적 조성물
|
US11981671B2
(en)
|
2021-06-21 |
2024-05-14 |
Incyte Corporation |
Bicyclic pyrazolyl amines as CDK2 inhibitors
|
US11932648B2
(en)
|
2021-06-28 |
2024-03-19 |
Blueprint Medicines Corporation |
CDK2 inhibitors
|
AR127108A1
(es)
|
2021-09-21 |
2023-12-20 |
Chiesi Farm Spa |
Derivados de amino piridazinilo como inhibidores de alk5
|
CN116023380B
(zh)
*
|
2021-10-26 |
2024-01-23 |
沈阳药科大学 |
一类吡唑并嘧啶衍生物及制备方法和应用
|
US11976073B2
(en)
|
2021-12-10 |
2024-05-07 |
Incyte Corporation |
Bicyclic amines as CDK2 inhibitors
|
AU2023207775A1
(en)
|
2022-01-11 |
2024-08-22 |
Chiesi Farmaceutici S.P.A. |
Pyridazinyl amino derivatives as alk5 inhibitors
|