ATE339416T1 - Inhibitoren von c-jun-n-terminalen-kinasen (jnk) und anderen proteinkinasen - Google Patents
Inhibitoren von c-jun-n-terminalen-kinasen (jnk) und anderen proteinkinasenInfo
- Publication number
- ATE339416T1 ATE339416T1 AT02762067T AT02762067T ATE339416T1 AT E339416 T1 ATE339416 T1 AT E339416T1 AT 02762067 T AT02762067 T AT 02762067T AT 02762067 T AT02762067 T AT 02762067T AT E339416 T1 ATE339416 T1 AT E339416T1
- Authority
- AT
- Austria
- Prior art keywords
- kinases
- jnk
- jun
- inhibitors
- terminal
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/18—Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P13/12—Drugs for disorders of the urinary system of the kidneys
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
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- A61P21/04—Drugs for disorders of the muscular or neuromuscular system for myasthenia gravis
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US28362101P | 2001-04-13 | 2001-04-13 | |
US29297401P | 2001-05-23 | 2001-05-23 | |
US32944001P | 2001-10-15 | 2001-10-15 |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE339416T1 true ATE339416T1 (de) | 2006-10-15 |
Family
ID=27403408
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT02762067T ATE339416T1 (de) | 2001-04-13 | 2002-04-10 | Inhibitoren von c-jun-n-terminalen-kinasen (jnk) und anderen proteinkinasen |
Country Status (12)
Country | Link |
---|---|
US (2) | US6642227B2 (de) |
EP (1) | EP1389206B1 (de) |
JP (1) | JP2004535381A (de) |
AR (1) | AR035824A1 (de) |
AT (1) | ATE339416T1 (de) |
AU (1) | AU2002338642A1 (de) |
CA (1) | CA2443487A1 (de) |
DE (1) | DE60214701T2 (de) |
ES (1) | ES2271322T3 (de) |
MX (1) | MXPA03009378A (de) |
TW (1) | TWI235752B (de) |
WO (1) | WO2002083667A2 (de) |
Families Citing this family (92)
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EP1317452B1 (de) * | 2000-09-15 | 2006-05-17 | Vertex Pharmaceuticals Incorporated | Pyrazolverbindungen als protein-kinasehemmer |
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ATE339418T1 (de) * | 2001-06-01 | 2006-10-15 | Vertex Pharma | Thiazolverbindungen, die sich als inhibitoren von proteinkinasen eignen |
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2002
- 2002-04-10 DE DE60214701T patent/DE60214701T2/de not_active Expired - Lifetime
- 2002-04-10 EP EP02762067A patent/EP1389206B1/de not_active Expired - Lifetime
- 2002-04-10 MX MXPA03009378A patent/MXPA03009378A/es unknown
- 2002-04-10 JP JP2002581422A patent/JP2004535381A/ja not_active Withdrawn
- 2002-04-10 CA CA002443487A patent/CA2443487A1/en not_active Abandoned
- 2002-04-10 US US10/121,035 patent/US6642227B2/en not_active Expired - Fee Related
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MXPA03009378A (es) | 2004-01-29 |
WO2002083667A2 (en) | 2002-10-24 |
DE60214701T2 (de) | 2007-09-13 |
ES2271322T3 (es) | 2007-04-16 |
TWI235752B (en) | 2005-07-11 |
US7084159B2 (en) | 2006-08-01 |
CA2443487A1 (en) | 2002-10-24 |
JP2004535381A (ja) | 2004-11-25 |
EP1389206B1 (de) | 2006-09-13 |
AU2002338642A1 (en) | 2002-10-28 |
DE60214701D1 (de) | 2006-10-26 |
US20040023963A1 (en) | 2004-02-05 |
AR035824A1 (es) | 2004-07-14 |
US6642227B2 (en) | 2003-11-04 |
EP1389206A2 (de) | 2004-02-18 |
US20030096816A1 (en) | 2003-05-22 |
WO2002083667A3 (en) | 2003-01-03 |
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