SK286635B6 - N-substituované 2-kyanopyrolidíny, farmaceutický prostriedok, ktorý ich obsahuje a ich použitie na výrobu liečiva - Google Patents

N-substituované 2-kyanopyrolidíny, farmaceutický prostriedok, ktorý ich obsahuje a ich použitie na výrobu liečiva Download PDF

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Publication number
SK286635B6
SK286635B6 SK789-2001A SK7892001A SK286635B6 SK 286635 B6 SK286635 B6 SK 286635B6 SK 7892001 A SK7892001 A SK 7892001A SK 286635 B6 SK286635 B6 SK 286635B6
Authority
SK
Slovakia
Prior art keywords
amino
acetyl
adamantyl
cyanopyrrolidine
pharmaceutically acceptable
Prior art date
Application number
SK789-2001A
Other languages
English (en)
Slovak (sk)
Other versions
SK7892001A3 (en
Inventor
Edwin Bernard Villhauer
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22777194&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SK286635(B6) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of SK7892001A3 publication Critical patent/SK7892001A3/sk
Publication of SK286635B6 publication Critical patent/SK286635B6/sk

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
SK789-2001A 1998-12-10 1999-12-09 N-substituované 2-kyanopyrolidíny, farmaceutický prostriedok, ktorý ich obsahuje a ich použitie na výrobu liečiva SK286635B6 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US20906898A 1998-12-10 1998-12-10
PCT/EP1999/009708 WO2000034241A1 (en) 1998-12-10 1999-12-09 N-substituted 2-cyanopyrrolidines

Publications (2)

Publication Number Publication Date
SK7892001A3 SK7892001A3 (en) 2001-11-06
SK286635B6 true SK286635B6 (sk) 2009-02-05

Family

ID=22777194

Family Applications (1)

Application Number Title Priority Date Filing Date
SK789-2001A SK286635B6 (sk) 1998-12-10 1999-12-09 N-substituované 2-kyanopyrolidíny, farmaceutický prostriedok, ktorý ich obsahuje a ich použitie na výrobu liečiva

Country Status (34)

Country Link
US (1) US6166063A (OSRAM)
EP (1) EP1137635B1 (OSRAM)
JP (2) JP3681110B2 (OSRAM)
KR (2) KR20050047561A (OSRAM)
CN (1) CN1160330C (OSRAM)
AR (1) AR023719A1 (OSRAM)
AT (1) ATE307112T1 (OSRAM)
BR (1) BRPI9915985B8 (OSRAM)
CA (1) CA2350609C (OSRAM)
CO (1) CO5150173A1 (OSRAM)
CY (3) CY1105355T1 (OSRAM)
CZ (1) CZ299151B6 (OSRAM)
DE (3) DE69927844T2 (OSRAM)
DK (1) DK1137635T3 (OSRAM)
ES (1) ES2251847T3 (OSRAM)
FR (1) FR08C0005I2 (OSRAM)
HK (1) HK1040394B (OSRAM)
HU (1) HU226769B1 (OSRAM)
ID (1) ID28796A (OSRAM)
IL (2) IL143091A0 (OSRAM)
LU (2) LU91409I2 (OSRAM)
MY (1) MY123244A (OSRAM)
NL (2) NL300333I2 (OSRAM)
NO (3) NO318741B1 (OSRAM)
NZ (1) NZ511935A (OSRAM)
PE (1) PE20001317A1 (OSRAM)
PL (1) PL199443B1 (OSRAM)
RU (1) RU2251544C2 (OSRAM)
SK (1) SK286635B6 (OSRAM)
TR (1) TR200101478T2 (OSRAM)
TW (1) TW509674B (OSRAM)
UY (1) UY25843A1 (OSRAM)
WO (1) WO2000034241A1 (OSRAM)
ZA (1) ZA200104581B (OSRAM)

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