JP2010520168A5 - - Google Patents

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Publication number
JP2010520168A5
JP2010520168A5 JP2009551208A JP2009551208A JP2010520168A5 JP 2010520168 A5 JP2010520168 A5 JP 2010520168A5 JP 2009551208 A JP2009551208 A JP 2009551208A JP 2009551208 A JP2009551208 A JP 2009551208A JP 2010520168 A5 JP2010520168 A5 JP 2010520168A5
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JP
Japan
Prior art keywords
formula
compound
inhibitor
examples
chain
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JP2009551208A
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English (en)
Japanese (ja)
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JP2010520168A (ja
JP5930573B2 (ja
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Priority claimed from US11/685,881 external-priority patent/US7732162B2/en
Application filed filed Critical
Priority claimed from PCT/EP2008/052411 external-priority patent/WO2008104580A1/en
Publication of JP2010520168A publication Critical patent/JP2010520168A/ja
Publication of JP2010520168A5 publication Critical patent/JP2010520168A5/ja
Application granted granted Critical
Publication of JP5930573B2 publication Critical patent/JP5930573B2/ja
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JP2009551208A 2007-03-01 2008-02-28 グルタミニルシクラーゼ阻害剤の新規使用 Active JP5930573B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US89226507P 2007-03-01 2007-03-01
US60/892,265 2007-03-01
US11/685,881 2007-03-14
US11/685,881 US7732162B2 (en) 2003-05-05 2007-03-14 Inhibitors of glutaminyl cyclase for treating neurodegenerative diseases
PCT/EP2008/052411 WO2008104580A1 (en) 2007-03-01 2008-02-28 New use of glutaminyl cyclase inhibitors

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2014038631A Division JP2014148508A (ja) 2007-03-01 2014-02-28 グルタミニルシクラーゼ阻害剤の新規使用

Publications (3)

Publication Number Publication Date
JP2010520168A JP2010520168A (ja) 2010-06-10
JP2010520168A5 true JP2010520168A5 (enExample) 2012-04-12
JP5930573B2 JP5930573B2 (ja) 2016-06-15

Family

ID=39345241

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2009551208A Active JP5930573B2 (ja) 2007-03-01 2008-02-28 グルタミニルシクラーゼ阻害剤の新規使用

Country Status (12)

Country Link
EP (2) EP2481408A3 (enExample)
JP (1) JP5930573B2 (enExample)
KR (1) KR20090115951A (enExample)
CN (1) CN101668525A (enExample)
AU (1) AU2008220785B2 (enExample)
CA (1) CA2679446C (enExample)
EA (1) EA200901140A1 (enExample)
IL (1) IL200315A (enExample)
MX (1) MX2009009234A (enExample)
NZ (1) NZ579310A (enExample)
WO (1) WO2008104580A1 (enExample)
ZA (1) ZA200905537B (enExample)

Families Citing this family (12)

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US9108948B2 (en) 2006-06-23 2015-08-18 Abbvie Inc. Cyclopropyl amine derivatives
BRPI0808170A2 (pt) * 2007-03-01 2014-07-08 Probiodrug Ag Uso de inibidores de glutaminil ciclase
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UA108742C2 (uk) * 2009-09-23 2015-06-10 Фармацевтична композиція для лікування запальних захворювань, опосередкованих mcp-1
JP2013519891A (ja) * 2010-02-18 2013-05-30 プロビオドルグ エージー ピログルタミン酸修飾mcp−1を決定することにより炎症性疾患を診断する方法及びグルタミニルシクラーゼの阻害剤のスクリーニング方法
WO2012037258A1 (en) 2010-09-16 2012-03-22 Abbott Laboratories Processes for preparing 1,2-substituted cyclopropyl derivatives
CN105384691B (zh) * 2015-10-26 2018-06-29 深圳大学 一种谷氨酰胺酰基环化酶抑制剂的制备方法及应用
CN105384692B (zh) * 2015-10-26 2018-06-29 深圳大学 一种谷氨酰胺酰基环化酶抑制剂
EP3747437A1 (en) * 2017-07-24 2020-12-09 Stichting Het Nederlands Kanker Instituut- Antoni van Leeuwenhoek Ziekenhuis Treating pathological conditions by direct and indirect targeting of sirpa - cd47 interaction
KR102230832B1 (ko) * 2019-06-17 2021-03-24 (주) 메디프론디비티 N-치환된 티오우레아 또는 우레아 유도체 및 이를 유효성분으로 함유하는 글루타미닐 사이클레이즈 활성 관련 질환의 예방 또는 치료용 약학적 조성물
CN118019737A (zh) 2021-06-24 2024-05-10 英矽智能科技知识产权有限公司 用于治疗疾病的β-内酰胺衍生物

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