ES2536433T3 - Derivados de 1,2,4-triazolo[4,3-a]piridina y su uso como moduladores alostéricos positivos de receptores mGluR2 - Google Patents
Derivados de 1,2,4-triazolo[4,3-a]piridina y su uso como moduladores alostéricos positivos de receptores mGluR2 Download PDFInfo
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- ES2536433T3 ES2536433T3 ES11781524.1T ES11781524T ES2536433T3 ES 2536433 T3 ES2536433 T3 ES 2536433T3 ES 11781524 T ES11781524 T ES 11781524T ES 2536433 T3 ES2536433 T3 ES 2536433T3
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP10190327 | 2010-11-08 | ||
| EP10190327 | 2010-11-08 | ||
| PCT/EP2011/069641 WO2012062751A1 (en) | 2010-11-08 | 2011-11-08 | 1,2,4-TRIAZOLO[4,3-a]PYRIDINE DERIVATIVES AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 RECEPTORS |
Publications (1)
| Publication Number | Publication Date |
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| ES2536433T3 true ES2536433T3 (es) | 2015-05-25 |
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| Country | Link |
|---|---|
| US (1) | US9012448B2 (enExample) |
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| CA (1) | CA2814998C (enExample) |
| ES (1) | ES2536433T3 (enExample) |
| WO (1) | WO2012062751A1 (enExample) |
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| AR059898A1 (es) | 2006-03-15 | 2008-05-07 | Janssen Pharmaceutica Nv | Derivados de 3-ciano-piridona 1,4-disustituida y su uso como moduladores alostericos de los receptores mglur2 |
| TW200845978A (en) | 2007-03-07 | 2008-12-01 | Janssen Pharmaceutica Nv | 3-cyano-4-(4-tetrahydropyran-phenyl)-pyridin-2-one derivatives |
| TW200900065A (en) | 2007-03-07 | 2009-01-01 | Janssen Pharmaceutica Nv | 3-cyano-4-(4-pyridinyloxy-phenyl)-pyridin-2-one derivatives |
| US8722894B2 (en) | 2007-09-14 | 2014-05-13 | Janssen Pharmaceuticals, Inc. | 1,3-disubstituted-4-phenyl-1H-pyridin-2-ones |
| NZ584152A (en) | 2007-09-14 | 2011-11-25 | Ortho Mcneil Janssen Pharm | 1,3-disubstituted 4-(aryl-x-phenyl)-1h-pyridin-2-ones |
| SI2203439T1 (sl) | 2007-09-14 | 2011-05-31 | Ortho Mcneil Janssen Pharm | 1',3'-disubstituirani 4-fenil-3,4,5,6-tetrahidro-2H-1'H-(1,4')bipiridinil-2'-oni |
| RU2492170C9 (ru) | 2007-11-14 | 2013-12-27 | Орто-Макнейл-Янссен Фармасьютикалз, Инк. | Имидазо[1,2-а]пиридиновые производные и их применение в качестве положительных аллостерических модуляторов рецепторов mglur2 |
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| US20140088151A1 (en) | 2011-05-03 | 2014-03-27 | Douglas C. Beshore | Alhydroxymethyl biaryl benzotriazole derivatives |
| EP2705024B1 (en) | 2011-05-03 | 2015-12-16 | Merck Sharp & Dohme Corp. | Alkyne benzotriazole derivatives |
-
2011
- 2011-11-08 JP JP2013537166A patent/JP5852665B2/ja not_active Expired - Fee Related
- 2011-11-08 WO PCT/EP2011/069641 patent/WO2012062751A1/en not_active Ceased
- 2011-11-08 EP EP20110781524 patent/EP2643320B1/en not_active Not-in-force
- 2011-11-08 ES ES11781524.1T patent/ES2536433T3/es active Active
- 2011-11-08 CN CN201180053638.6A patent/CN103261195B/zh not_active Expired - Fee Related
- 2011-11-08 AU AU2011328195A patent/AU2011328195B2/en not_active Ceased
- 2011-11-08 CA CA2814998A patent/CA2814998C/en not_active Expired - Fee Related
- 2011-11-08 US US13/884,149 patent/US9012448B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| JP5852665B2 (ja) | 2016-02-03 |
| CA2814998A1 (en) | 2012-05-18 |
| US20130252952A1 (en) | 2013-09-26 |
| CN103261195A (zh) | 2013-08-21 |
| AU2011328195A1 (en) | 2013-05-02 |
| US9012448B2 (en) | 2015-04-21 |
| CN103261195B (zh) | 2015-09-02 |
| WO2012062751A1 (en) | 2012-05-18 |
| EP2643320A1 (en) | 2013-10-02 |
| CA2814998C (en) | 2019-10-29 |
| EP2643320B1 (en) | 2015-03-04 |
| AU2011328195B2 (en) | 2015-04-02 |
| JP2013541578A (ja) | 2013-11-14 |
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