AR044743A1 - Herbicida, metodo de emplearlo, derivados de tienopirimidina sustituida,compuestos intermediarios, y procedimientos que se utilizan para producirlos, - Google Patents
Herbicida, metodo de emplearlo, derivados de tienopirimidina sustituida,compuestos intermediarios, y procedimientos que se utilizan para producirlos,Info
- Publication number
- AR044743A1 AR044743A1 ARP030103503A ARP030103503A AR044743A1 AR 044743 A1 AR044743 A1 AR 044743A1 AR P030103503 A ARP030103503 A AR P030103503A AR P030103503 A ARP030103503 A AR P030103503A AR 044743 A1 AR044743 A1 AR 044743A1
- Authority
- AR
- Argentina
- Prior art keywords
- alkyl
- substituted
- fluorine
- containing fluorine
- formula
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C255/00—Carboxylic acid nitriles
- C07C255/01—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms
- C07C255/32—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring
- C07C255/40—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring the carbon skeleton being further substituted by doubly-bound oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/76—Esters of carboxylic acids having a carboxyl group bound to a carbon atom of a six-membered aromatic ring
- C07C69/84—Esters of carboxylic acids having a carboxyl group bound to a carbon atom of a six-membered aromatic ring of monocyclic hydroxy carboxylic acids, the hydroxy groups and the carboxyl groups of which are bound to carbon atoms of a six-membered aromatic ring
- C07C69/92—Esters of carboxylic acids having a carboxyl group bound to a carbon atom of a six-membered aromatic ring of monocyclic hydroxy carboxylic acids, the hydroxy groups and the carboxyl groups of which are bound to carbon atoms of a six-membered aromatic ring with etherified hydroxyl groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/30—Hetero atoms other than halogen
- C07D333/36—Nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Abstract
Un herbicida que comprende, como ingrediente activo, un derivado de tienopirimidina sustituida que se representa a través de la fórmula (1), donde A representa según lo indica el grupo de fórmulas (2) ó (3), donde R1 representa hidrógeno o alquilo que puede ser sustituido, y R2 representa hidrógeno, halógeno o alquilo que puede ser sustituido; donde R1 y R2 tienen los mismos significados que se describieron; Q1 representa hidrógeno, halógeno, ciano, hidroxilo, carboxilo o -X1R3, donde X1 es un enlace simple, -O-, -SOn- donde n representa un entero de 0 a 2, -OSOn- donde n tiene el mismo significado que se describió previamente, -CO-, -CO2-, -OCO2- o -OC(O)-, y R3 representa alquilo que puede ser sustituido, alquenilo que puede ser sustituido, alquinilo que puede ser sustituido, amino que puede ser sustituido, arilo que puede ser sustituido o un grupo heterocíclico que puede ser sustituido; Q2 representa hidrógeno, halógeno, hidroxilo o -X2R4, donde X2 es un enlace simple, -O-, -SOn-, donde n tiene el mismo signficado que se describió previamente, -OSOn- donde n tiene el mismo significado que se descrbió previamente, -CO-, -CO2-, -OCO2- o -OC(O)-; y R4 representa alquilo que puede ser sustituido, alquenilo que puede ser sustituido, alquinilo que puede ser sustituido, amino que puede ser sustituido, arilo que puede ser sustituido o un grupo heterocíclico que puede ser sustituido; un método herbicida, que comprende realizar un tratamiento del suelo, un tratamiento foliar del terreno o un tratamiento de riego con una cantidad eficaz del herbicida según cualquiera de las reivindicaciones 1 a 5. Un derivado de tienopirimidina sustituida representado por la fórmula (1), un método para producir un derivado de tienopirimidina sustituida representado por la fórmula (4), que comprende hacer reaccionar un compuesto de la fórmula (5), donde Q2a representa: arilo sustituido que tiene uno o más sustituyentes que son iguales o diferentes y que se seleccionan del grupo que consta de alquilo (C1-6) que contiene flúor, alcoxi (C1-6) que contiene flúor y alquil(C1-6)tio que contiene flúor; ariloxi sustituido que tiene uno o más sustituyentes que son iguales o diferentes y que se seleccionan del grupo que consta de alquilo (C1-6) que contiene flúor, alcoxi (C1-6) que contiene flúor y alquil(C1-6)tio que contiene flúor; ariltio sustituido que tiene uno o más sustituyentes que son iguales o diferentes y que se seleccionan del grupo que consta de alquilo (C1-6) que contiene flúor, alcoxi (C1-6) que contiene flúor y alquil(C1-6)tio que contiene flúor; arilsulfinilo sustituido que tiene uno o más sustituyentes que son iguales o diferentes y que se seleccionan del grupo que consta de alquilo (C1-6) que contiene flúor, alcoxi (C1-6) que contiene flúor y alquil(C1-6)tio que contiene flúor; arilsulfonilo sustituido que tiene uno o más sustituyentes que son iguales o diferentes y que se seleccionan del grupo que consta de alquilo (C1-6) que contiene flúor, alcoxi (C1-6) que contiene flúor y alquil(C1-6)tio que contiene flúor; con un compuesto representado por la fórmula: R3X1aH, donde X1a es un enlace simple, -O- o -S-. Un procedimiento para elaborar un derivado de tieno[2,3-d]pirimidina sustituida representado por la fórmula (6), que comprende realizar una reacción de acople del derivado de 2,4-dihalogenotieno[2,3-d]pirimidina representado por la fórmula (7), donde R1 representa hidrógeno, alquilo (C1-6) o haloalquilo(C1-6); R2 representa hidrógeno, halógeno, alquilo (C1-6) o haloalquilo (C1-6); e Y representa halógeno que son iguales o diferentes; Q2a-L, donde Q2a representa arilo sustituido que tiene uno o más sustituyentes que son iguales o diferentes y que se seleccionan del grupo que consta de alquilo (C1-6) que contiene flúor, alcoxi (C1-6) que contiene flúor y alquil(C1-6)tio que contiene flúor; y L representa un grupo saliente. Un derivado de 2-amino-3-(benzoilo sustituido)tiofeno representado por la fórmula (8), donde R1 representa hidrógeno, alquilo (C1-6) o haloalquilo (C1-6); R5 representa hidrógeno, halógeno, alquilo (C1-6) o haloalquilo (C1-6); R6 representa alquilo (C1-6) que contiene flúor, alcoxi (C1-6) que contiene flúor o alquil(C1-6)tio que contiene flúor. Un derivado de ureidotiofeno representado por la fórmula (9), donde R1 representa hidrógeno, alquilo (C1-6) o haloalquilo (C1-6); R2 representa hidrógeno, halógeno, alquilo (C1-6) o haloalquilo (C1-6); y w representa arilo o arilo sustituido que tiene uno o más sustituyentes que son iguales o diferentes y que se seleccionan del grupo que consta de halógeno, ciano, nitro, alquilo (C1-6), haloalquilo (C1-6), alcoxi (C1-6), haloalcoxi (C1-6) y haloalquil(C1-6)tio. Un derivado de benzoilacetonitrilo sustituido representado pro la fórmula (10), donde R5 representa hidrógeno, halógeno, alquilo (C1-6) o haloalquilo (C1-6); R6 representa alquilo (C1-6) que contienen flúor, alcoxi C1-6) que contiene flúor y alquil(C1-6)tio que contiene flúor, y donde, cuando R6 es alquilo (C1-6) que contiene flúor, R5 no es hidrógeno. Un compuesto que es benzoato de 3-(trifluorometoxi)etilo.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
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JP2002281271 | 2002-09-26 |
Publications (1)
Publication Number | Publication Date |
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AR044743A1 true AR044743A1 (es) | 2005-10-05 |
Family
ID=32040508
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP030103503A AR044743A1 (es) | 2002-09-26 | 2003-09-25 | Herbicida, metodo de emplearlo, derivados de tienopirimidina sustituida,compuestos intermediarios, y procedimientos que se utilizan para producirlos, |
Country Status (7)
Country | Link |
---|---|
US (1) | US20070010402A1 (es) |
EP (1) | EP1544202A4 (es) |
AR (1) | AR044743A1 (es) |
AU (1) | AU2003272898B2 (es) |
CA (1) | CA2500207A1 (es) |
TW (1) | TW200410975A (es) |
WO (1) | WO2004029060A1 (es) |
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-
2003
- 2003-09-25 TW TW092126472A patent/TW200410975A/zh unknown
- 2003-09-25 AR ARP030103503A patent/AR044743A1/es unknown
- 2003-09-26 WO PCT/JP2003/012356 patent/WO2004029060A1/ja active Application Filing
- 2003-09-26 US US10/529,474 patent/US20070010402A1/en not_active Abandoned
- 2003-09-26 CA CA002500207A patent/CA2500207A1/en not_active Abandoned
- 2003-09-26 AU AU2003272898A patent/AU2003272898B2/en not_active Expired - Fee Related
- 2003-09-26 EP EP03753959A patent/EP1544202A4/en not_active Withdrawn
Also Published As
Publication number | Publication date |
---|---|
AU2003272898A1 (en) | 2004-04-19 |
WO2004029060A1 (ja) | 2004-04-08 |
AU2003272898B2 (en) | 2009-08-13 |
EP1544202A4 (en) | 2007-07-18 |
US20070010402A1 (en) | 2007-01-11 |
EP1544202A1 (en) | 2005-06-22 |
TW200410975A (en) | 2004-07-01 |
CA2500207A1 (en) | 2004-04-08 |
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