DZ3191A1 - Composés d'indazole et compositions pharmaceutiques inhibant les protéines kinases, et procédés d'utilisation de ceux-ci. - Google Patents

Composés d'indazole et compositions pharmaceutiques inhibant les protéines kinases, et procédés d'utilisation de ceux-ci.

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Publication number
DZ3191A1
DZ3191A1 DZ003191A DZ003191A DZ3191A1 DZ 3191 A1 DZ3191 A1 DZ 3191A1 DZ 003191 A DZ003191 A DZ 003191A DZ 003191 A DZ003191 A DZ 003191A DZ 3191 A1 DZ3191 A1 DZ 3191A1
Authority
DZ
Algeria
Prior art keywords
methods
same
pharmaceutical compositions
protein kinases
inhibiting protein
Prior art date
Application number
DZ003191A
Other languages
English (en)
French (fr)
Inventor
Robert Steven Kania
Steven Lee Bender
Allen J Borchardt
John F Braganza
Stephan James Cripps
Ye Hua
Michael David Johnson
Theodore Otto Johnson Jr
Hiep The Luu
Cynthia Louise Palmer
Siegfried Heinz Reich
Anna Maria Tempczyk-Russell
Min Teng
Christine Thomas
Michael David Varney
Michael Brennan Wallace
Michael Raymond Collins
Original Assignee
Agouron Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22498654&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DZ3191(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Agouron Pharma filed Critical Agouron Pharma
Application granted granted Critical
Publication of DZ3191A1 publication Critical patent/DZ3191A1/xx

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    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
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    • A61P19/00Drugs for skeletal disorders
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
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    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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    • A61P3/00Drugs for disorders of the metabolism
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    • A61P3/00Drugs for disorders of the metabolism
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P35/00Antineoplastic agents
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    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
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    • C07D491/04Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
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  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Ophthalmology & Optometry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Dermatology (AREA)
  • Obesity (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
DZ003191A 1999-07-02 2000-06-30 Composés d'indazole et compositions pharmaceutiques inhibant les protéines kinases, et procédés d'utilisation de ceux-ci. DZ3191A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US14213099P 1999-07-02 1999-07-02
PCT/US2000/018263 WO2001002369A2 (en) 1999-07-02 2000-06-30 Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use

Publications (1)

Publication Number Publication Date
DZ3191A1 true DZ3191A1 (fr) 2001-01-11

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ID=22498654

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DZ003191A DZ3191A1 (fr) 1999-07-02 2000-06-30 Composés d'indazole et compositions pharmaceutiques inhibant les protéines kinases, et procédés d'utilisation de ceux-ci.

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EP (2) EP1218348B1 (pm)
JP (2) JP3878849B2 (pm)
KR (1) KR100529639B1 (pm)
CN (2) CN1137884C (pm)
AP (1) AP1486A (pm)
AR (2) AR035554A1 (pm)
AT (1) ATE376543T1 (pm)
AU (1) AU777701B2 (pm)
BE (1) BE2013C015I2 (pm)
BG (1) BG66070B1 (pm)
BR (1) BRPI0012352B8 (pm)
CA (1) CA2383630C (pm)
CO (1) CO5190686A1 (pm)
CR (2) CR6517A (pm)
CY (3) CY1107148T1 (pm)
CZ (1) CZ301667B6 (pm)
DE (2) DE60037211T2 (pm)
DK (2) DK1614683T3 (pm)
DZ (1) DZ3191A1 (pm)
EA (1) EA004460B1 (pm)
EE (1) EE05585B1 (pm)
ES (2) ES2293906T3 (pm)
FR (1) FR13C0010I2 (pm)
GE (1) GEP20063885B (pm)
GT (1) GT200000107A (pm)
HR (1) HRP20020109B1 (pm)
HU (1) HU228502B1 (pm)
IL (1) IL146710A0 (pm)
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LU (1) LU92154I2 (pm)
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MY (2) MY137622A (pm)
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PE (1) PE20010306A1 (pm)
PL (1) PL212108B1 (pm)
PT (2) PT1614683E (pm)
RS (1) RS50339B (pm)
SI (2) SI1218348T1 (pm)
SK (1) SK286936B6 (pm)
SV (1) SV2002000121A (pm)
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UY (1) UY26231A1 (pm)
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PE20010306A1 (es) * 1999-07-02 2001-03-29 Agouron Pharma Compuestos de indazol y composiciones farmaceuticas que los contienen utiles para la inhibicion de proteina kinasa
DZ3377A1 (fr) 1999-12-24 2001-07-05 Aventis Pharma Ltd Azaindoles
JP2003522174A (ja) 2000-02-07 2003-07-22 ブリストル−マイヤーズ スクイブ カンパニー サイクリン依存性キナーゼの3−アミノピラゾール阻害剤
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WO2002012228A1 (en) 2000-08-09 2002-02-14 Astrazeneca Ab Cinnoline compounds
EP1313726A1 (en) 2000-08-09 2003-05-28 AstraZeneca AB Quinoline derivatives having vegf inhibiting activity
WO2002018383A2 (en) 2000-09-01 2002-03-07 Chiron Corporation Aza heterocyclic derivatives and their therapeutic use
AU2001293275B2 (en) 2000-09-11 2005-04-14 Novartis Vaccines And Diagnostic Inc. Quinolinone derivatives as tyrosine kinase inhibitors
WO2002032872A1 (en) 2000-10-20 2002-04-25 Eisai Co., Ltd. Nitrogenous aromatic ring compounds
TWI243164B (en) 2001-02-13 2005-11-11 Aventis Pharma Gmbh Acylated indanyl amines and their use as pharmaceuticals
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JPWO2004050088A1 (ja) * 2002-12-03 2006-03-30 協和醗酵工業株式会社 Jnk阻害剤
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