CN1469875A - 可用作蛋白激酶抑制剂的吡唑化合物 - Google Patents

可用作蛋白激酶抑制剂的吡唑化合物 Download PDF

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Publication number
CN1469875A
CN1469875A CNA018174329A CN01817432A CN1469875A CN 1469875 A CN1469875 A CN 1469875A CN A018174329 A CNA018174329 A CN A018174329A CN 01817432 A CN01817432 A CN 01817432A CN 1469875 A CN1469875 A CN 1469875A
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ring
optionally substituted
aliphatic group
group
halogen
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Chinese (zh)
Inventor
D
D·拜宾顿
θ�̩��
R·克奈格泰尔
C
J·M·C·戈里克
李磐
R·戴维斯
J-D·凯瑞尔
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Vertex Pharmaceuticals Inc
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Vertex Pharmaceuticals Inc
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27398347&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CN1469875(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Vertex Pharmaceuticals Inc filed Critical Vertex Pharmaceuticals Inc
Publication of CN1469875A publication Critical patent/CN1469875A/zh
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  • Chemical & Material Sciences (AREA)
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  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Endocrinology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Hematology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Biomedical Technology (AREA)
  • Obesity (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pulmonology (AREA)
  • Oncology (AREA)
  • Psychiatry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Emergency Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
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  • Dermatology (AREA)
  • Transplantation (AREA)
  • Urology & Nephrology (AREA)
CNA018174329A 2000-09-15 2001-09-14 可用作蛋白激酶抑制剂的吡唑化合物 Pending CN1469875A (zh)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US23279500P 2000-09-15 2000-09-15
US60/232,795 2000-09-15
US25788700P 2000-12-21 2000-12-21
US60/257,887 2000-12-21
US28694901P 2001-04-27 2001-04-27
US60/286,949 2001-04-27

Publications (1)

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CN1469875A true CN1469875A (zh) 2004-01-21

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CNA018174329A Pending CN1469875A (zh) 2000-09-15 2001-09-14 可用作蛋白激酶抑制剂的吡唑化合物
CNB018174272A Expired - Fee Related CN100355750C (zh) 2000-09-15 2001-09-14 可用作蛋白激酶抑制剂的吡唑化合物
CNA018174337A Pending CN1473161A (zh) 2000-09-15 2001-09-14 可用作蛋白激酶抑制剂的吡唑化合物

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CNB018174272A Expired - Fee Related CN100355750C (zh) 2000-09-15 2001-09-14 可用作蛋白激酶抑制剂的吡唑化合物
CNA018174337A Pending CN1473161A (zh) 2000-09-15 2001-09-14 可用作蛋白激酶抑制剂的吡唑化合物

Country Status (23)

Country Link
US (7) US7098330B2 (https=)
EP (8) EP1317450B1 (https=)
JP (9) JP4922539B2 (https=)
KR (4) KR20030032035A (https=)
CN (3) CN1469875A (https=)
AP (1) AP2003002762A0 (https=)
AT (8) ATE346064T1 (https=)
AU (9) AU2001294558A1 (https=)
BR (1) BR0114088A (https=)
CA (8) CA2422299C (https=)
DE (8) DE60110616T3 (https=)
DK (1) DK1318997T3 (https=)
ES (3) ES2266258T3 (https=)
HU (4) HUP0302172A2 (https=)
IL (6) IL154747A0 (https=)
MX (8) MXPA03002297A (https=)
NO (4) NO326850B1 (https=)
NZ (4) NZ525014A (https=)
PE (1) PE20020451A1 (https=)
PL (1) PL361676A1 (https=)
PT (2) PT1318997E (https=)
TW (1) TWI303636B (https=)
WO (8) WO2002022601A1 (https=)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN104271578A (zh) * 2012-05-03 2015-01-07 霍夫曼-拉罗奇有限公司 作为lrrk2调节剂用于治疗帕金森病的吡唑氨基嘧啶衍生物
CN104271569A (zh) * 2012-05-03 2015-01-07 霍夫曼-拉罗奇有限公司 作为lrrk2调节剂的吡唑氨基嘧啶衍生物
CN105367555A (zh) * 2014-08-07 2016-03-02 广东东阳光药业有限公司 取代的杂芳基化合物及其组合物和用途
CN112638910A (zh) * 2018-08-27 2021-04-09 株式会社大熊制药 新的杂环胺衍生物及包含其的药物组合物

Families Citing this family (408)

* Cited by examiner, † Cited by third party
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CN104271569B (zh) * 2012-05-03 2016-08-24 霍夫曼-拉罗奇有限公司 作为lrrk2调节剂的吡唑氨基嘧啶衍生物
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