CA2400567C - Tamper-resistant oral opioid agonist formulations - Google Patents

Tamper-resistant oral opioid agonist formulations Download PDF

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Publication number
CA2400567C
CA2400567C CA002400567A CA2400567A CA2400567C CA 2400567 C CA2400567 C CA 2400567C CA 002400567 A CA002400567 A CA 002400567A CA 2400567 A CA2400567 A CA 2400567A CA 2400567 C CA2400567 C CA 2400567C
Authority
CA
Canada
Prior art keywords
dosage form
antagonist
opioid
naltrexone
oral dosage
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
CA002400567A
Other languages
English (en)
French (fr)
Other versions
CA2400567A1 (en
Inventor
Benjamin Oshlack
Curtis Wright
J. David Haddox
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Euro Celtique SA
Original Assignee
Euro Celtique SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
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Application filed by Euro Celtique SA filed Critical Euro Celtique SA
Publication of CA2400567A1 publication Critical patent/CA2400567A1/en
Application granted granted Critical
Publication of CA2400567C publication Critical patent/CA2400567C/en
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5084—Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
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    • A61K31/33—Heterocyclic compounds
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
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  • Dermatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Emergency Medicine (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Otolaryngology (AREA)
  • Addiction (AREA)
  • Pain & Pain Management (AREA)
  • Inorganic Chemistry (AREA)
  • Physics & Mathematics (AREA)
  • Nanotechnology (AREA)
  • Optics & Photonics (AREA)
  • Rheumatology (AREA)
  • Toxicology (AREA)
  • Psychiatry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CA002400567A 2000-02-08 2001-02-08 Tamper-resistant oral opioid agonist formulations Expired - Lifetime CA2400567C (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US18136900P 2000-02-08 2000-02-08
US60/181,369 2000-02-08
PCT/US2001/004346 WO2001058451A1 (en) 2000-02-08 2001-02-08 Tamper-resistant oral opioid agonist formulations

Publications (2)

Publication Number Publication Date
CA2400567A1 CA2400567A1 (en) 2001-08-16
CA2400567C true CA2400567C (en) 2008-01-15

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ID=22663996

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CA002400567A Expired - Lifetime CA2400567C (en) 2000-02-08 2001-02-08 Tamper-resistant oral opioid agonist formulations

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