KR20050047561A - Ｎ-치환된 2-시아노피롤리딘 - Google Patents

Ｎ-치환된 2-시아노피롤리딘 Download PDF

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Publication number
KR20050047561A
KR20050047561A KR1020057007771A KR20057007771A KR20050047561A KR 20050047561 A KR20050047561 A KR 20050047561A KR 1020057007771 A KR1020057007771 A KR 1020057007771A KR 20057007771 A KR20057007771 A KR 20057007771A KR 20050047561 A KR20050047561 A KR 20050047561A
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KR
South Korea
Prior art keywords
formula
amino
adamantyl
compounds
alkyl
Prior art date
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Ceased
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KR1020057007771A
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English (en)
Korean (ko)
Inventor
에드윈 버나드 빌하우어
Original Assignee
노파르티스 아게
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22777194&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=KR20050047561(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 노파르티스 아게 filed Critical 노파르티스 아게
Publication of KR20050047561A publication Critical patent/KR20050047561A/ko
Ceased legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
KR1020057007771A 1998-12-10 1999-12-09 Ｎ-치환된 2-시아노피롤리딘 Ceased KR20050047561A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US20906898A 1998-12-10 1998-12-10
US09/209,068 1998-12-10

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
KR10-2001-7007227A Division KR100509311B1 (ko) 1998-12-10 1999-12-09 Ｎ-치환된 2-시아노피롤리딘

Publications (1)

Publication Number Publication Date
KR20050047561A true KR20050047561A (ko) 2005-05-20

Family

ID=22777194

Family Applications (2)

Application Number Title Priority Date Filing Date
KR1020057007771A Ceased KR20050047561A (ko) 1998-12-10 1999-12-09 Ｎ-치환된 2-시아노피롤리딘
KR10-2001-7007227A Expired - Lifetime KR100509311B1 (ko) 1998-12-10 1999-12-09 Ｎ-치환된 2-시아노피롤리딘

Family Applications After (1)

Application Number Title Priority Date Filing Date
KR10-2001-7007227A Expired - Lifetime KR100509311B1 (ko) 1998-12-10 1999-12-09 Ｎ-치환된 2-시아노피롤리딘

Country Status (34)

Country Link
US (1) US6166063A (https=)
EP (1) EP1137635B1 (https=)
JP (2) JP3681110B2 (https=)
KR (2) KR20050047561A (https=)
CN (1) CN1160330C (https=)
AR (1) AR023719A1 (https=)
AT (1) ATE307112T1 (https=)
BR (1) BRPI9915985B8 (https=)
CA (1) CA2350609C (https=)
CO (1) CO5150173A1 (https=)
CY (3) CY1105355T1 (https=)
CZ (1) CZ299151B6 (https=)
DE (3) DE122008000007I1 (https=)
DK (1) DK1137635T3 (https=)
ES (1) ES2251847T3 (https=)
FR (1) FR08C0005I2 (https=)
HK (1) HK1040394B (https=)
HU (1) HU226769B1 (https=)
ID (1) ID28796A (https=)
IL (2) IL143091A0 (https=)
LU (2) LU91409I2 (https=)
MY (1) MY123244A (https=)
NL (2) NL300333I2 (https=)
NO (3) NO318741B1 (https=)
NZ (1) NZ511935A (https=)
PE (1) PE20001317A1 (https=)
PL (1) PL199443B1 (https=)
RU (1) RU2251544C2 (https=)
SK (1) SK286635B6 (https=)
TR (1) TR200101478T2 (https=)
TW (1) TW509674B (https=)
UY (1) UY25843A1 (https=)
WO (1) WO2000034241A1 (https=)
ZA (1) ZA200104581B (https=)

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* Cited by examiner, † Cited by third party
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