JPWO2019152374A5 - - Google Patents

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JPWO2019152374A5
JPWO2019152374A5 JP2020562089A JP2020562089A JPWO2019152374A5 JP WO2019152374 A5 JPWO2019152374 A5 JP WO2019152374A5 JP 2020562089 A JP2020562089 A JP 2020562089A JP 2020562089 A JP2020562089 A JP 2020562089A JP WO2019152374 A5 JPWO2019152374 A5 JP WO2019152374A5
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formula
salt
reaction
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JP2021512163A (ja
JP7393348B2 (ja
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JP2020562089A 2018-01-30 2019-01-29 (1-(3-フルオロ-2(トリフルオロメチル)イソニコチニル)ピぺリジン―4-オン)を作製するためのプロセス及び中間体 Active JP7393348B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2023175953A JP2024023173A (ja) 2018-01-30 2023-10-11 (1-(3-フルオロ-2(トリフルオロメチル)イソニコチニル)ピぺリジン―4-オン)を作製するためのプロセス及び中間体

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862623664P 2018-01-30 2018-01-30
US62/623,664 2018-01-30
PCT/US2019/015582 WO2019152374A1 (en) 2018-01-30 2019-01-29 Processes for preparing (1 -(3-fluoro-2-(trifluoromethyl)isonicotinyl)piperidine-4-one)

Related Child Applications (1)

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JP2023175953A Division JP2024023173A (ja) 2018-01-30 2023-10-11 (1-(3-フルオロ-2(トリフルオロメチル)イソニコチニル)ピぺリジン―4-オン)を作製するためのプロセス及び中間体

Publications (3)

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JP2021512163A JP2021512163A (ja) 2021-05-13
JPWO2019152374A5 true JPWO2019152374A5 (sl) 2022-02-07
JP7393348B2 JP7393348B2 (ja) 2023-12-06

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JP2020562089A Active JP7393348B2 (ja) 2018-01-30 2019-01-29 (1-(3-フルオロ-2(トリフルオロメチル)イソニコチニル)ピぺリジン―4-オン)を作製するためのプロセス及び中間体
JP2023175953A Pending JP2024023173A (ja) 2018-01-30 2023-10-11 (1-(3-フルオロ-2(トリフルオロメチル)イソニコチニル)ピぺリジン―4-オン)を作製するためのプロセス及び中間体

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JP2023175953A Pending JP2024023173A (ja) 2018-01-30 2023-10-11 (1-(3-フルオロ-2(トリフルオロメチル)イソニコチニル)ピぺリジン―4-オン)を作製するためのプロセス及び中間体

Country Status (32)

Country Link
US (1) US10899736B2 (sl)
EP (2) EP4086245A1 (sl)
JP (2) JP7393348B2 (sl)
KR (1) KR20200129099A (sl)
CN (1) CN112105608B (sl)
AR (1) AR114810A1 (sl)
AU (1) AU2019213665B2 (sl)
BR (1) BR112020015470A2 (sl)
CA (1) CA3089832A1 (sl)
CL (1) CL2020001983A1 (sl)
CO (1) CO2020009994A2 (sl)
CR (1) CR20200379A (sl)
DK (1) DK3746429T3 (sl)
EA (1) EA202091830A1 (sl)
ES (1) ES2912469T3 (sl)
HR (1) HRP20220510T1 (sl)
IL (1) IL276302B2 (sl)
LT (1) LT3746429T (sl)
MA (1) MA51771B1 (sl)
MD (1) MD3746429T2 (sl)
MX (1) MX2020007973A (sl)
PE (1) PE20211310A1 (sl)
PH (1) PH12020551145A1 (sl)
PL (1) PL3746429T3 (sl)
PT (1) PT3746429T (sl)
RS (1) RS63312B1 (sl)
SG (1) SG11202007164UA (sl)
SI (1) SI3746429T1 (sl)
TW (1) TWI797242B (sl)
UA (1) UA127488C2 (sl)
WO (1) WO2019152374A1 (sl)
ZA (1) ZA202004692B (sl)

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MA52655A (fr) 2018-03-30 2021-02-17 Incyte Corp Biomarqueurs pour maladie cutanée inflammatoire
US11372003B2 (en) 2018-04-13 2022-06-28 Incyte Corporation Biomarkers for graft-versus-host disease
AU2019374072A1 (en) 2018-10-31 2021-05-27 Incyte Corporation Combination therapy for treatment of hematological diseases
SG11202109563WA (en) 2019-03-05 2021-09-29 Incyte Corp Jak1 pathway inhibitors for the treatment of chronic lung allograft dysfunction
US11992490B2 (en) 2019-10-16 2024-05-28 Incyte Corporation Use of JAK1 inhibitors for the treatment of cutaneous lupus erythematosus and Lichen planus (LP)
CN110683978A (zh) * 2019-10-30 2020-01-14 西安医学院 一种3-腈基亚甲基氮杂环丁烷-1-碳酸叔丁酯的制备方法
IL300555A (en) 2020-08-18 2023-04-01 Incyte Corp Process and intermediates for preparing a JAK inhibitor
PE20231308A1 (es) 2020-08-18 2023-08-24 Incyte Corp Proceso e intermedios para preparar un inhibidor de jak1
KR20230118118A (ko) 2020-12-08 2023-08-10 인사이트 코포레이션 백반증의 치료를 위한 jak1 경로 저해제
CN112625030A (zh) * 2020-12-25 2021-04-09 杭州澳赛诺生物科技有限公司 一种一锅法合成n-保护3-溴代吡唑的合成方法
EP4370504A1 (en) 2021-07-12 2024-05-22 Incyte Corporation Process and intermediates for preparing baricitinib

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