JP2011506330A5 - - Google Patents

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Publication number
JP2011506330A5
JP2011506330A5 JP2010537037A JP2010537037A JP2011506330A5 JP 2011506330 A5 JP2011506330 A5 JP 2011506330A5 JP 2010537037 A JP2010537037 A JP 2010537037A JP 2010537037 A JP2010537037 A JP 2010537037A JP 2011506330 A5 JP2011506330 A5 JP 2011506330A5
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composition
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JP2010537037A
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JP2011506330A (ja
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Priority claimed from PCT/US2008/085456 external-priority patent/WO2009073757A1/en
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Publication of JP2011506330A5 publication Critical patent/JP2011506330A5/ja
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JP2010537037A 2007-12-07 2008-12-04 3−(6−(1−(2,2−ジフルオロベンゾ[d][1,3]ジオキソル−5−イル)シクロプロパンカルボキサミド)−3−メチルピリジン−2−イル)安息香酸の固体状形態 Withdrawn JP2011506330A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US1216207P 2007-12-07 2007-12-07
PCT/US2008/085456 WO2009073757A1 (en) 2007-12-07 2008-12-04 Solid forms of 3-(6-(1-(2,2-difluorobenzo[d][1,3] dioxol-5-yl) cyclopropanecarboxamido)-3-methylpyridin-2-yl) benzoic acid

Related Child Applications (2)

Application Number Title Priority Date Filing Date
JP2013194966A Division JP2013253111A (ja) 2007-12-07 2013-09-20 3−(6−(1−(2,2−ジフルオロベンゾ[d][1,3]ジオキソル−5−イル)シクロプロパンカルボキサミド)−3−メチルピリジン−2−イル)安息香酸の固体状形態
JP2014028062A Division JP2014088447A (ja) 2007-12-07 2014-02-18 3−(6−(1−(2,2−ジフルオロベンゾ[d][1,3]ジオキソル−5−イル)シクロプロパンカルボキサミド)−3−メチルピリジン−2−イル)安息香酸の固体状形態

Publications (2)

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JP2011506330A JP2011506330A (ja) 2011-03-03
JP2011506330A5 true JP2011506330A5 (enExample) 2013-01-10

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ID=40344271

Family Applications (6)

Application Number Title Priority Date Filing Date
JP2010537037A Withdrawn JP2011506330A (ja) 2007-12-07 2008-12-04 3−(6−(1−(2,2−ジフルオロベンゾ[d][1,3]ジオキソル−5−イル)シクロプロパンカルボキサミド)−3−メチルピリジン−2−イル)安息香酸の固体状形態
JP2013194966A Pending JP2013253111A (ja) 2007-12-07 2013-09-20 3−(6−(1−(2,2−ジフルオロベンゾ[d][1,3]ジオキソル−5−イル)シクロプロパンカルボキサミド)−3−メチルピリジン−2−イル)安息香酸の固体状形態
JP2014028062A Pending JP2014088447A (ja) 2007-12-07 2014-02-18 3−(6−(1−(2,2−ジフルオロベンゾ[d][1,3]ジオキソル−5−イル)シクロプロパンカルボキサミド)−3−メチルピリジン−2−イル)安息香酸の固体状形態
JP2015099613A Pending JP2015145426A (ja) 2007-12-07 2015-05-15 3−(6−(1−(2,2−ジフルオロベンゾ[d][1,3]ジオキソル−5−イル)シクロプロパンカルボキサミド)−3−メチルピリジン−2−イル)安息香酸の固体状形態
JP2016207622A Active JP6227741B2 (ja) 2007-12-07 2016-10-24 3−(6−(1−(2,2−ジフルオロベンゾ[d][1,3]ジオキソル−5−イル)シクロプロパンカルボキサミド)−3−メチルピリジン−2−イル)安息香酸の固体状形態
JP2017112429A Pending JP2017149778A (ja) 2007-12-07 2017-06-07 3−(6−(1−(2,2−ジフルオロベンゾ[d][1,3]ジオキソル−5−イル)シクロプロパンカルボキサミド)−3−メチルピリジン−2−イル)安息香酸の固体状形態

Family Applications After (5)

Application Number Title Priority Date Filing Date
JP2013194966A Pending JP2013253111A (ja) 2007-12-07 2013-09-20 3−(6−(1−(2,2−ジフルオロベンゾ[d][1,3]ジオキソル−5−イル)シクロプロパンカルボキサミド)−3−メチルピリジン−2−イル)安息香酸の固体状形態
JP2014028062A Pending JP2014088447A (ja) 2007-12-07 2014-02-18 3−(6−(1−(2,2−ジフルオロベンゾ[d][1,3]ジオキソル−5−イル)シクロプロパンカルボキサミド)−3−メチルピリジン−2−イル)安息香酸の固体状形態
JP2015099613A Pending JP2015145426A (ja) 2007-12-07 2015-05-15 3−(6−(1−(2,2−ジフルオロベンゾ[d][1,3]ジオキソル−5−イル)シクロプロパンカルボキサミド)−3−メチルピリジン−2−イル)安息香酸の固体状形態
JP2016207622A Active JP6227741B2 (ja) 2007-12-07 2016-10-24 3−(6−(1−(2,2−ジフルオロベンゾ[d][1,3]ジオキソル−5−イル)シクロプロパンカルボキサミド)−3−メチルピリジン−2−イル)安息香酸の固体状形態
JP2017112429A Pending JP2017149778A (ja) 2007-12-07 2017-06-07 3−(6−(1−(2,2−ジフルオロベンゾ[d][1,3]ジオキソル−5−イル)シクロプロパンカルボキサミド)−3−メチルピリジン−2−イル)安息香酸の固体状形態

Country Status (28)

Country Link
US (8) US8507534B2 (enExample)
EP (3) EP3683218B1 (enExample)
JP (6) JP2011506330A (enExample)
KR (3) KR20100101130A (enExample)
CN (2) CN103626744B (enExample)
AU (1) AU2008333845C1 (enExample)
BR (1) BRPI0821039B8 (enExample)
CA (2) CA2706920C (enExample)
CL (1) CL2010000607A1 (enExample)
CY (3) CY1118630T1 (enExample)
DK (2) DK2225230T3 (enExample)
EA (1) EA201070698A1 (enExample)
ES (3) ES2790830T3 (enExample)
HR (2) HRP20170241T2 (enExample)
HU (3) HUE049642T2 (enExample)
IL (2) IL206203A (enExample)
LT (3) LT2225230T (enExample)
MX (2) MX367154B (enExample)
NO (2) NO2017009I2 (enExample)
NZ (4) NZ614151A (enExample)
PL (2) PL3170818T3 (enExample)
PT (2) PT3170818T (enExample)
RS (2) RS55559B1 (enExample)
SG (1) SG186638A1 (enExample)
SI (2) SI3170818T1 (enExample)
UA (1) UA102534C2 (enExample)
WO (1) WO2009073757A1 (enExample)
ZA (1) ZA201003623B (enExample)

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US20100074949A1 (en) 2008-08-13 2010-03-25 William Rowe Pharmaceutical composition and administration thereof
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BRPI0919550A2 (pt) 2008-09-29 2019-09-10 Vertex Pharma unidades de dosagem de ácido 3-(6-(1-(2,2-difluorobenzo]d][1,3]dioxol-5-il)ciclopropanocarboxamido)-3-metilpiridin-2-il)benzoico
SI2349263T1 (sl) * 2008-10-23 2014-09-30 Vertex Pharmaceuticals Incorporated Modulatorji cistiäśno-fibroznega transmembranskega regulatorja prevodnosti
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MA51039A (fr) 2017-12-08 2020-10-14 Vertex Pharma Procédés pour préparer des modulateurs du régulateur de la conductance transmembranaire de la mucoviscidose
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SI3752510T1 (sl) 2018-02-15 2023-03-31 Vertex Pharmaceuticals Incorporated Makrocikli kot modulatorji regulatorja transmembranske prevodnosti pri cistični fibrozi, farmacevtski sestavki iz le-teh, njihova uporaba pri zdravljenju cistične fibroze in postopek za njihovo proizvodnjo
EP3774825A1 (en) 2018-04-13 2021-02-17 Vertex Pharmaceuticals Incorporated Modulators of cystic fibrosis transmembrane conductance regulator, pharmaceutical compositions, methods of treatment, and process for making the modulator
AR118555A1 (es) 2019-04-03 2021-10-20 Vertex Pharma Agentes moduladores del regulador de la conductancia transmembrana de la fibrosis quística
WO2020214921A1 (en) 2019-04-17 2020-10-22 Vertex Pharmaceuticals Incorporated Solid forms of modulators of cftr
TWI867024B (zh) 2019-08-14 2024-12-21 美商維泰克斯製藥公司 囊腫纖維化跨膜傳導調節蛋白之調節劑
CA3150162A1 (en) 2019-08-14 2021-02-18 Vertex Pharmaceuticals Incorporated Crystalline forms of cftr modulators
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BR112022002606A2 (pt) 2019-08-14 2022-05-03 Vertex Pharma Moduladores do regulador de condutância transmembrana da fibrose cística
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CR20230120A (es) 2020-08-07 2023-09-01 Vertex Pharma Moduladores del regulador de la conductancia transmembrana de la fibrosis quística
US20230277550A1 (en) 2020-08-20 2023-09-07 The Board Of Trustees Of The Leland Stanford Junior University Methods for Treating Respiratory Diseases Characterized by Mucus Hypersecretion
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