JP2009084270A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2009084270A5 JP2009084270A5 JP2008225403A JP2008225403A JP2009084270A5 JP 2009084270 A5 JP2009084270 A5 JP 2009084270A5 JP 2008225403 A JP2008225403 A JP 2008225403A JP 2008225403 A JP2008225403 A JP 2008225403A JP 2009084270 A5 JP2009084270 A5 JP 2009084270A5
- Authority
- JP
- Japan
- Prior art keywords
- xinafoate
- xinafoate salt
- disease
- indicated
- dry powder
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US97003007P | 2007-09-05 | 2007-09-05 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2009084270A JP2009084270A (ja) | 2009-04-23 |
| JP2009084270A5 true JP2009084270A5 (enExample) | 2011-10-06 |
Family
ID=40293576
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008225403A Pending JP2009084270A (ja) | 2007-09-05 | 2008-09-03 | 塩形態 |
Country Status (17)
| Country | Link |
|---|---|
| US (3) | US8193181B2 (enExample) |
| EP (1) | EP2215087B1 (enExample) |
| JP (1) | JP2009084270A (enExample) |
| KR (2) | KR20120120453A (enExample) |
| CN (1) | CN101861314B (enExample) |
| AR (1) | AR068369A1 (enExample) |
| AU (1) | AU2008294473B2 (enExample) |
| BR (1) | BRPI0816278A2 (enExample) |
| CA (1) | CA2697495C (enExample) |
| ES (1) | ES2452965T3 (enExample) |
| IL (1) | IL203973A (enExample) |
| MX (1) | MX2010002518A (enExample) |
| NZ (1) | NZ583582A (enExample) |
| RU (1) | RU2458925C2 (enExample) |
| TW (1) | TWI371277B (enExample) |
| WO (1) | WO2009031011A2 (enExample) |
| ZA (1) | ZA201002356B (enExample) |
Families Citing this family (29)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5913093B2 (ja) | 2009-05-21 | 2016-04-27 | アストラゼネカ アクチボラグ | 新規ピリミジン誘導体と、癌とさらなる疾患の治療におけるそれらの使用 |
| GB0908772D0 (en) * | 2009-05-21 | 2009-07-01 | Astrazeneca Ab | New salts 756 |
| WO2012154518A1 (en) | 2011-05-10 | 2012-11-15 | Merck Sharp & Dohme Corp. | Bipyridylaminopyridines as syk inhibitors |
| JP2014513687A (ja) | 2011-05-10 | 2014-06-05 | メルク・シャープ・アンド・ドーム・コーポレーション | Ｓｙｋ阻害薬としてのピリジルアミノピリジン |
| EP2706853B1 (en) | 2011-05-10 | 2017-06-14 | Merck Sharp & Dohme Corp. | Aminopyrimidines as syk inhibitors |
| US8987456B2 (en) | 2011-10-05 | 2015-03-24 | Merck Sharp & Dohme Corp. | 3-pyridyl carboxamide-containing spleen tyrosine kinase (SYK) inhibitors |
| EP2763976B1 (en) | 2011-10-05 | 2016-05-18 | Merck Sharp & Dohme Corp. | 2-pyridyl carboxamide-containing spleen tyrosine kinase (syk) inhibitors |
| WO2013052391A1 (en) | 2011-10-05 | 2013-04-11 | Merck Sharp & Dohme Corp. | PHENYL CARBOXAMIDE-CONTAINING SPLEEN TYROSINE KINASE (Syk) INHIBITORS |
| EP2768480A1 (en) * | 2011-10-21 | 2014-08-27 | Rigel Pharmaceuticals, Inc. | Method and device for administering xinafoate salt of n4-(2,2-difluoro-4h-benzo [1,4]oxazin-3-one) -6-yl]-5-fluoro-n2- [3- (methylaminocarbonylmethyleneoxy) phenyl]2,4-pyrimidinediamine |
| WO2013192128A1 (en) | 2012-06-20 | 2013-12-27 | Merck Sharp & Dohme Corp. | Imidazolyl analogs as syk inhibitors |
| US9242984B2 (en) | 2012-06-20 | 2016-01-26 | Merck Sharp & Dohme Corp. | Pyrazolyl derivatives as Syk inhibitors |
| EP2863916B1 (en) | 2012-06-22 | 2018-07-18 | Merck Sharp & Dohme Corp. | Substituted pyridine spleen tyrosine kinase (syk) inhibitors |
| WO2013192088A1 (en) | 2012-06-22 | 2013-12-27 | Merck Sharp & Dohme Corp. | SUBSTITUTED DIAZINE AND TRIAZINE SPLEEN TYROSINE KINASE (Syk) INHIBITORS |
| WO2014031438A2 (en) | 2012-08-20 | 2014-02-27 | Merck Sharp & Dohme Corp. | SUBSTITUTED PHENYL SPLEEN TYROSINE KINASE (Syk) INHIBITORS |
| EP2900665B1 (en) | 2012-09-28 | 2018-01-03 | Merck Sharp & Dohme Corp. | Triazolyl derivatives as syk inhibitors |
| US9624210B2 (en) | 2012-12-12 | 2017-04-18 | Merck Sharp & Dohme Corp. | Amino-pyrimidine-containing spleen tyrosine kinase (Syk) inhibitors |
| EP2934525B1 (en) | 2012-12-21 | 2019-05-08 | Merck Sharp & Dohme Corp. | Thiazole-substituted aminopyridines as spleen tyrosine kinase inhibitors |
| JP6649246B2 (ja) * | 2013-03-14 | 2020-02-19 | アラーガン、インコーポレイテッドＡｌｌｅｒｇａｎ，Ｉｎｃｏｒｐｏｒａｔｅｄ | タンパク質の徐放性送達の組成物及び製造プロセス中のタンパク質の安定化方法 |
| EP2988744A4 (en) | 2013-04-26 | 2016-11-02 | Merck Sharp & Dohme | THIAZOLSUBSTITUTED AMINOHETEROARYLE AS MILZTYROSINKINASE INHIBITOR |
| EP2988749B1 (en) | 2013-04-26 | 2019-08-14 | Merck Sharp & Dohme Corp. | Thiazole-substituted aminopyrimidines as spleen tyrosine kinase inhibitors |
| WO2015094997A1 (en) | 2013-12-20 | 2015-06-25 | Merck Sharp & Dohme Corp. | Thiazole-substituted aminoheteroaryls as spleen tyrosine kinase inhibitors |
| US9670196B2 (en) | 2013-12-20 | 2017-06-06 | Merck Sharp & Dohme Corp. | Thiazole-substituted aminoheteroaryls as Spleen Tyrosine Kinase inhibitors |
| EP3083559B1 (en) | 2013-12-20 | 2021-03-10 | Merck Sharp & Dohme Corp. | Thiazole-substituted aminoheteroaryls as spleen tyrosine kinase inhibitors |
| EP3116506B1 (en) | 2014-03-13 | 2019-04-17 | Merck Sharp & Dohme Corp. | 2-pyrazine carboxamides as spleen tyrosine kinase inhibitors |
| WO2018189566A1 (en) * | 2017-04-10 | 2018-10-18 | Dorian Bevec | Use of a chemical compound as a therapeutic agent |
| CA3105585A1 (en) * | 2018-07-18 | 2020-01-23 | Astrazeneca Ab | A xinafoate salt of a jak inhibiting compound |
| BR112021018168B1 (pt) | 2019-03-21 | 2023-11-28 | Onxeo | Composição farmacêutica, combinação e kit compreendendo uma molécula dbait e um inibidor de quinase para o tratamento de câncer |
| CA3159348A1 (en) | 2019-11-08 | 2021-05-14 | Inserm (Institut National De La Sante Et De La Recherche Medicale) | Methods for the treatment of cancers that have acquired resistance to kinase inhibitors |
| WO2021148581A1 (en) | 2020-01-22 | 2021-07-29 | Onxeo | Novel dbait molecule and its use |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5376645A (en) | 1990-01-23 | 1994-12-27 | University Of Kansas | Derivatives of cyclodextrins exhibiting enhanced aqueous solubility and the use thereof |
| KR0166088B1 (ko) | 1990-01-23 | 1999-01-15 | . | 수용해도가 증가된 시클로덱스트린 유도체 및 이의 용도 |
| GB9711643D0 (en) | 1997-06-05 | 1997-07-30 | Janssen Pharmaceutica Nv | Glass thermoplastic systems |
| GB9808802D0 (en) | 1998-04-24 | 1998-06-24 | Glaxo Group Ltd | Pharmaceutical formulations |
| TWI329105B (en) | 2002-02-01 | 2010-08-21 | Rigel Pharmaceuticals Inc | 2,4-pyrimidinediamine compounds and their uses |
| GB0208609D0 (en) * | 2002-04-13 | 2002-05-22 | Glaxo Group Ltd | Compositions |
| EP1546120A4 (en) * | 2002-10-04 | 2006-11-22 | Pharmacia Corp | PHARMACEUTICAL COMPOSITIONS FOR THE TREATMENT OF PARKINSON'S DISEASE |
| JP4886511B2 (ja) * | 2003-07-30 | 2012-02-29 | ライジェル ファーマシューティカルズ， インコーポレイテッド | ２，４−ピリミジンジアミン化合物による自己免疫疾患の治療または予防方法 |
| EP1896026B1 (en) * | 2005-06-15 | 2013-10-09 | Boehringer Ingelheim International GmbH | Process for preparing tiotropium salts, tiotropium salts as such and pharmaceutical compositions thereof |
| BRPI0713951B8 (pt) * | 2006-06-30 | 2021-05-25 | Novartis Ag | derivados de quinazolina, e composição farmacêutica |
-
2008
- 2008-08-27 ES ES08806983.6T patent/ES2452965T3/es active Active
- 2008-08-27 CN CN200880105757XA patent/CN101861314B/zh not_active Expired - Fee Related
- 2008-08-27 BR BRPI0816278A patent/BRPI0816278A2/pt not_active Application Discontinuation
- 2008-08-27 NZ NZ583582A patent/NZ583582A/en not_active IP Right Cessation
- 2008-08-27 KR KR1020127024371A patent/KR20120120453A/ko not_active Withdrawn
- 2008-08-27 RU RU2010108162/04A patent/RU2458925C2/ru active
- 2008-08-27 CA CA2697495A patent/CA2697495C/en not_active Expired - Fee Related
- 2008-08-27 AU AU2008294473A patent/AU2008294473B2/en not_active Ceased
- 2008-08-27 US US12/676,075 patent/US8193181B2/en not_active Expired - Fee Related
- 2008-08-27 WO PCT/IB2008/002288 patent/WO2009031011A2/en not_active Ceased
- 2008-08-27 EP EP08806983.6A patent/EP2215087B1/en not_active Not-in-force
- 2008-08-27 MX MX2010002518A patent/MX2010002518A/es active IP Right Grant
- 2008-08-27 KR KR1020107007283A patent/KR101225233B1/ko not_active Expired - Fee Related
- 2008-09-03 JP JP2008225403A patent/JP2009084270A/ja active Pending
- 2008-09-04 AR ARP080103848A patent/AR068369A1/es unknown
- 2008-09-04 TW TW097133970A patent/TWI371277B/zh not_active IP Right Cessation
-
2010
- 2010-02-15 IL IL203973A patent/IL203973A/en active IP Right Grant
- 2010-04-01 ZA ZA2010/02356A patent/ZA201002356B/en unknown
-
2012
- 2012-05-09 US US13/467,850 patent/US8486935B2/en not_active Expired - Fee Related
-
2013
- 2013-06-18 US US13/920,434 patent/US20130281446A1/en not_active Abandoned
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2009084270A5 (enExample) | ||
| CA2697495A1 (en) | Xinafoate salt of n4-[(2,2-difluoro-4h-benzo[1,4]oxazin-3-one)-6-yl]-5-fluoro-n2-[3-(methylaminocarbonylmethyleneoxy)phenyl]-2,4-pyrimidinediamine | |
| AU2014219283C1 (en) | Benzothiophene derivatives and compositions thereof as selective estrogen receptor degraders | |
| CN101260112B (zh) | 含噻吩并[3.2-c]吡啶的乙酰肼衍生物及其制备方法和用途 | |
| ES2437346T3 (es) | Procedimiento para la producción de derivado de diamina | |
| TW200528097A (en) | Novel thiazolidin-4-one derivatives | |
| JP2019510787A5 (enExample) | ||
| JP2006517572A5 (enExample) | ||
| CN104039765B (zh) | 多奈哌齐双羟萘酸盐、制备方法及其应用 | |
| KR101823451B1 (ko) | 퀴논계 화합물, 이의 광학 이성질체 및 이의 제조 방법과 의약 용도 | |
| JP2017538676A (ja) | ミトコンドリア透過性遷移孔（ｍｔＰＴＰ）の小分子阻害剤 | |
| CN103102348B (zh) | 噁二唑类化合物及其制备方法、药物组合物及其用途 | |
| JP2015508092A5 (enExample) | ||
| BRPI0612266A2 (pt) | composição fermacêutica, e, uso da mesma | |
| JP2007522162A5 (enExample) | ||
| WO2010103312A1 (en) | Hydroxymorpholiness and their use for the treatment of inflammatory disorders and pain | |
| CN116947756B (zh) | 环丁烯二酮基喹啉类化合物及其制备方法、药物组合物和应用 | |
| HU229137B1 (en) | 8,8a-dihydro-indeno[1,2-d]thiazole derivatives having sulphoneamid- or sulphone substitutents in the 2 position, method for production thereof and use thereof as a medicament | |
| TWI423972B (zh) | 治療呼吸系融合細胞病毒感染之多環劑 | |
| KR20140003379A (ko) | 스핑고신 1-포스페이트(ｓ１ｐ) 수용체들에 대한 리간드들로서의 5-(바이페닐-4-일)-3-페닐-1,2,4-옥사디아졸릴 유도체들 | |
| JP2007518798A5 (enExample) | ||
| EP1844017A1 (en) | An amorphous and three crystalline forms of rimonabant hydrochloride | |
| JP2008520611A5 (enExample) | ||
| CN107207407B (zh) | 用于治疗疾病和病症的组合物和方法 | |
| JP2015504913A (ja) | 安定な非晶質のラルテグラビルカリウムプレミックス、及び、その調製方法 |