IL143091A0 - N-substituted 2-cyanopyrrolidines - Google Patents

N-substituted 2-cyanopyrrolidines

Info

Publication number
IL143091A0
IL143091A0 IL14309199A IL14309199A IL143091A0 IL 143091 A0 IL143091 A0 IL 143091A0 IL 14309199 A IL14309199 A IL 14309199A IL 14309199 A IL14309199 A IL 14309199A IL 143091 A0 IL143091 A0 IL 143091A0
Authority
IL
Israel
Prior art keywords
cyanopyrrolidines
substituted
Prior art date
Application number
IL14309199A
Other languages
English (en)
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22777194&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL143091(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of IL143091A0 publication Critical patent/IL143091A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IL14309199A 1998-12-10 1999-12-09 N-substituted 2-cyanopyrrolidines IL143091A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US20906898A 1998-12-10 1998-12-10
PCT/EP1999/009708 WO2000034241A1 (en) 1998-12-10 1999-12-09 N-substituted 2-cyanopyrrolidines

Publications (1)

Publication Number Publication Date
IL143091A0 true IL143091A0 (en) 2002-04-21

Family

ID=22777194

Family Applications (2)

Application Number Title Priority Date Filing Date
IL14309199A IL143091A0 (en) 1998-12-10 1999-12-09 N-substituted 2-cyanopyrrolidines
IL143091A IL143091A (en) 1998-12-10 2001-05-10 N-substituted 2-cyanopyrrolidines, pharmaceutical compositions comprising them and use thereof in the preparation of medicaments for treating conditions mediated by dpp-iv inhibition

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL143091A IL143091A (en) 1998-12-10 2001-05-10 N-substituted 2-cyanopyrrolidines, pharmaceutical compositions comprising them and use thereof in the preparation of medicaments for treating conditions mediated by dpp-iv inhibition

Country Status (34)

Country Link
US (1) US6166063A (fa)
EP (1) EP1137635B1 (fa)
JP (2) JP3681110B2 (fa)
KR (2) KR20050047561A (fa)
CN (1) CN1160330C (fa)
AR (1) AR023719A1 (fa)
AT (1) ATE307112T1 (fa)
BR (1) BRPI9915985B8 (fa)
CA (1) CA2350609C (fa)
CO (1) CO5150173A1 (fa)
CY (3) CY1105355T1 (fa)
CZ (1) CZ299151B6 (fa)
DE (3) DE69927844T2 (fa)
DK (1) DK1137635T3 (fa)
ES (1) ES2251847T3 (fa)
FR (1) FR08C0005I2 (fa)
HK (1) HK1040394B (fa)
HU (1) HU226769B1 (fa)
ID (1) ID28796A (fa)
IL (2) IL143091A0 (fa)
LU (2) LU91409I2 (fa)
MY (1) MY123244A (fa)
NL (2) NL300333I2 (fa)
NO (3) NO318741B1 (fa)
NZ (1) NZ511935A (fa)
PE (1) PE20001317A1 (fa)
PL (1) PL199443B1 (fa)
RU (1) RU2251544C2 (fa)
SK (1) SK286635B6 (fa)
TR (1) TR200101478T2 (fa)
TW (1) TW509674B (fa)
UY (1) UY25843A1 (fa)
WO (1) WO2000034241A1 (fa)
ZA (1) ZA200104581B (fa)

Families Citing this family (309)

* Cited by examiner, † Cited by third party
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