AU777701B2 - Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use - Google Patents

Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use Download PDF

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Publication number
AU777701B2
AU777701B2 AU57852/00A AU5785200A AU777701B2 AU 777701 B2 AU777701 B2 AU 777701B2 AU 57852/00 A AU57852/00 A AU 57852/00A AU 5785200 A AU5785200 A AU 5785200A AU 777701 B2 AU777701 B2 AU 777701B2
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Australia
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found
calc
indazole
nmr
mmol
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Expired, expires
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AU57852/00A
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AU5785200A (en
Inventor
Steven Lee Bender
Allen J. Borchardt
John F. Braganza
Michael Raymond Collins
Stephan James Cripps
Ye Hua
Michael David Johnson
Theodore Otto Johnson Jr.
Robert Steven Kania
Hiep The Luu
Cynthia Louise Palmer
Siegfried Heinz Reich
Anna Maria Tempczyk-Russell
Min Teng
Christine Thomas
Michael David Varney
Michael Brennan Wallace
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Agouron Pharmaceuticals LLC
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Agouron Pharmaceuticals LLC
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Application filed by Agouron Pharmaceuticals LLC filed Critical Agouron Pharmaceuticals LLC
Publication of AU5785200A publication Critical patent/AU5785200A/en
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    • C07D209/04—Indoles; Hydrogenated indoles
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Diabetes (AREA)
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  • Cardiology (AREA)
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  • Dermatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
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  • Obesity (AREA)
  • Pain & Pain Management (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Vascular Medicine (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AU57852/00A 1999-07-02 2000-06-30 Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use Expired AU777701B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US14213099P 1999-07-02 1999-07-02
US60/142130 1999-07-02
PCT/US2000/018263 WO2001002369A2 (en) 1999-07-02 2000-06-30 Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use

Publications (2)

Publication Number Publication Date
AU5785200A AU5785200A (en) 2001-01-22
AU777701B2 true AU777701B2 (en) 2004-10-28

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AU57852/00A Expired AU777701B2 (en) 1999-07-02 2000-06-30 Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use

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JP (2) JP3878849B2 (enExample)
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BE (1) BE2013C015I2 (enExample)
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PE20010306A1 (es) * 1999-07-02 2001-03-29 Agouron Pharma Compuestos de indazol y composiciones farmaceuticas que los contienen utiles para la inhibicion de proteina kinasa
WO2001047922A2 (en) 1999-12-24 2001-07-05 Aventis Pharma Limited Azaindoles
AU2001229727B2 (en) 2000-02-07 2004-10-14 Bristol-Myers Squibb Co. 3-aminopyrazole inhibitors of cyclin dependent kinases
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ATE287886T1 (de) 2000-04-25 2005-02-15 Bristol Myers Squibb Co Verwendung von 5-thio, sulfinyl- und sulfonylpyrazolo 3,4-b) pyridinen als cyclin- abhängige kinase-hemmer
AU7652101A (en) 2000-08-09 2002-02-18 Astrazeneca Ab Cinnoline compounds
BR0113056A (pt) 2000-08-09 2003-07-08 Astrazeneca Ab Composto, processo papa a preparação do mesmo, composição farmacêutica, e, método para produzir um efeito antiangiogênico e/ou redutor da permeabilidade vascular em um animal de sangue quente, e, uso de um composto
ES2334641T3 (es) 2000-09-01 2010-03-15 Novartis Vaccines And Diagnostics, Inc. Derivados aza heterociclicos y su uso terapeutico.
NZ524717A (en) 2000-09-11 2004-09-24 Chiron Corp Quinolinone derivatives
HU230302B1 (hu) 2000-10-20 2015-12-28 Eisai R&D Management Co., Ltd. Nitrogéntartalmú aromás származékok és ezeket tartalmazó gyógyászati készítmények
TWI243164B (en) 2001-02-13 2005-11-11 Aventis Pharma Gmbh Acylated indanyl amines and their use as pharmaceuticals
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