DE602008003055D1 - Zyklokondensierte Azaindole, die als Kinase-Hemmer wirken - Google Patents
Zyklokondensierte Azaindole, die als Kinase-Hemmer wirkenInfo
- Publication number
- DE602008003055D1 DE602008003055D1 DE602008003055T DE602008003055T DE602008003055D1 DE 602008003055 D1 DE602008003055 D1 DE 602008003055D1 DE 602008003055 T DE602008003055 T DE 602008003055T DE 602008003055 T DE602008003055 T DE 602008003055T DE 602008003055 D1 DE602008003055 D1 DE 602008003055D1
- Authority
- DE
- Germany
- Prior art keywords
- cyclocondensed
- azaindoles
- act
- kinase inhibitors
- kinase
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Active
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/06—Peri-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/16—Peri-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP07109338 | 2007-05-31 |
Publications (1)
Publication Number | Publication Date |
---|---|
DE602008003055D1 true DE602008003055D1 (de) | 2010-12-02 |
Family
ID=39731692
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE602008003055T Active DE602008003055D1 (de) | 2007-05-31 | 2008-05-14 | Zyklokondensierte Azaindole, die als Kinase-Hemmer wirken |
Country Status (2)
Country | Link |
---|---|
EP (1) | EP2002836B1 (de) |
DE (1) | DE602008003055D1 (de) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2010114905A1 (en) * | 2009-03-31 | 2010-10-07 | Arqule, Inc. | Peri-fused pyrazolo-pyrimidine compounds |
PL2440558T3 (pl) | 2009-06-08 | 2015-10-30 | Takeda Pharmaceuticals Co | Związki dihydropirolonaftyrydynony jako inhibitory JAK |
AU2014360455B2 (en) * | 2013-12-06 | 2018-05-10 | Genentech, Inc. | Serine/threonine kinase inhibitors |
KR102351270B1 (ko) * | 2016-06-16 | 2022-01-14 | 하얼빈 젠바오 파마슈티컬 컴퍼니, 리미티드 | Akt 억제제인 디히드로피라졸로아제핀계 화합물 |
FR3067349B1 (fr) | 2017-06-12 | 2020-12-04 | Cisbio Bioassays | Nouveaux agents mono et di-antennes complexants hydrosolubles et complexes de lanthanide correspondants |
FR3067712B1 (fr) | 2017-06-14 | 2019-08-02 | Cisbio Bioassays | Nouveaux agents complexants de type trimethoxyphenyl pyridine hydrosolubles et complexes de lanthanide correspondants |
JP6906105B2 (ja) * | 2017-06-16 | 2021-07-21 | 成都先導薬物開発股▲ふん▼有限公司Hitgen Ltd. | Rockを阻害する化合物及びその使用 |
PT3725791T (pt) * | 2017-12-13 | 2023-04-04 | Harbin Zhenbao Pharmaceutical Co Ltd | Sal que serve como inibidor de akt e seu cristal |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PE20010306A1 (es) | 1999-07-02 | 2001-03-29 | Agouron Pharma | Compuestos de indazol y composiciones farmaceuticas que los contienen utiles para la inhibicion de proteina kinasa |
US6335342B1 (en) | 2000-06-19 | 2002-01-01 | Pharmacia & Upjohn S.P.A. | Azaindole derivatives, process for their preparation, and their use as antitumor agents |
GB0117395D0 (en) * | 2001-07-17 | 2001-09-05 | Glaxo Group Ltd | Chemical compounds |
EP1452525A4 (de) | 2001-10-30 | 2005-01-26 | Nippon Shinyaku Co Ltd | Amidderivate und arzneimittel |
GB0330042D0 (en) * | 2003-12-24 | 2004-01-28 | Pharmacia Italia Spa | Pyrrolo [2,3-b] pyridine derivatives active as kinase inhibitors process for their preparation and pharmaceutical compositions them |
US20080015212A1 (en) * | 2004-12-02 | 2008-01-17 | Barnett Stanley F | Inhibitors Of Akt Activity |
US7579356B2 (en) * | 2005-05-04 | 2009-08-25 | Janssen Pharmaceutica Nv | Thia-tetraazaacenaphthylene kinase inhibitors |
-
2008
- 2008-05-14 EP EP08156203A patent/EP2002836B1/de not_active Not-in-force
- 2008-05-14 DE DE602008003055T patent/DE602008003055D1/de active Active
Also Published As
Publication number | Publication date |
---|---|
EP2002836B1 (de) | 2010-10-20 |
EP2002836A1 (de) | 2008-12-17 |
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