MX2021012250A - Formas solidas de (e)-3-[2-(2-tienil)vinil]-1h-pirazol. - Google Patents

Formas solidas de (e)-3-[2-(2-tienil)vinil]-1h-pirazol.

Info

Publication number
MX2021012250A
MX2021012250A MX2021012250A MX2021012250A MX2021012250A MX 2021012250 A MX2021012250 A MX 2021012250A MX 2021012250 A MX2021012250 A MX 2021012250A MX 2021012250 A MX2021012250 A MX 2021012250A MX 2021012250 A MX2021012250 A MX 2021012250A
Authority
MX
Mexico
Prior art keywords
pyrazole
thienyl
vinyl
solid forms
compositions
Prior art date
Application number
MX2021012250A
Other languages
English (en)
Inventor
An-Hu Li
Satish Kumar Sakilam
Dong Sung Lim
Original Assignee
Angion Biomedica Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Angion Biomedica Corp filed Critical Angion Biomedica Corp
Publication of MX2021012250A publication Critical patent/MX2021012250A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/4155—1,2-Diazoles non condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

La presente descripción proporciona formas sólidas de (E)-3-[2-(2-tienil)vinil]-1H-pirazol, composiciones de las mismas, y métodos de preparación y uso de las mismas.
MX2021012250A 2019-04-11 2020-04-10 Formas solidas de (e)-3-[2-(2-tienil)vinil]-1h-pirazol. MX2021012250A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201962832519P 2019-04-11 2019-04-11
PCT/US2020/027710 WO2020210657A1 (en) 2019-04-11 2020-04-10 Solid forms of (e)-3-[2-(2-thienyl)vinyl]-1h-pyrazole

Publications (1)

Publication Number Publication Date
MX2021012250A true MX2021012250A (es) 2022-01-18

Family

ID=72751396

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2021012250A MX2021012250A (es) 2019-04-11 2020-04-10 Formas solidas de (e)-3-[2-(2-tienil)vinil]-1h-pirazol.

Country Status (13)

Country Link
US (2) US10875849B2 (es)
EP (1) EP3927702A4 (es)
JP (1) JP2022526827A (es)
KR (1) KR20220004083A (es)
CN (1) CN114026085A (es)
AU (1) AU2020272036A1 (es)
BR (1) BR112021020367A2 (es)
CA (1) CA3133803A1 (es)
EA (1) EA202192786A1 (es)
IL (1) IL287118A (es)
MX (1) MX2021012250A (es)
SG (1) SG11202110406SA (es)
WO (1) WO2020210657A1 (es)

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SG11202110406SA (en) 2019-04-11 2021-10-28 Angion Biomedica Corp Solid forms of (e)-3-[2-(2-thienyl)vinyl]-1h-pyrazole
US20230000828A1 (en) * 2019-10-31 2023-01-05 Angion Biomedica Corp. Improving renal function after kidney transplantation
US11358963B2 (en) 2020-03-05 2022-06-14 Ankh Life Sciences Limited Low-temperature synthesis of thymoquinone and harmaline compounds
EP4228626A2 (en) * 2020-10-14 2023-08-23 Angion Biomedica Corp. Preparation of terevalefim and formulations thereof

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Also Published As

Publication number Publication date
US20210078984A1 (en) 2021-03-18
JP2022526827A (ja) 2022-05-26
US10875849B2 (en) 2020-12-29
EP3927702A1 (en) 2021-12-29
CN114026085A (zh) 2022-02-08
EA202192786A1 (ru) 2022-01-11
BR112021020367A2 (pt) 2021-12-07
SG11202110406SA (en) 2021-10-28
IL287118A (en) 2021-12-01
KR20220004083A (ko) 2022-01-11
CA3133803A1 (en) 2020-10-15
WO2020210657A1 (en) 2020-10-15
EP3927702A4 (en) 2022-05-11
AU2020272036A1 (en) 2021-11-04
US20200369654A1 (en) 2020-11-26
US11370783B2 (en) 2022-06-28

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