KR20090125814A - 3-시아노-4-(4-테트라하이드로피란-페닐)-피리딘-2-온 유도체 - Google Patents
3-시아노-4-(4-테트라하이드로피란-페닐)-피리딘-2-온 유도체 Download PDFInfo
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- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
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| WOPCT/EP/2007/052442 | 2007-03-15 | ||
| EP07116403 | 2007-09-14 | ||
| EP07116403.2 | 2007-09-14 |
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| JO3368B1 (ar) | 2013-06-04 | 2019-03-13 | Janssen Pharmaceutica Nv | مركبات 6، 7- ثاني هيدرو بيرازولو [5،1-a] بيرازين- 4 (5 يد)- اون واستخدامها بصفة منظمات تفارغية سلبية لمستقبلات ميجلور 2 |
| DK3013813T3 (da) | 2013-06-27 | 2019-06-03 | Pfizer | Heteroaromatiske forbindelser og anvendelse deraf som dopamin-d1-ligander |
| JO3367B1 (ar) | 2013-09-06 | 2019-03-13 | Janssen Pharmaceutica Nv | مركبات 2،1، 4- ثلاثي زولو [3،4-a] بيريدين واستخدامها بصفة منظمات تفارغية موجبة لمستقبلات ميجلور 2 |
| PT3096790T (pt) | 2014-01-21 | 2019-10-15 | Janssen Pharmaceutica Nv | Combinações compreendendo moduladores alostéricos positivos ou agonistas ortostéricos do recetor glutamatérgico metabotrópico do subtipo 2 e seu uso |
| EA202192105A3 (ru) | 2014-02-04 | 2022-02-28 | Янссен Фармацевтика Нв | Комбинации, содержащие положительные аллостерические модуляторы или ортостерические агонисты метаботропного глутаматергического рецептора 2 подтипа, и их применение |
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-
2008
- 2008-03-06 TW TW097107754A patent/TW200845978A/zh unknown
- 2008-03-07 CA CA2680104A patent/CA2680104C/en not_active Expired - Fee Related
- 2008-03-07 EP EP08717515A patent/EP2134708B1/en active Active
- 2008-03-07 PL PL08717515T patent/PL2134708T3/pl unknown
- 2008-03-07 AR ARP080100961A patent/AR065654A1/es not_active Application Discontinuation
- 2008-03-07 KR KR1020097020927A patent/KR20090125814A/ko not_active Withdrawn
- 2008-03-07 JP JP2009552216A patent/JP5357061B2/ja not_active Expired - Fee Related
- 2008-03-07 AT AT08717515T patent/ATE509020T1/de active
- 2008-03-07 DK DK08717515.4T patent/DK2134708T3/da active
- 2008-03-07 US US12/529,568 patent/US8906939B2/en not_active Expired - Fee Related
- 2008-03-07 EA EA200901160A patent/EA017294B1/ru not_active IP Right Cessation
- 2008-03-07 AU AU2008223796A patent/AU2008223796B2/en not_active Ceased
- 2008-03-07 WO PCT/EP2008/052768 patent/WO2008107481A1/en not_active Ceased
- 2008-03-07 CN CN2008800073170A patent/CN101711244B/zh not_active Expired - Fee Related
- 2008-03-07 MX MX2009009424A patent/MX2009009424A/es active IP Right Grant
- 2008-03-07 BR BRPI0808509-9A patent/BRPI0808509A2/pt not_active IP Right Cessation
- 2008-03-07 NZ NZ579988A patent/NZ579988A/en not_active IP Right Cessation
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Also Published As
| Publication number | Publication date |
|---|---|
| WO2008107481A8 (en) | 2008-12-24 |
| EA017294B1 (ru) | 2012-11-30 |
| US8906939B2 (en) | 2014-12-09 |
| AU2008223796A1 (en) | 2008-09-12 |
| MX2009009424A (es) | 2010-02-09 |
| JP5357061B2 (ja) | 2013-12-04 |
| IL200329A0 (en) | 2010-04-29 |
| TW200845978A (en) | 2008-12-01 |
| EP2134708A1 (en) | 2009-12-23 |
| BRPI0808509A2 (pt) | 2014-08-19 |
| PL2134708T3 (pl) | 2011-10-31 |
| AR065654A1 (es) | 2009-06-24 |
| AU2008223796B2 (en) | 2011-03-17 |
| CA2680104A1 (en) | 2008-09-12 |
| CN101711244B (zh) | 2013-01-16 |
| CA2680104C (en) | 2016-05-31 |
| WO2008107481A1 (en) | 2008-09-12 |
| DK2134708T3 (da) | 2011-08-29 |
| NZ579988A (en) | 2011-09-30 |
| JP2010520265A (ja) | 2010-06-10 |
| EP2134708B1 (en) | 2011-05-11 |
| EA200901160A1 (ru) | 2010-04-30 |
| CN101711244A (zh) | 2010-05-19 |
| ATE509020T1 (de) | 2011-05-15 |
| US20100087487A1 (en) | 2010-04-08 |
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