JP2005525291A5 - - Google Patents
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- JP2005525291A5 JP2005525291A5 JP2003520733A JP2003520733A JP2005525291A5 JP 2005525291 A5 JP2005525291 A5 JP 2005525291A5 JP 2003520733 A JP2003520733 A JP 2003520733A JP 2003520733 A JP2003520733 A JP 2003520733A JP 2005525291 A5 JP2005525291 A5 JP 2005525291A5
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- JP
- Japan
- Prior art keywords
- alkyl
- solvate
- salt
- compound
- formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE0102764A SE0102764D0 (sv) | 2001-08-17 | 2001-08-17 | Compounds |
| PCT/GB2002/003745 WO2003015774A1 (en) | 2001-08-17 | 2002-08-15 | Compounds effecting glucokinase |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2005168987A Division JP4441446B2 (ja) | 2001-08-17 | 2005-06-09 | グルコキナーゼ化合物 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2005525291A JP2005525291A (ja) | 2005-08-25 |
| JP2005525291A5 true JP2005525291A5 (https=) | 2006-01-05 |
| JP3987829B2 JP3987829B2 (ja) | 2007-10-10 |
Family
ID=20285065
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003520733A Expired - Fee Related JP3987829B2 (ja) | 2001-08-17 | 2002-08-15 | グルコキナーゼ化合物 |
| JP2005168987A Expired - Fee Related JP4441446B2 (ja) | 2001-08-17 | 2005-06-09 | グルコキナーゼ化合物 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2005168987A Expired - Fee Related JP4441446B2 (ja) | 2001-08-17 | 2005-06-09 | グルコキナーゼ化合物 |
Country Status (31)
| Country | Link |
|---|---|
| US (3) | US7390908B2 (https=) |
| EP (12) | EP1661568B1 (https=) |
| JP (2) | JP3987829B2 (https=) |
| KR (1) | KR100920439B1 (https=) |
| CN (4) | CN101584691A (https=) |
| AR (1) | AR037898A1 (https=) |
| AT (11) | ATE397928T1 (https=) |
| AU (1) | AU2002321462B2 (https=) |
| BR (1) | BR0212008A (https=) |
| CA (1) | CA2457410C (https=) |
| CO (1) | CO5560563A2 (https=) |
| CY (5) | CY1105746T1 (https=) |
| DE (11) | DE60227122D1 (https=) |
| DK (5) | DK1661569T3 (https=) |
| ES (10) | ES2308609T3 (https=) |
| HU (1) | HUP0401213A3 (https=) |
| IL (2) | IL160219A0 (https=) |
| IS (1) | IS7150A (https=) |
| MX (1) | MXPA04001500A (https=) |
| MY (1) | MY146279A (https=) |
| NO (1) | NO20040686L (https=) |
| NZ (1) | NZ531193A (https=) |
| PL (1) | PL368970A1 (https=) |
| PT (5) | PT1669068E (https=) |
| RU (1) | RU2329043C9 (https=) |
| SE (1) | SE0102764D0 (https=) |
| SI (5) | SI1669068T1 (https=) |
| TW (1) | TWI333855B (https=) |
| UA (1) | UA83182C2 (https=) |
| WO (1) | WO2003015774A1 (https=) |
| ZA (1) | ZA200401015B (https=) |
Families Citing this family (146)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE0102300D0 (sv) * | 2001-06-26 | 2001-06-26 | Astrazeneca Ab | Compounds |
| SE0102299D0 (sv) | 2001-06-26 | 2001-06-26 | Astrazeneca Ab | Compounds |
| SE0102764D0 (sv) | 2001-08-17 | 2001-08-17 | Astrazeneca Ab | Compounds |
| WO2004024705A1 (ja) * | 2002-09-10 | 2004-03-25 | Takeda Pharmaceutical Company Limited | 5員複素環化合物 |
| JP2004123732A (ja) * | 2002-09-10 | 2004-04-22 | Takeda Chem Ind Ltd | 5員複素環化合物 |
| BR0314864A (pt) | 2002-10-03 | 2005-08-02 | Novartis Ag | Compostos orgânicos |
| GB0226930D0 (en) | 2002-11-19 | 2002-12-24 | Astrazeneca Ab | Chemical compounds |
| GB0226931D0 (en) | 2002-11-19 | 2002-12-24 | Astrazeneca Ab | Chemical compounds |
| PL378117A1 (pl) | 2003-02-11 | 2006-03-06 | Prosidion Limited | Tricyklopodstawione związki amidowe |
| NZ540791A (en) | 2003-02-13 | 2009-09-25 | Banyu Pharma Co Ltd | Novel 2-pyridinecarboxamide derivatives |
| US7432287B2 (en) | 2003-02-26 | 2008-10-07 | Banyu Pharmeceutical Co., Ltd. | Heteroarylcarbamoylbenzene derivative |
| JP2006525361A (ja) * | 2003-05-02 | 2006-11-09 | エラン ファーマシューティカルズ,インコーポレイテッド | ブラジキニンb1受容体アンタゴニストとしての選択された置換ピラゾール誘導体および関連化合物 |
| JP2006526015A (ja) * | 2003-05-02 | 2006-11-16 | エラン ファーマシューティカルズ,インコーポレイテッド | 炎症疾患治療のためのブラジキニンb1受容体アンタゴニストとしての4−ブロモ−5−(2−クロロ−ベンゾイルアミノ)−1h−ピラゾール−3−カルボン酸アミド誘導体および関連化合物 |
| RU2344132C2 (ru) * | 2003-06-20 | 2009-01-20 | Ф.Хоффманн-Ля Рош Аг | 2-аминобензотиазолы в качестве обратных агонистов рецепторов cb1 |
| ES2222822B1 (es) * | 2003-07-28 | 2005-12-16 | Laboratorios Farmaceuticos Rovi, S.A. | Diamidas de aminoacidos en posicion no alfa utiles como adyuvantes para la administracion de agentes biologicos activos. |
| MXPA06003951A (es) | 2003-10-07 | 2006-06-27 | Renovis Inc | Derivados de amida como ligandos del canal de ion y composiciones farmaceuticas y sus metodos de uso. |
| GB0325402D0 (en) * | 2003-10-31 | 2003-12-03 | Astrazeneca Ab | Compounds |
| GB0328178D0 (en) * | 2003-12-05 | 2004-01-07 | Astrazeneca Ab | Compounds |
| KR20070007104A (ko) * | 2004-02-18 | 2007-01-12 | 아스트라제네카 아베 | 화합물 |
| BRPI0507746A (pt) | 2004-02-18 | 2007-07-10 | Astrazeneca Ab | composto ou um sal, pró-droga ou solvato do mesmo, composição farmacêutica, método de tratar doenças mediadas por glk, e, processo para a preparação de um composto |
| EP1734963A4 (en) | 2004-04-02 | 2008-06-18 | Merck & Co Inc | METHOD FOR TREATING PEOPLE WITH METABOLIC AND ANTHROPOMETRIC DISORDER |
| BRPI0509573A (pt) | 2004-04-02 | 2007-09-25 | Novartis Ag | derivados de sulfonamida-tiazolpiridina como ativadores de glicocinase úteis para o tratamento de diabetes do tipo 2 |
| US7781451B2 (en) | 2004-04-02 | 2010-08-24 | Novartis Ag | Thiazolopyridine derivatives, pharmaceut ical conditions containing them and methods of treating glucokinase mediated conditions |
| TW200600086A (en) * | 2004-06-05 | 2006-01-01 | Astrazeneca Ab | Chemical compound |
| RU2403246C2 (ru) * | 2004-06-05 | 2010-11-10 | Астразенека Аб | Гетероарилбензамидные производные для применения в качестве активаторов глюкокиназы (glk) в лечении диабета |
| KR100739367B1 (ko) * | 2004-07-14 | 2007-07-16 | 크리스탈지노믹스(주) | 설파마이드 유도체 및 이를 함유하는 지방대사 촉진용약학적 조성물 |
| GB0423043D0 (en) * | 2004-10-16 | 2004-11-17 | Astrazeneca Ab | Compounds |
| GB0423044D0 (en) * | 2004-10-16 | 2004-11-17 | Astrazeneca Ab | Compounds |
| KR20070085371A (ko) | 2004-10-16 | 2007-08-27 | 아스트라제네카 아베 | 페녹시 벤즈아미드 화합물의 제조 방법 |
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| GB0510852D0 (en) * | 2005-05-27 | 2005-07-06 | Astrazeneca Ab | Chemical compounds |
| TW200714597A (en) * | 2005-05-27 | 2007-04-16 | Astrazeneca Ab | Chemical compounds |
| JP2009500442A (ja) * | 2005-07-09 | 2009-01-08 | アストラゼネカ アクチボラグ | 2型糖尿病を処置するためのグルコキナーゼのモジュレーターとしての2−ヘテロシクリルオキシベンゾイルアミノヘテロシクリル化合物 |
| EP2027113A1 (en) * | 2005-07-09 | 2009-02-25 | AstraZeneca AB | Heteroaryl benzamide derivatives for use as glk activators in the treatment of diabetes |
| KR101346902B1 (ko) * | 2005-07-09 | 2014-01-02 | 아스트라제네카 아베 | 당뇨병 치료에 있어 glk 활성화제로서 사용하기 위한헤테로아릴 벤즈아미드 유도체 |
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| GT200600428A (es) | 2005-09-30 | 2007-05-21 | Compuestos organicos | |
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