JP2005525291A5 - - Google Patents
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- JP2005525291A5 JP2005525291A5 JP2003520733A JP2003520733A JP2005525291A5 JP 2005525291 A5 JP2005525291 A5 JP 2005525291A5 JP 2003520733 A JP2003520733 A JP 2003520733A JP 2003520733 A JP2003520733 A JP 2003520733A JP 2005525291 A5 JP2005525291 A5 JP 2005525291A5
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- Japan
- Prior art keywords
- alkyl
- solvate
- salt
- compound
- formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE0102764A SE0102764D0 (sv) | 2001-08-17 | 2001-08-17 | Compounds |
| PCT/GB2002/003745 WO2003015774A1 (en) | 2001-08-17 | 2002-08-15 | Compounds effecting glucokinase |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2005168987A Division JP4441446B2 (ja) | 2001-08-17 | 2005-06-09 | グルコキナーゼ化合物 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2005525291A JP2005525291A (ja) | 2005-08-25 |
| JP2005525291A5 true JP2005525291A5 (https=) | 2006-01-05 |
| JP3987829B2 JP3987829B2 (ja) | 2007-10-10 |
Family
ID=20285065
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003520733A Expired - Fee Related JP3987829B2 (ja) | 2001-08-17 | 2002-08-15 | グルコキナーゼ化合物 |
| JP2005168987A Expired - Fee Related JP4441446B2 (ja) | 2001-08-17 | 2005-06-09 | グルコキナーゼ化合物 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2005168987A Expired - Fee Related JP4441446B2 (ja) | 2001-08-17 | 2005-06-09 | グルコキナーゼ化合物 |
Country Status (31)
| Country | Link |
|---|---|
| US (3) | US7390908B2 (https=) |
| EP (12) | EP1661567B1 (https=) |
| JP (2) | JP3987829B2 (https=) |
| KR (1) | KR100920439B1 (https=) |
| CN (4) | CN101704797A (https=) |
| AR (1) | AR037898A1 (https=) |
| AT (11) | ATE397928T1 (https=) |
| AU (1) | AU2002321462B2 (https=) |
| BR (1) | BR0212008A (https=) |
| CA (1) | CA2457410C (https=) |
| CO (1) | CO5560563A2 (https=) |
| CY (5) | CY1105746T1 (https=) |
| DE (11) | DE60228770D1 (https=) |
| DK (5) | DK1529530T5 (https=) |
| ES (10) | ES2309862T3 (https=) |
| HU (1) | HUP0401213A3 (https=) |
| IL (2) | IL160219A0 (https=) |
| IS (1) | IS7150A (https=) |
| MX (1) | MXPA04001500A (https=) |
| MY (1) | MY146279A (https=) |
| NO (1) | NO20040686L (https=) |
| NZ (1) | NZ531193A (https=) |
| PL (1) | PL368970A1 (https=) |
| PT (5) | PT1661569E (https=) |
| RU (1) | RU2329043C9 (https=) |
| SE (1) | SE0102764D0 (https=) |
| SI (5) | SI1568367T1 (https=) |
| TW (1) | TWI333855B (https=) |
| UA (1) | UA83182C2 (https=) |
| WO (1) | WO2003015774A1 (https=) |
| ZA (1) | ZA200401015B (https=) |
Families Citing this family (147)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE0102300D0 (sv) * | 2001-06-26 | 2001-06-26 | Astrazeneca Ab | Compounds |
| SE0102299D0 (sv) | 2001-06-26 | 2001-06-26 | Astrazeneca Ab | Compounds |
| SE0102764D0 (sv) | 2001-08-17 | 2001-08-17 | Astrazeneca Ab | Compounds |
| US7368578B2 (en) | 2002-09-10 | 2008-05-06 | Takeda Pharmaceutical Company Limited | Five-membered heterocyclic compounds |
| JP2004123732A (ja) * | 2002-09-10 | 2004-04-22 | Takeda Chem Ind Ltd | 5員複素環化合物 |
| BR0314864A (pt) | 2002-10-03 | 2005-08-02 | Novartis Ag | Compostos orgânicos |
| GB0226931D0 (en) | 2002-11-19 | 2002-12-24 | Astrazeneca Ab | Chemical compounds |
| GB0226930D0 (en) | 2002-11-19 | 2002-12-24 | Astrazeneca Ab | Chemical compounds |
| PL378117A1 (pl) | 2003-02-11 | 2006-03-06 | Prosidion Limited | Tricyklopodstawione związki amidowe |
| EP1598349B1 (en) | 2003-02-13 | 2011-07-27 | Msd K.K. | Novel 2-pyridinecarboxamide derivatives |
| NZ541824A (en) | 2003-02-26 | 2010-04-30 | Banyu Pharma Co Ltd | Heteroarylcarbamoylbenzene derivatives as glucokinase activators |
| ATE410161T1 (de) | 2003-05-02 | 2008-10-15 | Elan Pharm Inc | 4-bromo-5-(2-chloro-benzoylamino)-1h-pyrazol-3- carbonsäureamid-derivate und verwandte verbindungen als bradykinin b1 rezeptor antagonisten zur behandlung von entzündlichen erkrankungen |
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| BRPI0415179A (pt) | 2003-10-07 | 2006-11-28 | Renovis Inc | derivados de amida como ligandos de canal de ìon e composições farmacêuticas e métodos de empregar as mesmas |
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| GB0328178D0 (en) * | 2003-12-05 | 2004-01-07 | Astrazeneca Ab | Compounds |
| KR20070007104A (ko) * | 2004-02-18 | 2007-01-12 | 아스트라제네카 아베 | 화합물 |
| DE602005013491D1 (de) * | 2004-02-18 | 2009-05-07 | Astrazeneca Ab | Benzamidderivate und deren verwendung als glucokinaseaktivierende mittel |
| US7750020B2 (en) | 2004-04-02 | 2010-07-06 | Novartis Ag | Sulfonamide-thiazolpyridine derivatives as glucokinase activators useful the treatment of Type 2 diabetes |
| AU2005229415B2 (en) | 2004-04-02 | 2009-05-14 | Novartis Ag | Thiazolopyridine derivatives, pharmaceutical conditions containing them and methods of treating glucokinase mediated conditions |
| US20080125403A1 (en) | 2004-04-02 | 2008-05-29 | Merck & Co., Inc. | Method of Treating Men with Metabolic and Anthropometric Disorders |
| RU2403246C2 (ru) * | 2004-06-05 | 2010-11-10 | Астразенека Аб | Гетероарилбензамидные производные для применения в качестве активаторов глюкокиназы (glk) в лечении диабета |
| TW200600086A (en) | 2004-06-05 | 2006-01-01 | Astrazeneca Ab | Chemical compound |
| KR100739367B1 (ko) * | 2004-07-14 | 2007-07-16 | 크리스탈지노믹스(주) | 설파마이드 유도체 및 이를 함유하는 지방대사 촉진용약학적 조성물 |
| GB0423043D0 (en) * | 2004-10-16 | 2004-11-17 | Astrazeneca Ab | Compounds |
| KR20070085371A (ko) | 2004-10-16 | 2007-08-27 | 아스트라제네카 아베 | 페녹시 벤즈아미드 화합물의 제조 방법 |
| GB0423044D0 (en) * | 2004-10-16 | 2004-11-17 | Astrazeneca Ab | Compounds |
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| EP1884513A4 (en) * | 2005-05-23 | 2010-04-28 | Japan Tobacco Inc | PYRAZOLE COMPOUND AND THERAPEUTIC AGENT FOR DIABETES COMPRISING THE SAME |
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| CA2614746C (en) | 2005-07-09 | 2011-05-10 | Astrazeneca Ab | Heteroaryl benzamide derivatives for use as glk activators in the treatment of diabetes |
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| US20080234273A1 (en) * | 2005-07-09 | 2008-09-25 | Mckerrecher Darren | Heteroaryl Benzamide Derivatives for Use as Glk Activators in the Treatment of Diabetes |
| EP1910317B1 (en) | 2005-07-20 | 2013-07-03 | Eli Lilly And Company | 1-amino linked compounds |
| US9202182B2 (en) * | 2005-08-11 | 2015-12-01 | International Business Machines Corporation | Method and system for analyzing business architecture |
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| GT200600429A (es) | 2005-09-30 | 2007-04-30 | Compuestos organicos | |
| GT200600428A (es) | 2005-09-30 | 2007-05-21 | Compuestos organicos | |
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| US8034822B2 (en) | 2006-03-08 | 2011-10-11 | Takeda San Diego, Inc. | Glucokinase activators |
| JP5190448B2 (ja) * | 2006-04-20 | 2013-04-24 | ファイザー・プロダクツ・インク | グルコキナーゼ仲介疾患を予防および治療するための縮合フェニルアミド複素環化合物 |
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| US7910747B2 (en) | 2006-07-06 | 2011-03-22 | Bristol-Myers Squibb Company | Phosphonate and phosphinate pyrazolylamide glucokinase activators |
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