TW201100417A - 1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors - Google Patents

1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors Download PDF

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Publication number
TW201100417A
TW201100417A TW099115165A TW99115165A TW201100417A TW 201100417 A TW201100417 A TW 201100417A TW 099115165 A TW099115165 A TW 099115165A TW 99115165 A TW99115165 A TW 99115165A TW 201100417 A TW201100417 A TW 201100417A
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group
alkyl
substituted
independently selected
compound
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TW099115165A
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English (en)
Chinese (zh)
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Jose Maria Cid-Nunez
Lucas Olivares Ana Isabel De
Andres Avelino Trabanco-Suarez
Gregor James Macdonald
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Ortho Mcneil Janssen Pharm
Addex Pharmaceuticals Sa
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
TW099115165A 2009-05-12 2010-05-12 1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors TW201100417A (en)

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Application Number Priority Date Filing Date Title
EP09160067 2009-05-12

Publications (1)

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TW201100417A true TW201100417A (en) 2011-01-01

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US (1) US8946205B2 (enExample)
EP (1) EP2430031B1 (enExample)
JP (1) JP5707390B2 (enExample)
KR (1) KR20120035158A (enExample)
CN (1) CN102439015B (enExample)
AR (1) AR076859A1 (enExample)
AU (1) AU2010246607B2 (enExample)
BR (1) BRPI1010831A2 (enExample)
CA (1) CA2760259C (enExample)
CL (1) CL2011002837A1 (enExample)
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ES (1) ES2409006T3 (enExample)
IL (1) IL215910A (enExample)
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MY (1) MY153912A (enExample)
NZ (1) NZ596053A (enExample)
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TW (1) TW201100417A (enExample)
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US8765767B2 (en) 2012-03-16 2014-07-01 Bristol-Myers Squibb Company Positive allosteric modulators of mGluR2
JO3368B1 (ar) 2013-06-04 2019-03-13 Janssen Pharmaceutica Nv مركبات 6، 7- ثاني هيدرو بيرازولو [5،1-a] بيرازين- 4 (5 يد)- اون واستخدامها بصفة منظمات تفارغية سلبية لمستقبلات ميجلور 2
JO3367B1 (ar) 2013-09-06 2019-03-13 Janssen Pharmaceutica Nv مركبات 2،1، 4- ثلاثي زولو [3،4-a] بيريدين واستخدامها بصفة منظمات تفارغية موجبة لمستقبلات ميجلور 2
WO2015042243A1 (en) 2013-09-19 2015-03-26 Bristol-Myers Squibb Company Triazolopyridine ether derivatives and their use in neurological and pyschiatric disorders
PT3096790T (pt) 2014-01-21 2019-10-15 Janssen Pharmaceutica Nv Combinações compreendendo moduladores alostéricos positivos ou agonistas ortostéricos do recetor glutamatérgico metabotrópico do subtipo 2 e seu uso
EA202192105A3 (ru) 2014-02-04 2022-02-28 Янссен Фармацевтика Нв Комбинации, содержащие положительные аллостерические модуляторы или ортостерические агонисты метаботропного глутаматергического рецептора 2 подтипа, и их применение
US10138237B2 (en) 2014-12-11 2018-11-27 Janssen Pharmaceutica Nv 1,2,4-triazolo[4,3-a]pyridine compounds and their use as positive allosteric modulators of mGluR2 receptors
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