PL3070090T3 - Zastosowanie soli inhibitora kinazy janusowej (r)-3-(4-(7h-pirolo[2,3- d]pirymidyn-4-ylo)-1h-pirazol-1-ilo)-3-cyklopentylopropanonitrylu - Google Patents

Zastosowanie soli inhibitora kinazy janusowej (r)-3-(4-(7h-pirolo[2,3- d]pirymidyn-4-ylo)-1h-pirazol-1-ilo)-3-cyklopentylopropanonitrylu

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Publication number
PL3070090T3
PL3070090T3 PL16152794T PL16152794T PL3070090T3 PL 3070090 T3 PL3070090 T3 PL 3070090T3 PL 16152794 T PL16152794 T PL 16152794T PL 16152794 T PL16152794 T PL 16152794T PL 3070090 T3 PL3070090 T3 PL 3070090T3
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PL
Poland
Prior art keywords
cyclopentylpropanenitrile
pyrrolo
pyrazol
pyrimidin
salts
Prior art date
Application number
PL16152794T
Other languages
English (en)
Inventor
Hui-Yin Li
James D. Rodgers
Original Assignee
Incyte Holdings Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40029273&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL3070090(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Incyte Holdings Corporation filed Critical Incyte Holdings Corporation
Publication of PL3070090T3 publication Critical patent/PL3070090T3/pl

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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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PL16152794T 2007-06-13 2008-06-12 Zastosowanie soli inhibitora kinazy janusowej (r)-3-(4-(7h-pirolo[2,3- d]pirymidyn-4-ylo)-1h-pirazol-1-ilo)-3-cyklopentylopropanonitrylu PL3070090T3 (pl)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US94370507P 2007-06-13 2007-06-13
PCT/US2008/066662 WO2008157208A2 (en) 2007-06-13 2008-06-12 Salts of the janus kinase inhibitor (r)-3-(4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl)-3-cyclopentylpropanenitrile
EP16152794.0A EP3070090B1 (en) 2007-06-13 2008-06-12 Use of salts of the janus kinase inhibitor (r)-3-(4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h- pyrazol-1-yl)-3- cyclopentylpropanenitrile
EP13198120.1A EP2740731B1 (en) 2007-06-13 2008-06-12 Crystalline salts of the janus kinase inhibitor (r)-3-(4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl)-3-cyclopentylpropanenitrile
EP08770794.9A EP2173752B2 (en) 2007-06-13 2008-06-12 Salts of the janus kinase inhibitor (r)-3-(4-(7h-pyrrolo(2,3-d)pyrimidin-4-yl)-1h-pyrazol-1-yl)-3-cyclopentylpropanenitrile

Publications (1)

Publication Number Publication Date
PL3070090T3 true PL3070090T3 (pl) 2019-07-31

Family

ID=40029273

Family Applications (3)

Application Number Title Priority Date Filing Date
PL16152794T PL3070090T3 (pl) 2007-06-13 2008-06-12 Zastosowanie soli inhibitora kinazy janusowej (r)-3-(4-(7h-pirolo[2,3- d]pirymidyn-4-ylo)-1h-pirazol-1-ilo)-3-cyklopentylopropanonitrylu
PL08770794.9T PL2173752T5 (pl) 2007-06-13 2008-06-12 Sole (r)-3-(4-(7h-pirolo(2,3-d)pirymidyn-4-ylo)-1h-pirazol-1-ilo)-3-cyklopentylopropanonitrylu inhibitora kinazy janusowej
PL13198120.1T PL2740731T3 (pl) 2007-06-13 2008-06-12 Krystaliczne sole (R)-3-(4-(7H-pirolo[2,3-d]pirymidyn-4-ylo)-1H-pirazol-1-ilo)-3-cyklopentylopropanonitrylu jako inhibitory kinazy Janusowej

Family Applications After (2)

Application Number Title Priority Date Filing Date
PL08770794.9T PL2173752T5 (pl) 2007-06-13 2008-06-12 Sole (r)-3-(4-(7h-pirolo(2,3-d)pirymidyn-4-ylo)-1h-pirazol-1-ilo)-3-cyklopentylopropanonitrylu inhibitora kinazy janusowej
PL13198120.1T PL2740731T3 (pl) 2007-06-13 2008-06-12 Krystaliczne sole (R)-3-(4-(7H-pirolo[2,3-d]pirymidyn-4-ylo)-1H-pirazol-1-ilo)-3-cyklopentylopropanonitrylu jako inhibitory kinazy Janusowej

Country Status (41)

Country Link
US (10) US20080312259A1 (pl)
EP (6) EP2740731B1 (pl)
JP (1) JP5475653B2 (pl)
KR (2) KR20150036210A (pl)
CN (2) CN103524509B (pl)
AU (1) AU2008266183B2 (pl)
BR (1) BRPI0814254B8 (pl)
CA (1) CA2689663C (pl)
CO (1) CO6251256A2 (pl)
CR (1) CR11151A (pl)
CU (2) CU24179B1 (pl)
CY (3) CY1115145T1 (pl)
DK (3) DK2740731T3 (pl)
DO (1) DOP2009000280A (pl)
EA (1) EA019784B1 (pl)
EC (1) ECSP099802A (pl)
ES (4) ES2467665T5 (pl)
GE (1) GEP20125533B (pl)
GT (1) GT200900314A (pl)
HR (3) HRP20140541T4 (pl)
HU (2) HUE029236T2 (pl)
IL (5) IL202524A (pl)
LT (1) LT3070090T (pl)
MA (1) MA31517B1 (pl)
ME (1) ME00960B (pl)
MX (2) MX2009013402A (pl)
MY (1) MY154969A (pl)
NI (1) NI200900216A (pl)
NO (1) NO2019025I1 (pl)
NZ (1) NZ581803A (pl)
PL (3) PL3070090T3 (pl)
PT (2) PT3070090T (pl)
RS (3) RS54878B1 (pl)
SG (3) SG182198A1 (pl)
SI (3) SI3070090T1 (pl)
SM (1) SMP201000002B (pl)
TN (1) TN2009000514A1 (pl)
TR (1) TR201903488T4 (pl)
UA (1) UA99467C2 (pl)
WO (1) WO2008157208A2 (pl)
ZA (1) ZA200908826B (pl)

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WO2005105814A1 (en) * 2004-04-28 2005-11-10 Incyte Corporation Tetracyclic inhibitors of janus kinases
US8604042B2 (en) 2005-11-01 2013-12-10 Targegen, Inc. Bi-aryl meta-pyrimidine inhibitors of kinases
NZ592990A (en) 2005-11-01 2013-01-25 Targegen Inc Bi-aryl meta-pyrimidine inhibitors of kinases
US8133900B2 (en) 2005-11-01 2012-03-13 Targegen, Inc. Use of bi-aryl meta-pyrimidine inhibitors of kinases
DK3184526T3 (en) 2005-12-13 2019-01-14 Incyte Holdings Corp PYRROLO [2,3-D] PYRIMIDINE DERIVATIVES AS A JANUS-KINASE INHIBITOR
EP2121692B1 (en) 2006-12-22 2013-04-10 Incyte Corporation Substituted heterocycles as janus kinase inhibitors
CL2008001709A1 (es) 2007-06-13 2008-11-03 Incyte Corp Compuestos derivados de pirrolo [2,3-b]pirimidina, moduladores de quinasas jak; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como cancer, psoriasis, artritis reumatoide, entre otras.
DK2740731T3 (en) 2007-06-13 2016-04-11 Incyte Holdings Corp CRYSTALLINE SALTS OF JANUSKINASEINHIBITOREN (R) -3- (4- (7H-pyrrolo [2,3-d] pyrimidin-4-yl) -1H-pyrazol-1-yl) -3-CYCLOPENTYLPROPANNITRIL
WO2009064835A1 (en) * 2007-11-16 2009-05-22 Incyte Corporation 4-pyrazolyl-n-arylpyrimidin-2-amines and 4-pyrazolyl-n-heteroarylpyrimidin-2-amines as janus kinase inhibitors
BRPI0909040B8 (pt) 2008-03-11 2021-05-25 Incyte Holdings Corp derivados de azetidina e ciclobutano, seus usos, e composição
JOP20190230A1 (ar) * 2009-01-15 2017-06-16 Incyte Corp طرق لاصلاح مثبطات انزيم jak و المركبات الوسيطة المتعلقة به
CN102395576A (zh) 2009-02-27 2012-03-28 埃姆比特生物科学公司 调控jak激酶的喹唑啉衍生物和其使用方法
MY156727A (en) 2009-05-22 2016-03-15 Incyte Corp N-(hetero)aryl-pyrrolidine derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines and pyrrol-3-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors
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