PH12012502411A1 - Method of modulating stress-activated protein kinase system - Google Patents
Method of modulating stress-activated protein kinase systemInfo
- Publication number
- PH12012502411A1 PH12012502411A1 PH1/2012/502411A PH12012502411A PH12012502411A1 PH 12012502411 A1 PH12012502411 A1 PH 12012502411A1 PH 12012502411 A PH12012502411 A PH 12012502411A PH 12012502411 A1 PH12012502411 A1 PH 12012502411A1
- Authority
- PH
- Philippines
- Prior art keywords
- protein kinase
- activated protein
- modulating
- sapk
- kinase system
- Prior art date
Links
- 102000001253 Protein Kinase Human genes 0.000 title abstract 3
- 108060006633 protein kinase Proteins 0.000 title abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 3
- 230000005764 inhibitory process Effects 0.000 abstract 2
- 102000002574 p38 Mitogen-Activated Protein Kinases Human genes 0.000 abstract 2
- 108010068338 p38 Mitogen-Activated Protein Kinases Proteins 0.000 abstract 2
- 230000002401 inhibitory effect Effects 0.000 abstract 1
- ISWRGOKTTBVCFA-UHFFFAOYSA-N pirfenidone Chemical class C1=C(C)C=CC(=O)N1C1=CC=CC=C1 ISWRGOKTTBVCFA-UHFFFAOYSA-N 0.000 abstract 1
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- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- 2007-11-09 TN TNP2007000416A patent/TNSN07416A1/en unknown
- 2007-11-09 NI NI200700289A patent/NI200700289A/es unknown
- 2007-11-30 MA MA30442A patent/MA29499B1/fr unknown
-
2010
- 2010-05-28 US US12/790,099 patent/US20100240704A1/en not_active Abandoned
-
2012
- 2012-03-26 JP JP2012069833A patent/JP2012125254A/ja not_active Withdrawn
- 2012-03-26 JP JP2012069834A patent/JP5735931B2/ja not_active Expired - Fee Related
- 2012-06-20 US US13/528,624 patent/US8741936B2/en active Active
-
2014
- 2014-04-28 US US14/263,787 patent/US9527816B2/en not_active Expired - Fee Related
-
2016
- 2016-12-21 US US15/387,537 patent/US10010536B2/en active Active
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