NO328134B1 - Vannfrie aripiprazol krystaller B og hydrat A av aripiprazol samt fremgangsmater for fremstilling og anvendelse derav, samt farmsoytisk preparat. - Google Patents
Vannfrie aripiprazol krystaller B og hydrat A av aripiprazol samt fremgangsmater for fremstilling og anvendelse derav, samt farmsoytisk preparat. Download PDFInfo
- Publication number
- NO328134B1 NO328134B1 NO20030247A NO20030247A NO328134B1 NO 328134 B1 NO328134 B1 NO 328134B1 NO 20030247 A NO20030247 A NO 20030247A NO 20030247 A NO20030247 A NO 20030247A NO 328134 B1 NO328134 B1 NO 328134B1
- Authority
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- Norway
- Prior art keywords
- aripiprazole
- crystals
- hydrate
- approx
- hours
- Prior art date
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
- C07D215/22—Oxygen atoms attached in position 2 or 4
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
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- Y10T428/00—Stock material or miscellaneous articles
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- Y10T428/2982—Particulate matter [e.g., sphere, flake, etc.]
Landscapes
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- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
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- Chemical Kinetics & Catalysis (AREA)
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Quinoline Compounds (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2001290645 | 2001-09-25 | ||
| JP2001348276 | 2001-11-14 | ||
| CA 2379005 CA2379005A1 (en) | 2001-09-25 | 2002-03-27 | Low hygroscopic aripiprazole drug substance and processes for the preparation thereof |
| PCT/JP2002/009858 WO2003026659A1 (en) | 2001-09-25 | 2002-09-25 | Low hygroscopic aripiprazole drug substance and processes for the preparation thereof |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO20030247D0 NO20030247D0 (no) | 2003-01-17 |
| NO20030247L NO20030247L (no) | 2003-01-17 |
| NO328134B1 true NO328134B1 (no) | 2009-12-14 |
Family
ID=27171631
Family Applications (7)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20030247A NO328134B1 (no) | 2001-09-25 | 2003-01-17 | Vannfrie aripiprazol krystaller B og hydrat A av aripiprazol samt fremgangsmater for fremstilling og anvendelse derav, samt farmsoytisk preparat. |
| NO20081632A NO336262B1 (no) | 2001-09-25 | 2008-04-02 | Vannfrie aripiprazol-krystaller F, fremgangsmåte for fremstilling derav samt farmasøytisk preparat |
| NO20081633A NO20081633L (no) | 2001-09-25 | 2008-04-02 | Lav hygroskopisk Aripiprazol medikament forbindelse og fremgangsmate for fremstilling derav |
| NO20081631A NO336263B1 (no) | 2001-09-25 | 2008-04-02 | Vannfrie aripiprazol-krystaller E, fremgangsmåte for fremstilling derav, samt farmasøytisk preparat |
| NO20081627A NO336265B1 (no) | 2001-09-25 | 2008-04-02 | Vannfrie aripiprazol-krystaller D, fremgangsmåte for fremstilling derav, samt farmasøytisk preparat |
| NO20081626A NO336264B1 (no) | 2001-09-25 | 2008-04-02 | Vannfrie aripiprazol-krystaller C, fremgangsmåte for fremstilling derav samt farmasøytisk preparat |
| NO20091689A NO336679B1 (no) | 2001-09-25 | 2009-04-28 | Fremgangsmåte for fremstilling av et fast oralt preparat av granuler, fremgangsmåte for fremstilling av et fast oral preparat, og farmasøytisk fast oralt preparat |
Family Applications After (6)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20081632A NO336262B1 (no) | 2001-09-25 | 2008-04-02 | Vannfrie aripiprazol-krystaller F, fremgangsmåte for fremstilling derav samt farmasøytisk preparat |
| NO20081633A NO20081633L (no) | 2001-09-25 | 2008-04-02 | Lav hygroskopisk Aripiprazol medikament forbindelse og fremgangsmate for fremstilling derav |
| NO20081631A NO336263B1 (no) | 2001-09-25 | 2008-04-02 | Vannfrie aripiprazol-krystaller E, fremgangsmåte for fremstilling derav, samt farmasøytisk preparat |
| NO20081627A NO336265B1 (no) | 2001-09-25 | 2008-04-02 | Vannfrie aripiprazol-krystaller D, fremgangsmåte for fremstilling derav, samt farmasøytisk preparat |
| NO20081626A NO336264B1 (no) | 2001-09-25 | 2008-04-02 | Vannfrie aripiprazol-krystaller C, fremgangsmåte for fremstilling derav samt farmasøytisk preparat |
| NO20091689A NO336679B1 (no) | 2001-09-25 | 2009-04-28 | Fremgangsmåte for fremstilling av et fast oralt preparat av granuler, fremgangsmåte for fremstilling av et fast oral preparat, og farmasøytisk fast oralt preparat |
Country Status (23)
| Country | Link |
|---|---|
| US (20) | US20040058935A1 (zh) |
| EP (6) | EP1330249B1 (zh) |
| JP (3) | JP3760264B2 (zh) |
| CN (16) | CN101423493A (zh) |
| AR (2) | AR033485A1 (zh) |
| AT (5) | ATE322269T1 (zh) |
| AU (1) | AU2002334413C1 (zh) |
| BR (1) | BR0205391A (zh) |
| CA (6) | CA2689052C (zh) |
| CY (1) | CY1118195T1 (zh) |
| DE (5) | DE60236383D1 (zh) |
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