IL154175A0 - 17. beta.-carbothioate 17. alpha-arylcarbonyloxyloxy androstane derivatives as anti-inflammatory agents - Google Patents

17. beta.-carbothioate 17. alpha-arylcarbonyloxyloxy androstane derivatives as anti-inflammatory agents

Info

Publication number
IL154175A0
IL154175A0 IL15417501A IL15417501A IL154175A0 IL 154175 A0 IL154175 A0 IL 154175A0 IL 15417501 A IL15417501 A IL 15417501A IL 15417501 A IL15417501 A IL 15417501A IL 154175 A0 IL154175 A0 IL 154175A0
Authority
IL
Israel
Prior art keywords
arylcarbonyloxyloxy
carbothioate
beta
alpha
inflammatory agents
Prior art date
Application number
IL15417501A
Other languages
English (en)
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26244792&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL154175(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GBGB0019172.6A external-priority patent/GB0019172D0/en
Priority claimed from GBGB0108800.4A external-priority patent/GB0108800D0/en
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of IL154175A0 publication Critical patent/IL154175A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/04—Antipruritics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/14—Decongestants or antiallergics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
    • A61P5/44—Glucocorticosteroids; Drugs increasing or potentiating the activity of glucocorticosteroids

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Endocrinology (AREA)
  • Otolaryngology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Diabetes (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IL15417501A 2000-08-05 2001-08-03 17. beta.-carbothioate 17. alpha-arylcarbonyloxyloxy androstane derivatives as anti-inflammatory agents IL154175A0 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0019172.6A GB0019172D0 (en) 2000-08-05 2000-08-05 Novel compounds
GBGB0108800.4A GB0108800D0 (en) 2001-04-07 2001-04-07 Novel compounds
PCT/GB2001/003499 WO2002012266A1 (en) 2000-08-05 2001-08-03 17.beta.-carbothioate 17.alpha.-arylcarbonyloxyloxy androstane derivative as anti-inflammatory agents

Publications (1)

Publication Number Publication Date
IL154175A0 true IL154175A0 (en) 2003-07-31

Family

ID=26244792

Family Applications (4)

Application Number Title Priority Date Filing Date
IL15417501A IL154175A0 (en) 2000-08-05 2001-08-03 17. beta.-carbothioate 17. alpha-arylcarbonyloxyloxy androstane derivatives as anti-inflammatory agents
IL15414801A IL154148A0 (en) 2000-08-05 2001-08-03 6.alpha.,9.alpha.-difluoro-17.alpha.-'(2-furanylcarboxyl) oxyl-11.beta.-hydroxy-16.alpha.-methyl-3-oxo-androst-1,4-diene-17-carbothioic acid s-fluoromethyl ester as an anti-inflammatory agent
IL154148A IL154148A (en) 2000-08-05 2003-01-27 S - Fluoro methyl ester of α6, α9 - difluoro - α 17 '(2 - phenylcarboxyl) Waxi - ß11 - hydroxy - α 16 - methyl - 3 - oxo-androst - 1,4 - dian - 17 - battoic acid as an anti-inflammatory factor
IL188364A IL188364A (en) 2000-08-05 2007-12-24 Pharmaceutical preparation containing S-fluoro-methyl ester of 6 alpha, 9 alpha-difluoro-17 alpha-[(2-furanylcarbonyl) oxy] -11 beta-hydroxy-16 alpha-methyl-3-oxo-androstate-4,1-diane-17-beta-fatty acid As an anti-inflammatory factor

Family Applications After (3)

Application Number Title Priority Date Filing Date
IL15414801A IL154148A0 (en) 2000-08-05 2001-08-03 6.alpha.,9.alpha.-difluoro-17.alpha.-'(2-furanylcarboxyl) oxyl-11.beta.-hydroxy-16.alpha.-methyl-3-oxo-androst-1,4-diene-17-carbothioic acid s-fluoromethyl ester as an anti-inflammatory agent
IL154148A IL154148A (en) 2000-08-05 2003-01-27 S - Fluoro methyl ester of α6, α9 - difluoro - α 17 '(2 - phenylcarboxyl) Waxi - ß11 - hydroxy - α 16 - methyl - 3 - oxo-androst - 1,4 - dian - 17 - battoic acid as an anti-inflammatory factor
IL188364A IL188364A (en) 2000-08-05 2007-12-24 Pharmaceutical preparation containing S-fluoro-methyl ester of 6 alpha, 9 alpha-difluoro-17 alpha-[(2-furanylcarbonyl) oxy] -11 beta-hydroxy-16 alpha-methyl-3-oxo-androstate-4,1-diane-17-beta-fatty acid As an anti-inflammatory factor

Country Status (36)

Country Link
US (3) US7498321B2 (enExample)
EP (5) EP2067784A3 (enExample)
JP (3) JP4436041B2 (enExample)
KR (3) KR100889426B1 (enExample)
CN (4) CN1294142C (enExample)
AP (1) AP1422A (enExample)
AR (3) AR032471A1 (enExample)
AT (2) ATE416184T1 (enExample)
AU (4) AU7576001A (enExample)
BG (1) BG66241B1 (enExample)
BR (2) BRPI0113042B8 (enExample)
CA (3) CA2417825C (enExample)
CO (2) CO5310534A1 (enExample)
CY (4) CY1107899T1 (enExample)
CZ (2) CZ2003353A3 (enExample)
DE (3) DE122008000029I1 (enExample)
DK (3) DK1775305T3 (enExample)
DZ (1) DZ3468A1 (enExample)
EA (1) EA005992B1 (enExample)
ES (4) ES2523930T3 (enExample)
FR (1) FR08C0014I2 (enExample)
HK (2) HK1056180B (enExample)
HU (3) HU230328B1 (enExample)
IL (4) IL154175A0 (enExample)
LU (1) LU91429I2 (enExample)
MA (1) MA25899A1 (enExample)
MX (2) MXPA03001097A (enExample)
NL (1) NL300343I2 (enExample)
NO (4) NO324747B1 (enExample)
NZ (2) NZ523958A (enExample)
OA (1) OA12394A (enExample)
PL (2) PL359917A1 (enExample)
PT (3) PT1775305E (enExample)
SI (3) SI1775305T1 (enExample)
SK (1) SK287576B6 (enExample)
WO (2) WO2002012266A1 (enExample)

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CY1116145T1 (el) 2017-02-08
CN1468252A (zh) 2004-01-14
NO20075376L (no) 2007-10-22
MXPA03001096A (es) 2003-05-27
DK1775305T3 (en) 2014-11-17
EP1305329B1 (en) 2007-12-05
JP4436041B2 (ja) 2010-03-24
EA200300082A1 (ru) 2003-08-28
OA12394A (en) 2004-07-09

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