WO1999010349A1
(fr)
|
1997-08-22 |
1999-03-04 |
Zeneca Limited |
Derives d'oxindolylquinazoline utiles comme inhibiteurs d'angiogenese
|
RS49779B
(sr)
*
|
1998-01-12 |
2008-06-05 |
Glaxo Group Limited, |
Biciklična heteroaromatična jedinjenja kao inhibitori protein tirozin kinaze
|
AU756556B2
(en)
|
1998-10-08 |
2003-01-16 |
Astrazeneca Ab |
Quinazoline derivatives
|
GB2345486A
(en)
*
|
1999-01-11 |
2000-07-12 |
Glaxo Group Ltd |
Heteroaromatic protein tyrosine kinase inhibitors
|
DK1553097T3
(da)
|
1999-02-10 |
2010-12-13 |
Astrazeneca Ab |
Quinazolinderivat som angiogeneseinhibitor og mellemprodukter dertil
|
GB9910580D0
(en)
|
1999-05-08 |
1999-07-07 |
Zeneca Ltd |
Chemical compounds
|
GB9910579D0
(en)
|
1999-05-08 |
1999-07-07 |
Zeneca Ltd |
Chemical compounds
|
MXPA01012899A
(es)
|
1999-06-21 |
2002-07-30 |
Boehringer Ingelheim Pharma |
Heterociclos biciclicos, medicamentos que contienen estos compuestos, su empleo y procedimientos para su preparacion.
|
EP1192151B1
(fr)
*
|
1999-07-09 |
2007-11-07 |
Glaxo Group Limited |
Anilino-quinazolines comme inhibiteurs de la proteine tyrosine kinase
|
US6933299B1
(en)
|
1999-07-09 |
2005-08-23 |
Smithkline Beecham Corporation |
Anilinoquinazolines as protein tyrosine kinase inhibitors
|
ES2334879T3
(es)
|
1999-09-21 |
2010-03-17 |
Astrazeneca Ab |
Derivados de quinazolina y su uso como productos farmaceuticos.
|
UA74803C2
(uk)
|
1999-11-11 |
2006-02-15 |
Осі Фармасьютікалз, Інк. |
Стійкий поліморф гідрохлориду n-(3-етинілфеніл)-6,7-біс(2-метоксіетокси)-4-хіназолінаміну, спосіб його одержання (варіанти) та фармацевтичне застосування
|
JP2003520855A
(ja)
*
|
2000-01-28 |
2003-07-08 |
アストラゼネカ アクチボラグ |
化学的化合物
|
GB0002952D0
(en)
*
|
2000-02-09 |
2000-03-29 |
Pharma Mar Sa |
Process for producing kahalalide F compounds
|
US6521618B2
(en)
|
2000-03-28 |
2003-02-18 |
Wyeth |
3-cyanoquinolines, 3-cyano-1,6-naphthyridines, and 3-cyano-1,7-naphthyridines as protein kinase inhibitors
|
AR035851A1
(es)
*
|
2000-03-28 |
2004-07-21 |
Wyeth Corp |
3-cianoquinolinas, 3-ciano-1,6-naftiridinas y 3-ciano-1,7-naftiridinas como inhibidoras de proteina quinasas
|
CA2409139A1
(fr)
|
2000-05-02 |
2001-11-08 |
Array Biopharma, Inc. |
Procede de reduction de sulfones cyano-substituees en sulfones aminoalkylene-substituees
|
EA005525B1
(ru)
|
2000-06-22 |
2005-04-28 |
Пфайзер Продактс Инк. |
Замещенные бициклические производные для лечения аномального роста клеток
|
HUP0301236A2
(hu)
|
2000-06-28 |
2003-10-28 |
Astrazeneca Ab, |
Szubsztituált kinazolinszármazékok és felhasználásuk inhibitorokként
|
DE60126611T2
(de)
*
|
2000-06-30 |
2007-11-22 |
Glaxo Group Ltd., Greenford |
Ditosylatsalze von chinazolinverbindungen
|
EP1792902A1
(fr)
*
|
2000-06-30 |
2007-06-06 |
Glaxo Group Limited |
Procédés pour la préparation de 5-(6-quinazolinyl)-furane-2-carbaldéhydes
|
MXPA03000252A
(es)
|
2000-08-09 |
2003-06-06 |
Astrazeneca Ab |
Derivados de quinolina que tienen actividad de inhibicion de fcev.
|
PL359920A1
(en)
|
2000-09-20 |
2004-09-06 |
Merck Patent Gmbh |
4-amino-quinazolines
|
EP1506962B1
(fr)
|
2000-10-20 |
2008-07-02 |
Eisai R&D Management Co., Ltd. |
Hétérocycles aromatiques contenant de l'azote
|
US7776315B2
(en)
|
2000-10-31 |
2010-08-17 |
Boehringer Ingelheim Pharma Gmbh & Co. Kg |
Pharmaceutical compositions based on anticholinergics and additional active ingredients
|
AU2001295791A1
(en)
|
2000-11-02 |
2002-05-15 |
Astrazeneca Ab |
4-substituted quinolines as antitumor agents
|
US7067532B2
(en)
|
2000-11-02 |
2006-06-27 |
Astrazeneca |
Substituted quinolines as antitumor agents
|
US7019012B2
(en)
|
2000-12-20 |
2006-03-28 |
Boehringer Ingelheim International Pharma Gmbh & Co. Kg |
Quinazoline derivatives and pharmaceutical compositions containing them
|
WO2002053596A2
(fr)
|
2001-01-05 |
2002-07-11 |
Pfizer Inc. |
Anticorps anti-recepteur du facteur de croissance insulinoide i
|
EP1488809A1
(fr)
|
2001-01-16 |
2004-12-22 |
Glaxo Group Limited |
combinaison pharmaceutique contenant de l'amino-4 quinazoline et un autre agent antineoplasique pour le traitement du cancer
|
DE60203260T2
(de)
|
2001-01-16 |
2006-02-02 |
Glaxo Group Ltd., Greenford |
Pharmazeutische kombination, die ein 4-chinazolinamin und paclitaxel, carboplatin oder vinorelbin enthält, zur behandlung von krebs
|
AU2002252338B2
(en)
*
|
2001-03-15 |
2007-09-13 |
Rhode Island Hospital, A Lifespan Partner |
Taurine compounds
|
US20030125344A1
(en)
*
|
2001-03-23 |
2003-07-03 |
Bayer Corporation |
Rho-kinase inhibitors
|
PT1370552E
(pt)
*
|
2001-03-23 |
2007-04-30 |
Bayer Pharmaceuticals Corp |
Inibidores de rho-quinase
|
ATE330956T1
(de)
|
2001-04-13 |
2006-07-15 |
Pfizer Prod Inc |
Bizyklisch substituierte 4- aminopyridopyrimidinderivate
|
WO2002092578A1
(fr)
*
|
2001-05-14 |
2002-11-21 |
Astrazeneca Ab |
Derives de quinazoline
|
AU2002345792A1
(en)
|
2001-06-21 |
2003-01-08 |
Pfizer Inc. |
Thienopyridine and thienopyrimidine anticancer agents
|
US20090197852A9
(en)
*
|
2001-08-06 |
2009-08-06 |
Johnson Robert G Jr |
Method of treating breast cancer using 17-AAG or 17-AG or a prodrug of either in combination with a HER2 inhibitor
|
US7829566B2
(en)
|
2001-09-17 |
2010-11-09 |
Werner Mederski |
4-amino-quinazolines
|
AR039067A1
(es)
|
2001-11-09 |
2005-02-09 |
Pfizer Prod Inc |
Anticuerpos para cd40
|
WO2003059913A1
(fr)
|
2002-01-10 |
2003-07-24 |
Bayer Healthcare Ag |
Inhibiteurs de la rho-kinase
|
CN1627944A
(zh)
|
2002-01-17 |
2005-06-15 |
神经能质公司 |
取代的喹唑啉-4-基胺类似物作为辣椒辣素调节剂
|
JP4469179B2
(ja)
|
2002-01-23 |
2010-05-26 |
バイエル ファーマセチカル コーポレーション |
Rhoキナーゼ阻害剤としてのピリミジン誘導体
|
WO2003062227A1
(fr)
|
2002-01-23 |
2003-07-31 |
Bayer Pharmaceuticals Corporation |
Inhibiteurs de kinase rho
|
NZ534171A
(en)
|
2002-02-01 |
2007-06-29 |
Astrazeneca Ab |
Quinazoline compounds for the treatment of diseases associated with angiogenesis and/or increased vascular permeability
|
EP1481971B1
(fr)
*
|
2002-02-06 |
2011-11-16 |
Ube Industries, Ltd. |
Procede relatif a l'elaboration d'un compose 4-aminoquinazoline
|
US20050176740A1
(en)
*
|
2002-04-08 |
2005-08-11 |
Spector Neil L. |
Cancer treatment method comprising administering an erb-family inhibitor and a raf and/or ras inhibitor
|
DE10221018A1
(de)
|
2002-05-11 |
2003-11-27 |
Boehringer Ingelheim Pharma |
Verwendung von Hemmern der EGFR-vermittelten Signaltransduktion zur Behandlung von gutartiger Prostatahyperplasie (BPH)/Prostatahypertrophie
|
WO2003101491A1
(fr)
*
|
2002-06-03 |
2003-12-11 |
Mitsubishi Pharma Corporation |
Moyens preventifs et/ou therapeutiques destines a des sujets presentant l'expression ou l'activation de her2 et/ou egfr
|
UA77303C2
(en)
|
2002-06-14 |
2006-11-15 |
Pfizer |
Derivatives of thienopyridines substituted by benzocondensed heteroarylamide useful as therapeutic agents, pharmaceutical compositions and methods for their use
|
US20040048887A1
(en)
*
|
2002-07-09 |
2004-03-11 |
Boehringer Ingelheim Pharma Gmbh & Co. Kg |
Pharmaceutical compositions based on anticholinergics and EGFR kinase inhibitors
|
EP1528925B1
(fr)
|
2002-07-09 |
2009-04-22 |
Astrazeneca AB |
Derives de quinazoline utilises dans le traitement du cancer
|
GB0215823D0
(en)
|
2002-07-09 |
2002-08-14 |
Astrazeneca Ab |
Quinazoline derivatives
|
JP4703183B2
(ja)
*
|
2002-07-15 |
2011-06-15 |
シンフォニー エボルーション, インク. |
受容体型キナーゼモジュレーターおよびその使用方法
|
GB0304367D0
(en)
*
|
2003-02-26 |
2003-04-02 |
Pharma Mar Sau |
Methods for treating psoriasis
|
GB0225579D0
(en)
|
2002-11-02 |
2002-12-11 |
Astrazeneca Ab |
Chemical compounds
|
US8505468B2
(en)
*
|
2002-11-19 |
2013-08-13 |
Sharp Kabushiki Kaisha |
Substrate accommodating tray
|
MXPA05006123A
(es)
*
|
2002-12-13 |
2005-09-30 |
Neurogen Corp |
Analogos de quinazolin-4-ilamina 2-sustituida como moduladores de receptores de capsaicina.
|
EA008501B1
(ru)
|
2002-12-19 |
2007-06-29 |
Пфайзер Инк. |
2-(1н-индазол-6-иламино)бензамидные соединения как ингибиторы протеинкиназ, полезные для лечения офтальмологических заболеваний
|
WO2004056812A1
(fr)
*
|
2002-12-23 |
2004-07-08 |
Astrazeneca Ab |
Derives de 4-(pyridin-4-ylamino)-quinazoline utilises comme agents anticancereux
|
WO2004060400A1
(fr)
*
|
2003-01-06 |
2004-07-22 |
Mitsubishi Pharma Corp |
Recepteur antipsychotique du facteur de croissance epitheliale a ciblage moleculaire
|
US7223749B2
(en)
|
2003-02-20 |
2007-05-29 |
Boehringer Ingelheim International Gmbh |
Bicyclic heterocycles, pharmaceutical compositions containing these compounds, their use and processes for preparing them
|
AP2114A
(en)
|
2003-02-26 |
2010-03-04 |
Sugen Inc |
Aminoheteroaryl compounds as protein kinase inhibitors
|
BRPI0410634A
(pt)
|
2003-05-30 |
2006-06-13 |
Astrazeneca Uk Ltd |
processo
|
TW200510373A
(en)
|
2003-07-14 |
2005-03-16 |
Neurogen Corp |
Substituted quinolin-4-ylamine analogues
|
US7329664B2
(en)
|
2003-07-16 |
2008-02-12 |
Neurogen Corporation |
Substituted (7-pyridyl-4-phenylamino-quinazolin-2-yl)-methanol analogues
|
KR101254371B1
(ko)
|
2003-07-18 |
2013-05-02 |
암젠 프레몬트 인코포레이티드 |
간세포 성장인자에 결합하는 분리된 항체
|
EP1653986A4
(fr)
|
2003-08-01 |
2007-03-14 |
Smithkline Beecham Corp |
Traitement des cancers exprimant p95 sp erbb2 /sp
|
BRPI0413876A
(pt)
|
2003-08-29 |
2006-10-24 |
Pfizer |
tienopiridin-fenilacetamidas e seus derivados úteis como agentes antiangiogênicos
|
GB0321066D0
(en)
*
|
2003-09-09 |
2003-10-08 |
Pharma Mar Sau |
New antitumoral compounds
|
AR045563A1
(es)
|
2003-09-10 |
2005-11-02 |
Warner Lambert Co |
Anticuerpos dirigidos a m-csf
|
PL2213661T3
(pl)
|
2003-09-26 |
2011-12-30 |
Exelixis Inc |
Modulatory c-Met i sposoby ich zastosowania
|
DE10349113A1
(de)
|
2003-10-17 |
2005-05-12 |
Boehringer Ingelheim Pharma |
Verfahren zur Herstellung von Aminocrotonylverbindungen
|
EP1682123A1
(fr)
*
|
2003-11-07 |
2006-07-26 |
SmithKline Beecham (Cork) Limited |
Methode de traitement du cancer
|
WO2005044788A1
(fr)
|
2003-11-11 |
2005-05-19 |
Eisai Co., Ltd. |
Derive d'uree et son procede de production
|
GB0326459D0
(en)
|
2003-11-13 |
2003-12-17 |
Astrazeneca Ab |
Quinazoline derivatives
|
JP4936897B2
(ja)
*
|
2003-12-18 |
2012-05-23 |
ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ |
抗増殖剤としてのピリド−およびピリミドピリミジン誘導体
|
GB0330002D0
(en)
|
2003-12-24 |
2004-01-28 |
Astrazeneca Ab |
Quinazoline derivatives
|
JP2007532658A
(ja)
*
|
2004-04-16 |
2007-11-15 |
スミスクライン ビーチャム コーポレーション |
がんの治療方法
|
NZ550796A
(en)
|
2004-05-06 |
2010-07-30 |
Warner Lambert Co |
4-phenylamino-quinazolin-6-yl-amides
|
MXPA06013635A
(es)
*
|
2004-06-03 |
2007-02-28 |
Smithkline Beecam Cork Ltd |
Metodo para el tratamiento de cancer.
|
BRPI0511765A
(pt)
*
|
2004-06-04 |
2008-01-08 |
Smithkline Beechman Cork Ltd |
métodos de tratar cáncer de mama, de pulmão, e colo-retal em um mamìfero
|
US7452887B2
(en)
*
|
2004-06-04 |
2008-11-18 |
Amphora Discovery Corporation |
Quinoline- and isoquinoline-based compounds exhibiting ATP-utilizing enzyme inhibitory activity, and compositions, and uses thereof
|
US20100226931A1
(en)
*
|
2004-06-24 |
2010-09-09 |
Nicholas Valiante |
Compounds for immunopotentiation
|
EP2277595A3
(fr)
|
2004-06-24 |
2011-09-28 |
Novartis Vaccines and Diagnostics, Inc. |
Composés pour potentialiser l'immunité
|
US20060035893A1
(en)
|
2004-08-07 |
2006-02-16 |
Boehringer Ingelheim International Gmbh |
Pharmaceutical compositions for treatment of respiratory and gastrointestinal disorders
|
AU2005276135B2
(en)
|
2004-08-26 |
2011-04-28 |
Pfizer Inc. |
Enantiomerically pure aminoheteroaryl compounds as protein kinase inhibitors
|
KR20070053205A
(ko)
|
2004-09-17 |
2007-05-23 |
에자이 알앤드디 매니지먼트 가부시키가이샤 |
의약 조성물
|
TW200621251A
(en)
|
2004-10-12 |
2006-07-01 |
Neurogen Corp |
Substituted biaryl quinolin-4-ylamine analogues
|
US7652009B2
(en)
|
2004-11-30 |
2010-01-26 |
Amgem Inc. |
Substituted heterocycles and methods of use
|
GB0427131D0
(en)
*
|
2004-12-10 |
2005-01-12 |
Glaxosmithkline Biolog Sa |
Novel combination
|
JP4881875B2
(ja)
|
2004-12-14 |
2012-02-22 |
アストラゼネカ アクチボラグ |
抗腫瘍剤としてのピラゾロピリミジン化合物
|
JP5291345B2
(ja)
*
|
2004-12-17 |
2013-09-18 |
スミスクライン ビーチャム (コーク) リミテッド |
癌治療法
|
US7812022B2
(en)
*
|
2004-12-21 |
2010-10-12 |
Glaxosmithkline Llc |
2-pyrimidinyl pyrazolopyridine ErbB kinase inhibitors
|
ATE430747T1
(de)
*
|
2004-12-21 |
2009-05-15 |
Smithkline Beecham Corp |
2-pyrimidinyl-pyrazolopyridin-erbb- kinaseinhibitoren
|
PE20060777A1
(es)
|
2004-12-24 |
2006-10-06 |
Boehringer Ingelheim Int |
Derivados de indolinona para el tratamiento o la prevencion de enfermedades fibroticas
|
JP2008526997A
(ja)
*
|
2005-01-14 |
2008-07-24 |
ニューロジェン・コーポレーション |
ヘテロアリール置換キノリン−4−イルアミン類縁体
|
PT2301531T
(pt)
|
2005-02-18 |
2018-07-30 |
Abraxis Bioscience Llc |
Combinações e modos de administração de agentes terapêuticos e terapia de combinação
|
US8735394B2
(en)
|
2005-02-18 |
2014-05-27 |
Abraxis Bioscience, Llc |
Combinations and modes of administration of therapeutic agents and combination therapy
|
US20060216288A1
(en)
*
|
2005-03-22 |
2006-09-28 |
Amgen Inc |
Combinations for the treatment of cancer
|
KR20080003390A
(ko)
|
2005-03-31 |
2008-01-07 |
어젠시스 인코포레이티드 |
161p2f10b 단백질과 결합하는 항체 및 관련 분자
|
PE20061430A1
(es)
*
|
2005-04-19 |
2007-01-25 |
Smithkline Beecham Cork Ltd |
Composicion farmaceutica que comprende compuestos de 4-quinazolinaminas
|
MX2007013304A
(es)
|
2005-04-26 |
2007-12-13 |
Pfizer |
Anticuerpos de p-caderina.
|
US9006240B2
(en)
|
2005-08-02 |
2015-04-14 |
Eisai R&D Management Co., Ltd. |
Method for assay on the effect of vascularization inhibitor
|
TWI453218B
(zh)
|
2005-09-07 |
2014-09-21 |
Amgen Fremont Inc |
針對類活化素受體激酶-1之人類單株抗體
|
EP1928861B1
(fr)
|
2005-09-20 |
2010-11-17 |
AstraZeneca AB |
Composés de 4- (ih-indazol-5-yl-amino)-quinazoline utilisés comme inhibiteurs des recepteurs erbb des tyrosines kinases pour traiter le cancer
|
EP1926996B1
(fr)
|
2005-09-20 |
2011-11-09 |
OSI Pharmaceuticals, Inc. |
Marqueurs biologiques prédictifs d'une réaction anticancéreuse aux inhibiteurs kinase du récepteur du facteur de croissance 1 analogue à l'insuline
|
UA96139C2
(uk)
|
2005-11-08 |
2011-10-10 |
Дженентек, Інк. |
Антитіло до нейропіліну-1 (nrp1)
|
JP5688877B2
(ja)
|
2005-11-11 |
2015-03-25 |
ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング |
癌疾患の治療用キナゾリン誘導体
|
US7807673B2
(en)
*
|
2005-12-05 |
2010-10-05 |
Glaxosmithkline Llc |
2-pyrimidinyl pyrazolopyridine ErbB kinase inhibitors
|
CN101003514A
(zh)
|
2006-01-20 |
2007-07-25 |
上海艾力斯医药科技有限公司 |
喹唑啉衍生物、其制备方法及用途
|
JO2660B1
(en)
|
2006-01-20 |
2012-06-17 |
نوفارتيس ايه جي |
Pi-3 inhibitors and methods of use
|
AR059066A1
(es)
|
2006-01-27 |
2008-03-12 |
Amgen Inc |
Combinaciones del inhibidor de la angiopoyetina -2 (ang2) y el inhibidor del factor de crecimiento endotelial vascular (vegf)
|
AU2007211684A1
(en)
*
|
2006-01-31 |
2007-08-09 |
F. Hoffmann-La Roche Ag |
7H-pyrido[3,4-d]pyrimidin-8-ones, their manufacture and use as protein kinase inhibitors
|
PE20070978A1
(es)
*
|
2006-02-14 |
2007-11-15 |
Novartis Ag |
COMPUESTOS HETEROCICLICOS COMO INHIBIDORES DE FOSFATIDILINOSITOL 3-QUINASAS (PI3Ks)
|
AR060358A1
(es)
*
|
2006-04-06 |
2008-06-11 |
Novartis Vaccines & Diagnostic |
Quinazolinas para la inhibicion de pdk 1
|
US20090203718A1
(en)
*
|
2006-04-13 |
2009-08-13 |
Smithkline Beecham (Cork) Ltd. |
Cancer treatment method
|
AU2007240496A1
(en)
|
2006-04-19 |
2007-11-01 |
Novartis Ag |
Indazole compounds and methods for inhibition of CDC7
|
MX2008013990A
(es)
|
2006-05-09 |
2009-01-29 |
Pfizer Prod Inc |
Derivados de cicloalquilamino acidos.
|
NL2000613C2
(nl)
|
2006-05-11 |
2007-11-20 |
Pfizer Prod Inc |
Triazoolpyrazinederivaten.
|
EP2036557B1
(fr)
|
2006-05-18 |
2015-10-21 |
Eisai R&D Management Co., Ltd. |
Agent antitumoral destiné au cancer de la thyroïde
|
DE602006004196D1
(de)
*
|
2006-06-01 |
2009-01-22 |
Cellzome Ag |
Verfahren zur Identifizierung von mit ZAP-70 wechselwirkenden Molekülen und zur ZAP-70-Reinigung
|
WO2008005469A2
(fr)
|
2006-06-30 |
2008-01-10 |
Schering Corporation |
Biomarqueur igfbp2
|
PE20121506A1
(es)
|
2006-07-14 |
2012-11-26 |
Amgen Inc |
Compuestos triazolopiridinas como inhibidores de c-met
|
US8217177B2
(en)
|
2006-07-14 |
2012-07-10 |
Amgen Inc. |
Fused heterocyclic derivatives and methods of use
|
US20110053964A1
(en)
*
|
2006-08-22 |
2011-03-03 |
Roger Tung |
4-aminoquinazoline derivatives and methods of use thereof
|
CA2661223A1
(fr)
|
2006-08-22 |
2008-02-28 |
Concert Pharmaceuticals Inc. |
Derives de 4-aminoquinazoline et leurs procedes d'utilisation
|
CN101511793B
(zh)
|
2006-08-28 |
2011-08-03 |
卫材R&D管理有限公司 |
针对未分化型胃癌的抗肿瘤剂
|
KR20090074202A
(ko)
|
2006-09-18 |
2009-07-06 |
베링거 인겔하임 인터내셔날 게엠베하 |
Egfr 돌연변이를 갖는 암을 치료하는 방법
|
JP2010505811A
(ja)
*
|
2006-10-04 |
2010-02-25 |
ファイザー・プロダクツ・インク |
カルシウム受容体アンタゴニストとしてのピリド[4,3−d]ピリミジン−4(3H)−オン誘導体
|
WO2008044045A1
(fr)
|
2006-10-12 |
2008-04-17 |
Astex Therapeutics Limited |
Combinaisons pharmaceutiques
|
US8916552B2
(en)
|
2006-10-12 |
2014-12-23 |
Astex Therapeutics Limited |
Pharmaceutical combinations
|
WO2008054633A1
(fr)
*
|
2006-10-31 |
2008-05-08 |
Janssen Pharmaceutica N.V. |
Dérivés d'hydrazone en tant qu'inhibiteurs de kinase
|
WO2008063888A2
(fr)
|
2006-11-22 |
2008-05-29 |
Plexxikon, Inc. |
Composés modulant l'activité de c-fms et/ou de c-kit et utilisations associées
|
CA2672828A1
(fr)
|
2006-12-13 |
2008-06-26 |
Schering Corporation |
Procedes de traitements
|
CA2672438A1
(fr)
|
2006-12-20 |
2008-07-03 |
Amgen Inc. |
Heterocycles substitues et leurs methodes d'utilisation
|
WO2008086014A2
(fr)
|
2007-01-09 |
2008-07-17 |
Amgen Inc. |
Dérivés de bis-aryl amide et procédés d'utilisation
|
EP2119707B1
(fr)
|
2007-01-29 |
2015-01-14 |
Eisai R&D Management Co., Ltd. |
Composition destinée au traitement d'un cancer de l'estomac de type indifférencié
|
CN101245050A
(zh)
|
2007-02-14 |
2008-08-20 |
上海艾力斯医药科技有限公司 |
4-苯胺喹唑啉衍生物的盐
|
AU2008219166B2
(en)
|
2007-02-16 |
2013-05-16 |
Amgen Inc. |
Nitrogen-containing heterocyclyl ketones and their use as c-Met inhibitors
|
ES2529790T3
(es)
|
2007-04-13 |
2015-02-25 |
Dana-Farber Cancer Institute, Inc. |
Métodos de tratamiento de cáncer resistente a agentes terapéuticos de ERBB
|
KR20120011093A
(ko)
*
|
2007-05-09 |
2012-02-06 |
화이자 인코포레이티드 |
치환된 헤테로사이클릭 유도체 및 조성물 및 항균제로서의 이의 약학적 용도
|
US20110245496A1
(en)
*
|
2007-06-11 |
2011-10-06 |
Andrew Simon Craig |
Quinazoline Salt Compounds
|
UY31137A1
(es)
*
|
2007-06-14 |
2009-01-05 |
Smithkline Beecham Corp |
Derivados de quinazolina como inhibidores de la pi3 quinasa
|
PT2188313T
(pt)
|
2007-08-21 |
2017-12-12 |
Amgen Inc |
Proteínas de ligação ao antigénio c-fms humano
|
PL2185574T3
(pl)
|
2007-09-07 |
2013-09-30 |
Agensys Inc |
Przeciwciała i powiązane cząsteczki, które wiążą się do białek 24P4C12
|
US20090215802A1
(en)
*
|
2007-09-13 |
2009-08-27 |
Protia, Llc |
Deuterium-enriched lapatinib
|
MX2010004259A
(es)
*
|
2007-10-19 |
2010-08-31 |
Pharma Mar Sa |
Tratamientos antitumorales mejorados.
|
EP2212432A4
(fr)
|
2007-10-22 |
2011-10-19 |
Schering Corp |
Anticorps anti-vegf entièrement humains et leurs procédés d'utilisation
|
GEP20125603B
(en)
|
2007-10-29 |
2012-08-10 |
Nacto Pharma Ltd |
Novel 4-(tetrazol-5-yl)-quinazoline derivatives as anti cancer agents
|
EP2218712B1
(fr)
|
2007-11-09 |
2015-07-01 |
Eisai R&D Management Co., Ltd. |
Combinaison d'une substance antiangiogénique et d'un complexe de platine antitumoral
|
AR069798A1
(es)
|
2007-12-20 |
2010-02-17 |
Novartis Ag |
Derivados de 1, 3-tiazol, metodos para su preparacion, composiciones farmaceuticas que los comprenden y su uso en la manufactura de medicamentos para el tratamiento de enfermedades mediadas por la fosfatidilinositol 3-cinasa.
|
CN101492445A
(zh)
*
|
2008-01-22 |
2009-07-29 |
孙飘扬 |
杂芳族化合物、其制备方法以及其用途
|
WO2009095480A1
(fr)
*
|
2008-01-30 |
2009-08-06 |
Pharma Mar, S.A. |
Traitements antitumoraux améliorés
|
US20110015135A1
(en)
*
|
2008-03-07 |
2011-01-20 |
Pharma Mar S.A. |
Antitumoral Treatments
|
KR20210131473A
(ko)
|
2008-03-18 |
2021-11-02 |
제넨테크, 인크. |
항-her2 항체-약물 접합체와 화학요법제의 병용물, 및 사용 방법
|
WO2009137714A2
(fr)
|
2008-05-07 |
2009-11-12 |
Teva Pharmaceutical Industries Ltd. |
Formes de ditosylate de lapatinib et procédés pour leur préparation
|
US20090306106A1
(en)
*
|
2008-05-15 |
2009-12-10 |
Leonid Metsger |
Forms of crystalline lapatinib and processes for preparation thereof
|
CN101584696A
(zh)
|
2008-05-21 |
2009-11-25 |
上海艾力斯医药科技有限公司 |
包含喹唑啉衍生物的组合物及制备方法、用途
|
US20100197915A1
(en)
*
|
2008-08-06 |
2010-08-05 |
Leonid Metsger |
Lapatinib intermediates
|
EP2158913A1
(fr)
|
2008-08-25 |
2010-03-03 |
Ratiopharm GmbH |
Composition pharmaceutique comportant de la N-[3-chhloro-4-[3-fluorophenyl)methoxy)phenyl]6-[5[[[2-(methylsulfonyl)ethyl]amino]methyl]-2-furyl]-4-quinazolinamine
|
EP2158912A1
(fr)
|
2008-08-25 |
2010-03-03 |
Ratiopharm GmbH |
Composition pharmaceutique comportant de la N-[3-chhloro-4-[3-fluorophenyl)methoxy)phenyl]6-[5[[[2-(methylsulfonyl)ethyl]amino]methyl]-2-furyl]-4-quinazolinamine
|
US20100087459A1
(en)
*
|
2008-08-26 |
2010-04-08 |
Leonid Metsger |
Forms of lapatinib compounds and processes for the preparation thereof
|
CA2737597C
(fr)
|
2008-10-16 |
2017-03-14 |
University Of Pittsburgh-Of The Commonwealth System Of Higher Education |
Anticorps entierement humains diriges contre un antigene associe au melanome de masse moleculaire elevee et leurs utilisations
|
EP2358666A1
(fr)
|
2008-11-03 |
2011-08-24 |
Natco Pharma Limited |
Nouveau procédé de préparation de lapatinib et de ses sels de qualité pharmaceutique
|
EP2349235A1
(fr)
|
2008-11-07 |
2011-08-03 |
Triact Therapeutics, Inc. |
Utilisation de dérivés de butane catécholique dans la thérapie du cancer
|
JP5677318B2
(ja)
|
2009-01-16 |
2015-02-25 |
エクセリクシス, インク. |
N−(4−{[6,7−ビス(メチルオキシ)キノリン−4−イル]オキシ}フェニル)−n’−(4−フルオロフェニル)シクロプロパン−1,1−ジカルボキサミドのリンゴ酸塩およびその結晶質形態
|
CN101787017A
(zh)
*
|
2009-01-23 |
2010-07-28 |
岑均达 |
光学纯喹唑啉类化合物
|
SG172857A1
(en)
|
2009-02-09 |
2011-08-29 |
Supergen Inc |
Pyrrolopyrimidinyl axl kinase inhibitors
|
JP2012518657A
(ja)
|
2009-02-25 |
2012-08-16 |
オーエスアイ・ファーマシューティカルズ,エルエルシー |
併用抗癌治療
|
JP2012519170A
(ja)
|
2009-02-26 |
2012-08-23 |
オーエスアイ・ファーマシューティカルズ,エルエルシー |
生体内の腫瘍細胞のemtステータスをモニターするためのinsitu法
|
WO2010098866A1
(fr)
|
2009-02-27 |
2010-09-02 |
Supergen, Inc. |
Inhibiteurs cyclopentathiophène/cyclohexathiophène de l'adn méthyltransférase
|
US8465912B2
(en)
|
2009-02-27 |
2013-06-18 |
OSI Pharmaceuticals, LLC |
Methods for the identification of agents that inhibit mesenchymal-like tumor cells or their formation
|
WO2010099363A1
(fr)
|
2009-02-27 |
2010-09-02 |
Osi Pharmaceuticals, Inc. |
Méthodes d'identification d'agents qui inhibent les cellules cancéreuses mésenchymateuses ou leur formation
|
WO2010099138A2
(fr)
|
2009-02-27 |
2010-09-02 |
Osi Pharmaceuticals, Inc. |
Procédés pour l'identification d'agents qui inhibent les cellules tumorales de type mésenchymateuses ou leur formation
|
EP2403339B1
(fr)
|
2009-03-06 |
2017-01-18 |
Merck Sharp & Dohme Corp. |
Thérapie de combinaison anti-cancer avec un inhibiteur de akt et d'autres agents anti-cancer
|
WO2010107968A1
(fr)
|
2009-03-18 |
2010-09-23 |
Osi Pharmaceuticals, Inc. |
Plurithérapie contre le cancer comprenant l'administration d'un inhibiteur de l'egfr et d'un inhibiteur de l'igf-1r
|
ES2572728T3
(es)
*
|
2009-03-20 |
2016-06-02 |
F. Hoffmann-La Roche Ag |
Anticuerpos anti-HER biespecíficos
|
US8530492B2
(en)
|
2009-04-17 |
2013-09-10 |
Nektar Therapeutics |
Oligomer-protein tyrosine kinase inhibitor conjugates
|
WO2010120388A1
(fr)
|
2009-04-17 |
2010-10-21 |
Nektar Therapeutics |
Conjugués inhibiteur de protéine tyrosine kinase-oligomère
|
US8293753B2
(en)
|
2009-07-02 |
2012-10-23 |
Novartis Ag |
Substituted 2-carboxamide cycloamino ureas
|
PT2451445T
(pt)
|
2009-07-06 |
2019-07-10 |
Boehringer Ingelheim Int |
Processo para secagem de bibw2992, dos seus sais e de formulações farmacêuticas sólidas compreendendo este ingrediente ativo
|
UA108618C2
(uk)
|
2009-08-07 |
2015-05-25 |
|
Застосування c-met-модуляторів в комбінації з темозоломідом та/або променевою терапією для лікування раку
|
ME02492B
(fr)
|
2009-08-21 |
2017-02-20 |
Novartis Ag |
Procédé de traitement du cancer
|
EP2473500A2
(fr)
|
2009-09-01 |
2012-07-11 |
Pfizer Inc. |
Dérivés de benzimidazole
|
US8916574B2
(en)
|
2009-09-28 |
2014-12-23 |
Qilu Pharmaceutical Co., Ltd. |
4-(substituted anilino)-quinazoline derivatives useful as tyrosine kinase inhibitors
|
WO2011039759A1
(fr)
*
|
2009-09-29 |
2011-04-07 |
Natco Pharma Limited |
Nouveau procédé de préparation de lapatinib et de ses sels pharmaceutiquement acceptables
|
JP2013510564A
(ja)
|
2009-11-13 |
2013-03-28 |
パンガエア ビオテック、ソシエダッド、リミターダ |
肺癌におけるチロシンキナーゼ阻害剤に対する応答を予測するための分子バイオマーカー
|
CN102079759B
(zh)
*
|
2009-12-01 |
2014-09-17 |
天津药物研究院 |
6位取代的喹唑啉类衍生物、其制备方法和用途
|
AR079256A1
(es)
|
2009-12-04 |
2012-01-04 |
Genentech Inc |
Metodo para el tratamiento del cancer de mama metastasico con trastuzumab-mcc-dm1
|
EP2519526B1
(fr)
|
2009-12-31 |
2014-03-26 |
Centro Nacional de Investigaciones Oncológicas (CNIO) |
Nouveaux composés
|
EP2526102B1
(fr)
|
2010-01-22 |
2017-03-08 |
Fundación Centro Nacional de Investigaciones Oncológicas Carlos III |
Inhibiteurs de la PI3 kinase
|
KR20120127495A
(ko)
|
2010-02-12 |
2012-11-21 |
화이자 인코포레이티드 |
8-플루오로-2-{4-[(메틸아미노)메틸]페닐}-1,3,4,5-테트라하이드로-6h-아제피노[5,4,3-cd]인돌-6-온의 염 및 다형체
|
SG183361A1
(en)
|
2010-02-18 |
2012-09-27 |
Ct Nac Investigaciones Oncologicas Cnio |
Triazolo [4, 5 - b] pyridin derivatives
|
WO2011109572A2
(fr)
|
2010-03-03 |
2011-09-09 |
OSI Pharmaceuticals, LLC |
Marqueurs biologiques prédictifs d'une réponse anticancéreuse aux inhibiteurs de kinase du récepteur du facteur de croissance insulinique 1
|
WO2011109584A2
(fr)
|
2010-03-03 |
2011-09-09 |
OSI Pharmaceuticals, LLC |
Marqueurs biologiques prédictifs d'une réponse anticancéreuse aux inhibiteurs de kinase du récepteur du facteur de croissance insulinique 1
|
US8563719B2
(en)
*
|
2010-03-23 |
2013-10-22 |
Scinopharm Taiwan, Ltd. |
Process and intermediates for preparing lapatinib
|
US8710221B2
(en)
|
2010-03-23 |
2014-04-29 |
Scinopharm Taiwan, Ltd. |
Process and intermediates for preparing lapatinib
|
SG10201906075VA
(en)
|
2010-03-29 |
2019-08-27 |
Abraxis Bioscience Llc |
Methods of treating cancer
|
KR20130028727A
(ko)
|
2010-03-29 |
2013-03-19 |
아브락시스 바이오사이언스, 엘엘씨 |
치료제의 약물 전달 및 유효성 향상 방법
|
WO2011121317A1
(fr)
|
2010-04-01 |
2011-10-06 |
Centro Nacional De Investigaciones Oncologicas (Cnio) |
Imidazo[1,2-b][1,2,3]thiadiazoles en tant qu'inhibiteurs de la kinase protéique ou de la kinase lipidique
|
WO2011146712A1
(fr)
|
2010-05-21 |
2011-11-24 |
Glaxosmithkline Llc |
Combinaison
|
WO2011146710A1
(fr)
|
2010-05-21 |
2011-11-24 |
Glaxosmithkline Llc |
Combinaison
|
KR20190130050A
(ko)
|
2010-06-04 |
2019-11-20 |
아브락시스 바이오사이언스, 엘엘씨 |
췌장암의 치료 방법
|
ES2611479T3
(es)
|
2010-06-16 |
2017-05-09 |
University Of Pittsburgh- Of The Commonwealth System Of Higher Education |
Anticuerpos contra endoplasmina y su uso
|
WO2011161217A2
(fr)
|
2010-06-23 |
2011-12-29 |
Palacký University in Olomouc |
Ciblage du vegfr2
|
AU2011270165B2
(en)
|
2010-06-25 |
2015-12-24 |
Eisai R&D Management Co., Ltd. |
Antitumor agent using compounds having kinase inhibitory effect in combination
|
NZ605449A
(en)
|
2010-07-09 |
2015-03-27 |
Genentech Inc |
Anti-neuropilin antibodies and methods of use
|
CN102344445B
(zh)
*
|
2010-07-23 |
2015-11-25 |
岑均达 |
光学纯喹唑啉类化合物
|
CN102344444B
(zh)
*
|
2010-07-23 |
2015-07-01 |
岑均达 |
光学纯喹唑啉类化合物
|
AR082418A1
(es)
|
2010-08-02 |
2012-12-05 |
Novartis Ag |
Formas cristalinas de 1-(4-metil-5-[2-(2,2,2-trifluoro-1,1-dimetil-etil)-piridin-4-il]-tiazol-2-il)-amida de 2-amida del acido (s)-pirrolidin-1,2-dicarboxilico
|
MX2013002084A
(es)
|
2010-08-31 |
2013-05-09 |
Genentech Inc |
Biomarcadores y metodos de tratamiento.
|
JP5802756B2
(ja)
|
2010-10-20 |
2015-11-04 |
ファイザー・インク |
スムーズンド受容体モジュレーターとしてのピリジン−2−誘導体
|
WO2012052745A1
(fr)
|
2010-10-21 |
2012-04-26 |
Centro Nacional De Investigaciones Oncológicas (Cnio) |
Combinaisons d'inhibiteurs de pi3k avec un second agent antitumoral
|
EA201390611A1
(ru)
|
2010-11-24 |
2014-01-30 |
Глаксо Груп Лимитед |
Мультиспецифические антигенсвязывающие белки, направленные на hgf
|
CN102558160B
(zh)
*
|
2010-12-20 |
2015-09-23 |
天津药物研究院 |
4-取代对甲磺酰胺苯胺基-喹唑啉衍生物及其制备方法和用途
|
CN102558159A
(zh)
*
|
2010-12-20 |
2012-07-11 |
天津药物研究院 |
4-取代间甲磺酰胺苯胺基-喹唑啉衍生物及其制备方法和用途
|
EP2468883A1
(fr)
|
2010-12-22 |
2012-06-27 |
Pangaea Biotech S.L. |
Biomarqueurs moléculaires pour la prédiction de la réponse aux inhibiteurs de la tyrosine kinase dans le cancer du poumon
|
EP2655364A4
(fr)
|
2010-12-23 |
2014-06-11 |
Apotex Pharmachem Inc |
Procédé pour la préparation de lapatinib et de son sel ditosylate
|
US9134297B2
(en)
|
2011-01-11 |
2015-09-15 |
Icahn School Of Medicine At Mount Sinai |
Method and compositions for treating cancer and related methods
|
WO2012098387A1
(fr)
|
2011-01-18 |
2012-07-26 |
Centro Nacional De Investigaciones Oncológicas (Cnio) |
Dérivés de triazolo[4,3-b]pyridazines au cycle 6,7 fusionné utilisés en tant qu'inhibiteurs de pim
|
WO2012104776A1
(fr)
|
2011-01-31 |
2012-08-09 |
Novartis Ag |
Dérivés hétérocycliques inédits
|
WO2012116040A1
(fr)
|
2011-02-22 |
2012-08-30 |
OSI Pharmaceuticals, LLC |
Marqueurs biologiques prédictifs d'une réponse anticancéreuse aux inhibiteurs de la kinase du récepteur du facteur de croissance 1 analogue à l'insuline dans le carcinome hépatocellulaire
|
EP2492688A1
(fr)
|
2011-02-23 |
2012-08-29 |
Pangaea Biotech, S.A. |
Biomarqueurs moléculaires pour la prédiction de la réponse à un traitement antitumoral dans le cancer du poumon
|
AU2012225735B2
(en)
|
2011-03-04 |
2016-03-10 |
Glaxosmithkline Intellectual Property Development Limited |
Amino-quinolines as kinase inhibitors
|
CN103998040B
(zh)
|
2011-03-04 |
2017-03-29 |
江苏康缘药业股份有限公司 |
炔基取代的喹唑啉化合物及其使用方法
|
AU2012225232B2
(en)
|
2011-03-09 |
2016-05-12 |
Richard G. Pestell |
Prostate cancer cell lines, gene signatures and uses thereof
|
CN103648500B
(zh)
|
2011-03-17 |
2016-05-04 |
宾夕法尼亚大学理事会 |
双功能酶制钳型分子的方法和用途
|
WO2012125904A1
(fr)
|
2011-03-17 |
2012-09-20 |
The Trustees Of The University Of Pennsylvania |
Composés imitant des mutations qui se lient au domaine kinase de l'egfr
|
WO2012129145A1
(fr)
|
2011-03-18 |
2012-09-27 |
OSI Pharmaceuticals, LLC |
Polythérapie du cancer du poumon non à petites cellules (nsclc)
|
EP2937349B1
(fr)
|
2011-03-23 |
2016-12-28 |
Amgen Inc. |
Doubles inhibiteurs tricycliques fusionnés de cdk 4/6 et flt3
|
RU2631240C2
(ru)
|
2011-04-01 |
2017-09-20 |
Дженентек, Инк. |
Комбинации соединений-ингибиторов акт и абиратерона, и способы применения
|
US9150644B2
(en)
|
2011-04-12 |
2015-10-06 |
The United States Of America, As Represented By The Secretary, Department Of Health And Human Services |
Human monoclonal antibodies that bind insulin-like growth factor (IGF) I and II
|
CN103402519B
(zh)
|
2011-04-18 |
2015-11-25 |
卫材R&D管理有限公司 |
肿瘤治疗剂
|
CA2830972C
(fr)
|
2011-04-19 |
2018-11-20 |
Pfizer Inc. |
Combinaisons d'anticorps anti-4-1bb et d'anticorps induisant une cytotoxicite a mediation cellulaire dependante d'un anticorps (adcc) pour le traitement du cancer
|
US9896730B2
(en)
|
2011-04-25 |
2018-02-20 |
OSI Pharmaceuticals, LLC |
Use of EMT gene signatures in cancer drug discovery, diagnostics, and treatment
|
WO2012155339A1
(fr)
|
2011-05-17 |
2012-11-22 |
江苏康缘药业股份有限公司 |
Dérivés de la 4-phénylamino-6-buténamide-7-alkyloxy quinazoline, leur procédé de préparation et leur utilisation
|
CA2872979C
(fr)
|
2011-05-19 |
2020-02-18 |
Joaquin Pastor Fernandez |
Composes macrocycliques en tant qu'inhibiteurs de proteine kinases
|
EP2524918A1
(fr)
|
2011-05-19 |
2012-11-21 |
Centro Nacional de Investigaciones Oncológicas (CNIO) |
Imidazopyrazines en tant qu'inhibiteurs de kinase
|
ITMI20110894A1
(it)
*
|
2011-05-20 |
2012-11-21 |
Italiana Sint Spa |
Impurezza del lapatinib e suoi sali
|
JP5414739B2
(ja)
|
2011-05-25 |
2014-02-12 |
三菱電機株式会社 |
半導体テスト治具
|
JP6038128B2
(ja)
|
2011-06-03 |
2016-12-07 |
エーザイ・アール・アンド・ディー・マネジメント株式会社 |
レンバチニブ化合物に対する甲状腺癌対象及び腎臓癌対象の反応性を予測及び評価するためのバイオマーカー
|
WO2013004984A1
(fr)
|
2011-07-07 |
2013-01-10 |
Centro Nacional De Investigaciones Oncologicas (Cnio) |
Composés tricycliques pour l'utilisation en tant qu'inhibiteurs de kinase
|
WO2013005057A1
(fr)
|
2011-07-07 |
2013-01-10 |
Centro Nacional De Investigaciones Oncológicas (Cnio) |
Nouveaux composés
|
WO2013005041A1
(fr)
|
2011-07-07 |
2013-01-10 |
Centro Nacional De Investigaciones Oncológicas (Cnio) |
Composés hétérocycliques tricycliques en tant qu'inhibiteurs de kinases
|
PL3409278T3
(pl)
|
2011-07-21 |
2021-02-22 |
Sumitomo Pharma Oncology, Inc. |
Heterocykliczne inhibitory kinazy białkowej
|
US9499530B2
(en)
|
2011-08-01 |
2016-11-22 |
Hangzhou Minsheng Institutes For Pharma Research |
Quinazoline derivative, composition having the derivative, and use of the derivative in preparing medicament
|
WO2013025939A2
(fr)
|
2011-08-16 |
2013-02-21 |
Indiana University Research And Technology Corporation |
Composés et méthodes de traitement du cancer par l'inhibition du récepteur de l'urokinase
|
TWI547494B
(zh)
|
2011-08-18 |
2016-09-01 |
葛蘭素史克智慧財產發展有限公司 |
作為激酶抑制劑之胺基喹唑啉類
|
US20130084286A1
(en)
|
2011-08-31 |
2013-04-04 |
Thomas E. Januario |
Diagnostic markers
|
JP5914667B2
(ja)
|
2011-09-22 |
2016-05-11 |
ファイザー・インク |
ピロロピリミジンおよびプリン誘導体
|
AU2012321248A1
(en)
|
2011-09-30 |
2014-04-24 |
Genentech, Inc. |
Diagnostic methylation markers of epithelial or mesenchymal phenotype and response to EGFR kinase inhibitor in tumours or tumour cells
|
CA2848842C
(fr)
|
2011-10-04 |
2020-09-29 |
King's College London |
Anticorps ige anti-hmw-maa
|
EA023935B1
(ru)
|
2011-10-28 |
2016-07-29 |
Новартис Аг |
Производные пурина и их применение для лечения заболевания
|
MX2014005570A
(es)
|
2011-11-08 |
2014-05-30 |
Pfizer |
El uso de anticuerpos anti factor estimulante de la colonia de macrofagos para tratar trastornos inflamatorios.
|
WO2013080218A1
(fr)
|
2011-11-28 |
2013-06-06 |
Fresenius Kabi Oncology Ltd. |
Nouveaux intermédiaires et procédé de préparation de lapatinib et de ses sels pharmaceutiquement acceptables
|
EP2809805A1
(fr)
|
2012-01-31 |
2014-12-10 |
SmithKline Beecham (Cork) Limited |
Méthode de traitement du cancer
|
AR090263A1
(es)
|
2012-03-08 |
2014-10-29 |
Hoffmann La Roche |
Terapia combinada de anticuerpos contra el csf-1r humano y las utilizaciones de la misma
|
JP2015512425A
(ja)
|
2012-04-03 |
2015-04-27 |
ノバルティス アーゲー |
チロシンキナーゼ阻害剤との組合せ製品及びそれらの使用
|
WO2013152252A1
(fr)
|
2012-04-06 |
2013-10-10 |
OSI Pharmaceuticals, LLC |
Polythérapie antinéoplasique
|
EP2861302A4
(fr)
|
2012-05-14 |
2016-08-24 |
Prostagene Llc |
Utilisation de modulateurs de ccr5 dans le traitement du cancer
|
SG11201406550QA
(en)
|
2012-05-16 |
2014-11-27 |
Novartis Ag |
Dosage regimen for a pi-3 kinase inhibitor
|
WO2013190089A1
(fr)
|
2012-06-21 |
2013-12-27 |
Pangaea Biotech, S.L. |
Biomarqueurs moléculaires permettant de prédire l'issue dans le cancer du poumon
|
US9505749B2
(en)
|
2012-08-29 |
2016-11-29 |
Amgen Inc. |
Quinazolinone compounds and derivatives thereof
|
TWI592417B
(zh)
|
2012-09-13 |
2017-07-21 |
葛蘭素史克智慧財產發展有限公司 |
胺基喹唑啉激酶抑制劑之前藥
|
DK2909181T3
(da)
|
2012-10-16 |
2017-11-20 |
Tolero Pharmaceuticals Inc |
PKM2-modulatorer og fremgangsmåder til anvendelse deraf
|
CZ2012712A3
(cs)
|
2012-10-17 |
2014-04-30 |
Zentiva, K.S. |
Nový způsob výroby klíčového intermediátu výroby lapatinibu
|
CN102942561A
(zh)
*
|
2012-11-06 |
2013-02-27 |
深圳海王药业有限公司 |
4-氨基喹唑啉杂环化合物及其用途
|
US9260426B2
(en)
|
2012-12-14 |
2016-02-16 |
Arrien Pharmaceuticals Llc |
Substituted 1H-pyrrolo [2, 3-b] pyridine and 1H-pyrazolo [3, 4-b] pyridine derivatives as salt inducible kinase 2 (SIK2) inhibitors
|
AU2013364953A1
(en)
|
2012-12-21 |
2015-04-30 |
Eisai R&D Management Co., Ltd. |
Amorphous form of quinoline derivative, and method for producing same
|
CN103896889B
(zh)
*
|
2012-12-27 |
2016-05-25 |
上海创诺制药有限公司 |
拉帕替尼中间体及其制备方法和应用
|
CA2900652C
(fr)
|
2013-02-15 |
2021-05-04 |
Kala Pharmaceuticals, Inc. |
Composes therapeutiques et utilisations de ceux-ci
|
ES2635620T3
(es)
|
2013-02-19 |
2017-10-04 |
Hexal Ag |
Composición farmacéutica que comprende n-[3-cloro-4-(3-fluorobenciloxi)fenil]-6-[5({[2-(metilsulfonil)etil]amino} metil)-2-furil]quinazolin-4-amina o una sal, solvato o sal solvatada farmacéuticamente aceptables de la misma
|
BR112015020139A2
(pt)
|
2013-02-20 |
2017-07-18 |
Kala Pharmaceuticals Inc |
compostos terapêuticos e usos dos mesmos
|
US9688688B2
(en)
|
2013-02-20 |
2017-06-27 |
Kala Pharmaceuticals, Inc. |
Crystalline forms of 4-((4-((4-fluoro-2-methyl-1H-indol-5-yl)oxy)-6-methoxyquinazolin-7-yl)oxy)-1-(2-oxa-7-azaspiro[3.5]nonan-7-yl)butan-1-one and uses thereof
|
ES2654100T3
(es)
|
2013-02-21 |
2018-02-12 |
Glaxosmithkline Intellectual Property Development Limited |
Quinazolinas como inhibidores de quinasa
|
EP2958592A1
(fr)
|
2013-02-22 |
2015-12-30 |
F. Hoffmann-La Roche AG |
Méthodes de traitement du cancer et de prévention de résistance aux médicaments
|
CN103159747A
(zh)
*
|
2013-02-26 |
2013-06-19 |
常州鸿创高分子科技有限公司 |
一种二对甲苯磺酸拉帕替尼的合成方法
|
US9834575B2
(en)
|
2013-02-26 |
2017-12-05 |
Triact Therapeutics, Inc. |
Cancer therapy
|
US9468681B2
(en)
|
2013-03-01 |
2016-10-18 |
California Institute Of Technology |
Targeted nanoparticles
|
US9925240B2
(en)
|
2013-03-06 |
2018-03-27 |
Genentech, Inc. |
Methods of treating and preventing cancer drug resistance
|
MX2015012062A
(es)
|
2013-03-14 |
2016-05-05 |
Tolero Pharmaceuticals Inc |
Inhibidores de jak2 y alk2 y metodos para su uso.
|
BR112015022604A2
(pt)
|
2013-03-14 |
2017-10-24 |
Genentech Inc |
usos de um modulador de modificador de cromatina e um antagonista de egfr
|
KR20150130451A
(ko)
|
2013-03-15 |
2015-11-23 |
제넨테크, 인크. |
암 치료 방법 및 항암제 내성 예방을 위한 방법
|
EP2976085A1
(fr)
|
2013-03-21 |
2016-01-27 |
INSERM - Institut National de la Santé et de la Recherche Médicale |
Méthode et composition pharmaceutique pour l'utilisation dans le traitement de maladies hépatiques chroniques associées à une faible expression d'hepcidine
|
WO2014170910A1
(fr)
|
2013-04-04 |
2014-10-23 |
Natco Pharma Limited |
Procédé de préparation du lapatinib
|
US9206188B2
(en)
|
2013-04-18 |
2015-12-08 |
Arrien Pharmaceuticals Llc |
Substituted pyrrolo[2,3-b]pyridines as ITK and JAK inhibitors
|
MX368099B
(es)
|
2013-05-14 |
2019-09-19 |
Eisai R&D Man Co Ltd |
Biomarcadores para predecir y evaluar el grado de respuesta de sujetos con cancer de endometrio a compuestos de tipo lenvatinib.
|
HU231012B1
(hu)
|
2013-05-24 |
2019-11-28 |
Egis Gyógyszergyár Nyilvánosan Működő Részvénytársaság |
Lapatinib sók
|
US9714235B2
(en)
*
|
2013-07-18 |
2017-07-25 |
Shanghai Fochon Pharmaceutical Co., Ltd. |
Quinazoline derivatives, compositions thereof, and use as pharmaceuticals
|
CA2923667A1
(fr)
|
2013-09-09 |
2015-03-12 |
Triact Therapeutics, Inc. |
Traitement du cancer
|
CN105764511B
(zh)
|
2013-10-04 |
2019-01-11 |
艾普托斯生物科学公司 |
用于治疗癌症的组合物和方法
|
NZ719185A
(en)
|
2013-11-01 |
2017-11-24 |
Kala Pharmaceuticals Inc |
Crystalline forms of therapeutic compounds and uses thereof
|
US9890173B2
(en)
|
2013-11-01 |
2018-02-13 |
Kala Pharmaceuticals, Inc. |
Crystalline forms of therapeutic compounds and uses thereof
|
CN103554091B
(zh)
*
|
2013-11-05 |
2016-05-18 |
沈阳工业大学 |
喹唑啉衍生物及其制备方法和用途
|
UA115388C2
(uk)
|
2013-11-21 |
2017-10-25 |
Пфайзер Інк. |
2,6-заміщені пуринові похідні та їх застосування в лікуванні проліферативних захворювань
|
ES2899167T3
(es)
|
2013-12-06 |
2022-03-10 |
Novartis Ag |
Régimen posológico para un inhibidor de fosfatidilinositol 3-cinasas selectivo para la isoforma alfa
|
US9242965B2
(en)
|
2013-12-31 |
2016-01-26 |
Boehringer Ingelheim International Gmbh |
Process for the manufacture of (E)-4-N,N-dialkylamino crotonic acid in HX salt form and use thereof for synthesis of EGFR tyrosine kinase inhibitors
|
EP3636649B1
(fr)
|
2014-01-24 |
2024-02-14 |
Turning Point Therapeutics, Inc. |
Macrocycles de diaryle en tant que modulateurs de kinases de protéines
|
US20160361309A1
(en)
|
2014-02-26 |
2016-12-15 |
Glaxosmithkline Intellectual Property (No.2) Limited |
Methods of treating cancer patients responding to ezh2 inhibitor gsk126
|
JP2017516458A
(ja)
|
2014-03-24 |
2017-06-22 |
ジェネンテック, インコーポレイテッド |
c−met拮抗剤による癌治療及びc−met拮抗剤のHGF発現との相関
|
WO2015156674A2
(fr)
|
2014-04-10 |
2015-10-15 |
Stichting Het Nederlands Kanker Instituut |
Méthode de traitement du cancer
|
WO2015155624A1
(fr)
|
2014-04-10 |
2015-10-15 |
Pfizer Inc. |
Dérivés de dihydropyrrolopyrimidine
|
EP2937346A1
(fr)
|
2014-04-24 |
2015-10-28 |
F.I.S.- Fabbrica Italiana Sintetici S.p.A. |
Co-cristaux de lapatinib
|
HUE046518T2
(hu)
|
2014-04-30 |
2020-03-30 |
Pfizer |
Cikloalkilcsoporthoz kapcsolt diheterociklusos származékok
|
US9388239B2
(en)
|
2014-05-01 |
2016-07-12 |
Consejo Nacional De Investigation Cientifica |
Anti-human VEGF antibodies with unusually strong binding affinity to human VEGF-A and cross reactivity to human VEGF-B
|
WO2016001789A1
(fr)
|
2014-06-30 |
2016-01-07 |
Pfizer Inc. |
Dérivés de pyrimidine en tant qu'inhibiteurs de pi3k destinés à être utilisés dans le traitement du cancer
|
JP6811706B2
(ja)
|
2014-07-31 |
2021-01-13 |
ザ ホンコン ユニヴァーシティ オブ サイエンス アンド テクノロジー |
Epha4に対するヒトモノクローナル抗体及びそれらの使用
|
PT3524595T
(pt)
|
2014-08-28 |
2022-09-19 |
Eisai R&D Man Co Ltd |
Derivado de quinolina altamente puro e método para produção do mesmo
|
WO2016059600A1
(fr)
|
2014-10-17 |
2016-04-21 |
Novartis Ag |
Combinaison de ceritinib et d'un inhibiteur d'egfr
|
CN107531665B
(zh)
|
2014-12-15 |
2021-03-30 |
密歇根大学董事会 |
Egfr和pi3k的小分子抑制剂
|
ES2746839T3
(es)
|
2014-12-18 |
2020-03-09 |
Pfizer |
Derivados de pirimidina y triazina y su uso como inhibidores de AXL
|
RU2739942C2
(ru)
|
2014-12-24 |
2020-12-30 |
Дженентек, Инк. |
Терапевтические, диагностические и прогностические способы для рака мочевого пузыря
|
CN105801565B
(zh)
*
|
2014-12-30 |
2020-04-03 |
天津法莫西医药科技有限公司 |
N-[3-氯-4-[(3-氟苯基)甲氧基]苯基]-6-[(5-甲酰基)呋喃-2-基]-4-喹唑啉胺制备方法
|
JP7041515B2
(ja)
|
2015-01-08 |
2022-03-24 |
ザ ボード オブ トラスティーズ オブ ザ レランド スタンフォード ジュニア ユニバーシティー |
骨、骨髄、及び軟骨の誘導を提供する因子及び細胞
|
MA41414A
(fr)
|
2015-01-28 |
2017-12-05 |
Centre Nat Rech Scient |
Protéines de liaison agonistes d' icos
|
AU2016214923A1
(en)
*
|
2015-02-03 |
2017-08-24 |
Trillium Therapeutics Inc. |
Novel fluorinated derivatives as EGFR inhibitors useful for treating cancers
|
SI3263106T1
(sl)
|
2015-02-25 |
2024-02-29 |
Eisai R&D Management Co., Ltd. |
Postopek zatiranja grenkobe derivata kinolina
|
AU2015384801B2
(en)
|
2015-03-04 |
2022-01-06 |
Eisai R&D Management Co., Ltd. |
Combination of a PD-1 antagonist and a VEGFR/FGFR/RET tyrosine kinase inhibitor for treating cancer
|
WO2016172214A1
(fr)
|
2015-04-20 |
2016-10-27 |
Tolero Pharmaceuticals, Inc. |
Prédiction de la réaction à l'alvocidib par identification de profil mitochondrial
|
MX2017013956A
(es)
|
2015-05-01 |
2018-09-05 |
Cocrystal Pharma Inc |
Analogos de nucleosidos para el tratamiento de la familia de virus flaviviridae y cancer.
|
EP4086264B1
(fr)
|
2015-05-18 |
2023-10-25 |
Sumitomo Pharma Oncology, Inc. |
Promédicaments de l'alvocidib à biodisponibilité augmentée
|
CN106279307B
(zh)
*
|
2015-05-19 |
2019-07-26 |
正大天晴药业集团股份有限公司 |
芳氨代葡萄糖衍生物、其制备方法及抗肿瘤用途
|
AU2016279474B2
(en)
|
2015-06-16 |
2021-09-09 |
Eisai R&D Management Co., Ltd. |
Anticancer agent
|
CN107922609B
(zh)
|
2015-07-01 |
2020-04-24 |
加州理工学院 |
基于阳离子粘酸聚合物的递送系统
|
RU2732405C2
(ru)
|
2015-07-02 |
2020-09-16 |
Тёрнинг Поинт Терапьютикс, Инк. |
Хиральные диарильные макроциклы в качестве модуляторов протеинкиназ
|
WO2017009751A1
(fr)
|
2015-07-15 |
2017-01-19 |
Pfizer Inc. |
Dérivés de pyrimidine
|
EP3325488B1
(fr)
|
2015-07-21 |
2020-06-24 |
Turning Point Therapeutics, Inc. |
Macrocycle diaryle chiral et son utilisation dans le traitement du cancer
|
MX2018001289A
(es)
|
2015-08-03 |
2018-04-30 |
Tolero Pharmaceuticals Inc |
Terapias de combinacion para el tratamiento del cancer.
|
EP3331919A1
(fr)
|
2015-08-07 |
2018-06-13 |
GlaxoSmithKline Intellectual Property Development Limited |
Polythérapie comprenant des anticorps anti-ctla-4
|
US11124483B2
(en)
|
2015-09-02 |
2021-09-21 |
The Regents Of The University Of California |
HER3 ligands and uses thereof
|
CN106632276B
(zh)
*
|
2015-10-28 |
2021-06-15 |
上海天慈生物谷生物工程有限公司 |
一种治疗乳腺癌药物的制备方法
|
EP3370719A1
(fr)
|
2015-11-02 |
2018-09-12 |
Novartis AG |
Schéma posologique pour un inhibiteur de la phosphatidylinositol 3-kinase
|
JP2019505476A
(ja)
|
2015-12-01 |
2019-02-28 |
グラクソスミスクライン、インテレクチュアル、プロパティー、ディベロップメント、リミテッドGlaxosmithkline Intellectual Property Development Limited |
組合せ処置およびその方法
|
MX2018006781A
(es)
|
2015-12-03 |
2018-11-09 |
Agios Pharmaceuticals Inc |
Inhibidores de mat2a para el tratamiento del cancer que no expresen mtap.
|
KR20230042756A
(ko)
|
2016-03-15 |
2023-03-29 |
오리존 지노믹스 에스.에이. |
고형 종양의 치료에 사용하기 위한 lsd1 억제제의 조합물
|
US10689400B2
(en)
|
2016-07-28 |
2020-06-23 |
Turning Point Therapeutics, Inc. |
Macrocycle kinase inhibitors
|
WO2018025221A1
(fr)
|
2016-08-04 |
2018-02-08 |
Glaxosmithkline Intellectual Property Development Limited |
Polythérapie à base d'anticorps anti-icos et anti-pd-1
|
WO2018048746A1
(fr)
|
2016-09-08 |
2018-03-15 |
Kala Pharmaceuticals, Inc. |
Formes cristallines de composés thérapeutiques et leurs utilisations
|
CA3036340A1
(fr)
|
2016-09-08 |
2018-03-15 |
Kala Pharmaceuticals, Inc. |
Formes cristallines de composes therapeutiques et leurs utilisations
|
US10253036B2
(en)
|
2016-09-08 |
2019-04-09 |
Kala Pharmaceuticals, Inc. |
Crystalline forms of therapeutic compounds and uses thereof
|
WO2018060833A1
(fr)
|
2016-09-27 |
2018-04-05 |
Novartis Ag |
Schéma posologique pour l'alpelisib, un inhibiteur de la phosphatidylinositol 3-kinase spécifique de l'isoforme alpha
|
US11279694B2
(en)
|
2016-11-18 |
2022-03-22 |
Sumitomo Dainippon Pharma Oncology, Inc. |
Alvocidib prodrugs and their use as protein kinase inhibitors
|
KR20190099260A
(ko)
|
2016-12-19 |
2019-08-26 |
톨레로 파마수티컬스, 인크. |
프로파일링 펩티드 및 감도 프로파일링을 위한 방법
|
CR20190338A
(es)
|
2016-12-22 |
2019-09-09 |
Amgen Inc |
Inhibidores de kras g12c y métodos para su uso
|
TWI808958B
(zh)
|
2017-01-25 |
2023-07-21 |
美商特普醫葯公司 |
涉及二芳基巨環化合物之組合療法
|
JOP20190272A1
(ar)
|
2017-05-22 |
2019-11-21 |
Amgen Inc |
مثبطات kras g12c وطرق لاستخدامها
|
SG11202000356VA
(en)
|
2017-07-28 |
2020-02-27 |
Turning Point Therapeutics Inc |
Macrocyclic compounds and uses thereof
|
CN116003405A
(zh)
|
2017-09-08 |
2023-04-25 |
美国安进公司 |
Kras g12c的抑制剂及其使用方法
|
US11497756B2
(en)
|
2017-09-12 |
2022-11-15 |
Sumitomo Pharma Oncology, Inc. |
Treatment regimen for cancers that are insensitive to BCL-2 inhibitors using the MCL-1 inhibitor alvocidib
|
WO2019075367A1
(fr)
|
2017-10-13 |
2019-04-18 |
Tolero Pharmaceuticals, Inc. |
Activateurs de pkm2 en combinaison avec des espèces réactives de l'oxygène pour le traitement du cancer
|
WO2019126136A2
(fr)
|
2017-12-18 |
2019-06-27 |
Sterngreene, Inc. |
Composés de pyrimidine utiles en tant qu'inhibiteurs de tyrosine kinase
|
HRP20221502T1
(hr)
|
2017-12-19 |
2023-03-31 |
Turning Point Therapeutics, Inc. |
Makrociklički spojevi za liječenje bolesti
|
WO2019213526A1
(fr)
|
2018-05-04 |
2019-11-07 |
Amgen Inc. |
Inhibiteurs de kras g12c et leurs procédés d'utilisation
|
MX2020010836A
(es)
|
2018-05-04 |
2021-01-08 |
Amgen Inc |
Inhibidores de kras g12c y métodos para su uso.
|
CA3099045A1
(fr)
|
2018-05-10 |
2019-11-14 |
Amgen Inc. |
Inhibiteurs de kras g12c pour le traitement du cancer
|
EP3802535B1
(fr)
|
2018-06-01 |
2022-12-14 |
Amgen, Inc |
Inhibiteurs de kras g12c et leurs procédés d'utilisation
|
WO2019241157A1
(fr)
|
2018-06-11 |
2019-12-19 |
Amgen Inc. |
Inhibiteurs de kras g12c pour le traitement du cancer
|
MX2020012261A
(es)
|
2018-06-12 |
2021-03-31 |
Amgen Inc |
Inhibidores de kras g12c que comprenden un anillo de piperazina y uso de estos en el tratamiento del cancer.
|
CA3099440A1
(fr)
|
2018-06-13 |
2019-12-19 |
California Institute Of Technology |
Nanoparticules permettant de traverser la barriere hematoencephalique et methodes de traitement faisant appel a celle-ci
|
CN112351985B
(zh)
*
|
2018-06-27 |
2023-12-15 |
奥斯考泰克公司 |
吡啶并嘧啶酮衍生物用作axl抑制剂
|
WO2020023910A1
(fr)
|
2018-07-26 |
2020-01-30 |
Tolero Pharmaceuticals, Inc. |
Procédés de traitement de maladies associées à l'expression anormale d'acvr1 et inhibiteurs d'acvr1 destinés à être utilisés dans ceux-ci
|
AU2019352741A1
(en)
|
2018-10-04 |
2021-05-06 |
Assistance Publique-Hôpitaux De Paris (Aphp) |
EGFR inhibitors for treating keratodermas
|
JP7516029B2
(ja)
|
2018-11-16 |
2024-07-16 |
アムジエン・インコーポレーテツド |
Kras g12c阻害剤化合物の重要な中間体の改良合成法
|
JP7377679B2
(ja)
|
2018-11-19 |
2023-11-10 |
アムジエン・インコーポレーテツド |
がん治療のためのkrasg12c阻害剤及び1種以上の薬学的に活性な追加の薬剤を含む併用療法
|
US11053226B2
(en)
|
2018-11-19 |
2021-07-06 |
Amgen Inc. |
KRAS G12C inhibitors and methods of using the same
|
MX2021006544A
(es)
|
2018-12-04 |
2021-07-07 |
Sumitomo Pharma Oncology Inc |
Inhibidores de cinasa dependiente de ciclina 9 (cdk9) y polimorfos de los mismos para uso como agentes para el tratamiento de cancer.
|
CN113474337A
(zh)
|
2018-12-19 |
2021-10-01 |
奥瑞生物药品公司 |
作为fgfr抑制剂用于治疗癌症的7-((3,5-二甲氧基苯基)氨基)喹喔啉衍生物
|
JP2022515198A
(ja)
|
2018-12-19 |
2022-02-17 |
アレイ バイオファーマ インコーポレイテッド |
FGFRチロシンキナーゼの阻害剤としての置換ピラゾロ[1,5-a]ピリジン化合物
|
MX2021007104A
(es)
|
2018-12-20 |
2021-08-11 |
Amgen Inc |
Inhibidores de kif18a.
|
AR117490A1
(es)
|
2018-12-20 |
2021-08-11 |
Amgen Inc |
Inhibidores de kif18a
|
WO2020132653A1
(fr)
|
2018-12-20 |
2020-06-25 |
Amgen Inc. |
Amides d'hétéroaryle utiles en tant qu'inhibiteurs de kif18a
|
JP2022513967A
(ja)
|
2018-12-20 |
2022-02-09 |
アムジエン・インコーポレーテツド |
Kif18a阻害剤として有用なヘテロアリールアミド
|
BR112021014662A2
(pt)
|
2019-02-01 |
2021-09-21 |
Glaxosmithkline Intellectual Property Development Limited |
Tratamentos de combinação para o câncer que compreendem belantamab mafodotin e um anticorpo anti ox40 e usos e métodos dos mesmos
|
KR20210146290A
(ko)
|
2019-02-12 |
2021-12-03 |
스미토모 다이니폰 파마 온콜로지, 인크. |
헤테로시클릭 단백질 키나제 억제제를 포함하는 제제
|
KR20210146288A
(ko)
|
2019-03-01 |
2021-12-03 |
레볼루션 메디슨즈, 인크. |
이환식 헤테로사이클릴 화합물 및 이의 용도
|
WO2020180768A1
(fr)
|
2019-03-01 |
2020-09-10 |
Revolution Medicines, Inc. |
Composés hétéroaryle bicycliques et leurs utilisations
|
WO2020191326A1
(fr)
|
2019-03-20 |
2020-09-24 |
Sumitomo Dainippon Pharma Oncology, Inc. |
Traitement de la leucémie myéloïde aiguë (aml) après échec du vénétoclax
|
KR20210141621A
(ko)
|
2019-03-22 |
2021-11-23 |
스미토모 다이니폰 파마 온콜로지, 인크. |
Pkm2 조정제를 포함하는 조성물 및 그를 사용한 치료 방법
|
EP3738593A1
(fr)
|
2019-05-14 |
2020-11-18 |
Amgen, Inc |
Dosage d'inhibiteur de kras pour le traitement de cancers
|
CA3140392A1
(fr)
|
2019-05-21 |
2020-11-26 |
Amgen Inc. |
Formes a l'etat solide
|
JP2022539178A
(ja)
|
2019-06-26 |
2022-09-07 |
グラクソスミスクライン、インテレクチュアル、プロパティー、ディベロップメント、リミテッド |
Il1rap結合タンパク質
|
JP2022542967A
(ja)
|
2019-08-02 |
2022-10-07 |
アムジエン・インコーポレーテツド |
Kif18a阻害剤
|
EP4007756A1
(fr)
|
2019-08-02 |
2022-06-08 |
Amgen Inc. |
Inhibiteurs de kif18a
|
MX2022001302A
(es)
|
2019-08-02 |
2022-03-02 |
Amgen Inc |
Inhibidores de kif18a.
|
MX2022001296A
(es)
|
2019-08-02 |
2022-02-22 |
Amgen Inc |
Inhibidores de kif18a.
|
WO2021043961A1
(fr)
|
2019-09-06 |
2021-03-11 |
Glaxosmithkline Intellectual Property Development Limited |
Schéma posologique pour le traitement du cancer avec un anticorps agoniste anti-icos et une chimiothérapie
|
WO2021046289A1
(fr)
|
2019-09-06 |
2021-03-11 |
Glaxosmithkline Intellectual Property Development Limited |
Schéma posologique pour le traitement du cancer avec un anticorps agoniste anti-cos et de l'ipilimumab
|
EP4048671A1
(fr)
|
2019-10-24 |
2022-08-31 |
Amgen Inc. |
Dérivés de pyridopyrimidine utiles en tant qu'inhibiteurs de kras g12c et de kras g12d dans le traitement du cancer
|
MX2022005357A
(es)
|
2019-11-04 |
2022-06-02 |
Revolution Medicines Inc |
Inhibidores de ras.
|
CA3159561A1
(fr)
|
2019-11-04 |
2021-05-14 |
Revolution Medicines, Inc. |
Inhibiteurs de ras
|
CR20220243A
(es)
|
2019-11-04 |
2022-08-04 |
Revolution Medicines Inc |
Inhibidores de ras
|
BR112022008858A2
(pt)
|
2019-11-08 |
2022-09-06 |
Revolution Medicines Inc |
Composto, composição farmacêutica e métodos para inibir sos1 em um sujeito, para inibir a interação de sos1 e uma proteína, para tratar ou prevenir uma doença e para tratar ou prevenir câncer
|
IL292315A
(en)
|
2019-11-14 |
2022-06-01 |
Amgen Inc |
Improved synthesis of a kras g12c inhibitory compound
|
US20230192682A1
(en)
|
2019-11-14 |
2023-06-22 |
Amgen Inc. |
Improved synthesis of kras g12c inhibitor compound
|
WO2021108683A1
(fr)
|
2019-11-27 |
2021-06-03 |
Revolution Medicines, Inc. |
Inhibiteurs de ras covalents et leurs utilisations
|
BR112022010086A2
(pt)
|
2020-01-07 |
2022-09-06 |
Revolution Medicines Inc |
Dosagem do inibidor de shp2 e métodos de tratamento de câncer
|
WO2021152495A1
(fr)
|
2020-01-28 |
2021-08-05 |
Glaxosmithkline Intellectual Property Development Limited |
Traitements combinés et utilisations et méthodes associées
|
WO2021155006A1
(fr)
|
2020-01-31 |
2021-08-05 |
Les Laboratoires Servier Sas |
Inhibiteurs de kinases dépendantes des cyclines et leurs utilisations
|
CA3174455A1
(fr)
*
|
2020-03-02 |
2021-09-10 |
Turning Point Therapeutics, Inc. |
Utilisations therapeutiques de composes macrocycliques
|
IL299131A
(en)
|
2020-06-18 |
2023-02-01 |
Revolution Medicines Inc |
Methods for delaying, preventing and treating acquired resistance to RAS inhibitors
|
AU2021344830A1
(en)
|
2020-09-03 |
2023-04-06 |
Revolution Medicines, Inc. |
Use of SOS1 inhibitors to treat malignancies with SHP2 mutations
|
CN116457358A
(zh)
|
2020-09-15 |
2023-07-18 |
锐新医药公司 |
作为ras抑制剂以治疗癌症的吲哚衍生物
|
EP4267250A1
(fr)
|
2020-12-22 |
2023-11-01 |
Qilu Regor Therapeutics Inc. |
Inhibiteurs de sos1 et utilisations associées
|
EP4267554A1
(fr)
|
2020-12-22 |
2023-11-01 |
Mekanistic Therapeutics LLC |
Composés d'hétéroaryle d'aminobenzyle substitués utilisés en tant qu'inhibiteurs d'egfr et/ou de pi3k
|
BR112023021111A2
(pt)
|
2021-04-13 |
2023-12-19 |
Nuvalent Inc |
Composto, composição farmacêutica, método de tratamento de câncer, método para inibir seletivamente her2, método de regulação de um nível de her2, método para aumentar um nível de her2, método de diminuição da fosforilação de her2
|
EP4334324A1
(fr)
|
2021-05-05 |
2024-03-13 |
Revolution Medicines, Inc. |
Inhibiteurs de ras covalents et leurs utilisations
|
IL308195A
(en)
|
2021-05-05 |
2024-01-01 |
Revolution Medicines Inc |
RAS inhibitors for cancer treatment
|
CN118234731A
(zh)
|
2021-05-05 |
2024-06-21 |
锐新医药公司 |
Ras抑制剂
|
AR127308A1
(es)
|
2021-10-08 |
2024-01-10 |
Revolution Medicines Inc |
Inhibidores ras
|
TW202340214A
(zh)
|
2021-12-17 |
2023-10-16 |
美商健臻公司 |
做為shp2抑制劑之吡唑并吡𠯤化合物
|
EP4227307A1
(fr)
|
2022-02-11 |
2023-08-16 |
Genzyme Corporation |
Composés pyrazolopyrazine en tant qu'inhibiteurs de shp2
|
WO2023172940A1
(fr)
|
2022-03-08 |
2023-09-14 |
Revolution Medicines, Inc. |
Méthodes de traitement du cancer du poumon réfractaire immunitaire
|
WO2023240263A1
(fr)
|
2022-06-10 |
2023-12-14 |
Revolution Medicines, Inc. |
Inhibiteurs de ras macrocycliques
|
WO2024081916A1
(fr)
|
2022-10-14 |
2024-04-18 |
Black Diamond Therapeutics, Inc. |
Méthodes de traitement de cancers à l'aide de dérivés d'isoquinoline ou de 6-aza-quinoléine
|