LU91017I2 - Cialis-tadalafil et les sels et solvates physiologiquement acceptables de celui-ci - Google Patents

Cialis-tadalafil et les sels et solvates physiologiquement acceptables de celui-ci

Info

Publication number
LU91017I2
LU91017I2 LU91017C LU91017C LU91017I2 LU 91017 I2 LU91017 I2 LU 91017I2 LU 91017 C LU91017 C LU 91017C LU 91017 C LU91017 C LU 91017C LU 91017 I2 LU91017 I2 LU 91017I2
Authority
LU
Luxembourg
Prior art keywords
3alkyl
alkyl
represents hydrogen
ring
solvates
Prior art date
Application number
LU91017C
Other languages
English (en)
French (fr)
Original Assignee
Icos Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10749089&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=LU91017(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Icos Corp filed Critical Icos Corp
Publication of LU91017I2 publication Critical patent/LU91017I2/fr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12—Antidiarrhoeals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/14—Decongestants or antiallergics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/16—Otologicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Immunology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Indole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
LU91017C 1994-01-21 2003-03-26 Cialis-tadalafil et les sels et solvates physiologiquement acceptables de celui-ci LU91017I2 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB9401090A GB9401090D0 (en) 1994-01-21 1994-01-21 Chemical compounds
PCT/EP1995/000183 WO1995019978A1 (en) 1994-01-21 1995-01-19 Tetracyclic derivatives, process of preparation and use

Publications (1)

Publication Number Publication Date
LU91017I2 true LU91017I2 (fr) 2003-05-26

Family

ID=10749089

Family Applications (1)

Application Number Title Priority Date Filing Date
LU91017C LU91017I2 (fr) 1994-01-21 2003-03-26 Cialis-tadalafil et les sels et solvates physiologiquement acceptables de celui-ci

Country Status (48)

Country Link
US (5) US5859006A (OSRAM)
EP (1) EP0740668B1 (OSRAM)
JP (3) JP3808095B2 (OSRAM)
KR (1) KR100357411B1 (OSRAM)
CN (2) CN1045777C (OSRAM)
AP (1) AP556A (OSRAM)
AT (1) ATE169018T1 (OSRAM)
AU (2) AU689205B2 (OSRAM)
BG (1) BG62733B1 (OSRAM)
BR (1) BR9506559C8 (OSRAM)
CA (1) CA2181377C (OSRAM)
CO (1) CO4340684A1 (OSRAM)
CZ (1) CZ286566B6 (OSRAM)
DE (2) DE69503753T2 (OSRAM)
DK (1) DK0740668T3 (OSRAM)
EE (1) EE03231B1 (OSRAM)
EG (1) EG25852A (OSRAM)
ES (1) ES2122543T3 (OSRAM)
FI (1) FI113176B (OSRAM)
GB (1) GB9401090D0 (OSRAM)
HR (1) HRP950023B1 (OSRAM)
HU (1) HU222494B1 (OSRAM)
IL (1) IL112384A (OSRAM)
IN (1) IN183942B (OSRAM)
IS (1) IS1888B (OSRAM)
LU (1) LU91017I2 (OSRAM)
LV (1) LV11690B (OSRAM)
MA (1) MA23433A1 (OSRAM)
MX (1) MX9602904A (OSRAM)
MY (1) MY114663A (OSRAM)
NL (1) NL300124I2 (OSRAM)
NO (2) NO306465B1 (OSRAM)
NZ (1) NZ279199A (OSRAM)
OA (1) OA10584A (OSRAM)
PE (1) PE49495A1 (OSRAM)
PL (1) PL179744B1 (OSRAM)
RO (1) RO117794B1 (OSRAM)
RU (1) RU2142463C1 (OSRAM)
SA (1) SA95150475B1 (OSRAM)
SG (1) SG49184A1 (OSRAM)
SI (1) SI0740668T1 (OSRAM)
SK (1) SK280879B6 (OSRAM)
SV (1) SV1995000002A (OSRAM)
TN (1) TNSN95004A1 (OSRAM)
TW (1) TW378210B (OSRAM)
UY (1) UY23893A1 (OSRAM)
WO (1) WO1995019978A1 (OSRAM)
ZA (1) ZA95424B (OSRAM)

Families Citing this family (219)

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US6060477A (en) 1995-06-07 2000-05-09 Cell Pathways, Inc. Method of treating a patient having precancerous lesions with phenyl cycloamino pyrimidinone derivatives
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SG49184A1 (en) 1998-05-18
CN1224720A (zh) 1999-08-04
LV11690B (en) 1997-06-20
CA2181377C (en) 2002-05-28
US6127542A (en) 2000-10-03
EG25852A (en) 2012-09-10
CN1070492C (zh) 2001-09-05
IL112384A0 (en) 1995-03-30
JP2009102386A (ja) 2009-05-14
DE10399006I2 (de) 2004-05-06
BR9506559A (pt) 1997-10-28
US6025494A (en) 2000-02-15
AU7391298A (en) 1998-08-20
JP3808095B2 (ja) 2006-08-09
ATE169018T1 (de) 1998-08-15
IS1888B (is) 2003-09-01
SK94096A3 (en) 1997-04-09
CN1143963A (zh) 1997-02-26
CZ286566B6 (cs) 2000-05-17
DE69503753D1 (de) 1998-09-03
HUT74943A (en) 1997-03-28
LV11690A (lv) 1997-02-20
IL112384A (en) 1998-08-16
JPH09508113A (ja) 1997-08-19
ZA95424B (en) 1995-09-27
FI113176B (fi) 2004-03-15
TNSN95004A1 (fr) 1996-02-06
CO4340684A1 (es) 1996-07-30
MA23433A1 (fr) 1995-10-01
NL300124I1 (nl) 2003-07-01
EE03231B1 (et) 1999-10-15
FI962927A0 (fi) 1996-07-19
SA95150475B1 (ar) 2005-07-31
SV1995000002A (es) 1995-10-04
NO2003002I2 (no) 2005-03-21
HU9601982D0 (en) 1996-09-30
NO963015D0 (no) 1996-07-19
SK280879B6 (sk) 2000-08-14
PL315559A1 (en) 1996-11-12
BG62733B1 (bg) 2000-06-30
MX9602904A (es) 1997-12-31
DE10399006I1 (de) 2003-07-31
BG100727A (bg) 1997-02-28
OA10584A (en) 2002-08-26
TW378210B (en) 2000-01-01
DE69503753T2 (de) 1999-01-21
IN183942B (OSRAM) 2000-05-20
NO306465B1 (no) 1999-11-08
NO2003002I1 (no) 2003-01-22
CA2181377A1 (en) 1995-07-27
AP9500712A0 (en) 1995-01-31
GB9401090D0 (en) 1994-03-16
FI962927A7 (fi) 1996-07-19
US6369059B1 (en) 2002-04-09
IS4252A (is) 1995-07-22
HRP950023A2 (en) 1998-04-30
SI0740668T1 (en) 1999-02-28
MY114663A (en) 2002-12-31
AU707055B2 (en) 1999-07-01
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US20020119976A1 (en) 2002-08-29
NZ279199A (en) 1998-01-26

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