KR20220103810A - Jak1 억제제용 지속 방출 복용 형태 - Google Patents

Jak1 억제제용 지속 방출 복용 형태 Download PDF

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Publication number
KR20220103810A
KR20220103810A KR1020227023370A KR20227023370A KR20220103810A KR 20220103810 A KR20220103810 A KR 20220103810A KR 1020227023370 A KR1020227023370 A KR 1020227023370A KR 20227023370 A KR20227023370 A KR 20227023370A KR 20220103810 A KR20220103810 A KR 20220103810A
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South Korea
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sustained release
dosage forms
fluoro
acetonitrile
pyrrolo
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KR1020227023370A
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Korean (ko)
Inventor
크리쉬나스와미 옐레스와람
바브니쉬 파리크
딜립 피. 모디
트럽티 셰트
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인사이트 코포레이션
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Dermatology (AREA)
  • Neurology (AREA)
  • Hematology (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Endocrinology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Inorganic Chemistry (AREA)
  • Transplantation (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Oncology (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
KR1020227023370A 2013-08-07 2014-08-06 Jak1 억제제용 지속 방출 복용 형태 Ceased KR20220103810A (ko)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US201361863325P 2013-08-07 2013-08-07
US61/863,325 2013-08-07
US201361913066P 2013-12-06 2013-12-06
US61/913,066 2013-12-06
KR1020217018433A KR102419714B1 (ko) 2013-08-07 2014-08-06 Jak1 억제제용 지속 방출 복용 형태
PCT/US2014/049940 WO2015021153A1 (en) 2013-08-07 2014-08-06 Sustained release dosage forms for a jak1 inhibitor

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
KR1020217018433A Division KR102419714B1 (ko) 2013-08-07 2014-08-06 Jak1 억제제용 지속 방출 복용 형태

Publications (1)

Publication Number Publication Date
KR20220103810A true KR20220103810A (ko) 2022-07-22

Family

ID=51383933

Family Applications (3)

Application Number Title Priority Date Filing Date
KR1020227023370A Ceased KR20220103810A (ko) 2013-08-07 2014-08-06 Jak1 억제제용 지속 방출 복용 형태
KR1020167006096A Ceased KR20160045081A (ko) 2013-08-07 2014-08-06 Jak1 억제제용 지속 방출 복용 형태
KR1020217018433A Active KR102419714B1 (ko) 2013-08-07 2014-08-06 Jak1 억제제용 지속 방출 복용 형태

Family Applications After (2)

Application Number Title Priority Date Filing Date
KR1020167006096A Ceased KR20160045081A (ko) 2013-08-07 2014-08-06 Jak1 억제제용 지속 방출 복용 형태
KR1020217018433A Active KR102419714B1 (ko) 2013-08-07 2014-08-06 Jak1 억제제용 지속 방출 복용 형태

Country Status (31)

Country Link
US (5) US9655854B2 (https=)
EP (2) EP3721873A1 (https=)
JP (6) JP6334700B2 (https=)
KR (3) KR20220103810A (https=)
CN (3) CN116036089A (https=)
AU (3) AU2014305989B2 (https=)
BR (1) BR122020001831A8 (https=)
CA (2) CA3155500A1 (https=)
CL (1) CL2016000292A1 (https=)
CR (3) CR20230316A (https=)
CY (1) CY1123314T1 (https=)
DK (1) DK3030227T3 (https=)
EA (1) EA201690357A1 (https=)
ES (1) ES2792549T3 (https=)
HR (1) HRP20200955T1 (https=)
HU (1) HUE049345T2 (https=)
IL (2) IL277554B2 (https=)
LT (1) LT3030227T (https=)
MX (2) MX376856B (https=)
MY (2) MY203694A (https=)
PE (2) PE20160223A1 (https=)
PH (3) PH12019502074B1 (https=)
PL (1) PL3030227T3 (https=)
PT (1) PT3030227T (https=)
RS (1) RS60469B1 (https=)
SG (3) SG10201801069QA (https=)
SI (1) SI3030227T1 (https=)
SM (1) SMT202000315T1 (https=)
TW (3) TWI730935B (https=)
UA (1) UA120499C2 (https=)
WO (1) WO2015021153A1 (https=)

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