JP2018534296A5 - - Google Patents

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Publication number
JP2018534296A5
JP2018534296A5 JP2018521907A JP2018521907A JP2018534296A5 JP 2018534296 A5 JP2018534296 A5 JP 2018534296A5 JP 2018521907 A JP2018521907 A JP 2018521907A JP 2018521907 A JP2018521907 A JP 2018521907A JP 2018534296 A5 JP2018534296 A5 JP 2018534296A5
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JP
Japan
Prior art keywords
pyrrolidin
heptaen
fluoro
carboxamide
mutation
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Pending
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JP2018521907A
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English (en)
Japanese (ja)
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JP2018534296A (ja
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Priority claimed from PCT/US2016/058951 external-priority patent/WO2017075107A1/en
Publication of JP2018534296A publication Critical patent/JP2018534296A/ja
Publication of JP2018534296A5 publication Critical patent/JP2018534296A5/ja
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JP2018521907A 2015-10-26 2016-10-26 Ｔｒｋ阻害薬耐性がんにおける点変異およびそれに関連する方法 Pending JP2018534296A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201562246580P 2015-10-26 2015-10-26
US62/246,580 2015-10-26
US201662287778P 2016-01-27 2016-01-27
US62/287,778 2016-01-27
US201662323586P 2016-04-15 2016-04-15
US62/323,586 2016-04-15
PCT/US2016/058951 WO2017075107A1 (en) 2015-10-26 2016-10-26 Point mutations in trk inhibitor-resistant cancer and methods relating to the same

Publications (2)

Publication Number Publication Date
JP2018534296A JP2018534296A (ja) 2018-11-22
JP2018534296A5 true JP2018534296A5 (enExample) 2019-12-26

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JP2018521907A Pending JP2018534296A (ja) 2015-10-26 2016-10-26 Ｔｒｋ阻害薬耐性がんにおける点変異およびそれに関連する方法

Country Status (17)

Country Link
US (6) US10724102B2 (enExample)
EP (1) EP3368039A1 (enExample)
JP (1) JP2018534296A (enExample)
KR (1) KR20180102544A (enExample)
CN (1) CN108697708A (enExample)
AU (1) AU2016344058A1 (enExample)
BR (1) BR112018008357A2 (enExample)
CA (1) CA3003153A1 (enExample)
CL (1) CL2018001110A1 (enExample)
IL (1) IL258877A (enExample)
MX (1) MX2018005087A (enExample)
PH (1) PH12018500902A1 (enExample)
RU (1) RU2744852C2 (enExample)
SG (1) SG11201803438XA (enExample)
SV (1) SV2018005677A (enExample)
TN (2) TN2019000271A1 (enExample)
WO (1) WO2017075107A1 (enExample)

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