IN2015DN01132A - - Google Patents

Info

Publication number
IN2015DN01132A
IN2015DN01132A IN1132DEN2015A IN2015DN01132A IN 2015DN01132 A IN2015DN01132 A IN 2015DN01132A IN 1132DEN2015 A IN1132DEN2015 A IN 1132DEN2015A IN 2015DN01132 A IN2015DN01132 A IN 2015DN01132A
Authority
IN
India
Prior art keywords
group
methyl
quinazolinylmethyl
denotes
quinolinylmethyl
Prior art date
Application number
Other languages
English (en)
Inventor
Frank Himmelsbach
Elke Langkopf
Matthias Eckhardt
Michael Mark
Roland Maier
Ralf R H Lotz
Mohammad Tadayyon
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=31947613&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IN2015DN01132(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from DE10238243A external-priority patent/DE10238243A1/de
Priority claimed from DE10312353A external-priority patent/DE10312353A1/de
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Publication of IN2015DN01132A publication Critical patent/IN2015DN01132A/en

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
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    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/286Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02Inorganic compounds
    • AHUMAN NECESSITIES
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    • A61K9/0087Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • AHUMAN NECESSITIES
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    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
    • C07D473/06Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
    • C07D473/06Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
    • C07D473/12Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3 with methyl radicals in positions 1, 3, and 7, e.g. caffeine

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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
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  • Diabetes (AREA)
  • Hematology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Epidemiology (AREA)
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  • Oncology (AREA)
  • Reproductive Health (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Communicable Diseases (AREA)
  • Pain & Pain Management (AREA)
  • Virology (AREA)
  • Urology & Nephrology (AREA)
  • Molecular Biology (AREA)
  • Dermatology (AREA)
  • Cardiology (AREA)
  • Emergency Medicine (AREA)
  • Psychiatry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
IN1132DEN2015 2002-08-21 2013-08-18 IN2015DN01132A (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE10238243A DE10238243A1 (de) 2002-08-21 2002-08-21 8-[3-Amino-piperidin-1-yl]-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
DE10312353A DE10312353A1 (de) 2003-03-20 2003-03-20 8-[3-Amino-piperidin-1-yl]-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
PCT/EP2003/009127 WO2004018468A2 (fr) 2002-08-21 2003-08-18 8-[3-amino-piperidin-1-yl]-xanthines, leur production et leur utilisation comme medicament

Publications (1)

Publication Number Publication Date
IN2015DN01132A true IN2015DN01132A (fr) 2015-06-26

Family

ID=31947613

Family Applications (2)

Application Number Title Priority Date Filing Date
IN1133DEN2015 IN2015DN01133A (fr) 2002-08-21 2013-08-18
IN1132DEN2015 IN2015DN01132A (fr) 2002-08-21 2013-08-18

Family Applications Before (1)

Application Number Title Priority Date Filing Date
IN1133DEN2015 IN2015DN01133A (fr) 2002-08-21 2013-08-18

Country Status (38)

Country Link
EP (6) EP2308878A3 (fr)
JP (6) JP4233524B2 (fr)
KR (2) KR101111101B1 (fr)
CN (4) CN107674077A (fr)
AR (3) AR041025A1 (fr)
AT (1) ATE453644T1 (fr)
AU (2) AU2003253418B2 (fr)
BE (1) BE2011C038I2 (fr)
BR (2) BRPI0313648B8 (fr)
CA (1) CA2496249C (fr)
CY (3) CY1109928T1 (fr)
DE (2) DE50312295D1 (fr)
DK (1) DK1532149T3 (fr)
EA (3) EA024251B1 (fr)
EC (2) ECSP055617A (fr)
EG (1) EG25011A (fr)
ES (1) ES2339112T3 (fr)
FR (1) FR11C0052I2 (fr)
HK (6) HK1081552A1 (fr)
HR (2) HRP20050157B1 (fr)
HU (1) HUS1100028I1 (fr)
IL (1) IL166964A (fr)
IN (2) IN2015DN01133A (fr)
LU (2) LU91889I2 (fr)
ME (1) ME00396B (fr)
MX (1) MXPA05001684A (fr)
MY (2) MY137619A (fr)
NO (4) NO333970B1 (fr)
PE (1) PE20040897A1 (fr)
PL (2) PL403104A1 (fr)
PT (1) PT1532149E (fr)
RS (2) RS20120139A3 (fr)
SA (1) SA03240448B1 (fr)
SI (1) SI1532149T1 (fr)
TW (3) TWI319320B (fr)
UA (1) UA84275C2 (fr)
UY (1) UY27946A1 (fr)
WO (1) WO2004018468A2 (fr)

Families Citing this family (175)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2270047T3 (es) * 2002-05-31 2007-04-01 Schering Corporation Proceso para preparar inhibidores de la fosfodiesterasa v de xantina y sus precursores.
GB0215293D0 (en) 2002-07-03 2002-08-14 Rega Foundation Viral inhibitors
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