HK1134076A1 - - Google Patents

Info

Publication number
HK1134076A1
HK1134076A1 HK10100903.4A HK10100903A HK1134076A1 HK 1134076 A1 HK1134076 A1 HK 1134076A1 HK 10100903 A HK10100903 A HK 10100903A HK 1134076 A1 HK1134076 A1 HK 1134076A1
Authority
HK
Hong Kong
Application number
HK10100903.4A
Inventor
Frank Himmelsbach
Elke Langkopf
Matthias Eckhardt
Michael Mark
Roland Maier
Ralf Richard Hermann Lotz
Mohammad Tadayyon
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=31947613&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1134076(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from DE10238243A external-priority patent/DE10238243A1/de
Priority claimed from DE10312353A external-priority patent/DE10312353A1/de
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Publication of HK1134076A1 publication Critical patent/HK1134076A1/xx

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
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    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
    • C07D473/06—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
    • C07D473/12—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3 with methyl radicals in positions 1, 3, and 7, e.g. caffeine
HK10100903.4A 2002-08-21 2010-01-28 HK1134076A1 (xx)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10238243A DE10238243A1 (de) 2002-08-21 2002-08-21 8-[3-Amino-piperidin-1-yl]-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
DE10312353A DE10312353A1 (de) 2003-03-20 2003-03-20 8-[3-Amino-piperidin-1-yl]-xanthine, deren Herstellung und deren Verwendung als Arzneimittel

Publications (1)

Publication Number Publication Date
HK1134076A1 true HK1134076A1 (xx) 2010-04-16

Family

ID=31947613

Family Applications (6)

Application Number Title Priority Date Filing Date
HK06101985.9A HK1081552A1 (en) 2002-08-21 2006-02-16 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments
HK10100903.4A HK1134076A1 (xx) 2002-08-21 2010-01-28
HK10100904.3A HK1134077A1 (en) 2002-08-21 2010-01-28 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments 8-[3---1-]-
HK13110418.8A HK1183028A1 (zh) 2002-08-21 2013-09-09 -氨基-哌啶- -基 -黃嘌呤化合物，其製備方法及作為藥物製劑的用途
HK16103474.1A HK1215439A1 (zh) 2002-08-21 2016-03-24 -氨基-哌啶- -基 -黃嘌呤化合物，其製備方法及作為藥物製劑的用途
HK18109982.1A HK1250708A1 (zh) 2002-08-21 2018-08-02 8-[3-氨基-呱啶-1-基]-黃嘌呤化合物，其製備方法及作為藥物製劑的用途

Family Applications Before (1)

Application Number Title Priority Date Filing Date
HK06101985.9A HK1081552A1 (en) 2002-08-21 2006-02-16 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments

Family Applications After (4)

Application Number Title Priority Date Filing Date
HK10100904.3A HK1134077A1 (en) 2002-08-21 2010-01-28 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments 8-[3---1-]-
HK13110418.8A HK1183028A1 (zh) 2002-08-21 2013-09-09 -氨基-哌啶- -基 -黃嘌呤化合物，其製備方法及作為藥物製劑的用途
HK16103474.1A HK1215439A1 (zh) 2002-08-21 2016-03-24 -氨基-哌啶- -基 -黃嘌呤化合物，其製備方法及作為藥物製劑的用途
HK18109982.1A HK1250708A1 (zh) 2002-08-21 2018-08-02 8-[3-氨基-呱啶-1-基]-黃嘌呤化合物，其製備方法及作為藥物製劑的用途

Country Status (38)

Country Link
EP (6) EP2058311A3 (xx)
JP (6) JP4233524B2 (xx)
KR (2) KR101111101B1 (xx)
CN (4) CN100522962C (xx)
AR (3) AR041025A1 (xx)
AT (1) ATE453644T1 (xx)
AU (2) AU2003253418B2 (xx)
BE (1) BE2011C038I2 (xx)
BR (2) BRPI0313648B8 (xx)
CA (1) CA2496249C (xx)
CY (3) CY1109928T1 (xx)
DE (2) DE50312295D1 (xx)
DK (1) DK1532149T3 (xx)
EA (3) EA016166B1 (xx)
EC (2) ECSP055617A (xx)
EG (1) EG25011A (xx)
ES (1) ES2339112T3 (xx)
FR (1) FR11C0052I2 (xx)
HK (6) HK1081552A1 (xx)
HR (2) HRP20050157B1 (xx)
HU (1) HUS1100028I1 (xx)
IL (1) IL166964A (xx)
IN (2) IN2015DN01133A (xx)
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